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PL357109A1 - Niepeptydylowe inhibitory zależnego od VLA-4 wiązania komórek, użyteczne w leczeniu chorób zapalnych, autoimmunologicznych i chorób układu oddechowego - Google Patents

Niepeptydylowe inhibitory zależnego od VLA-4 wiązania komórek, użyteczne w leczeniu chorób zapalnych, autoimmunologicznych i chorób układu oddechowego

Info

Publication number
PL357109A1
PL357109A1 PL00357109A PL35710900A PL357109A1 PL 357109 A1 PL357109 A1 PL 357109A1 PL 00357109 A PL00357109 A PL 00357109A PL 35710900 A PL35710900 A PL 35710900A PL 357109 A1 PL357109 A1 PL 357109A1
Authority
PL
Poland
Prior art keywords
vla
autoimmune
cell binding
dependent cell
respiratory diseases
Prior art date
Application number
PL00357109A
Other languages
English (en)
Inventor
Louis Stanley Chupak
Allen Jacob Duplantier
Wan Fang Lau
Anthony John Milici
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of PL357109A1 publication Critical patent/PL357109A1/pl

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    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P25/00—Drugs for disorders of the nervous system
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    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
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    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
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    • C07C233/00—Carboxylic acid amides
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    • C07C233/47—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
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    • C07C311/06—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by carboxyl groups
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    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
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    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/08—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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PL00357109A 1999-12-28 2000-12-15 Niepeptydylowe inhibitory zależnego od VLA-4 wiązania komórek, użyteczne w leczeniu chorób zapalnych, autoimmunologicznych i chorób układu oddechowego PL357109A1 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17326099P 1999-12-28 1999-12-28
PCT/IB2000/001893 WO2001051487A1 (en) 1999-12-28 2000-12-15 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases

Publications (1)

Publication Number Publication Date
PL357109A1 true PL357109A1 (pl) 2004-07-12

Family

ID=22631221

Family Applications (1)

Application Number Title Priority Date Filing Date
PL00357109A PL357109A1 (pl) 1999-12-28 2000-12-15 Niepeptydylowe inhibitory zależnego od VLA-4 wiązania komórek, użyteczne w leczeniu chorób zapalnych, autoimmunologicznych i chorób układu oddechowego

Country Status (35)

Country Link
US (4) US20020049236A1 (pl)
EP (1) EP1244656A1 (pl)
JP (1) JP2003519697A (pl)
KR (1) KR20020067050A (pl)
CN (1) CN1413210A (pl)
AP (1) AP2002002565A0 (pl)
AR (1) AR029216A1 (pl)
AU (1) AU2018301A (pl)
BG (1) BG106867A (pl)
BR (1) BR0016818A (pl)
CA (1) CA2396087A1 (pl)
CO (1) CO5261616A1 (pl)
CR (1) CR6682A (pl)
CZ (1) CZ20022072A3 (pl)
EA (1) EA004673B1 (pl)
EE (1) EE200200372A (pl)
GT (1) GT200000226A (pl)
HU (1) HUP0203897A3 (pl)
IL (1) IL149758A0 (pl)
IS (1) IS6382A (pl)
MA (1) MA26861A1 (pl)
NO (1) NO20023085D0 (pl)
NZ (1) NZ518886A (pl)
OA (1) OA12126A (pl)
PA (1) PA8509301A1 (pl)
PE (1) PE20010987A1 (pl)
PL (1) PL357109A1 (pl)
SK (1) SK8692002A3 (pl)
SV (1) SV2002000246A (pl)
TN (1) TNSN00256A1 (pl)
TR (1) TR200201668T2 (pl)
UY (1) UY26512A1 (pl)
WO (1) WO2001051487A1 (pl)
YU (1) YU41202A (pl)
ZA (1) ZA200205142B (pl)

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US20020049236A1 (en) 2002-04-25
IL149758A0 (en) 2002-11-10
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