Cimetidine | Histamine H2 receptor | target |
Cimetidine | Cytochrome P450 1A2 | enzyme |
Cimetidine | Cytochrome P450 2D6 | enzyme |
Cimetidine | Cytochrome P450 2C19 | enzyme |
Cimetidine | Cytochrome P450 3A4 | enzyme |
Cimetidine | Cytochrome P450 3A5 | enzyme |
Cimetidine | P-glycoprotein 1 | transporter |
Cimetidine | Solute carrier family 22 member 2 | transporter |
Cimetidine | Solute carrier family 22 member 1 | transporter |
Cimetidine | Solute carrier family 22 member 3 | transporter |
Cimetidine | Solute carrier family 22 member 5 | transporter |
Cimetidine | Solute carrier family 22 member 6 | transporter |
Cimetidine | Solute carrier family 22 member 8 | transporter |
Cimetidine | Multidrug and toxin extrusion protein 1 | transporter |
Cimetidine | Solute carrier family 22 member 4 | transporter |
Cimetidine | Solute carrier family 22 member 11 | transporter |
Cimetidine | Solute carrier family 22 member 7 | transporter |
Cimetidine | Cytochrome P450 11B1, mitochondrial | enzyme |
Cimetidine | Cytochrome P450 2C8 | enzyme |
Cimetidine | Cytochrome P450 2C9 | enzyme |
Cimetidine | Cytochrome P450 2E1 | enzyme |
Cimetidine | Dimethylaniline monooxygenase [N-oxide-forming] 3 | enzyme |
Cimetidine | Dimethylaniline monooxygenase [N-oxide-forming] 1 | enzyme |
Cimetidine | Bile salt export pump | transporter |
Cimetidine | Multidrug and toxin extrusion protein 2 | transporter |
Cimetidine | Serum albumin | carrier |
Ranitidine | Histamine H2 receptor | target |
Ranitidine | Cytochrome P450 1A2 | enzyme |
Ranitidine | Cytochrome P450 2D6 | enzyme |
Ranitidine | Solute carrier family 22 member 1 | transporter |
Ranitidine | P-glycoprotein 1 | transporter |
Ranitidine | Solute carrier family 22 member 8 | transporter |
Ranitidine | Cytochrome P450 3A4 | enzyme |
Ranitidine | Acetylcholinesterase | target |
Ranitidine | Solute carrier family 22 member 2 | transporter |
Ranitidine | Acetylcholinesterase | enzyme |
Levofloxacin | DNA gyrase subunit A | target |
Levofloxacin | DNA topoisomerase 4 subunit A | target |
Levofloxacin | Solute carrier family 22 member 2 | transporter |
Levofloxacin | P-glycoprotein 1 | transporter |
Levofloxacin | Solute carrier family 22 member 4 | transporter |
Levofloxacin | Multidrug and toxin extrusion protein 1 | transporter |
Levofloxacin | Multidrug and toxin extrusion protein 2 | transporter |
Levofloxacin | Cytochrome P450 2C9 | enzyme |
Levofloxacin | Serum albumin | carrier |
Levofloxacin | Solute carrier organic anion transporter family member 4C1 | transporter |
Levofloxacin | Solute carrier family 22 member 1 | transporter |
Levofloxacin | Solute carrier organic anion transporter family member 1A2 | transporter |
Levofloxacin | DNA gyrase subunit A | target |
Levofloxacin | DNA gyrase subunit B | target |
Tafenoquine | Cytochrome P450 2D6 | enzyme |
Tafenoquine | Ferredoxin--NADP reductase, apicoplast | enzyme |
Tafenoquine | Solute carrier family 22 member 2 | transporter |
Tafenoquine | Multidrug and toxin extrusion protein 1 | transporter |
Tafenoquine | Multidrug and toxin extrusion protein 2 | transporter |
Propranolol | Beta-1 adrenergic receptor | target |
Propranolol | Beta-2 adrenergic receptor | target |
Propranolol | Beta-3 adrenergic receptor | target |
Propranolol | 5-hydroxytryptamine receptor 1A | target |
Propranolol | 5-hydroxytryptamine receptor 1B | target |
Propranolol | Cytochrome P450 1A2 | enzyme |
Propranolol | Cytochrome P450 2D6 | enzyme |
Propranolol | Alpha-1-acid glycoprotein 1 | carrier |
Propranolol | Cytochrome P450 2C19 | enzyme |
Propranolol | Cytochrome P450 3A4 | enzyme |
Propranolol | Cytochrome P450 3A5 | enzyme |
Propranolol | Cytochrome P450 3A7 | enzyme |
Propranolol | Solute carrier family 22 member 2 | transporter |
Propranolol | P-glycoprotein 1 | transporter |
Propranolol | Cytochrome P450 1A1 | enzyme |
Propranolol | Amine oxidase [flavin-containing] A | enzyme |
Propranolol | Serum albumin | carrier |
Oxprenolol | Beta-1 adrenergic receptor | target |
Oxprenolol | Beta-2 adrenergic receptor | target |
Oxprenolol | Solute carrier family 22 member 2 | transporter |
Oxprenolol | Cytochrome P450 2D6 | enzyme |
Oxprenolol | Beta-3 adrenergic receptor | target |
Metoprolol | Beta-1 adrenergic receptor | target |
Metoprolol | Cytochrome P450 2D6 | enzyme |
Metoprolol | Beta-2 adrenergic receptor | target |
Metoprolol | Solute carrier family 22 member 2 | transporter |
Metoprolol | Serum albumin | carrier |
Metoprolol | Cytochrome P450 3A4 | enzyme |
Metoprolol | Beta adrenergic receptor | target |
Quinine | Platelet glycoprotein IX | target |
Quinine | Intermediate conductance calcium-activated potassium channel protein 4 | target |
Quinine | Cytochrome P450 3A4 | enzyme |
Quinine | Cytochrome P450 3A5 | enzyme |
Quinine | Cytochrome P450 1A1 | enzyme |
Quinine | Cytochrome P450 2D6 | enzyme |
Quinine | Cytochrome P450 1A2 | enzyme |
Quinine | Cytochrome P450 2C8 | enzyme |
Quinine | Cytochrome P450 2C9 | enzyme |
Quinine | Cytochrome P450 2C19 | enzyme |
Quinine | Cytochrome P450 2E1 | enzyme |
Quinine | Cytochrome P450 3A7 | enzyme |
Quinine | Solute carrier family 22 member 2 | transporter |
Quinine | Solute carrier family 22 member 1 | transporter |
Quinine | Solute carrier family 22 member 5 | transporter |
Quinine | P-glycoprotein 1 | transporter |
Quinine | Solute carrier organic anion transporter family member 1A2 | transporter |
Quinine | Solute carrier family 22 member 4 | transporter |
Quinine | Fe(II)-protoporphyrin IX | target |
Quinine | Solute carrier organic anion transporter family member 1B1 | transporter |
Choline | Choline-phosphate cytidylyltransferase B | target |
Choline | Acetylcholinesterase | target |
Choline | Choline-phosphate cytidylyltransferase A | target |
Choline | Phospholipase D2 | target |
Choline | Cholinesterase | target |
Choline | Phospholipase D1 | target |
Choline | Phosphoethanolamine/phosphocholine phosphatase | target |
Choline | Solute carrier family 22 member 2 | transporter |
Choline | Solute carrier family 22 member 1 | transporter |
Choline | Solute carrier family 22 member 3 | transporter |
Choline | Solute carrier family 22 member 5 | transporter |
Choline | Solute carrier family 22 member 4 | transporter |
Choline | Choline/ethanolaminephosphotransferase 1 | enzyme |
Choline | Choline transporter-like protein 1 | transporter |
Choline | Choline transporter-like protein 4 | transporter |
Choline | Choline transporter-like protein 2 | transporter |
Choline | Choline transporter-like protein 3 | transporter |
Choline | Choline/ethanolamine kinase | enzyme |
Choline | Choline O-acetyltransferase | enzyme |
Choline | Choline kinase alpha | enzyme |
Choline | Choline dehydrogenase, mitochondrial | enzyme |
Choline | High affinity choline transporter 1 | transporter |
Choline | Neuronal acetylcholine receptor subunit alpha-7 | target |
Choline | Neuronal acetylcholine receptor subunit alpha-2 | target |
Dinoprostone | Prostaglandin E2 receptor EP2 subtype | target |
Dinoprostone | Prostaglandin E2 receptor EP1 subtype | target |
Dinoprostone | Prostaglandin E2 receptor EP4 subtype | target |
Dinoprostone | Prostaglandin E2 receptor EP3 subtype | target |
Dinoprostone | Solute carrier family 22 member 2 | transporter |
Dinoprostone | Multidrug resistance-associated protein 5 | transporter |
Dinoprostone | Solute carrier family 22 member 6 | transporter |
Dinoprostone | Solute carrier family 22 member 8 | transporter |
Dinoprostone | Solute carrier family 22 member 11 | transporter |
Dinoprostone | Solute carrier family 22 member 7 | transporter |
Dinoprostone | Multidrug resistance-associated protein 4 | transporter |
Dinoprostone | Solute carrier organic anion transporter family member 2B1 | transporter |
Dinoprostone | Solute carrier organic anion transporter family member 1A2 | transporter |
Dinoprostone | Organic solute transporter subunit alpha | transporter |
Dinoprostone | Organic solute transporter subunit beta | transporter |
Dinoprostone | Solute carrier organic anion transporter family member 2A1 | transporter |
Dinoprostone | Solute carrier organic anion transporter family member 4A1 | transporter |
Dinoprostone | Solute carrier organic anion transporter family member 1C1 | transporter |
Dinoprostone | Solute carrier organic anion transporter family member 3A1 | transporter |
Dinoprostone | Solute carrier organic anion transporter family member 1B1 | transporter |
Dinoprostone | Prostaglandin D2 receptor 2 | target |
Dinoprostone | Prostaglandin F2-alpha receptor | target |
Thiamine | Thiamin pyrophosphokinase 1 | target |
Thiamine | Solute carrier family 22 member 2 | transporter |
Thiamine | Solute carrier family 22 member 1 | transporter |
Thiamine | Solute carrier family 22 member 5 | transporter |
Thiamine | Cytochrome P450 4B1 | enzyme |
Thiamine | Thiamine transporter 1 | transporter |
Thiamine | Thiamine transporter 2 | transporter |
Thiamine | Thiamin pyrophosphokinase 1 | enzyme |
Thiamine | Ectonucleoside triphosphate diphosphohydrolase 5 | enzyme |
Thiamine | Thiamine-triphosphatase | enzyme |
Thiamine | Serum albumin | carrier |
Thiamine | Pyruvate dehydrogenase E1 component | target |
Quinidine | Sodium channel protein type 5 subunit alpha | target |
Quinidine | Alpha-1-acid glycoprotein 1 | carrier |
Quinidine | Potassium voltage-gated channel subfamily H member 2 | target |
Quinidine | Potassium channel subfamily K member 1 | target |
Quinidine | Potassium channel subfamily K member 6 | target |
Quinidine | Cytochrome P450 1A2 | enzyme |
Quinidine | Cytochrome P450 2E1 | enzyme |
Quinidine | Cytochrome P450 1A1 | enzyme |
Quinidine | Cytochrome P450 2D6 | enzyme |
Quinidine | Cytochrome P450 3A4 | enzyme |
Quinidine | Cytochrome P450 3A7 | enzyme |
Quinidine | Solute carrier family 22 member 2 | transporter |
Quinidine | Solute carrier family 22 member 1 | transporter |
Quinidine | Solute carrier family 22 member 5 | transporter |
Quinidine | P-glycoprotein 1 | transporter |
Quinidine | Solute carrier organic anion transporter family member 1A2 | transporter |
Quinidine | Solute carrier family 22 member 8 | transporter |
Quinidine | Canalicular multispecific organic anion transporter 1 | transporter |
Quinidine | Solute carrier family 22 member 4 | transporter |
Quinidine | Solute carrier organic anion transporter family member 1B1 | transporter |
Quinidine | Cytochrome P450 2B6 | enzyme |
Quinidine | Cytochrome P450 2C9 | enzyme |
Quinidine | Alpha-1A adrenergic receptor | target |
Quinidine | Alpha-1B adrenergic receptor | target |
Quinidine | Alpha-1D adrenergic receptor | target |
Quinidine | Bile salt export pump | transporter |
Quinidine | Cytochrome P450 2C8 | enzyme |
Quinidine | Serum albumin | carrier |
Procainamide | Sodium channel protein type 5 subunit alpha | target |
Procainamide | DNA (cytosine-5)-methyltransferase 1 | target |
Procainamide | Cytochrome P450 2D6 | enzyme |
Procainamide | Cholinesterase | enzyme |
Procainamide | Solute carrier family 22 member 2 | transporter |
Procainamide | Solute carrier family 22 member 1 | transporter |
Procainamide | Solute carrier family 22 member 3 | transporter |
Procainamide | Solute carrier family 22 member 5 | transporter |
Procainamide | Solute carrier family 22 member 4 | transporter |
Procainamide | Potassium voltage-gated channel subfamily H member 2 | target |
Procainamide | Multidrug and toxin extrusion protein 1 | transporter |
Procainamide | Multidrug and toxin extrusion protein 2 | transporter |
Norepinephrine | Phenylalanine-4-hydroxylase | target |
Norepinephrine | Alpha-1A adrenergic receptor | target |
Norepinephrine | Alpha-1B adrenergic receptor | target |
Norepinephrine | Alpha-1D adrenergic receptor | target |
Norepinephrine | Alpha-2A adrenergic receptor | target |
Norepinephrine | Alpha-2B adrenergic receptor | target |
Norepinephrine | Alpha-2C adrenergic receptor | target |
Norepinephrine | Beta-1 adrenergic receptor | target |
Norepinephrine | Beta-2 adrenergic receptor | target |
Norepinephrine | Beta-3 adrenergic receptor | target |
Norepinephrine | Solute carrier family 22 member 2 | transporter |
Norepinephrine | Solute carrier family 22 member 3 | transporter |
Norepinephrine | Solute carrier family 22 member 5 | transporter |
Norepinephrine | Solute carrier family 22 member 1 | transporter |
Norepinephrine | POU domain, class 5, transcription factor 1 | transporter |
Norepinephrine | Sodium-dependent noradrenaline transporter | transporter |
Norepinephrine | Synaptic vesicular amine transporter | target |
Norepinephrine | Chromaffin granule amine transporter | target |
Nicotine | Neuronal acetylcholine receptor subunit alpha-2 | target |
Nicotine | Neuronal acetylcholine receptor subunit beta-2 | target |
Nicotine | Neuronal acetylcholine receptor subunit alpha-7 | target |
Nicotine | Neuronal acetylcholine receptor subunit alpha-4 | target |
Nicotine | Neuronal acetylcholine receptor subunit alpha-10 | target |
Nicotine | Neuronal acetylcholine receptor subunit alpha-9 | target |
Nicotine | Cytochrome P450 2A6 | enzyme |
Nicotine | Cytochrome P450 2E1 | enzyme |
Nicotine | Cytochrome P450 2A13 | enzyme |
Nicotine | Cytochrome P450 2B6 | enzyme |
Nicotine | Neuronal acetylcholine receptor subunit beta-4 | target |
Nicotine | Neuronal acetylcholine receptor subunit alpha-3 | target |
Nicotine | Neuronal acetylcholine receptor subunit alpha-5 | target |
Nicotine | Neuronal acetylcholine receptor subunit alpha-6 | target |
Nicotine | Neuronal acetylcholine receptor subunit beta-3 | target |
Nicotine | Solute carrier family 22 member 2 | transporter |
Nicotine | Solute carrier family 22 member 1 | transporter |
Nicotine | Solute carrier family 22 member 3 | transporter |
Nicotine | Solute carrier family 22 member 5 | transporter |
Nicotine | Solute carrier family 22 member 4 | transporter |
Nicotine | Cytochrome P450 1A1 | enzyme |
Nicotine | Cytochrome P450 1A2 | enzyme |
Nicotine | Cytochrome P450 2C19 | enzyme |
Nicotine | Cytochrome P450 2C8 | enzyme |
Nicotine | Cytochrome P450 2C9 | enzyme |
Nicotine | Cytochrome P450 2D6 | enzyme |
Nicotine | Cytochrome P450 3A4 | enzyme |
Nicotine | Amine oxidase [flavin-containing] A | enzyme |
Nicotine | Amine oxidase [flavin-containing] B | enzyme |
Nicotine | Cytochrome P450 19A1 | target |
Nicotine | Choline O-acetyltransferase | target |
Imipramine | Sodium-dependent noradrenaline transporter | target |
Imipramine | Sodium-dependent serotonin transporter | target |
Imipramine | Cytochrome P450 1A2 | enzyme |
Imipramine | Cytochrome P450 2C19 | enzyme |
Imipramine | Cytochrome P450 2D6 | enzyme |
Imipramine | Histamine H1 receptor | target |
Imipramine | Alpha-1A adrenergic receptor | target |
Imipramine | 5-hydroxytryptamine receptor 2A | target |
Imipramine | Muscarinic acetylcholine receptor M1 | target |
Imipramine | Muscarinic acetylcholine receptor M2 | target |
Imipramine | Muscarinic acetylcholine receptor M3 | target |
Imipramine | Muscarinic acetylcholine receptor M4 | target |
Imipramine | Muscarinic acetylcholine receptor M5 | target |
Imipramine | Potassium voltage-gated channel subfamily D member 2 | target |
Imipramine | Potassium voltage-gated channel subfamily D member 3 | target |
Imipramine | Alpha-1D adrenergic receptor | target |
Imipramine | Alpha-1-acid glycoprotein 1 | carrier |
Imipramine | Solute carrier family 22 member 2 | transporter |
Imipramine | Solute carrier family 22 member 3 | transporter |
Imipramine | P-glycoprotein 1 | transporter |
Imipramine | Solute carrier family 22 member 4 | transporter |
Imipramine | Cytochrome P450 3A4 | enzyme |
Imipramine | Cytochrome P450 2B6 | enzyme |
Imipramine | Cytochrome P450 2C18 | enzyme |
Imipramine | Cytochrome P450 2E1 | enzyme |
Imipramine | Cytochrome P450 3A7 | enzyme |
Imipramine | 5-hydroxytryptamine receptor 2C | target |
Imipramine | Alpha-1B adrenergic receptor | target |
Imipramine | 5-hydroxytryptamine receptor 7 | target |
Imipramine | D(1) dopamine receptor | target |
Imipramine | Dopamine D2 receptor | target |
Imipramine | Potassium voltage-gated channel subfamily H member 2 | target |
Imipramine | Sodium-dependent dopamine transporter | target |
Imipramine | 5-hydroxytryptamine receptor 1A | target |
Imipramine | 5-hydroxytryptamine receptor 6 | target |
Imipramine | Potassium voltage-gated channel subfamily H member 1 | target |
Imipramine | Serum albumin | carrier |
Imipramine | Alpha-1-acid glycoprotein 2 | target |
Histamine | Histamine H1 receptor | target |
Histamine | Histamine H2 receptor | target |
Histamine | Histamine H3 receptor | target |
Histamine | Histamine N-methyltransferase | enzyme |
Histamine | Solute carrier family 22 member 2 | transporter |
Histamine | Solute carrier family 22 member 1 | transporter |
Histamine | Solute carrier family 22 member 3 | transporter |
Histamine | Solute carrier family 22 member 5 | transporter |
Histamine | Histamine H4 receptor | target |
Histamine | Synaptic vesicular amine transporter | target |
Guanidine | Ribonuclease pancreatic | target |
Guanidine | DNA | target |
Guanidine | Disks large homolog 4 | target |
Guanidine | Lysozyme | target |
Guanidine | Aldehyde dehydrogenase, mitochondrial | target |
Guanidine | Guanidinoacetate N-methyltransferase | target |
Guanidine | Arginase | target |
Guanidine | Solute carrier family 22 member 2 | transporter |
Guanidine | Solute carrier family 22 member 1 | transporter |
Guanidine | Solute carrier family 22 member 3 | transporter |
Guanidine | Solute carrier family 22 member 5 | transporter |
Guanidine | Solute carrier family 22 member 8 | transporter |
Guanidine | Solute carrier family 22 member 4 | transporter |
Guanidine | Multidrug and toxin extrusion protein 1 | transporter |
Guanidine | Multidrug and toxin extrusion protein 2 | transporter |
Grepafloxacin | DNA gyrase subunit A | target |
Grepafloxacin | DNA topoisomerase 4 subunit A | target |
Grepafloxacin | Cytochrome P450 3A4 | enzyme |
Grepafloxacin | Cytochrome P450 1A2 | enzyme |
Grepafloxacin | Solute carrier family 22 member 2 | transporter |
Grepafloxacin | Solute carrier family 22 member 5 | transporter |
Grepafloxacin | Canalicular multispecific organic anion transporter 1 | transporter |
Grepafloxacin | P-glycoprotein 1 | transporter |
Grepafloxacin | Multidrug resistance-associated protein 1 | transporter |
Grepafloxacin | Solute carrier family 22 member 6 | transporter |
Grepafloxacin | DNA gyrase subunit A | target |
Grepafloxacin | DNA gyrase subunit B | target |
Dopamine | Dopamine D1 receptor | target |
Dopamine | Dopamine beta-hydroxylase | target |
Dopamine | Amine oxidase [flavin-containing] A | enzyme |
Dopamine | Amine oxidase [flavin-containing] B | enzyme |
Dopamine | Catechol O-methyltransferase | enzyme |
Dopamine | Solute carrier family 22 member 2 | transporter |
Dopamine | Solute carrier family 22 member 1 | transporter |
Dopamine | Solute carrier family 22 member 3 | transporter |
Dopamine | Solute carrier family 22 member 5 | transporter |
Dopamine | POU domain, class 5, transcription factor 1 | transporter |
Dopamine | Dopamine D5 receptor | target |
Dopamine | Dopamine D2 receptor | target |
Dopamine | Dopamine D3 receptor | target |
Dopamine | Dopamine D4 receptor | target |
Dopamine | Sodium-dependent dopamine transporter | target |
Dopamine | Dopamine beta-hydroxylase | enzyme |
Dopamine | 5-hydroxytryptamine receptor 1A | target |
Dopamine | 5-hydroxytryptamine receptor 7 | target |
Dopamine | D(1) dopamine receptor | target |
Dopamine | Sodium-dependent noradrenaline transporter | target |
Dopamine | Sodium-dependent serotonin transporter | target |
Dopamine | 5-hydroxytryptamine receptor 3A | target |
Dopamine | 5-hydroxytryptamine receptor 3B | target |
Dopamine | Superoxide dismutase [Cu-Zn] | target |
Dopamine | Synaptic vesicular amine transporter | target |
Amantadine | Dopamine D2 receptor | target |
Amantadine | Matrix protein 2 | target |
Amantadine | Aromatic-L-amino-acid decarboxylase | enzyme |
Amantadine | Amine oxidase [flavin-containing] B | enzyme |
Amantadine | Solute carrier family 22 member 2 | transporter |
Amantadine | Solute carrier family 22 member 1 | transporter |
Amantadine | Glutamate receptor ionotropic, NMDA 3A | target |
Amantadine | Neuronal acetylcholine receptor subunit alpha-7 | target |
Amantadine | Neuronal acetylcholine receptor subunit alpha-4 | target |
Amantadine | Neuronal acetylcholine receptor subunit alpha-3 | target |
Progesterone | Progesterone receptor | target |
Progesterone | Estrogen receptor alpha | target |
Progesterone | Steroid 17-alpha-hydroxylase/17,20 lyase | target |
Progesterone | Cytochrome P450 2C19 | enzyme |
Progesterone | Cytochrome P450 2C9 | enzyme |
Progesterone | Cytochrome P450 3A4 | enzyme |
Progesterone | Cytochrome P450 3A5 | enzyme |
Progesterone | Cytochrome P450 3A7 | enzyme |
Progesterone | P-glycoprotein 1 | transporter |
Progesterone | Solute carrier family 22 member 2 | transporter |
Progesterone | Solute carrier family 22 member 1 | transporter |
Progesterone | Solute carrier family 22 member 3 | transporter |
Progesterone | Bile salt export pump | transporter |
Progesterone | Multidrug resistance-associated protein 1 | transporter |
Progesterone | Sodium/bile acid cotransporter | transporter |
Progesterone | Steroid 17-alpha-hydroxylase/17,20 lyase | enzyme |
Progesterone | Cytochrome P450 1A1 | enzyme |
Progesterone | Cytochrome P450 1B1 | enzyme |
Progesterone | Cytochrome P450 2A6 | enzyme |
Progesterone | Cytochrome P450 2D6 | enzyme |
Progesterone | Mineralocorticoid receptor | target |
Progesterone | Kappa-type opioid receptor | target |
Progesterone | Alpha-1-acid glycoprotein 1 | target |
Progesterone | Glucocorticoid receptor | target |
Progesterone | Androgen receptor | target |
Progesterone | Sex hormone-binding globulin | target |
Progesterone | Solute carrier organic anion transporter family member 1B1 | transporter |
Progesterone | ATP-binding cassette sub-family G member 2 | transporter |
Progesterone | Estrogen receptor beta | target |
Progesterone | Solute carrier organic anion transporter family member 1B3 | transporter |
Phenoxybenzamine | Alpha-1A adrenergic receptor | target |
Phenoxybenzamine | Calmodulin | target |
Phenoxybenzamine | Solute carrier family 22 member 2 | transporter |
Phenoxybenzamine | Solute carrier family 22 member 1 | transporter |
Phenoxybenzamine | Solute carrier family 22 member 3 | transporter |
Phenoxybenzamine | Alpha-2A adrenergic receptor | target |
Phenoxybenzamine | Alpha-2C adrenergic receptor | target |
Phenoxybenzamine | Alpha-2B adrenergic receptor | target |
Phenoxybenzamine | Beta-2 adrenergic receptor | target |
Phenoxybenzamine | Alpha-1B adrenergic receptor | target |
Phenoxybenzamine | Alpha-1D adrenergic receptor | target |
Phenoxybenzamine | Dopamine D2 receptor | target |
Estradiol | Estrogen receptor alpha | target |
Estradiol | Nuclear receptor subfamily 1 group I member 2 | target |
Estradiol | Sex hormone-binding globulin | carrier |
Estradiol | Estrogen receptor beta | target |
Estradiol | Cytochrome P450 1A2 | enzyme |
Estradiol | UDP-glucuronosyltransferase 1-1 | enzyme |
Estradiol | Serum albumin | carrier |
Estradiol | Fatty acid-binding protein, intestinal | carrier |
Estradiol | Cytochrome P450 3A4 | enzyme |
Estradiol | Cytochrome P450 3A5 | enzyme |
Estradiol | Cytochrome P450 3A7 | enzyme |
Estradiol | Solute carrier family 22 member 2 | transporter |
Estradiol | Solute carrier family 22 member 3 | transporter |
Estradiol | Multidrug resistance-associated protein 7 | transporter |
Estradiol | Solute carrier family 22 member 11 | transporter |
Estradiol | ATP-binding cassette sub-family G member 2 | transporter |
Estradiol | Solute carrier organic anion transporter family member 1B1 | transporter |
Estradiol | P-glycoprotein 1 | transporter |
Estradiol | Cytochrome P450 1A1 | enzyme |
Estradiol | Cytochrome P450 1B1 | enzyme |
Estradiol | Cytochrome P450 2C19 | enzyme |
Estradiol | Cytochrome P450 2C8 | enzyme |
Estradiol | Cytochrome P450 2C9 | enzyme |
Estradiol | Solute carrier family 22 member 8 | transporter |
Estradiol | Solute carrier organic anion transporter family member 1B3 | transporter |
Estradiol | Solute carrier organic anion transporter family member 1C1 | transporter |
Estradiol | Neuronal acetylcholine receptor subunit alpha-4 | target |
Estradiol | G-protein coupled estrogen receptor 1 | target |
Estradiol | ATP synthase subunit a | target |
Estradiol | Beclin-1 | target |
Estradiol | UDP-glucuronosyltransferase 2B15 | enzyme |
Estradiol | Catechol O-methyltransferase | enzyme |
Estradiol | UDP-glucuronosyltransferases (UGTs) | enzyme |
Estradiol | Cytochrome P450 19A1 | enzyme |
Phenformin | 5'-AMP-activated protein kinase catalytic subunit alpha-1 | target |
Phenformin | Cytochrome P450 2D6 | enzyme |
Phenformin | Solute carrier family 22 member 2 | transporter |
Phenformin | Solute carrier family 22 member 1 | transporter |
Phenformin | ATP-sensitive inward rectifier potassium channel 8 | target |
Phenformin | 5'-AMP-activated protein kinase subunit beta-1 | target |
Phenformin | 5'-AMP-activated protein kinase subunit gamma-1 | target |
Metformin | 5'-AMP-activated protein kinase subunit beta-1 | target |
Metformin | Solute carrier family 22 member 2 | transporter |
Metformin | Solute carrier family 22 member 1 | transporter |
Metformin | Multidrug and toxin extrusion protein 1 | transporter |
Metformin | Equilibrative nucleoside transporter 4 | transporter |
Metformin | Solute carrier family 22 member 3 | transporter |
Metformin | Multidrug and toxin extrusion protein 2 | transporter |
Metformin | Electron transfer flavoprotein-ubiquinone oxidoreductase, mitochondrial | target |
Metformin | Glycerol-3-phosphate dehydrogenase [NAD(+)], cytoplasmic | target |
Metformin | Acetyl-CoA carboxylase 2 | target |
Metformin | Multidrug and toxin extrusion protein 1 | target |
Desipramine | Muscarinic acetylcholine receptor M1 | target |
Desipramine | Sodium-dependent noradrenaline transporter | target |
Desipramine | Beta-2 adrenergic receptor | target |
Desipramine | Muscarinic acetylcholine receptor M2 | target |
Desipramine | Sodium-dependent serotonin transporter | target |
Desipramine | Histamine H1 receptor | target |
Desipramine | Beta-1 adrenergic receptor | target |
Desipramine | Cytochrome P450 2D6 | enzyme |
Desipramine | Muscarinic acetylcholine receptor M3 | target |
Desipramine | Muscarinic acetylcholine receptor M4 | target |
Desipramine | Muscarinic acetylcholine receptor M5 | target |
Desipramine | Alpha-1 adrenergic receptors | target |
Desipramine | 5-hydroxytryptamine receptor 2A | target |
Desipramine | Alpha-1-acid glycoprotein 1 | carrier |
Desipramine | Cytochrome P450 2B6 | enzyme |
Desipramine | Cytochrome P450 3A4 | enzyme |
Desipramine | Solute carrier family 22 member 2 | transporter |
Desipramine | Solute carrier family 22 member 1 | transporter |
Desipramine | Solute carrier family 22 member 3 | transporter |
Desipramine | Solute carrier family 22 member 5 | transporter |
Desipramine | P-glycoprotein 1 | transporter |
Desipramine | Solute carrier family 22 member 4 | transporter |
Desipramine | Cytochrome P450 1A2 | enzyme |
Desipramine | Cytochrome P450 2E1 | enzyme |
Desipramine | Sphingomyelin phosphodiesterase | target |
Desipramine | 5-hydroxytryptamine receptor 1A | target |
Desipramine | 5-hydroxytryptamine receptor 2C | target |
Desipramine | Dopamine D2 receptor | target |
Desipramine | Alpha-2 adrenergic receptors | target |
Famotidine | Histamine H2 receptor | target |
Famotidine | Solute carrier family 22 member 2 | transporter |
Famotidine | Solute carrier family 22 member 8 | transporter |
Famotidine | Multidrug and toxin extrusion protein 1 | transporter |
Famotidine | Cytochrome P450 1A2 | enzyme |
Famotidine | Solute carrier family 22 member 6 | transporter |
Probenecid | Solute carrier family 22 member 8 | target |
Probenecid | Solute carrier family 22 member 11 | target |
Probenecid | Serum albumin | carrier |
Probenecid | Solute carrier family 22 member 2 | transporter |
Probenecid | Solute carrier family 22 member 1 | transporter |
Probenecid | Canalicular multispecific organic anion transporter 2 | transporter |
Probenecid | Multidrug resistance-associated protein 4 | transporter |
Probenecid | Multidrug resistance-associated protein 5 | transporter |
Probenecid | Monocarboxylate transporter 2 | transporter |
Probenecid | Solute carrier family 22 member 5 | transporter |
Probenecid | Multidrug resistance-associated protein 6 | transporter |
Probenecid | Multidrug resistance-associated protein 1 | transporter |
Probenecid | Solute carrier organic anion transporter family member 1A2 | transporter |
Probenecid | Monocarboxylate transporter 1 | transporter |
Probenecid | Sodium/bile acid cotransporter | transporter |
Probenecid | Solute carrier family 22 member 6 | transporter |
Probenecid | Solute carrier family 22 member 10 | transporter |
Probenecid | Solute carrier family 22 member 8 | transporter |
Probenecid | Canalicular multispecific organic anion transporter 1 | transporter |
Probenecid | ATP-binding cassette sub-family C member 11 | transporter |
Probenecid | Solute carrier family 22 member 11 | transporter |
Probenecid | Solute carrier organic anion transporter family member 1C1 | transporter |
Probenecid | Solute carrier family 22 member 7 | transporter |
Probenecid | Solute carrier family 22 member 6 | target |
Probenecid | Pannexin-1 | target |
Probenecid | Cytochrome P450 2C8 | enzyme |
Probenecid | Cytochrome P450 3A4 | enzyme |
Probenecid | Solute carrier family 22 member 12 | transporter |
Probenecid | Solute carrier family 2, facilitated glucose transporter member 9 | transporter |
Probenecid | Taste receptor type 2 member 16 | target |
Probenecid | UDP-glucuronosyltransferase 1-1 | enzyme |
Probenecid | Cytochrome P450 2C9 | enzyme |
Aminohippuric acid | Solute carrier family 22 member 2 | transporter |
Aminohippuric acid | Solute carrier family 22 member 5 | transporter |
Aminohippuric acid | Solute carrier family 22 member 6 | transporter |
Aminohippuric acid | Solute carrier family 22 member 8 | transporter |
Aminohippuric acid | Canalicular multispecific organic anion transporter 1 | transporter |
Aminohippuric acid | Solute carrier family 22 member 4 | transporter |
Aminohippuric acid | Solute carrier family 22 member 11 | transporter |
Aminohippuric acid | Solute carrier organic anion transporter family member 3A1 | transporter |
Aminohippuric acid | Multidrug resistance-associated protein 1 | transporter |
Aminohippuric acid | Monocarboxylate transporter 1 | transporter |
Aminohippuric acid | Solute carrier family 22 member 7 | transporter |
Aminohippuric acid | Solute carrier family 22 member 8 | target |
Cisplatin | DNA | target |
Cisplatin | Canalicular multispecific organic anion transporter 2 | transporter |
Cisplatin | Multidrug resistance-associated protein 5 | transporter |
Cisplatin | Canalicular multispecific organic anion transporter 1 | transporter |
Cisplatin | Solute carrier family 22 member 2 | transporter |
Cisplatin | High affinity copper uptake protein 1 | transporter |
Cisplatin | Probable low affinity copper uptake protein 2 | transporter |
Cisplatin | Multidrug resistance-associated protein 6 | transporter |
Cisplatin | Copper-transporting ATPase 2 | transporter |
Cisplatin | Copper-transporting ATPase 1 | transporter |
Cisplatin | Prostaglandin G/H synthase 2 | enzyme |
Cisplatin | Myeloperoxidase | enzyme |
Cisplatin | Xanthine dehydrogenase/oxidase | enzyme |
Cisplatin | Arylamine N-acetyltransferase | enzyme |
Cisplatin | Cytochrome P450 2C9 | enzyme |
Cisplatin | Cytochrome P450 2B6 | enzyme |
Cisplatin | Cholinesterase | enzyme |
Cisplatin | Cytochrome P450 4A11 | enzyme |
Cisplatin | ATP-binding cassette sub-family G member 2 | transporter |
Cisplatin | Glutathione S-transferase theta-1 | enzyme |
Cisplatin | Metallothionein-1A | enzyme |
Cisplatin | Metallothionein-2 | enzyme |
Cisplatin | Superoxide dismutase [Cu-Zn] | enzyme |
Cisplatin | Glutathione S-transferase P | enzyme |
Cisplatin | NAD(P)H dehydrogenase [quinone] 1 | enzyme |
Cisplatin | Glutathione S-transferase Mu 1 | enzyme |
Cisplatin | DNA-3-methyladenine glycosylase | target |
Cisplatin | Alpha-2-macroglobulin | target |
Cisplatin | Serum albumin | carrier |
Cisplatin | Serotransferrin | target |
Cisplatin | Copper transport protein ATOX1 | target |
Quinacrine | DNA | target |
Quinacrine | 85/88 kDa calcium-independent phospholipase A2 | target |
Quinacrine | Cytosolic phospholipase A2 | target |
Quinacrine | Inactive phospholipase C-like protein 1 | target |
Quinacrine | Histamine N-methyltransferase | enzyme |
Quinacrine | Solute carrier family 22 member 2 | transporter |
Quinacrine | P-glycoprotein 1 | transporter |
Quinacrine | Cytochrome P450 3A4 | enzyme |
Quinacrine | Cytochrome P450 3A5 | enzyme |
Quinacrine | Phospholipase A2 | target |
Chlorpheniramine | Histamine H1 receptor | target |
Chlorpheniramine | Cytochrome P450 3A4 | enzyme |
Chlorpheniramine | Cytochrome P450 2D6 | enzyme |
Chlorpheniramine | Sodium-dependent serotonin transporter | target |
Chlorpheniramine | Sodium-dependent noradrenaline transporter | target |
Chlorpheniramine | Sodium-dependent dopamine transporter | target |
Chlorpheniramine | Cytochrome P450 3A5 | enzyme |
Chlorpheniramine | Cytochrome P450 3A7 | enzyme |
Chlorpheniramine | Solute carrier family 22 member 2 | transporter |
Chlorpheniramine | Solute carrier family 22 member 1 | transporter |
Amiloride | Amiloride-sensitive sodium channel subunit beta | target |
Amiloride | Acid-sensing ion channel 1 | target |
Amiloride | Amiloride-sensitive amine oxidase [copper-containing] | target |
Amiloride | Amiloride-sensitive sodium channel subunit alpha | target |
Amiloride | Amiloride-sensitive sodium channel subunit gamma | target |
Amiloride | Sodium/hydrogen exchanger 1 | target |
Amiloride | Acid-sensing ion channel 2 | target |
Amiloride | Amiloride-sensitive sodium channel subunit delta | target |
Amiloride | Urokinase-type plasminogen activator | target |
Amiloride | Solute carrier family 22 member 2 | transporter |
Amiloride | Solute carrier family 22 member 4 | transporter |
Amiloride | Amiloride-sensitive amine oxidase [copper-containing] | enzyme |
Amiloride | Amiloride-sensitive amine oxidase [copper-containing] | enzyme |
Disopyramide | Sodium channel protein type 5 subunit alpha | target |
Disopyramide | Alpha-1-acid glycoprotein 1 | carrier |
Disopyramide | Cytochrome P450 3A4 | enzyme |
Disopyramide | Muscarinic acetylcholine receptor M1 | target |
Disopyramide | Muscarinic acetylcholine receptor M2 | target |
Disopyramide | Muscarinic acetylcholine receptor M3 | target |
Disopyramide | Potassium voltage-gated channel subfamily D member 2 | target |
Disopyramide | Potassium voltage-gated channel subfamily D member 3 | target |
Disopyramide | Solute carrier family 22 member 2 | transporter |
Disopyramide | Solute carrier family 22 member 1 | transporter |
Disopyramide | Potassium voltage-gated channel subfamily H member 2 | target |
Disopyramide | Alpha-1-acid glycoprotein 2 | target |
Disopyramide | Cytochrome P450 1A2 | enzyme |
Diphenhydramine | Histamine H1 receptor | target |
Diphenhydramine | Cytochrome P450 2D6 | enzyme |
Diphenhydramine | Cytochrome P450 2C9 | enzyme |
Diphenhydramine | Cytochrome P450 2C19 | enzyme |
Diphenhydramine | Solute carrier family 22 member 2 | transporter |
Diphenhydramine | Solute carrier family 22 member 5 | transporter |
Diphenhydramine | Prostaglandin G/H synthase 1 | enzyme |
Diphenhydramine | Muscarinic acetylcholine receptor M2 | target |
Diphenhydramine | Histamine N-methyltransferase | target |
Imatinib | Platelet-derived growth factor receptor beta | target |
Imatinib | Tyrosine-protein kinase ABL1 | target |
Imatinib | Mast/stem cell growth factor receptor Kit | target |
Imatinib | Proto-oncogene tyrosine-protein kinase receptor Ret | target |
Imatinib | High affinity nerve growth factor receptor | target |
Imatinib | Macrophage colony-stimulating factor 1 receptor | target |
Imatinib | Platelet-derived growth factor receptor alpha | target |
Imatinib | Epithelial discoidin domain-containing receptor 1 | target |
Imatinib | Cytochrome P450 3A4 | enzyme |
Imatinib | Breakpoint cluster region protein | target |
Imatinib | Cytochrome P450 1A2 | enzyme |
Imatinib | Cytochrome P450 2D6 | enzyme |
Imatinib | Cytochrome P450 2C9 | enzyme |
Imatinib | Cytochrome P450 2C19 | enzyme |
Imatinib | Cytochrome P450 3A5 | enzyme |
Imatinib | Cytochrome P450 3A7 | enzyme |
Imatinib | Solute carrier family 22 member 1 | transporter |
Imatinib | P-glycoprotein 1 | transporter |
Imatinib | Solute carrier family 22 member 2 | transporter |
Imatinib | ATP-binding cassette sub-family G member 2 | transporter |
Imatinib | ATP-binding cassette sub-family A member 3 | transporter |
Imatinib | Serum albumin | carrier |
Imatinib | Alpha-1-acid glycoprotein 1 | carrier |
Imatinib | Bile salt export pump | transporter |
Imatinib | Cytochrome P450 2C8 | enzyme |
Imatinib | Canalicular multispecific organic anion transporter 1 | transporter |
Imatinib | Multidrug resistance-associated protein 1 | transporter |
Imatinib | Solute carrier family 22 member 5 | transporter |
Imatinib | Solute carrier organic anion transporter family member 1B3 | transporter |
Imatinib | Multidrug resistance-associated protein 4 | transporter |
Imatinib | Solute carrier organic anion transporter family member 1A2 | transporter |
Imatinib | Discoidin domain-containing receptor 2 | target |
Imatinib | Induced myeloid leukemia cell differentiation protein Mcl-1 | target |
Pimagedine | Nitric oxide synthase, inducible | target |
Pimagedine | Aldose reductase | target |
Pimagedine | Metalloproteinase inhibitor 3 | target |
Pimagedine | Solute carrier family 22 member 2 | transporter |
Pimagedine | Amiloride-sensitive amine oxidase [copper-containing] | target |
Pimagedine | C-C chemokine receptor type 2 | target |
Flurazepam | Cytochrome P450 3A4 | enzyme |
Flurazepam | P-glycoprotein 1 | transporter |
Flurazepam | Cytochrome P450 2E1 | enzyme |
Flurazepam | Cytochrome P450 2A6 | enzyme |
Flurazepam | Solute carrier family 22 member 2 | transporter |
Flurazepam | GABA(A) Receptor | target |
Flurazepam | GABA(A) Receptor Benzodiazepine Binding Site | target |
Dexchlorpheniramine maleate | Cytochrome P450 2D6 | enzyme |
Dexchlorpheniramine maleate | Histamine H1 receptor | target |
Dexchlorpheniramine maleate | Solute carrier family 22 member 1 | carrier |
Dexchlorpheniramine maleate | Solute carrier family 22 member 2 | carrier |
Dexchlorpheniramine maleate | Cytochrome P450 3A4 | enzyme |
Enasidenib | Cytochrome P450 1A2 | enzyme |
Enasidenib | Cytochrome P450 2B6 | enzyme |
Enasidenib | Isocitrate dehydrogenase [NADP], mitochondrial | target |
Enasidenib | Cytochrome P450 2C8 | enzyme |
Enasidenib | Cytochrome P450 2C9 | enzyme |
Enasidenib | Cytochrome P450 2C19 | enzyme |
Enasidenib | Cytochrome P450 2D6 | enzyme |
Enasidenib | Cytochrome P450 3A4 | enzyme |
Enasidenib | UDP-glucuronosyltransferase 1-1 | enzyme |
Enasidenib | UDP-glucuronosyltransferase 1-3 | enzyme |
Enasidenib | UDP-glucuronosyltransferase 1-4 | enzyme |
Enasidenib | UDP-glucuronosyltransferase 1-9 | enzyme |
Enasidenib | UDP-glucuronosyltransferase 2B7 | enzyme |
Enasidenib | UDP-glucuronosyltransferase 2B15 | enzyme |
Enasidenib | P-glycoprotein 1 | transporter |
Enasidenib | ATP-binding cassette sub-family G member 2 | transporter |
Enasidenib | Solute carrier family 22 member 6 | transporter |
Enasidenib | Solute carrier organic anion transporter family member 1B1 | transporter |
Enasidenib | Solute carrier family 22 member 2 | transporter |
Enasidenib | Solute carrier organic anion transporter family member 1B3 | transporter |
Enasidenib | Solute carrier family 22 member 8 | transporter |
Enasidenib | Serum albumin | carrier |
Enasidenib | Isocitrate dehydrogenase [NADP] cytoplasmic | target |
Enasidenib | Isocitrate dehydrogenase [NAD] subunit alpha, mitochondrial | target |
Enasidenib | Isocitrate dehydrogenase [NAD] subunit beta, mitochondrial | target |
Enasidenib | Isocitrate dehydrogenase [NAD] subunit gamma, mitochondrial | target |
Dolutegravir | UDP-glucuronosyltransferase 1-1 | enzyme |
Dolutegravir | Cytochrome P450 3A Subfamily | enzyme |
Dolutegravir | Integrase | target |
Dolutegravir | Solute carrier family 22 member 2 | transporter |
Dolutegravir | UDP-glucuronosyltransferase 1-3 | enzyme |
Dolutegravir | UDP-glucuronosyltransferase 1-9 | enzyme |
Dolutegravir | ATP-binding cassette sub-family G member 2 | transporter |
Dolutegravir | Solute carrier family 22 member 6 | transporter |
Dolutegravir | Solute carrier family 22 member 8 | transporter |
Dolutegravir | P-glycoprotein 1 | transporter |
Dolutegravir | Multidrug and toxin extrusion protein 1 | transporter |
Dolutegravir | Serum albumin | carrier |
Dolutegravir | alpha1-acid glycoprotein | carrier |
Dolutegravir | Gag-Pol polyprotein | target |
Baricitinib | Solute carrier family 22 member 8 | transporter |
Baricitinib | ATP-binding cassette sub-family G member 2 | transporter |
Baricitinib | Multidrug and toxin extrusion protein 2 | transporter |
Baricitinib | Cytochrome P450 3A4 | enzyme |
Baricitinib | Tyrosine-protein kinase JAK1 | target |
Baricitinib | Tyrosine-protein kinase JAK2 | target |
Baricitinib | Solute carrier family 22 member 6 | transporter |
Baricitinib | Solute carrier family 22 member 2 | transporter |
Baricitinib | Solute carrier organic anion transporter family member 1B3 | transporter |
Baricitinib | Tyrosine-protein kinase JAK3 | target |
Baricitinib | P-glycoprotein 1 | transporter |
Baricitinib | Non-receptor tyrosine-protein kinase TYK2 | target |
Estradiol acetate | Estrogen receptor alpha | target |
Estradiol acetate | Nuclear receptor subfamily 1 group I member 2 | target |
Estradiol acetate | Sex hormone-binding globulin | carrier |
Estradiol acetate | Estrogen receptor beta | target |
Estradiol acetate | Cytochrome P450 1A2 | enzyme |
Estradiol acetate | UDP-glucuronosyltransferase 1-1 | enzyme |
Estradiol acetate | Serum albumin | carrier |
Estradiol acetate | Fatty acid-binding protein, intestinal | carrier |
Estradiol acetate | Cytochrome P450 3A4 | enzyme |
Estradiol acetate | Cytochrome P450 3A5 | enzyme |
Estradiol acetate | Cytochrome P450 3A7 | enzyme |
Estradiol acetate | Solute carrier family 22 member 2 | transporter |
Estradiol acetate | Solute carrier family 22 member 1 | transporter |
Estradiol acetate | Solute carrier family 22 member 3 | transporter |
Estradiol acetate | Solute carrier organic anion transporter family member 2B1 | transporter |
Estradiol acetate | Solute carrier organic anion transporter family member 1A2 | transporter |
Estradiol acetate | Multidrug resistance-associated protein 7 | transporter |
Estradiol acetate | Solute carrier family 22 member 11 | transporter |
Estradiol acetate | ATP-binding cassette sub-family G member 2 | transporter |
Estradiol acetate | Solute carrier organic anion transporter family member 1B1 | transporter |
Estradiol acetate | P-glycoprotein 1 | transporter |
Estradiol acetate | Cytochrome P450 1A1 | enzyme |
Estradiol acetate | Cytochrome P450 1B1 | enzyme |
Estradiol acetate | Cytochrome P450 2C19 | enzyme |
Estradiol acetate | Cytochrome P450 2C8 | enzyme |
Estradiol acetate | Cytochrome P450 2C9 | enzyme |
Estradiol acetate | Solute carrier family 22 member 8 | transporter |
Estradiol acetate | Solute carrier organic anion transporter family member 1B3 | transporter |
Estradiol acetate | Solute carrier organic anion transporter family member 1C1 | transporter |
Estradiol acetate | Solute carrier organic anion transporter family member 4A1 | transporter |
Estradiol acetate | Neuronal acetylcholine receptor subunit alpha-4 | target |
Estradiol acetate | Nuclear receptor coactivator 2 | target |
Estradiol acetate | G-protein coupled estrogen receptor 1 | target |
Estradiol acetate | ATP synthase subunit a | target |
Estradiol acetate | Beclin-1 | target |
Estradiol acetate | Estradiol 17-beta-dehydrogenase 2 | target |
Estradiol acetate | Estrogen-related receptor gamma | target |
Estradiol benzoate | Estrogen receptor alpha | target |
Estradiol benzoate | Nuclear receptor subfamily 1 group I member 2 | target |
Estradiol benzoate | Sex hormone-binding globulin | carrier |
Estradiol benzoate | Estrogen receptor beta | target |
Estradiol benzoate | Cytochrome P450 1A2 | enzyme |
Estradiol benzoate | UDP-glucuronosyltransferase 1-1 | enzyme |
Estradiol benzoate | Serum albumin | carrier |
Estradiol benzoate | Fatty acid-binding protein, intestinal | carrier |
Estradiol benzoate | Cytochrome P450 3A4 | enzyme |
Estradiol benzoate | Cytochrome P450 3A5 | enzyme |
Estradiol benzoate | Cytochrome P450 3A7 | enzyme |
Estradiol benzoate | Solute carrier family 22 member 2 | transporter |
Estradiol benzoate | Solute carrier family 22 member 1 | transporter |
Estradiol benzoate | Solute carrier family 22 member 3 | transporter |
Estradiol benzoate | Solute carrier organic anion transporter family member 2B1 | transporter |
Estradiol benzoate | Solute carrier organic anion transporter family member 1A2 | transporter |
Estradiol benzoate | Multidrug resistance-associated protein 7 | transporter |
Estradiol benzoate | Solute carrier family 22 member 11 | transporter |
Estradiol benzoate | ATP-binding cassette sub-family G member 2 | transporter |
Estradiol benzoate | Solute carrier organic anion transporter family member 1B1 | transporter |
Estradiol benzoate | P-glycoprotein 1 | transporter |
Estradiol benzoate | Cytochrome P450 1A1 | enzyme |
Estradiol benzoate | Cytochrome P450 1B1 | enzyme |
Estradiol benzoate | Cytochrome P450 2C19 | enzyme |
Estradiol benzoate | Cytochrome P450 2C8 | enzyme |
Estradiol benzoate | Cytochrome P450 2C9 | enzyme |
Estradiol benzoate | Solute carrier family 22 member 8 | transporter |
Estradiol benzoate | Solute carrier organic anion transporter family member 1B3 | transporter |
Estradiol benzoate | Solute carrier organic anion transporter family member 1C1 | transporter |
Estradiol benzoate | Solute carrier organic anion transporter family member 4A1 | transporter |
Estradiol benzoate | Neuronal acetylcholine receptor subunit alpha-4 | target |
Estradiol benzoate | Nuclear receptor coactivator 2 | target |
Estradiol benzoate | G-protein coupled estrogen receptor 1 | target |
Estradiol benzoate | ATP synthase subunit a | target |
Estradiol benzoate | Beclin-1 | target |
Estradiol benzoate | Estradiol 17-beta-dehydrogenase 2 | target |
Estradiol benzoate | Estrogen-related receptor gamma | target |
Estradiol cypionate | Estrogen receptor alpha | target |
Estradiol cypionate | Nuclear receptor subfamily 1 group I member 2 | target |
Estradiol cypionate | Sex hormone-binding globulin | carrier |
Estradiol cypionate | Estrogen receptor beta | target |
Estradiol cypionate | Cytochrome P450 1A2 | enzyme |
Estradiol cypionate | UDP-glucuronosyltransferase 1-1 | enzyme |
Estradiol cypionate | Serum albumin | carrier |
Estradiol cypionate | Fatty acid-binding protein, intestinal | carrier |
Estradiol cypionate | Cytochrome P450 3A4 | enzyme |
Estradiol cypionate | Cytochrome P450 3A5 | enzyme |
Estradiol cypionate | Cytochrome P450 3A7 | enzyme |
Estradiol cypionate | Solute carrier family 22 member 2 | transporter |
Estradiol cypionate | Solute carrier family 22 member 1 | transporter |
Estradiol cypionate | Solute carrier family 22 member 3 | transporter |
Estradiol cypionate | Solute carrier organic anion transporter family member 2B1 | transporter |
Estradiol cypionate | Solute carrier organic anion transporter family member 1A2 | transporter |
Estradiol cypionate | Multidrug resistance-associated protein 7 | transporter |
Estradiol cypionate | Solute carrier family 22 member 11 | transporter |
Estradiol cypionate | ATP-binding cassette sub-family G member 2 | transporter |
Estradiol cypionate | Solute carrier organic anion transporter family member 1B1 | transporter |
Estradiol cypionate | P-glycoprotein 1 | transporter |
Estradiol cypionate | Cytochrome P450 1A1 | enzyme |
Estradiol cypionate | Cytochrome P450 1B1 | enzyme |
Estradiol cypionate | Cytochrome P450 2C19 | enzyme |
Estradiol cypionate | Cytochrome P450 2C8 | enzyme |
Estradiol cypionate | Cytochrome P450 2C9 | enzyme |
Estradiol cypionate | Solute carrier family 22 member 8 | transporter |
Estradiol cypionate | Solute carrier organic anion transporter family member 1B3 | transporter |
Estradiol cypionate | Solute carrier organic anion transporter family member 1C1 | transporter |
Estradiol cypionate | Solute carrier organic anion transporter family member 4A1 | transporter |
Estradiol cypionate | Neuronal acetylcholine receptor subunit alpha-4 | target |
Estradiol cypionate | Nuclear receptor coactivator 2 | target |
Estradiol cypionate | G-protein coupled estrogen receptor 1 | target |
Estradiol cypionate | ATP synthase subunit a | target |
Estradiol cypionate | Beclin-1 | target |
Estradiol cypionate | Estradiol 17-beta-dehydrogenase 2 | target |
Estradiol cypionate | Estrogen-related receptor gamma | target |
Estradiol dienanthate | Estrogen receptor alpha | target |
Estradiol dienanthate | Nuclear receptor subfamily 1 group I member 2 | target |
Estradiol dienanthate | Sex hormone-binding globulin | carrier |
Estradiol dienanthate | Estrogen receptor beta | target |
Estradiol dienanthate | Cytochrome P450 1A2 | enzyme |
Estradiol dienanthate | UDP-glucuronosyltransferase 1-1 | enzyme |
Estradiol dienanthate | Serum albumin | carrier |
Estradiol dienanthate | Fatty acid-binding protein, intestinal | carrier |
Estradiol dienanthate | Cytochrome P450 3A4 | enzyme |
Estradiol dienanthate | Cytochrome P450 3A5 | enzyme |
Estradiol dienanthate | Cytochrome P450 3A7 | enzyme |
Estradiol dienanthate | Solute carrier family 22 member 2 | transporter |
Estradiol dienanthate | Solute carrier family 22 member 1 | transporter |
Estradiol dienanthate | Solute carrier family 22 member 3 | transporter |
Estradiol dienanthate | Solute carrier organic anion transporter family member 2B1 | transporter |
Estradiol dienanthate | Solute carrier organic anion transporter family member 1A2 | transporter |
Estradiol dienanthate | Multidrug resistance-associated protein 7 | transporter |
Estradiol dienanthate | Solute carrier family 22 member 11 | transporter |
Estradiol dienanthate | ATP-binding cassette sub-family G member 2 | transporter |
Estradiol dienanthate | Solute carrier organic anion transporter family member 1B1 | transporter |
Estradiol dienanthate | P-glycoprotein 1 | transporter |
Estradiol dienanthate | Cytochrome P450 1A1 | enzyme |
Estradiol dienanthate | Cytochrome P450 1B1 | enzyme |
Estradiol dienanthate | Cytochrome P450 2C19 | enzyme |
Estradiol dienanthate | Cytochrome P450 2C8 | enzyme |
Estradiol dienanthate | Cytochrome P450 2C9 | enzyme |
Estradiol dienanthate | Solute carrier family 22 member 8 | transporter |
Estradiol dienanthate | Solute carrier organic anion transporter family member 1B3 | transporter |
Estradiol dienanthate | Solute carrier organic anion transporter family member 1C1 | transporter |
Estradiol dienanthate | Solute carrier organic anion transporter family member 4A1 | transporter |
Estradiol dienanthate | Neuronal acetylcholine receptor subunit alpha-4 | target |
Estradiol dienanthate | Nuclear receptor coactivator 2 | target |
Estradiol dienanthate | G-protein coupled estrogen receptor 1 | target |
Estradiol dienanthate | ATP synthase subunit a | target |
Estradiol dienanthate | Beclin-1 | target |
Estradiol dienanthate | Estradiol 17-beta-dehydrogenase 2 | target |
Estradiol dienanthate | Estrogen-related receptor gamma | target |
Estradiol valerate | Estrogen receptor alpha | target |
Estradiol valerate | Nuclear receptor subfamily 1 group I member 2 | target |
Estradiol valerate | Sex hormone-binding globulin | carrier |
Estradiol valerate | Estrogen receptor beta | target |
Estradiol valerate | Cytochrome P450 1A2 | enzyme |
Estradiol valerate | UDP-glucuronosyltransferase 1-1 | enzyme |
Estradiol valerate | Serum albumin | carrier |
Estradiol valerate | Fatty acid-binding protein, intestinal | carrier |
Estradiol valerate | Cytochrome P450 3A4 | enzyme |
Estradiol valerate | Cytochrome P450 3A5 | enzyme |
Estradiol valerate | Cytochrome P450 3A7 | enzyme |
Estradiol valerate | Solute carrier family 22 member 2 | transporter |
Estradiol valerate | Solute carrier family 22 member 1 | transporter |
Estradiol valerate | Solute carrier family 22 member 3 | transporter |
Estradiol valerate | Solute carrier organic anion transporter family member 2B1 | transporter |
Estradiol valerate | Solute carrier organic anion transporter family member 1A2 | transporter |
Estradiol valerate | Multidrug resistance-associated protein 7 | transporter |
Estradiol valerate | Solute carrier family 22 member 11 | transporter |
Estradiol valerate | ATP-binding cassette sub-family G member 2 | transporter |
Estradiol valerate | Solute carrier organic anion transporter family member 1B1 | transporter |
Estradiol valerate | P-glycoprotein 1 | transporter |
Estradiol valerate | Cytochrome P450 1A1 | enzyme |
Estradiol valerate | Cytochrome P450 1B1 | enzyme |
Estradiol valerate | Cytochrome P450 2C19 | enzyme |
Estradiol valerate | Cytochrome P450 2C8 | enzyme |
Estradiol valerate | Cytochrome P450 2C9 | enzyme |
Estradiol valerate | Solute carrier family 22 member 8 | transporter |
Estradiol valerate | Solute carrier organic anion transporter family member 1B3 | transporter |
Estradiol valerate | Solute carrier organic anion transporter family member 1C1 | transporter |
Estradiol valerate | Solute carrier organic anion transporter family member 4A1 | transporter |
Estradiol valerate | Neuronal acetylcholine receptor subunit alpha-4 | target |
Estradiol valerate | Nuclear receptor coactivator 2 | target |
Estradiol valerate | G-protein coupled estrogen receptor 1 | target |
Estradiol valerate | ATP synthase subunit a | target |
Estradiol valerate | Beclin-1 | target |
Estradiol valerate | Estradiol 17-beta-dehydrogenase 2 | target |
Estradiol valerate | Estrogen-related receptor gamma | target |
Apalutamide | Androgen receptor | target |
Apalutamide | Cytochrome P450 3A4 | enzyme |
Apalutamide | Cytochrome P450 2C8 | enzyme |
Apalutamide | Cytochrome P450 2C19 | enzyme |
Apalutamide | Cytochrome P450 2C9 | enzyme |
Apalutamide | P-glycoprotein 1 | transporter |
Apalutamide | ATP-binding cassette sub-family G member 2 | transporter |
Apalutamide | Solute carrier organic anion transporter family member 1B1 | transporter |
Apalutamide | Solute carrier family 22 member 2 | transporter |
Apalutamide | Solute carrier family 22 member 8 | transporter |
Apalutamide | Multidrug and toxin extrusion protein 2 | transporter |
Apalutamide | GABA(A) Receptor | target |
Apalutamide | Multidrug and toxin extrusion protein 1 | transporter |
Apalutamide | Serum albumin | carrier |
Isavuconazole | Cytochrome P450 3A4 | enzyme |
Isavuconazole | Cytochrome P450 3A5 | enzyme |
Isavuconazole | Cytochrome P450 2C8 | enzyme |
Isavuconazole | Cytochrome P450 2C9 | enzyme |
Isavuconazole | Cytochrome P450 2C19 | enzyme |
Isavuconazole | Cytochrome P450 2D6 | enzyme |
Isavuconazole | Cytochrome P450 2B6 | enzyme |
Isavuconazole | UDP-glucuronosyltransferase 1-9 | enzyme |
Isavuconazole | UDP-glucuronosyltransferase 1-8 | enzyme |
Isavuconazole | P-glycoprotein 1 | transporter |
Isavuconazole | ATP-binding cassette sub-family G member 2 | transporter |
Isavuconazole | Solute carrier family 22 member 2 | transporter |
Isavuconazole | Lanosterol 14-alpha demethylase | target |
Isavuconazole | Potassium voltage-gated channel subfamily H member 2 | target |
Isavuconazole | Voltage-dependent L-type calcium channel subunit alpha-1C | target |
Isavuconazole | G protein-activated inward rectifier potassium channel 2 | target |
Isavuconazole | G protein-activated inward rectifier potassium channel 3 | target |
Isavuconazole | ATP-sensitive inward rectifier potassium channel 11 | target |
Isavuconazole | Potassium voltage-gated channel subfamily A member 5 | target |
Isavuconazole | Potassium voltage-gated channel subfamily D member 3 | target |
Isavuconazole | Potassium voltage-gated channel subfamily KQT member 1 | target |
Isavuconazole | Sodium channel protein type 5 subunit alpha | target |
Choline salicylate | Choline-phosphate cytidylyltransferase B | target |
Choline salicylate | Acetylcholinesterase | target |
Choline salicylate | Choline-phosphate cytidylyltransferase A | target |
Choline salicylate | Phospholipase D2 | target |
Choline salicylate | Cholinesterase | target |
Choline salicylate | Phospholipase D1 | target |
Choline salicylate | Solute carrier family 22 member 2 | transporter |
Choline salicylate | Solute carrier family 22 member 1 | transporter |
Choline salicylate | Solute carrier family 22 member 3 | transporter |
Choline salicylate | Solute carrier family 22 member 5 | transporter |
Choline salicylate | Solute carrier family 22 member 4 | transporter |
Choline salicylate | Choline/ethanolaminephosphotransferase 1 | enzyme |
Choline salicylate | Choline transporter-like protein 1 | transporter |
Choline salicylate | Choline transporter-like protein 4 | transporter |
Choline salicylate | Choline transporter-like protein 3 | transporter |
Choline salicylate | Choline/ethanolamine kinase | enzyme |
Choline salicylate | Choline O-acetyltransferase | enzyme |
Choline salicylate | Choline kinase alpha | enzyme |
Choline salicylate | Choline dehydrogenase, mitochondrial | enzyme |
Choline salicylate | High affinity choline transporter 1 | transporter |
Choline salicylate | Neuronal acetylcholine receptor subunit alpha-7 | target |
Lenvatinib | Vascular endothelial growth factor receptor 1 | target |
Lenvatinib | Vascular endothelial growth factor receptor 2 | target |
Lenvatinib | Vascular endothelial growth factor receptor 3 | target |
Lenvatinib | Fibroblast growth factor receptor 1 | target |
Lenvatinib | Fibroblast growth factor receptor 2 | target |
Lenvatinib | Fibroblast growth factor receptor 3 | target |
Lenvatinib | Fibroblast growth factor receptor 4 | target |
Lenvatinib | Platelet-derived growth factor receptor alpha | target |
Lenvatinib | Proto-oncogene tyrosine-protein kinase receptor Ret | target |
Lenvatinib | Mast/stem cell growth factor receptor Kit | target |
Lenvatinib | P-glycoprotein 1 | transporter |
Lenvatinib | ATP-binding cassette sub-family G member 2 | transporter |
Lenvatinib | Cytochrome P450 3A4 | enzyme |
Lenvatinib | Aldehyde oxidase | enzyme |
Lenvatinib | Cytochrome P450 2C8 | enzyme |
Lenvatinib | Cytochrome P450 2C9 | enzyme |
Lenvatinib | Cytochrome P450 1A2 | enzyme |
Lenvatinib | Cytochrome P450 2B6 | enzyme |
Lenvatinib | Cytochrome P450 2C19 | enzyme |
Lenvatinib | Solute carrier family 22 member 6 | transporter |
Lenvatinib | Solute carrier family 22 member 8 | transporter |
Lenvatinib | Solute carrier family 22 member 2 | transporter |
Lenvatinib | Solute carrier organic anion transporter family member 1B1 | transporter |
Lenvatinib | Bile salt export pump | transporter |
Lenvatinib | Cytochrome P450 2D6 | enzyme |
Lenvatinib | Solute carrier organic anion transporter family member 1B3 | transporter |
Varenicline | Neuronal acetylcholine receptor subunit alpha-4 | target |
Varenicline | Neuronal acetylcholine receptor subunit alpha-7 | target |
Varenicline | Neuronal acetylcholine receptor subunit alpha-3 | target |
Varenicline | Neuronal acetylcholine receptor subunit alpha-6 | target |
Varenicline | Neuronal acetylcholine receptor subunit beta-2 | target |
Varenicline | Solute carrier family 22 member 2 | transporter |
Bupropion | Sodium-dependent dopamine transporter | target |
Bupropion | Sodium-dependent noradrenaline transporter | target |
Bupropion | Cytochrome P450 2B6 | enzyme |
Bupropion | Cytochrome P450 2D6 | enzyme |
Bupropion | Alpha-1-acid glycoprotein 1 | carrier |
Bupropion | Neuronal acetylcholine receptor subunit alpha-3 | target |
Bupropion | Cytochrome P450 2C9 | enzyme |
Bupropion | Cytochrome P450 2E1 | enzyme |
Bupropion | Solute carrier family 22 member 2 | transporter |
Bupropion | 5-hydroxytryptamine receptor 3A | target |
Bupropion | Sodium-dependent serotonin transporter | target |
Amiodarone | Beta adrenergic receptor | target |
Amiodarone | HERG human cardiac K+ channel | target |
Amiodarone | Cytochrome P450 2C8 | enzyme |
Amiodarone | Cytochrome P450 2C9 | enzyme |
Amiodarone | Cytochrome P450 2D6 | enzyme |
Amiodarone | Voltage-dependent T-type calcium channel subunit alpha-1I | target |
Amiodarone | Voltage gated L-type calcium channel | target |
Amiodarone | Cytochrome P450 3A4 | enzyme |
Amiodarone | Cytochrome P450 1A2 | enzyme |
Amiodarone | Cytochrome P450 1A1 | enzyme |
Amiodarone | P-glycoprotein 1 | transporter |
Amiodarone | Cytochrome P450 2C19 | enzyme |
Amiodarone | Cytochrome P450 2A6 | enzyme |
Amiodarone | Thyroid hormone receptor | target |
Amiodarone | Peroxisome proliferator-activated receptor gamma | target |
Amiodarone | Bile salt export pump | transporter |
Amiodarone | Solute carrier family 22 member 2 | transporter |
Amiodarone | Cytochrome P450 2J2 | enzyme |
Amiodarone | Peroxisome proliferator-activated receptor alpha | target |
Amiodarone | Peroxisome proliferator-activated receptor gamma coactivator 1-beta | target |
Amiodarone | Serum albumin | carrier |
Clopidogrel | P2Y purinoceptor 12 | target |
Clopidogrel | Cytochrome P450 3A4 | enzyme |
Clopidogrel | Cytochrome P450 2B6 | enzyme |
Clopidogrel | Cytochrome P450 3A5 | enzyme |
Clopidogrel | Cytochrome P450 2C19 | enzyme |
Clopidogrel | Cytochrome P450 2C9 | enzyme |
Clopidogrel | Cytochrome P450 1A2 | enzyme |
Clopidogrel | Cytochrome P450 2C8 | enzyme |
Clopidogrel | Liver carboxylesterase 1 | enzyme |
Clopidogrel | P-glycoprotein 1 | transporter |
Clopidogrel | Solute carrier family 22 member 1 | transporter |
Clopidogrel | Solute carrier family 22 member 2 | transporter |
Clopidogrel | Serum albumin | carrier |
Crizotinib | Cytochrome P450 3A4 | enzyme |
Crizotinib | Cytochrome P450 3A5 | enzyme |
Crizotinib | P-glycoprotein 1 | transporter |
Crizotinib | ALK tyrosine kinase receptor | target |
Crizotinib | Hepatocyte growth factor receptor | target |
Crizotinib | Cytochrome P450 2B6 | enzyme |
Crizotinib | Cytochrome P450 3A Subfamily | enzyme |
Crizotinib | Serum albumin | carrier |
Crizotinib | alpha1-acid glycoprotein | carrier |
Crizotinib | Proto-oncogene tyrosine-protein kinase ROS | target |
Crizotinib | Macrophage-stimulating protein receptor | target |
Lamotrigine | Voltage-gated sodium channel alpha subunit | target |
Lamotrigine | UDP-glucuronosyltransferases (UGTs) | enzyme |
Lamotrigine | P-glycoprotein 1 | transporter |
Lamotrigine | Dihydrofolate reductase | enzyme |
Lamotrigine | 5-hydroxytryptamine receptor 3A | target |
Lamotrigine | Voltage-dependent R-type calcium channel subunit alpha-1E (CACNA1E) | target |
Lamotrigine | Adenosine receptor A1 | target |
Lamotrigine | Adenosine receptor A2a | target |
Lamotrigine | Alpha-1A adrenergic receptor | target |
Lamotrigine | Alpha-2A adrenergic receptor | target |
Lamotrigine | Beta-1 adrenergic receptor | target |
Lamotrigine | D(1) dopamine receptor | target |
Lamotrigine | Dopamine D2 receptor | target |
Lamotrigine | GABA(A) Receptor | target |
Lamotrigine | GABA(A) Receptor Benzodiazepine Binding Site | target |
Lamotrigine | Histamine H1 receptor | target |
Lamotrigine | Kappa-type opioid receptor | target |
Lamotrigine | Acetylcholine receptor subunit alpha | target |
Lamotrigine | 5-hydroxytryptamine receptor 2A | target |
Lamotrigine | Solute carrier family 22 member 2 | transporter |
Lamotrigine | Serum albumin | carrier |
Lamotrigine | Solute carrier family 22 member 1 | transporter |
Lamotrigine | Glutamate receptor 1 | target |
Lamotrigine | Sodium channel protein type 11 subunit alpha | target |
Vandetanib | Vascular endothelial growth factor A | target |
Vandetanib | Epidermal growth factor receptor | target |
Vandetanib | Multidrug resistance-associated protein 1 | transporter |
Vandetanib | ATP-binding cassette sub-family G member 2 | transporter |
Vandetanib | Proto-oncogene tyrosine-protein kinase receptor Ret | target |
Vandetanib | Dimethylaniline monooxygenase [N-oxide-forming] 1 | enzyme |
Vandetanib | Dimethylaniline monooxygenase [N-oxide-forming] 3 | enzyme |
Vandetanib | Protein-tyrosine kinase 6 | target |
Vandetanib | Angiopoietin-1 receptor | target |
Vandetanib | Alpha-1-acid glycoprotein 1 | carrier |
Vandetanib | Serum albumin | carrier |
Vandetanib | Cytochrome P450 3A4 | enzyme |
Vandetanib | Solute carrier family 22 member 2 | transporter |
Vandetanib | P-glycoprotein 1 | transporter |
Vandetanib | Vascular endothelial growth factor receptor 2 | target |
Ranolazine | Cytochrome P450 3A4 | enzyme |
Ranolazine | Cytochrome P450 2D6 | enzyme |
Ranolazine | Bile salt export pump | transporter |
Ranolazine | P-glycoprotein 1 | transporter |
Ranolazine | Sodium channel protein | target |
Ranolazine | Inward rectifier potassium channel | target |
Ranolazine | Voltage gated L-type calcium channel | target |
Ranolazine | Alpha-1 adrenergic receptors | target |
Ranolazine | Beta-1 adrenergic receptor | target |
Ranolazine | Fatty acid | target |
Ranolazine | Alpha-1-acid glycoprotein 1 | carrier |
Ranolazine | Multidrug and toxin extrusion protein 1 | transporter |
Ranolazine | Multidrug and toxin extrusion protein 2 | transporter |
Ranolazine | Plasminogen | target |
Linagliptin | Dipeptidyl peptidase 4 | target |
Linagliptin | Cytochrome P450 3A4 | enzyme |
Linagliptin | P-glycoprotein 1 | transporter |
Linagliptin | Solute carrier family 22 member 1 | transporter |
Linagliptin | Solute carrier family 22 member 2 | transporter |
Linagliptin | Solute carrier family 22 member 3 | transporter |
Erdafitinib | Cytochrome P450 2C9 | enzyme |
Erdafitinib | Cytochrome P450 3A4 | enzyme |
Erdafitinib | Fibroblast growth factor receptor 1 | target |
Erdafitinib | Fibroblast growth factor receptor 2 | target |
Erdafitinib | Fibroblast growth factor receptor 3 | target |
Erdafitinib | Fibroblast growth factor receptor 4 | target |
Erdafitinib | P-glycoprotein 1 | transporter |
Erdafitinib | Solute carrier family 22 member 2 | transporter |
Erdafitinib | Proto-oncogene tyrosine-protein kinase receptor Ret | target |
Erdafitinib | Macrophage colony-stimulating factor 1 receptor | target |
Erdafitinib | Platelet-derived growth factor receptor alpha | target |
Erdafitinib | Platelet-derived growth factor receptor beta | target |
Erdafitinib | Mast/stem cell growth factor receptor Kit | target |
Erdafitinib | Vascular endothelial growth factor receptor 2 | target |
Erdafitinib | alpha1-acid glycoprotein | carrier |
Dronedarone | Alpha-1A adrenergic receptor | target |
Dronedarone | Beta-1 adrenergic receptor | target |
Dronedarone | Alpha-1B adrenergic receptor | target |
Dronedarone | Alpha-1D adrenergic receptor | target |
Dronedarone | Alpha-2A adrenergic receptor | target |
Dronedarone | Alpha-2B adrenergic receptor | target |
Dronedarone | Alpha-2C adrenergic receptor | target |
Dronedarone | Potassium voltage-gated channel subfamily H member 2 | target |
Dronedarone | Voltage-dependent L-type calcium channel subunit alpha-1C | target |
Dronedarone | Voltage-dependent L-type calcium channel subunit alpha-1D | target |
Dronedarone | Voltage-dependent L-type calcium channel subunit alpha-1F | target |
Dronedarone | Voltage-dependent L-type calcium channel subunit alpha-1S | target |
Dronedarone | Voltage-dependent L-type calcium channel subunit beta-1 | target |
Dronedarone | Voltage-dependent L-type calcium channel subunit beta-2 | target |
Dronedarone | Voltage-dependent L-type calcium channel subunit beta-3 | target |
Dronedarone | Voltage-dependent L-type calcium channel subunit beta-4 | target |
Dronedarone | Cytochrome P450 2D6 | enzyme |
Dronedarone | Cytochrome P450 3A4 | enzyme |
Dronedarone | P-glycoprotein 1 | transporter |
Dronedarone | Potassium channel subfamily K member 2 | target |
Dronedarone | Serum albumin | carrier |
Dronedarone | Solute carrier family 22 member 2 | transporter |
Dronedarone | Solute carrier family 22 member 1 | transporter |
Dronedarone | Solute carrier organic anion transporter family member 1B1 | transporter |
Dronedarone | Solute carrier organic anion transporter family member 1B3 | transporter |
Dronedarone | Solute carrier family 22 member 8 | transporter |
Dronedarone | Cytochrome P450 3A5 | enzyme |
Dronedarone | Cytochrome P450 2J2 | enzyme |
Dronedarone | Thyroid hormone receptor alpha | target |
Dronedarone | Sodium channel protein type 5 subunit alpha | target |
Dronedarone | G protein-activated inward rectifier potassium channel 1 | target |
Dronedarone | Potassium voltage-gated channel subfamily KQT member 1 | target |
Dronedarone | Inward rectifier potassium channel | target |
Dronedarone | Sodium/calcium exchanger 1 | target |
Dronedarone | Potassium voltage-gated channel subfamily D member 3 | target |
Dronedarone | Potassium voltage-gated channel subfamily A member 5 | target |
Abemaciclib | Multidrug and toxin extrusion protein 1 | transporter |
Abemaciclib | Multidrug and toxin extrusion protein 2 | transporter |
Abemaciclib | Cyclin-dependent kinase 4 | target |
Abemaciclib | Cyclin-dependent kinase 6 | target |
Abemaciclib | Serum albumin | carrier |
Abemaciclib | alpha1-acid glycoprotein | carrier |
Abemaciclib | Cytochrome P450 3A4 | enzyme |
Abemaciclib | P-glycoprotein 1 | transporter |
Abemaciclib | ATP-binding cassette sub-family G member 2 | transporter |
Abemaciclib | Solute carrier family 22 member 2 | transporter |
Abemaciclib | Cytochrome P450 1A2 | enzyme |
Abemaciclib | Cytochrome P450 2B6 | enzyme |
Abemaciclib | Cytochrome P450 2C8 | enzyme |
Abemaciclib | Cytochrome P450 2C9 | enzyme |
Abemaciclib | Cytochrome P450 2D6 | enzyme |
Ubrogepant | P-glycoprotein 1 | transporter |
Ubrogepant | ATP-binding cassette sub-family G member 2 | transporter |
Ubrogepant | Cytochrome P450 3A4 | enzyme |
Ubrogepant | Cytochrome P450 2C8 | enzyme |
Ubrogepant | Cytochrome P450 2C9 | enzyme |
Ubrogepant | Cytochrome P450 2D6 | enzyme |
Ubrogepant | Cytochrome P450 2C19 | enzyme |
Ubrogepant | Amine oxidase [flavin-containing] A | enzyme |
Ubrogepant | UDP-glucuronosyltransferase 1-1 | enzyme |
Ubrogepant | Solute carrier organic anion transporter family member 1B1 | transporter |
Ubrogepant | Solute carrier organic anion transporter family member 1B3 | transporter |
Ubrogepant | Solute carrier family 22 member 6 | transporter |
Ubrogepant | Solute carrier family 22 member 2 | transporter |
Ubrogepant | Calcitonin gene-related peptide type 1 receptor | target |
Salmeterol | Beta-2 adrenergic receptor | target |
Salmeterol | Cytochrome P450 3A4 | enzyme |
Salmeterol | Cytochrome P450 2C8 | enzyme |
Salmeterol | Cytochrome P450 3A5 | enzyme |
Salmeterol | Cytochrome P450 3A7 | enzyme |
Salmeterol | Beta-1 adrenergic receptor | target |
Salmeterol | Beta-3 adrenergic receptor | target |
Salmeterol | Serum albumin | carrier |
Salmeterol | alpha1-acid glycoprotein | carrier |
Salmeterol | Solute carrier family 22 member 1 | transporter |
Salmeterol | Solute carrier family 22 member 2 | transporter |
Salmeterol | Solute carrier family 22 member 3 | transporter |
Rimegepant | Calcitonin gene-related peptide type 1 receptor | target |
Rimegepant | P-glycoprotein 1 | transporter |
Rimegepant | ATP-binding cassette sub-family G member 2 | transporter |
Rimegepant | Solute carrier organic anion transporter family member 1B1 | transporter |
Rimegepant | Solute carrier family 22 member 8 | transporter |
Rimegepant | Solute carrier organic anion transporter family member 1B3 | transporter |
Rimegepant | Solute carrier family 22 member 2 | transporter |
Rimegepant | Multidrug and toxin extrusion protein 1 | transporter |
Rimegepant | Cytochrome P450 3A4 | enzyme |
Rimegepant | Cytochrome P450 2C9 | enzyme |
Osilodrostat | Cytochrome P450 11B1, mitochondrial | target |
Osilodrostat | Cytochrome P450 11B2, mitochondrial | target |
Osilodrostat | Cytochrome P450 3A4 | enzyme |
Osilodrostat | Cytochrome P450 2B6 | enzyme |
Osilodrostat | Cytochrome P450 2D6 | enzyme |
Osilodrostat | UDP-glucuronosyltransferase 1-4 | enzyme |
Osilodrostat | UDP-glucuronosyltransferase 2B7 | enzyme |
Osilodrostat | UDP-glucuronosyltransferase 2B10 | enzyme |
Osilodrostat | Cytochrome P450 3A5 | enzyme |
Osilodrostat | Cytochrome P450 1A2 | enzyme |
Osilodrostat | Cytochrome P450 2C19 | enzyme |
Osilodrostat | Cytochrome P450 2E1 | enzyme |
Osilodrostat | UDP-glucuronosyltransferase 1A1 | enzyme |
Osilodrostat | Solute carrier organic anion transporter family member 1B1 | transporter |
Osilodrostat | Solute carrier family 22 member 1 | transporter |
Osilodrostat | Solute carrier family 22 member 2 | transporter |
Osilodrostat | Solute carrier family 22 member 6 | transporter |
Osilodrostat | Solute carrier family 22 member 8 | transporter |
Osilodrostat | Multidrug and toxin extrusion protein 1 | transporter |
Cocaine | Sodium-dependent noradrenaline transporter | target |
Cocaine | Sodium channel protein | target |
Cocaine | Sodium-dependent serotonin transporter | target |
Cocaine | Sodium-dependent dopamine transporter | target |
Cocaine | Cytochrome P450 3A4 | enzyme |
Cocaine | Muscarinic acetylcholine receptor M1 | target |
Cocaine | Muscarinic acetylcholine receptor M2 | target |
Cocaine | Cytochrome P450 2D6 | enzyme |
Cocaine | Solute carrier family 22 member 2 | transporter |
Cocaine | Cytochrome P450 2C8 | enzyme |
Cocaine | Sigma non-opioid intracellular receptor 1 | target |
Cocaine | Liver carboxylesterase 1 | target |
Cocaine | Cholinesterase | enzyme |
Cocaine | Sodium-dependent dopamine transporter | transporter |
Cocaine | alpha1-acid glycoprotein | carrier |
Cocaine | Liver carboxylesterase 1 | enzyme |
Methylene blue | Guanylate cyclase soluble subunit alpha-2 | target |
Methylene blue | Nitric oxide synthase, brain | target |
Methylene blue | UDP-glucuronosyltransferase 1-4 | enzyme |
Methylene blue | UDP-glucuronosyltransferase 1-9 | enzyme |
Methylene blue | Cytochrome P450 1A2 | enzyme |
Methylene blue | Cytochrome P450 2B6 | enzyme |
Methylene blue | Cytochrome P450 2C8 | enzyme |
Methylene blue | Cytochrome P450 2C9 | enzyme |
Methylene blue | Cytochrome P450 2C19 | enzyme |
Methylene blue | Cytochrome P450 3A4 | enzyme |
Methylene blue | Cytochrome P450 3A5 | enzyme |
Methylene blue | Serum albumin | carrier |
Methylene blue | P-glycoprotein 1 | transporter |
Methylene blue | Solute carrier family 22 member 2 | transporter |
Methylene blue | Multidrug and toxin extrusion protein 2 | transporter |
Methylene blue | Multidrug and toxin extrusion protein 1 | transporter |
Methylene blue | Flavin reductase (NADPH) | enzyme |
Methylene blue | Cytochrome P450 2D6 | enzyme |
Tucatinib | Receptor tyrosine-protein kinase erbB-2 | target |
Tucatinib | ATP-binding cassette sub-family G member 2 | transporter |
Tucatinib | P-glycoprotein 1 | transporter |
Tucatinib | Solute carrier family 22 member 2 | transporter |
Tucatinib | Multidrug and toxin extrusion protein 1 | transporter |
Tucatinib | Multidrug and toxin extrusion protein 2 | transporter |
Tucatinib | Cytochrome P450 2C8 | enzyme |
Tucatinib | Cytochrome P450 3A Subfamily | enzyme |
Tucatinib | Receptor tyrosine-protein kinase erbB-2 | enzyme |
Tucatinib | Receptor tyrosine-protein kinase erbB-3 | target |
Pemigatinib | Cytochrome P450 3A4 | enzyme |
Pemigatinib | Fibroblast growth factor receptor 1 | target |
Pemigatinib | Fibroblast growth factor receptor 2 | target |
Pemigatinib | Fibroblast growth factor receptor 3 | target |
Pemigatinib | Fibroblast growth factor receptor 4 | target |
Pemigatinib | P-glycoprotein 1 | transporter |
Pemigatinib | ATP-binding cassette sub-family G member 2 | transporter |
Pemigatinib | Solute carrier family 22 member 2 | transporter |
Pemigatinib | Multidrug and toxin extrusion protein 1 | transporter |
Tirbanibulin | Proto-oncogene tyrosine-protein kinase Src | target |
Tirbanibulin | Tubulin beta chain | target |
Tirbanibulin | Cytochrome P450 3A4 | enzyme |
Tirbanibulin | Cytochrome P450 2C8 | enzyme |
Tirbanibulin | Cytochrome P450 1A2 | enzyme |
Tirbanibulin | Cytochrome P450 2B6 | enzyme |
Tirbanibulin | Cytochrome P450 2C9 | enzyme |
Tirbanibulin | Cytochrome P450 2C19 | enzyme |
Tirbanibulin | Cytochrome P450 2D6 | enzyme |
Tirbanibulin | Multidrug and toxin extrusion protein 1 | transporter |
Tirbanibulin | Multidrug and toxin extrusion protein 2 | transporter |
Tirbanibulin | Solute carrier organic anion transporter family member 1B1 | transporter |
Tirbanibulin | Solute carrier organic anion transporter family member 1B3 | transporter |
Tirbanibulin | Solute carrier family 22 member 1 | transporter |
Tirbanibulin | Solute carrier family 22 member 2 | transporter |
Trilaciclib | Solute carrier family 22 member 2 | transporter |
Trilaciclib | Multidrug and toxin extrusion protein 1 | transporter |
Trilaciclib | Multidrug and toxin extrusion protein 2 | transporter |
Trilaciclib | Cytochrome P450 1A2 | enzyme |
Trilaciclib | ATP-binding cassette sub-family G member 2 | transporter |
Trilaciclib | P-glycoprotein 1 | transporter |
Trilaciclib | Cyclin-dependent kinase 4 | target |
Trilaciclib | Cyclin-dependent kinase 6 | target |
Trilaciclib | Cyclin-dependent kinase 9 | target |
Trilaciclib | Cyclin-dependent kinase 2 | target |
Trilaciclib | Cyclin-dependent kinase 5 | target |
Trilaciclib | Cyclin-dependent kinase 7 | target |
Infigratinib | Cytochrome P450 3A4 | enzyme |
Infigratinib | Multidrug and toxin extrusion protein 1 | transporter |
Infigratinib | ATP-binding cassette sub-family G member 2 | transporter |
Infigratinib | Bile salt export pump | transporter |
Infigratinib | Solute carrier family 22 member 1 | transporter |
Infigratinib | Solute carrier family 22 member 2 | transporter |
Infigratinib | Multidrug and toxin extrusion protein 2 | transporter |
Infigratinib | P-glycoprotein 1 | transporter |
Infigratinib | Solute carrier organic anion transporter family member 1B1 | transporter |
Infigratinib | Solute carrier organic anion transporter family member 1B3 | transporter |
Infigratinib | Apolipoproteins | carrier |
Infigratinib | Dimethylaniline monooxygenase [N-oxide-forming] 3 | enzyme |
Infigratinib | Fibroblast growth factor receptor 1 | target |
Infigratinib | Fibroblast growth factor receptor 2 | target |
Infigratinib | Fibroblast growth factor receptor 3 | target |
Infigratinib | Fibroblast growth factor receptor 4 | target |
Romidepsin | Cytochrome P450 3A4 | enzyme |
Romidepsin | Cytochrome P450 3A5 | enzyme |
Romidepsin | P-glycoprotein 1 | transporter |
Romidepsin | Solute carrier organic anion transporter family member 1B3 | transporter |
Romidepsin | Cytochrome P450 1A1 | enzyme |
Romidepsin | Cytochrome P450 2B6 | enzyme |
Romidepsin | Cytochrome P450 2C19 | enzyme |
Romidepsin | Histone deacetylase 1 | target |
Romidepsin | Histone deacetylase 2 | target |
Romidepsin | Histone deacetylase 4 | target |
Romidepsin | Histone deacetylase 6 | target |
Romidepsin | Multidrug resistance-associated protein 1 | target |
Romidepsin | Bile salt export pump | transporter |
Romidepsin | Solute carrier organic anion transporter family member 1B1 | transporter |
Romidepsin | Solute carrier family 22 member 6 | transporter |
Romidepsin | Solute carrier family 22 member 2 | transporter |
Romidepsin | Histone deacetylase | target |
Fexinidazole | Cytochrome P450 1A2 | enzyme |
Fexinidazole | Cytochrome P450 2B6 | enzyme |
Fexinidazole | Cytochrome P450 2C19 | enzyme |
Fexinidazole | Cytochrome P450 3A4 | enzyme |
Fexinidazole | Cytochrome P450 3A5 | enzyme |
Fexinidazole | Dimethylaniline monooxygenase [N-oxide-forming] 3 | enzyme |
Fexinidazole | Cytochrome P450 2D6 | enzyme |
Fexinidazole | Solute carrier organic anion transporter family member 1B1 | transporter |
Fexinidazole | Solute carrier organic anion transporter family member 1B3 | transporter |
Fexinidazole | Solute carrier family 22 member 2 | transporter |
Fexinidazole | Solute carrier family 22 member 6 | transporter |
Fexinidazole | Solute carrier family 22 member 8 | transporter |
Fexinidazole | Multidrug and toxin extrusion protein 1 | transporter |
Fexinidazole | Multidrug and toxin extrusion protein 2 | transporter |
Levoketoconazole | Cytochrome P450 11B1, mitochondrial | target |
Levoketoconazole | Lanosterol 14-alpha demethylase | target |
Levoketoconazole | Cytochrome P450 3A4 | enzyme |
Levoketoconazole | Cytochrome P450 3A5 | enzyme |
Levoketoconazole | Steroid 21-hydroxylase | enzyme |
Levoketoconazole | P-glycoprotein 1 | transporter |
Levoketoconazole | Steroid 17-alpha-hydroxylase/17,20 lyase | target |
Levoketoconazole | Cytochrome P450 11B2, mitochondrial | target |
Levoketoconazole | Cholesterol side-chain cleavage enzyme, mitochondrial | target |
Levoketoconazole | Solute carrier family 22 member 2 | transporter |
Levoketoconazole | Multidrug and toxin extrusion protein 1 | transporter |
Levoketoconazole | Cytochrome P450 2B6 | enzyme |
Levoketoconazole | Cytochrome P450 2C8 | enzyme |
Levoketoconazole | Cytochrome P450 1A2 | enzyme |
Levoketoconazole | Cytochrome P450 7A1 | enzyme |
Levoketoconazole | Cytochrome P450 19A1 | enzyme |
Pacritinib | Cytochrome P450 3A4 | enzyme |
Pacritinib | Cytochrome P450 1A2 | enzyme |
Pacritinib | Tyrosine-protein kinase JAK2 | target |
Pacritinib | Receptor-type tyrosine-protein kinase FLT3 | target |
Pacritinib | P-glycoprotein 1 | transporter |
Pacritinib | ATP-binding cassette sub-family G member 2 | transporter |
Pacritinib | Solute carrier family 22 member 1 | transporter |
Pacritinib | Cytochrome P450 2C19 | enzyme |
Pacritinib | Solute carrier family 22 member 2 | transporter |
Pacritinib | Tyrosine-protein kinase JAK3 | target |
Olaparib | Poly [ADP-ribose] polymerase 1 | target |
Olaparib | Cytochrome P450 3A4 | enzyme |
Olaparib | Cytochrome P450 2B6 | enzyme |
Olaparib | Poly [ADP-ribose] polymerase 2 | target |
Olaparib | Poly [ADP-ribose] polymerase 3 | target |
Olaparib | Cytochrome P450 3A5 | enzyme |
Olaparib | P-glycoprotein 1 | transporter |
Olaparib | ATP-binding cassette sub-family G member 2 | transporter |
Olaparib | Aldo-keto reductase family 1 member C3 | target |
Olaparib | UDP-glucuronosyltransferase 1-1 | enzyme |
Olaparib | Serum albumin | carrier |
Olaparib | Alpha-1-acid glycoprotein 1 | carrier |
Dabrafenib | Cytochrome P450 3A4 | enzyme |
Dabrafenib | Cytochrome P450 2C8 | enzyme |
Dabrafenib | P-glycoprotein 1 | transporter |
Dabrafenib | ATP-binding cassette sub-family G member 2 | transporter |
Dabrafenib | Solute carrier organic anion transporter family member 1B1 | transporter |
Dabrafenib | Solute carrier organic anion transporter family member 1B3 | transporter |
Dabrafenib | Solute carrier family 22 member 6 | transporter |
Dabrafenib | Solute carrier family 22 member 8 | transporter |
Dabrafenib | Serine/threonine-protein kinase B-raf | target |
Dabrafenib | RAF proto-oncogene serine/threonine-protein kinase | target |
Dabrafenib | Serine/threonine-protein kinase SIK1 | target |
Dabrafenib | Serine/threonine-protein kinase Nek11 | target |
Dabrafenib | LIM domain kinase 1 | target |
Dabrafenib | Cytochrome P450 2B6 | enzyme |
Dabrafenib | Cytochrome P450 2C9 | enzyme |
Dabrafenib | Cytochrome P450 2C19 | enzyme |
Dabrafenib | Cytochrome P450 1A2 | enzyme |
Dabrafenib | Serum albumin | carrier |
Dabrafenib | Solute carrier organic anion transporter family member 1A2 | transporter |
Dabrafenib | Solute carrier family 22 member 2 | transporter |
Dabrafenib | UDP-glucuronosyltransferase 1-1 | enzyme |
Tepotinib | P-glycoprotein 1 | transporter |
Tepotinib | Cytochrome P450 3A4 | enzyme |
Tepotinib | Cytochrome P450 2C8 | enzyme |
Tepotinib | ATP-binding cassette sub-family G member 2 | transporter |
Tepotinib | Hepatocyte growth factor receptor | target |
Tepotinib | Nischarin | target |
Tepotinib | Melatonin receptor type 1B | target |
Tepotinib | Serum albumin | carrier |
Tepotinib | Alpha-1-acid glycoprotein 1 | carrier |
Tepotinib | Solute carrier family 22 member 1 | transporter |
Tepotinib | Solute carrier family 22 member 2 | transporter |
Tepotinib | Multidrug and toxin extrusion protein 1 | transporter |
Tepotinib | Multidrug and toxin extrusion protein 2 | transporter |
Tepotinib | Bile salt export pump | transporter |
Tepotinib | Cytochrome P450 2C9 | enzyme |
Amifampridine | Arylamine N-acetyltransferase 1 | enzyme |
Amifampridine | Arylamine N-acetyltransferase 2 | enzyme |
Amifampridine | Potassium voltage-gated channel subfamily A member 1 | target |
Amifampridine | Solute carrier family 22 member 2 | transporter |
Olutasidenib | Isocitrate dehydrogenase [NADP] cytoplasmic | target |
Olutasidenib | Cytochrome P450 3A4 | enzyme |
Olutasidenib | Cytochrome P450 2C8 | enzyme |
Olutasidenib | Cytochrome P450 2C9 | enzyme |
Olutasidenib | Cytochrome P450 1A2 | enzyme |
Olutasidenib | Cytochrome P450 2C19 | enzyme |
Olutasidenib | P-glycoprotein 1 | transporter |
Olutasidenib | ATP-binding cassette sub-family G member 2 | transporter |
Olutasidenib | Solute carrier organic anion transporter family member 1B1 | transporter |
Olutasidenib | Solute carrier organic anion transporter family member 1B3 | transporter |
Olutasidenib | Solute carrier family 22 member 8 | transporter |
Olutasidenib | Solute carrier family 22 member 2 | transporter |
Olutasidenib | Multidrug and toxin extrusion protein 1 | transporter |
Olutasidenib | Multidrug and toxin extrusion protein 2 | transporter |
Olutasidenib | Cytochrome P450 2B6 | enzyme |
Tezacaftor | Cytochrome P450 3A4 | enzyme |
Tezacaftor | Cytochrome P450 3A5 | enzyme |
Tezacaftor | Cystic fibrosis transmembrane conductance regulator | target |
Tezacaftor | P-glycoprotein 1 | transporter |
Tezacaftor | ATP-binding cassette sub-family G member 2 | transporter |
Tezacaftor | Solute carrier family 22 member 2 | transporter |
Tezacaftor | Solute carrier family 22 member 6 | transporter |
Tezacaftor | Solute carrier family 22 member 8 | transporter |
Tezacaftor | Solute carrier organic anion transporter family member 1B1 | transporter |
Tezacaftor | Cytochrome P450 1A2 | enzyme |
Tezacaftor | Cytochrome P450 2B6 | enzyme |
Tezacaftor | Cytochrome P450 2C8 | enzyme |
Tezacaftor | Cytochrome P450 2C9 | enzyme |
Tezacaftor | Cytochrome P450 2C19 | enzyme |
Tezacaftor | Cytochrome P450 2D6 | enzyme |
Tezacaftor | Solute carrier organic anion transporter family member 1B3 | transporter |
Encorafenib | Cytochrome P450 3A4 | enzyme |
Encorafenib | Cytochrome P450 2C19 | enzyme |
Encorafenib | Cytochrome P450 2D6 | enzyme |
Encorafenib | Serine/threonine-protein kinase B-raf | target |
Encorafenib | G1/S-specific cyclin-D1 | target |
Encorafenib | UDP-glucuronosyltransferase 1-1 | enzyme |
Encorafenib | Serum albumin | carrier |
Encorafenib | Cytochrome P450 1A2 | enzyme |
Encorafenib | Cytochrome P450 2B6 | enzyme |
Encorafenib | Cytochrome P450 2C8 | enzyme |
Encorafenib | Cytochrome P450 2C9 | enzyme |
Encorafenib | Cytochrome P450 3A5 | enzyme |
Encorafenib | Cytochrome P450 3A7 | enzyme |
Encorafenib | P-glycoprotein 1 | transporter |
Encorafenib | Solute carrier family 22 member 2 | transporter |
Encorafenib | ATP-binding cassette sub-family G member 2 | transporter |
Encorafenib | Solute carrier family 22 member 6 | transporter |
Encorafenib | Solute carrier family 22 member 8 | transporter |
Encorafenib | Solute carrier organic anion transporter family member 1B1 | transporter |
Encorafenib | Solute carrier organic anion transporter family member 1B3 | transporter |
Encorafenib | RAF proto-oncogene serine/threonine-protein kinase | target |
Encorafenib | Mitogen-activated protein kinase 8 | target |
Encorafenib | Mitogen-activated protein kinase 9 | target |
Encorafenib | Mitogen-activated protein kinase 10 | target |
Encorafenib | LIM domain kinase 1 | target |
Encorafenib | LIM domain kinase 2 | target |
Encorafenib | Dual specificity mitogen-activated protein kinase kinase 4 | target |
Encorafenib | Serine/threonine-protein kinase 36 | target |
Capivasertib | Cytochrome P450 3A4 | enzyme |
Capivasertib | UDP-glucuronosyltransferase 2B7 | enzyme |
Capivasertib | RAC-alpha serine/threonine-protein kinase | target |
Capivasertib | RAC-beta serine/threonine-protein kinase | target |
Capivasertib | RAC-gamma serine/threonine-protein kinase | target |
Capivasertib | ATP-binding cassette sub-family G member 2 | transporter |
Capivasertib | Solute carrier organic anion transporter family member 1B1 | transporter |
Capivasertib | Solute carrier organic anion transporter family member 1B3 | transporter |
Capivasertib | Solute carrier family 22 member 8 | transporter |
Capivasertib | Multidrug and toxin extrusion protein 1 | transporter |
Capivasertib | Multidrug and toxin extrusion protein 2 | transporter |
Capivasertib | Solute carrier family 22 member 2 | transporter |
Isavuconazonium | Cytochrome P450 3A4 | enzyme |
Isavuconazonium | P-glycoprotein 1 | transporter |
Isavuconazonium | Cytochrome P450 3A5 | enzyme |
Isavuconazonium | Cholinesterase | enzyme |
Isavuconazonium | Cytochrome P450 2C8 | enzyme |
Isavuconazonium | Cytochrome P450 2C9 | enzyme |
Isavuconazonium | Cytochrome P450 2C19 | enzyme |
Isavuconazonium | Cytochrome P450 2D6 | enzyme |
Isavuconazonium | Cytochrome P450 2B6 | enzyme |
Isavuconazonium | ATP-binding cassette sub-family G member 2 | transporter |
Isavuconazonium | Solute carrier family 22 member 2 | transporter |
Isavuconazonium | Lanosterol 14-alpha demethylase | target |
Isavuconazonium | Serum albumin | carrier |
Givinostat | Histone deacetylase | target |
Givinostat | Cytochrome P450 3A4 | enzyme |
Givinostat | Solute carrier family 22 member 2 | transporter |
Givinostat | Cytochrome P450 1A2 | enzyme |
Givinostat | Cytochrome P450 2B6 | enzyme |
Givinostat | Histone deacetylase 1 | target |
Givinostat | Tyrosine-protein kinase JAK2 | target |
Mavorixafor | C-X-C chemokine receptor type 4 | target |
Mavorixafor | Cytochrome P450 3A4 | enzyme |
Mavorixafor | Cytochrome P450 2D6 | enzyme |
Mavorixafor | Cytochrome P450 3A5 | enzyme |
Mavorixafor | Cytochrome P450 2C19 | enzyme |
Mavorixafor | Cytochrome P450 2B6 | enzyme |
Mavorixafor | Cytochrome P450 1A2 | enzyme |
Mavorixafor | Cytochrome P450 2C8 | enzyme |
Mavorixafor | Cytochrome P450 2C9 | enzyme |
Mavorixafor | P-glycoprotein 1 | transporter |
Mavorixafor | Solute carrier family 22 member 2 | transporter |
Mavorixafor | Multidrug and toxin extrusion protein 1 | transporter |
Sofpironium | Muscarinic acetylcholine receptor M3 | target |
Sofpironium | Cytochrome P450 2D6 | enzyme |
Sofpironium | Cytochrome P450 3A4 | enzyme |
Sofpironium | Muscarinic acetylcholine receptor | target |
Sofpironium | Solute carrier family 22 member 1 | transporter |
Sofpironium | Solute carrier family 22 member 2 | transporter |
Sofpironium | Multidrug and toxin extrusion protein 1 | transporter |