| Chlorpromazine | approved, investigational, vet_approved | unknown | target | binder | Details |
| Thalidomide | approved, investigational, withdrawn | yes | target | binder | Details |
| Imidafenacin | investigational | no | carrier | substrate | Details |
| Neratinib | approved, investigational | no | carrier | substrate | Details |
| Vancomycin | approved | no | carrier | substrate | Details |
| Abemaciclib | approved, investigational | unknown | carrier | binder | Details |
| Ibrutinib | approved | no | carrier | substrate | Details |
| Vinflunine | approved, investigational | no | carrier | substrate | Details |
| Patisiran | approved, investigational | unknown | carrier | ligand | Details |
| Atomoxetine | approved | no | carrier | binder | Details |
| Ipratropium | approved, experimental | no | carrier | binder | Details |
| Alprazolam | approved, illicit, investigational | unknown | carrier | binder | Details |
| Spironolactone | approved | unknown | carrier | binder | Details |
| Duloxetine | approved | unknown | carrier | ligand | Details |
| Oxycodone | approved, illicit, investigational | unknown | carrier | binder | Details |
| Fentanyl | approved, illicit, investigational, vet_approved | unknown | carrier | binder | Details |
| Irbesartan | approved, investigational | unknown | carrier | binder | Details |
| Solifenacin | approved | unknown | carrier | binder | Details |
| Labetalol | approved | unknown | carrier | substrate | Details |
| Nadolol | approved | unknown | carrier | binder | Details |
| Hydroxychloroquine | approved | unknown | carrier | binder | Details |
| Rifampin | approved | unknown | carrier | binder | Details |
| Istradefylline | approved, investigational | unknown | carrier | binder | Details |
| Flecainide | approved, withdrawn | unknown | carrier | binder | Details |
| Argatroban | approved, investigational | unknown | carrier | binder | Details |
| Asenapine | approved | unknown | carrier | binder | Details |
| Atazanavir | approved, investigational | no | carrier | binder | Details |
| Acalabrutinib | approved, investigational | unknown | carrier | binder | Details |
| Terbinafine | approved, investigational, vet_approved | unknown | carrier | binder | Details |
| Fexofenadine | approved, investigational | unknown | carrier | substrate | Details |
| Nifedipine | approved | unknown | carrier | binder | Details |
| Salmeterol | approved | unknown | carrier | binder | Details |
| Chloroquine | approved, investigational, vet_approved | unknown | carrier | binder | Details |
| Favipiravir | approved, investigational | unknown | carrier | carrier | Details |
| Cocaine | approved, illicit | unknown | carrier | binder | Details |
| Selumetinib | approved, investigational | unknown | carrier | carrier | Details |
| Ripretinib | approved | unknown | carrier | binder | Details |
| Indapamide | approved | unknown | carrier | binder | Details |
| Remoxipride | approved, withdrawn | unknown | carrier | binder | Details |
| Pindolol | approved, investigational | unknown | carrier | binder | Details |
| Benzocaine | approved, investigational | unknown | carrier | binder | Details |
| Glycopyrronium | approved, investigational, vet_approved | unknown | carrier | binder | Details |
| Macitentan | approved | no | carrier | binder | Details |
| Terfenadine | approved, withdrawn | unknown | carrier | binderregulator | Details |
| Carbinoxamine | approved | unknown | carrier | binderregulator | Details |
| Crizotinib | approved, investigational | unknown | carrier | binder | Details |
| Dolutegravir | approved | no | carrier | binder | Details |
| Erdafitinib | approved, investigational | no | carrier | binder | Details |
| Glasdegib | approved, investigational | no | carrier | binder | Details |
| Nirogacestat | approved, investigational | no | carrier | binder | Details |