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HK1172549A1 - Dpp iv inhibitor formulations iv - Google Patents

Dpp iv inhibitor formulations iv

Info

Publication number
HK1172549A1
HK1172549A1 HK12113310.2A HK12113310A HK1172549A1 HK 1172549 A1 HK1172549 A1 HK 1172549A1 HK 12113310 A HK12113310 A HK 12113310A HK 1172549 A1 HK1172549 A1 HK 1172549A1
Authority
HK
Hong Kong
Prior art keywords
dpp
inhibitor formulations
formulations
inhibitor
Prior art date
Application number
HK12113310.2A
Other languages
English (en)
Chinese (zh)
Inventor
安賈．科爾勞希
帕特里克．羅默
格爾德．塞費爾特
Original Assignee
勃林格殷格翰國際有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36972901&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1172549(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 勃林格殷格翰國際有限公司 filed Critical 勃林格殷格翰國際有限公司
Publication of HK1172549A1 publication Critical patent/HK1172549A1/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
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    • A61K9/2833—Organic macromolecular compounds
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    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Inorganic Chemistry (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Child & Adolescent Psychology (AREA)
  • Transplantation (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
HK12113310.2A 2006-05-04 2009-11-13 Dpp iv inhibitor formulations iv HK1172549A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP06009201A EP1852108A1 (en) 2006-05-04 2006-05-04 DPP IV inhibitor formulations

Publications (1)

Publication Number Publication Date
HK1172549A1 true HK1172549A1 (en) 2013-04-26

Family

ID=36972901

Family Applications (2)

Application Number Title Priority Date Filing Date
HK09110601.1A HK1130442A1 (en) 2006-05-04 2009-11-13 Dpp iv inhibitor formulations
HK12113310.2A HK1172549A1 (en) 2006-05-04 2009-11-13 Dpp iv inhibitor formulations iv

Family Applications Before (1)

Application Number Title Priority Date Filing Date
HK09110601.1A HK1130442A1 (en) 2006-05-04 2009-11-13 Dpp iv inhibitor formulations

Country Status (37)

Country Link
US (9) US20080107731A1 (pt)
EP (5) EP1852108A1 (pt)
JP (8) JP5478244B2 (pt)
KR (5) KR20140063896A (pt)
CN (2) CN101437493B (pt)
AR (2) AR060755A1 (pt)
AT (1) ATE480228T1 (pt)
AU (1) AU2007247193B2 (pt)
BR (2) BRPI0722388B1 (pt)
CA (1) CA2649922C (pt)
CL (2) CL2012002522A1 (pt)
CY (2) CY1111354T1 (pt)
DE (1) DE602007009091D1 (pt)
DK (3) DK2283819T3 (pt)
EA (2) EA029890B1 (pt)
EC (1) ECSP088800A (pt)
ES (3) ES2348576T3 (pt)
HK (2) HK1130442A1 (pt)
HR (2) HRP20100507T1 (pt)
HU (1) HUE025210T2 (pt)
IL (2) IL195030A (pt)
ME (2) ME01170B (pt)
MX (2) MX358617B (pt)
MY (2) MY146969A (pt)
NO (1) NO343067B1 (pt)
NZ (3) NZ572862A (pt)
PE (2) PE20110666A1 (pt)
PL (3) PL2277509T3 (pt)
PT (2) PT2023902E (pt)
RS (2) RS51466B (pt)
SG (1) SG171649A1 (pt)
SI (2) SI2283819T1 (pt)
TW (2) TWI474843B (pt)
UA (1) UA94942C2 (pt)
UY (1) UY30319A1 (pt)
WO (1) WO2007128724A1 (pt)
ZA (1) ZA200808361B (pt)

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US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US7495005B2 (en) * 2002-08-22 2009-02-24 Boehringer Ingelheim Pharma Gmbh & Co. Kg Xanthine derivatives, their preparation and their use in pharmaceutical compositions
US7482337B2 (en) * 2002-11-08 2009-01-27 Boehringer Ingelheim Pharma Gmbh & Co. Kg Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions
US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
US7439370B2 (en) 2004-05-10 2008-10-21 Boehringer Ingelheim International Gmbh Imidazole derivatives, their preparation and their use as intermediates for the preparation of pharmaceutical compositions and pesticides
DE102004030502A1 (de) 2004-06-24 2006-01-12 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Imidazole und Triazole, deren Herstellung und Verwendung als Arzneimittel
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
US7772191B2 (en) 2005-05-10 2010-08-10 Boehringer Ingelheim International Gmbh Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
BRPI0711558A2 (pt) * 2006-05-04 2011-11-08 Boeringer Ingelheim Internat Gmbh polimorfos
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
MX2008015489A (es) 2006-06-06 2009-01-13 Intra Cellular Therapies Inc Compuestos organicos.
JP2010500326A (ja) 2006-08-08 2010-01-07 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 糖尿病の治療のためのｄｐｐ−ｉｖ阻害剤としてのピロロ［３，２−ｄ］ピリミジン
EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
CL2008002427A1 (es) 2007-08-16 2009-09-11 Boehringer Ingelheim Int Composicion farmaceutica que comprende 1-cloro-4-(b-d-glucopiranos-1-il)-2-[4-((s)-tetrahidrofurano-3-iloxi)bencil]-benceno combinado con 1-[(4-metilquinazolin-2-il)metil]-3-metil-7-(2-butin-1-il)-8-(3-(r)-aminopiperidin-1-il)xantina; y su uso para tratar diabetes mellitus tipo 2.
MX2010006208A (es) 2007-12-06 2010-12-21 Intra Cellular Therapies Inc Compuestos organicos.
PE20091730A1 (es) 2008-04-03 2009-12-10 Boehringer Ingelheim Int Formulaciones que comprenden un inhibidor de dpp4
KR20190016601A (ko) 2008-08-06 2019-02-18 베링거 인겔하임 인터내셔날 게엠베하 메트포르민 요법이 부적합한 환자에서의 당뇨병 치료
UY32030A (es) 2008-08-06 2010-03-26 Boehringer Ingelheim Int "tratamiento para diabetes en pacientes inapropiados para terapia con metformina"
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AU2007247193A1 (en) 2007-11-15
KR20160128446A (ko) 2016-11-07
IL212841A0 (en) 2011-07-31
EA029890B1 (ru) 2018-05-31
US20210260068A1 (en) 2021-08-26
US20170312287A1 (en) 2017-11-02
IL195030A0 (en) 2009-08-03
JP2016104811A (ja) 2016-06-09
JP2020079316A (ja) 2020-05-28
EA200802184A1 (ru) 2009-06-30
KR101855323B1 (ko) 2018-05-09
JP6564720B2 (ja) 2019-08-21
ES2538818T3 (es) 2015-06-24
CN101437493A (zh) 2009-05-20
CN102526737A (zh) 2012-07-04
JP6100998B2 (ja) 2017-03-22
CA2649922A1 (en) 2007-11-15
EA016559B1 (ru) 2012-05-30
SI2283819T1 (sl) 2015-01-30
ES2527409T3 (es) 2015-01-23
JP2013227338A (ja) 2013-11-07
HRP20150003T1 (xx) 2015-03-13
HUE025210T2 (en) 2016-03-29
RS51466B (en) 2011-04-30
PL2283819T3 (pl) 2015-03-31
KR101710881B1 (ko) 2017-02-28
CN102526737B (zh) 2015-02-25
KR20140063896A (ko) 2014-05-27
ME01170B (me) 2013-03-20
CL2012002522A1 (es) 2012-12-21
US20190209571A1 (en) 2019-07-11

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