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MX9707453A - Derivados de quinazolina. - Google Patents

Derivados de quinazolina.

Info

Publication number
MX9707453A
MX9707453A MX9707453A MX9707453A MX9707453A MX 9707453 A MX9707453 A MX 9707453A MX 9707453 A MX9707453 A MX 9707453A MX 9707453 A MX9707453 A MX 9707453A MX 9707453 A MX9707453 A MX 9707453A
Authority
MX
Mexico
Prior art keywords
quinazoline derivatives
formula
produgs
pharmaceutically acceptable
acceptable salts
Prior art date
Application number
MX9707453A
Other languages
English (en)
Inventor
Rodney C Schnur
Lee D Arnold
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23636708&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX9707453(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of MX9707453A publication Critical patent/MX9707453A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Esta invencion se refiere a ciertos derivados de 4-(fenilamino substituido)quinazolina de la formula: (I) sus profarmacos y sales farmacéuticas aceptables en la que R1, R2, R3, R4, m y n se describen más adelante; los compuestos de la formula I, sus profármacos y sales farmaceuticamente aceptables son utiles para el tratamiento de enfermedades hiperproliferativas.
MX9707453A 1995-03-30 1995-06-06 Derivados de quinazolina. MX9707453A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US41330095A 1995-03-30 1995-03-30
PCT/IB1995/000436 WO1996030347A1 (en) 1995-03-30 1995-06-06 Quinazoline derivatives

Publications (1)

Publication Number Publication Date
MX9707453A true MX9707453A (es) 1997-12-31

Family

ID=23636708

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9707453A MX9707453A (es) 1995-03-30 1995-06-06 Derivados de quinazolina.

Country Status (44)

Country Link
EP (5) EP1110953B1 (es)
JP (1) JP3088018B2 (es)
KR (1) KR100232335B1 (es)
CN (1) CN1066142C (es)
AP (1) AP735A (es)
AR (1) AR002723A1 (es)
AT (2) ATE205483T1 (es)
AU (2) AU703638B2 (es)
BR (1) BR9601200B1 (es)
CA (1) CA2216796C (es)
CO (1) CO4410333A1 (es)
CZ (2) CZ294967B6 (es)
DE (3) DE69536015D1 (es)
DK (1) DK0817775T3 (es)
EG (1) EG24229A (es)
ES (2) ES2332984T3 (es)
FI (1) FI120646B (es)
FR (1) FR06C0010I2 (es)
GR (1) GR3037070T3 (es)
HK (1) HK1038740A1 (es)
HR (1) HRP960147B1 (es)
HU (2) HU229120B1 (es)
IL (7) IL129995A (es)
LU (1) LU91209I2 (es)
MA (1) MA23831A1 (es)
MX (1) MX9707453A (es)
MY (1) MY117896A (es)
NL (1) NL300214I2 (es)
NO (2) NO308740B1 (es)
NZ (1) NZ286263A (es)
OA (1) OA10277A (es)
PE (1) PE43897A1 (es)
PL (1) PL186843B1 (es)
PT (1) PT817775E (es)
RU (2) RU2694252C2 (es)
SA (1) SA96160707B1 (es)
SG (1) SG43262A1 (es)
SI (1) SI9600102A (es)
SK (2) SK283762B6 (es)
TR (1) TR199600265A1 (es)
TW (1) TW454000B (es)
UA (1) UA44254C2 (es)
WO (1) WO1996030347A1 (es)
ZA (1) ZA962522B (es)

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