DK0770615T3 - Fremgangsmåde til fremstilling af dihalogenazolopyrimidiner - Google Patents
Fremgangsmåde til fremstilling af dihalogenazolopyrimidinerInfo
- Publication number
- DK0770615T3 DK0770615T3 DK96307528T DK96307528T DK0770615T3 DK 0770615 T3 DK0770615 T3 DK 0770615T3 DK 96307528 T DK96307528 T DK 96307528T DK 96307528 T DK96307528 T DK 96307528T DK 0770615 T3 DK0770615 T3 DK 0770615T3
- Authority
- DK
- Denmark
- Prior art keywords
- dihalogenazolopyrimidines
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US802295P | 1995-10-27 | 1995-10-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0770615T3 true DK0770615T3 (da) | 2003-07-14 |
Family
ID=21729405
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK96307528T DK0770615T3 (da) | 1995-10-27 | 1996-10-16 | Fremgangsmåde til fremstilling af dihalogenazolopyrimidiner |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US5808066A (da) |
| EP (1) | EP0770615B1 (da) |
| JP (1) | JP4018182B2 (da) |
| KR (1) | KR100443182B1 (da) |
| AR (1) | AR004122A1 (da) |
| AT (1) | ATE243211T1 (da) |
| BR (1) | BR9605258A (da) |
| CA (1) | CA2188905C (da) |
| DE (1) | DE69628712T2 (da) |
| DK (1) | DK0770615T3 (da) |
| ES (1) | ES2202419T3 (da) |
| HU (1) | HU217773B (da) |
| IL (1) | IL119496A (da) |
| MX (1) | MX9604882A (da) |
| PT (1) | PT770615E (da) |
| RU (1) | RU2147584C1 (da) |
| SG (1) | SG55239A1 (da) |
| SI (1) | SI0770615T1 (da) |
| SK (1) | SK284071B6 (da) |
| TR (1) | TR199600792A2 (da) |
| UA (1) | UA48132C2 (da) |
| ZA (1) | ZA968957B (da) |
Families Citing this family (40)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6117876A (en) * | 1997-04-14 | 2000-09-12 | American Cyanamid Company | Fungicidal trifluorophenyl-triazolopyrimidines |
| AU750489B2 (en) * | 1998-02-11 | 2002-07-18 | Wyeth Holdings Corporation | Fungicidal 7-alkyl-triazolopyrimidines |
| US6117865A (en) * | 1998-09-10 | 2000-09-12 | American Cyanamid Company | Fungicidal trifluorophenyl-triazolopyrimidines |
| US6156925A (en) * | 1998-09-25 | 2000-12-05 | American Cyanamid Company | Process for the preparation of halogenated phenylmaloates |
| US6380202B1 (en) * | 1998-09-25 | 2002-04-30 | Basf Aktiengesellschaft | Fungicidal fluoro-substituted 7-heterocyclyl-triazolopyrimidines |
| US6242451B1 (en) * | 1998-09-25 | 2001-06-05 | Klaus-Juergen Pees | Fungicidal trihalophenyl-triazolopyrimidines |
| US6559151B2 (en) | 2000-05-08 | 2003-05-06 | Basf Aktiengesellschaft | 6-(2-trifluoromethyl-phenyl)-triazolopyrimidines |
| US7683071B2 (en) * | 2000-07-26 | 2010-03-23 | Taro Pharmaceuticals Industries Ltd. | Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid |
| US6756379B2 (en) | 2001-07-26 | 2004-06-29 | Taro Pharmaceutical Industries Ltd. | Non-sedating barbiturate compounds as neuroprotective agents |
| US6939873B2 (en) * | 2000-07-26 | 2005-09-06 | Taro Pharmaceuticals Industries Limited | Non-sedating barbituric acid derivatives |
| DE10063115A1 (de) * | 2000-12-18 | 2002-06-27 | Bayer Ag | Triazolopyrimidine |
| JP2002249492A (ja) * | 2000-12-22 | 2002-09-06 | Nippon Bayer Agrochem Co Ltd | トリアゾロピリミジン類 |
| DE10121101A1 (de) * | 2001-04-27 | 2002-10-31 | Bayer Ag | Triazolopyrimidine |
| ATE353901T1 (de) | 2001-07-05 | 2007-03-15 | Basf Ag | Fungizide triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel |
| WO2003008416A1 (en) | 2001-07-18 | 2003-01-30 | Basf Aktiengesellschaft | Substituted 6-(2-methoxyphenyl) triazolopyrimides as fungicides |
| UA76486C2 (en) | 2001-07-26 | 2006-08-15 | Basf Ag | 7-amino triazolopyrimidines, a process of praparation, a fungicidal preparations based thereon and a method to control phytopathogenic fungi |
| ES2287312T3 (es) | 2001-09-04 | 2007-12-16 | Sumitomo Chemical Company, Limited | Imidazo(1,2-a)pirimidinas y composiciones fungicidas que las contienen. |
| ATE384064T1 (de) | 2002-03-21 | 2008-02-15 | Basf Ag | Fungizide triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel |
| BR0317289A (pt) * | 2002-12-11 | 2005-11-08 | Taro Pharma Ind | Método para tratar distúrbios do movimento usando derivados do ácido barbitúrico |
| ATE398452T1 (de) * | 2003-09-24 | 2008-07-15 | Wyeth Corp | 6-aryl-7-halo-imidazoä1,2-aüpyrimidine als mittel gegen krebs |
| US7419982B2 (en) * | 2003-09-24 | 2008-09-02 | Wyeth Holdings Corporation | Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts |
| RU2006107579A (ru) * | 2003-09-24 | 2007-10-27 | Вайет Холдингз Корпорейшн (Us) | 6-[(замещенный)фенил]триазолопиримидины в качестве противораковых препаратов |
| MY179926A (en) * | 2003-12-08 | 2020-11-19 | Wyeth Corp | Process for the preparation of tubulin inhibitors |
| TW200533670A (en) * | 2003-12-19 | 2005-10-16 | Basf Ag | 6-(aminocarbonylphenyl)triazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds |
| DE102004007076A1 (de) * | 2004-02-13 | 2005-08-25 | Bayer Cropscience Ag | Imidazolopyrimidine |
| CN1930166B (zh) * | 2004-03-10 | 2011-05-25 | 巴斯福股份公司 | 5,6-二烷基-7-氨基三唑并嘧啶、其制备方法及其在防治致病性真菌中的用途以及包含这些化合物的组合物 |
| DE502005009861D1 (de) * | 2004-03-10 | 2010-08-19 | Basf Se | 5,6-dialkyl-7-amino-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel |
| PE20060020A1 (es) * | 2004-03-30 | 2006-03-10 | Basf Ag | 5-6-cicloalquil-7-amino-triazolopirimidinas para combatir hongos fitopatogenos y procedimientos para su obtencion |
| CA2572797A1 (en) * | 2004-07-02 | 2006-01-12 | Daniella Gutman | A process for preparing 1-methoxymethyl-5,5-diphenylbarbituric acid |
| EP1856118A1 (de) * | 2005-03-01 | 2007-11-21 | Basf Aktiengesellschaft | 5,6-dialkyl-7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel |
| EP1856121A1 (de) * | 2005-03-01 | 2007-11-21 | Basf Aktiengesellschaft | 5,6-dialkyl-7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel |
| JP2008536806A (ja) * | 2005-03-01 | 2008-09-11 | ビーエーエスエフ ソシエタス・ヨーロピア | ５，６−ジアルキル−７−アミノアゾロピリミジン、それらの製造方法、植物病原性菌類を防除するためのそれらの使用、および該化合物を含む薬剤 |
| EP1856122A2 (de) * | 2005-03-02 | 2007-11-21 | Basf Aktiengesellschaft | 2-substituierte 7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel |
| US20080176744A1 (en) * | 2005-03-10 | 2008-07-24 | Basf Aktiengesellschaft | Use of 4-Aminopyrimidines for Controlling Harmful Fungi, Novel 4-Aminopyrimidines, Processes for Their Preparation and Compositions Comprising Them |
| JP2008533099A (ja) * | 2005-03-18 | 2008-08-21 | ビーエーエスエフ ソシエタス・ヨーロピア | ５−ハロ−２，４，６−トリフルオロイソフタル酸の製造方法 |
| CN101208287A (zh) * | 2005-06-27 | 2008-06-25 | 巴斯福股份公司 | 生产取代的苯基丙二酸酯的方法，新的苯基丙二酸酯及其用途 |
| CN101208289A (zh) * | 2005-06-27 | 2008-06-25 | 巴斯福股份公司 | 生产取代的苯基丙二酸酯中间体化合物的方法及其在生产5,7-二羟基-6-(2,4,6-三氟苯基)[1,2,4]三唑并[1,5-a]嘧啶中的用途 |
| WO2008066704A2 (en) * | 2006-11-14 | 2008-06-05 | Taro Pharmaceuticals North America, Inc. | Method of improving bioavailability for non-sedating barbiturates |
| EP2111404A1 (de) * | 2007-01-11 | 2009-10-28 | Basf Se | Verfahren zur herstellung arylsubstituierter anellierter pyrimidine |
| WO2011082271A2 (en) * | 2009-12-30 | 2011-07-07 | Arqule, Inc. | Substituted triazolo-pyrimidine compounds |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3907799A (en) * | 1971-08-16 | 1975-09-23 | Icn Pharmaceuticals | Xanthine oxidase inhibitors |
| AU557300B2 (en) * | 1982-03-16 | 1986-12-18 | Farmitalia Carlo Erba S.P.A. | Substituted 1h-pyrazolo(1,5-alpha)pyrimidines and processes for their preparation |
| JPS5962593A (ja) * | 1982-09-30 | 1984-04-10 | Ss Pharmaceut Co Ltd | ３―置換―５，７―ジクロルトリアゾロピリミジン誘導体 |
| DE3522463A1 (de) * | 1985-06-22 | 1987-01-02 | Bayer Ag | Herbizide mittel |
| US4910306A (en) * | 1987-11-09 | 1990-03-20 | The Dow Chemical Company | Preparation of substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides |
| US4892945A (en) * | 1987-12-21 | 1990-01-09 | Ciba-Geigy Corporation | Isoindoline pigments containing at least one triazolopyrimidone radical |
| US5006656A (en) * | 1990-02-26 | 1991-04-09 | Dowelanco | Preparation of 5,7-dihydroxy-1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides |
| ATE174917T1 (de) * | 1991-04-22 | 1999-01-15 | Otsuka Pharma Co Ltd | Pyrazolo(1,5-a>pyrimidinderivate und sie enthaltende antiinflammatorische mittel |
| US5356897A (en) * | 1991-09-09 | 1994-10-18 | Fujisawa Pharmaceutical Co., Ltd. | 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines |
| US5177206A (en) * | 1991-10-08 | 1993-01-05 | Dowelanco | Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides |
| TW224044B (da) * | 1991-12-30 | 1994-05-21 | Shell Internat Res Schappej B V | |
| IL108731A (en) * | 1993-03-04 | 1997-03-18 | Shell Int Research | 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES |
| RU2066295C1 (ru) * | 1993-05-19 | 1996-09-10 | Институт структурной макрокинетики РАН | Способ получения порошкового материала на основе карбида титана |
| EP0628559B1 (en) * | 1993-06-10 | 2002-04-03 | Beiersdorf-Lilly GmbH | Pyrimidine compounds and their use as pharmaceuticals |
| AU681913B2 (en) * | 1993-10-18 | 1997-09-11 | Dow Agrosciences Llc | Process for preparing N-(2,6-dichloro-3-methylphenyl)-5-7-dihalo(1,2,4)triazolo(1, 5A)pyrimidine-2-sulfonamide by cyclization and halo-dehydroxylation |
-
1996
- 1996-09-30 RU RU96120421A patent/RU2147584C1/ru not_active IP Right Cessation
- 1996-10-03 TR TR96/00792A patent/TR199600792A2/xx unknown
- 1996-10-15 US US08/729,204 patent/US5808066A/en not_active Expired - Lifetime
- 1996-10-16 DE DE69628712T patent/DE69628712T2/de not_active Expired - Lifetime
- 1996-10-16 DK DK96307528T patent/DK0770615T3/da active
- 1996-10-16 EP EP96307528A patent/EP0770615B1/en not_active Expired - Lifetime
- 1996-10-16 ES ES96307528T patent/ES2202419T3/es not_active Expired - Lifetime
- 1996-10-16 PT PT96307528T patent/PT770615E/pt unknown
- 1996-10-16 AT AT96307528T patent/ATE243211T1/de not_active IP Right Cessation
- 1996-10-16 MX MX9604882A patent/MX9604882A/es not_active IP Right Cessation
- 1996-10-16 SI SI9630630T patent/SI0770615T1/xx unknown
- 1996-10-18 SG SG1996010896A patent/SG55239A1/en unknown
- 1996-10-23 JP JP29790396A patent/JP4018182B2/ja not_active Expired - Fee Related
- 1996-10-23 UA UA96104029A patent/UA48132C2/uk unknown
- 1996-10-24 ZA ZA9608957A patent/ZA968957B/xx unknown
- 1996-10-25 HU HU9602957A patent/HU217773B/hu not_active IP Right Cessation
- 1996-10-25 CA CA002188905A patent/CA2188905C/en not_active Expired - Fee Related
- 1996-10-25 AR ARP960104928A patent/AR004122A1/es active IP Right Grant
- 1996-10-25 BR BR9605258A patent/BR9605258A/pt not_active IP Right Cessation
- 1996-10-25 SK SK1377-96A patent/SK284071B6/sk unknown
- 1996-10-26 KR KR1019960048877A patent/KR100443182B1/ko not_active Expired - Fee Related
- 1996-10-27 IL IL11949696A patent/IL119496A/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| ES2202419T3 (es) | 2004-04-01 |
| JP4018182B2 (ja) | 2007-12-05 |
| HUP9602957A3 (en) | 1998-01-28 |
| EP0770615A1 (en) | 1997-05-02 |
| IL119496A (en) | 2001-07-24 |
| SK284071B6 (sk) | 2004-09-08 |
| SK137796A3 (en) | 1997-05-07 |
| MX9604882A (es) | 1997-04-30 |
| HU9602957D0 (en) | 1996-12-30 |
| CA2188905C (en) | 2005-12-06 |
| US5808066A (en) | 1998-09-15 |
| JPH09124651A (ja) | 1997-05-13 |
| TR199600792A2 (tr) | 1997-05-21 |
| SI0770615T1 (en) | 2003-12-31 |
| HUP9602957A2 (en) | 1997-06-30 |
| DE69628712T2 (de) | 2004-04-29 |
| PT770615E (pt) | 2003-10-31 |
| ATE243211T1 (de) | 2003-07-15 |
| RU2147584C1 (ru) | 2000-04-20 |
| KR970021081A (ko) | 1997-05-28 |
| ZA968957B (en) | 1998-04-24 |
| UA48132C2 (uk) | 2002-08-15 |
| SG55239A1 (en) | 1998-12-21 |
| CA2188905A1 (en) | 1997-04-28 |
| BR9605258A (pt) | 1998-07-21 |
| AR004122A1 (es) | 1998-09-30 |
| DE69628712D1 (de) | 2003-07-24 |
| EP0770615B1 (en) | 2003-06-18 |
| KR100443182B1 (ko) | 2005-04-19 |
| HU217773B (hu) | 2000-04-28 |
| IL119496A0 (en) | 1997-01-10 |
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