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DK1137635T3 - N-substituerede 2-cyanopyrrolidiner - Google Patents

N-substituerede 2-cyanopyrrolidiner

Info

Publication number
DK1137635T3
DK1137635T3 DK99959396T DK99959396T DK1137635T3 DK 1137635 T3 DK1137635 T3 DK 1137635T3 DK 99959396 T DK99959396 T DK 99959396T DK 99959396 T DK99959396 T DK 99959396T DK 1137635 T3 DK1137635 T3 DK 1137635T3
Authority
DK
Denmark
Prior art keywords
cyanopyrrolidines
substituted
Prior art date
Application number
DK99959396T
Other languages
English (en)
Inventor
Edwin Bernard Villhauer
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22777194&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1137635(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Application granted granted Critical
Publication of DK1137635T3 publication Critical patent/DK1137635T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
DK99959396T 1998-12-10 1999-12-09 N-substituerede 2-cyanopyrrolidiner DK1137635T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US20906898A 1998-12-10 1998-12-10

Publications (1)

Publication Number Publication Date
DK1137635T3 true DK1137635T3 (da) 2006-02-13

Family

ID=22777194

Family Applications (1)

Application Number Title Priority Date Filing Date
DK99959396T DK1137635T3 (da) 1998-12-10 1999-12-09 N-substituerede 2-cyanopyrrolidiner

Country Status (34)

Country Link
US (1) US6166063A (da)
EP (1) EP1137635B1 (da)
JP (2) JP3681110B2 (da)
KR (2) KR20050047561A (da)
CN (1) CN1160330C (da)
AR (1) AR023719A1 (da)
AT (1) ATE307112T1 (da)
BR (1) BRPI9915985B8 (da)
CA (1) CA2350609C (da)
CO (1) CO5150173A1 (da)
CY (3) CY1105355T1 (da)
CZ (1) CZ299151B6 (da)
DE (3) DE122008000017I1 (da)
DK (1) DK1137635T3 (da)
ES (1) ES2251847T3 (da)
FR (1) FR08C0005I2 (da)
HK (1) HK1040394B (da)
HU (1) HU226769B1 (da)
ID (1) ID28796A (da)
IL (2) IL143091A0 (da)
LU (2) LU91409I2 (da)
MY (1) MY123244A (da)
NL (2) NL300333I2 (da)
NO (3) NO318741B1 (da)
NZ (1) NZ511935A (da)
PE (1) PE20001317A1 (da)
PL (1) PL199443B1 (da)
RU (1) RU2251544C2 (da)
SK (1) SK286635B6 (da)
TR (1) TR200101478T2 (da)
TW (1) TW509674B (da)
UY (1) UY25843A1 (da)
WO (1) WO2000034241A1 (da)
ZA (1) ZA200104581B (da)

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* Cited by examiner, † Cited by third party
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