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PT770615E - Processo para a preparacao de di-haloazolopirimidinas - Google Patents

Processo para a preparacao de di-haloazolopirimidinas

Info

Publication number
PT770615E
PT770615E PT96307528T PT96307528T PT770615E PT 770615 E PT770615 E PT 770615E PT 96307528 T PT96307528 T PT 96307528T PT 96307528 T PT96307528 T PT 96307528T PT 770615 E PT770615 E PT 770615E
Authority
PT
Portugal
Prior art keywords
haloazolopyrimidines
preparation
Prior art date
Application number
PT96307528T
Other languages
English (en)
Inventor
Karl-Otto Stumm
Gunther Krummel
Klaus-Jurgen Pees
Peter Heinz Rudi Liers
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of PT770615E publication Critical patent/PT770615E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PT96307528T 1995-10-27 1996-10-16 Processo para a preparacao de di-haloazolopirimidinas PT770615E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US802295P 1995-10-27 1995-10-27

Publications (1)

Publication Number Publication Date
PT770615E true PT770615E (pt) 2003-10-31

Family

ID=21729405

Family Applications (1)

Application Number Title Priority Date Filing Date
PT96307528T PT770615E (pt) 1995-10-27 1996-10-16 Processo para a preparacao de di-haloazolopirimidinas

Country Status (22)

Country Link
US (1) US5808066A (pt)
EP (1) EP0770615B1 (pt)
JP (1) JP4018182B2 (pt)
KR (1) KR100443182B1 (pt)
AR (1) AR004122A1 (pt)
AT (1) ATE243211T1 (pt)
BR (1) BR9605258A (pt)
CA (1) CA2188905C (pt)
DE (1) DE69628712T2 (pt)
DK (1) DK0770615T3 (pt)
ES (1) ES2202419T3 (pt)
HU (1) HU217773B (pt)
IL (1) IL119496A (pt)
MX (1) MX9604882A (pt)
PT (1) PT770615E (pt)
RU (1) RU2147584C1 (pt)
SG (1) SG55239A1 (pt)
SI (1) SI0770615T1 (pt)
SK (1) SK284071B6 (pt)
TR (1) TR199600792A2 (pt)
UA (1) UA48132C2 (pt)
ZA (1) ZA968957B (pt)

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AU750489B2 (en) * 1998-02-11 2002-07-18 Wyeth Holdings Corporation Fungicidal 7-alkyl-triazolopyrimidines
US6117865A (en) * 1998-09-10 2000-09-12 American Cyanamid Company Fungicidal trifluorophenyl-triazolopyrimidines
US6156925A (en) * 1998-09-25 2000-12-05 American Cyanamid Company Process for the preparation of halogenated phenylmaloates
US6380202B1 (en) * 1998-09-25 2002-04-30 Basf Aktiengesellschaft Fungicidal fluoro-substituted 7-heterocyclyl-triazolopyrimidines
US6242451B1 (en) * 1998-09-25 2001-06-05 Klaus-Juergen Pees Fungicidal trihalophenyl-triazolopyrimidines
US6559151B2 (en) 2000-05-08 2003-05-06 Basf Aktiengesellschaft 6-(2-trifluoromethyl-phenyl)-triazolopyrimidines
US7683071B2 (en) * 2000-07-26 2010-03-23 Taro Pharmaceuticals Industries Ltd. Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid
US6756379B2 (en) 2001-07-26 2004-06-29 Taro Pharmaceutical Industries Ltd. Non-sedating barbiturate compounds as neuroprotective agents
US6939873B2 (en) * 2000-07-26 2005-09-06 Taro Pharmaceuticals Industries Limited Non-sedating barbituric acid derivatives
DE10063115A1 (de) * 2000-12-18 2002-06-27 Bayer Ag Triazolopyrimidine
JP2002249492A (ja) * 2000-12-22 2002-09-06 Nippon Bayer Agrochem Co Ltd トリアゾロピリミジン類
DE10121101A1 (de) * 2001-04-27 2002-10-31 Bayer Ag Triazolopyrimidine
ATE353901T1 (de) 2001-07-05 2007-03-15 Basf Ag Fungizide triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
WO2003008416A1 (en) 2001-07-18 2003-01-30 Basf Aktiengesellschaft Substituted 6-(2-methoxyphenyl) triazolopyrimides as fungicides
UA76486C2 (en) 2001-07-26 2006-08-15 Basf Ag 7-amino triazolopyrimidines, a process of praparation, a fungicidal preparations based thereon and a method to control phytopathogenic fungi
ES2287312T3 (es) 2001-09-04 2007-12-16 Sumitomo Chemical Company, Limited Imidazo(1,2-a)pirimidinas y composiciones fungicidas que las contienen.
ATE384064T1 (de) 2002-03-21 2008-02-15 Basf Ag Fungizide triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
BR0317289A (pt) * 2002-12-11 2005-11-08 Taro Pharma Ind Método para tratar distúrbios do movimento usando derivados do ácido barbitúrico
ATE398452T1 (de) * 2003-09-24 2008-07-15 Wyeth Corp 6-aryl-7-halo-imidazoä1,2-aüpyrimidine als mittel gegen krebs
US7419982B2 (en) * 2003-09-24 2008-09-02 Wyeth Holdings Corporation Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
RU2006107579A (ru) * 2003-09-24 2007-10-27 Вайет Холдингз Корпорейшн (Us) 6-[(замещенный)фенил]триазолопиримидины в качестве противораковых препаратов
MY179926A (en) * 2003-12-08 2020-11-19 Wyeth Corp Process for the preparation of tubulin inhibitors
TW200533670A (en) * 2003-12-19 2005-10-16 Basf Ag 6-(aminocarbonylphenyl)triazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
DE102004007076A1 (de) * 2004-02-13 2005-08-25 Bayer Cropscience Ag Imidazolopyrimidine
CN1930166B (zh) * 2004-03-10 2011-05-25 巴斯福股份公司 5,6-二烷基-7-氨基三唑并嘧啶、其制备方法及其在防治致病性真菌中的用途以及包含这些化合物的组合物
DE502005009861D1 (de) * 2004-03-10 2010-08-19 Basf Se 5,6-dialkyl-7-amino-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
PE20060020A1 (es) * 2004-03-30 2006-03-10 Basf Ag 5-6-cicloalquil-7-amino-triazolopirimidinas para combatir hongos fitopatogenos y procedimientos para su obtencion
CA2572797A1 (en) * 2004-07-02 2006-01-12 Daniella Gutman A process for preparing 1-methoxymethyl-5,5-diphenylbarbituric acid
EP1856118A1 (de) * 2005-03-01 2007-11-21 Basf Aktiengesellschaft 5,6-dialkyl-7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
EP1856121A1 (de) * 2005-03-01 2007-11-21 Basf Aktiengesellschaft 5,6-dialkyl-7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
JP2008536806A (ja) * 2005-03-01 2008-09-11 ビーエーエスエフ ソシエタス・ヨーロピア 5,6−ジアルキル−7−アミノアゾロピリミジン、それらの製造方法、植物病原性菌類を防除するためのそれらの使用、および該化合物を含む薬剤
EP1856122A2 (de) * 2005-03-02 2007-11-21 Basf Aktiengesellschaft 2-substituierte 7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
US20080176744A1 (en) * 2005-03-10 2008-07-24 Basf Aktiengesellschaft Use of 4-Aminopyrimidines for Controlling Harmful Fungi, Novel 4-Aminopyrimidines, Processes for Their Preparation and Compositions Comprising Them
JP2008533099A (ja) * 2005-03-18 2008-08-21 ビーエーエスエフ ソシエタス・ヨーロピア 5−ハロ−2,4,6−トリフルオロイソフタル酸の製造方法
CN101208287A (zh) * 2005-06-27 2008-06-25 巴斯福股份公司 生产取代的苯基丙二酸酯的方法,新的苯基丙二酸酯及其用途
CN101208289A (zh) * 2005-06-27 2008-06-25 巴斯福股份公司 生产取代的苯基丙二酸酯中间体化合物的方法及其在生产5,7-二羟基-6-(2,4,6-三氟苯基)[1,2,4]三唑并[1,5-a]嘧啶中的用途
WO2008066704A2 (en) * 2006-11-14 2008-06-05 Taro Pharmaceuticals North America, Inc. Method of improving bioavailability for non-sedating barbiturates
EP2111404A1 (de) * 2007-01-11 2009-10-28 Basf Se Verfahren zur herstellung arylsubstituierter anellierter pyrimidine
WO2011082271A2 (en) * 2009-12-30 2011-07-07 Arqule, Inc. Substituted triazolo-pyrimidine compounds

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AU557300B2 (en) * 1982-03-16 1986-12-18 Farmitalia Carlo Erba S.P.A. Substituted 1h-pyrazolo(1,5-alpha)pyrimidines and processes for their preparation
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US4910306A (en) * 1987-11-09 1990-03-20 The Dow Chemical Company Preparation of substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
US4892945A (en) * 1987-12-21 1990-01-09 Ciba-Geigy Corporation Isoindoline pigments containing at least one triazolopyrimidone radical
US5006656A (en) * 1990-02-26 1991-04-09 Dowelanco Preparation of 5,7-dihydroxy-1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
ATE174917T1 (de) * 1991-04-22 1999-01-15 Otsuka Pharma Co Ltd Pyrazolo(1,5-a>pyrimidinderivate und sie enthaltende antiinflammatorische mittel
US5356897A (en) * 1991-09-09 1994-10-18 Fujisawa Pharmaceutical Co., Ltd. 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines
US5177206A (en) * 1991-10-08 1993-01-05 Dowelanco Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides
TW224044B (pt) * 1991-12-30 1994-05-21 Shell Internat Res Schappej B V
IL108731A (en) * 1993-03-04 1997-03-18 Shell Int Research 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
RU2066295C1 (ru) * 1993-05-19 1996-09-10 Институт структурной макрокинетики РАН Способ получения порошкового материала на основе карбида титана
EP0628559B1 (en) * 1993-06-10 2002-04-03 Beiersdorf-Lilly GmbH Pyrimidine compounds and their use as pharmaceuticals
AU681913B2 (en) * 1993-10-18 1997-09-11 Dow Agrosciences Llc Process for preparing N-(2,6-dichloro-3-methylphenyl)-5-7-dihalo(1,2,4)triazolo(1, 5A)pyrimidine-2-sulfonamide by cyclization and halo-dehydroxylation

Also Published As

Publication number Publication date
ES2202419T3 (es) 2004-04-01
JP4018182B2 (ja) 2007-12-05
HUP9602957A3 (en) 1998-01-28
EP0770615A1 (en) 1997-05-02
IL119496A (en) 2001-07-24
SK284071B6 (sk) 2004-09-08
SK137796A3 (en) 1997-05-07
MX9604882A (es) 1997-04-30
HU9602957D0 (en) 1996-12-30
CA2188905C (en) 2005-12-06
US5808066A (en) 1998-09-15
JPH09124651A (ja) 1997-05-13
TR199600792A2 (tr) 1997-05-21
DK0770615T3 (da) 2003-07-14
SI0770615T1 (en) 2003-12-31
HUP9602957A2 (en) 1997-06-30
DE69628712T2 (de) 2004-04-29
ATE243211T1 (de) 2003-07-15
RU2147584C1 (ru) 2000-04-20
KR970021081A (ko) 1997-05-28
ZA968957B (en) 1998-04-24
UA48132C2 (uk) 2002-08-15
SG55239A1 (en) 1998-12-21
CA2188905A1 (en) 1997-04-28
BR9605258A (pt) 1998-07-21
AR004122A1 (es) 1998-09-30
DE69628712D1 (de) 2003-07-24
EP0770615B1 (en) 2003-06-18
KR100443182B1 (ko) 2005-04-19
HU217773B (hu) 2000-04-28
IL119496A0 (en) 1997-01-10

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