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OA12908A - Indole or benzimidazole derivatives for modulatingIKB-kinase. - Google Patents

Indole or benzimidazole derivatives for modulatingIKB-kinase. Download PDF

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Publication number
OA12908A
OA12908A OA1200500047A OA1200500047A OA12908A OA 12908 A OA12908 A OA 12908A OA 1200500047 A OA1200500047 A OA 1200500047A OA 1200500047 A OA1200500047 A OA 1200500047A OA 12908 A OA12908 A OA 12908A
Authority
OA
OAPI
Prior art keywords
alkyl
indole
compound
carboxamide
hydrogen atom
Prior art date
Application number
OA1200500047A
Other languages
English (en)
Inventor
Olaf Ritzeler
Gerhard Jaehne
Original Assignee
Aventis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Publication of OA12908A publication Critical patent/OA12908A/en

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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
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    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Life Sciences & Earth Sciences (AREA)
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  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Rheumatology (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Pain & Pain Management (AREA)
  • Neurosurgery (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Obesity (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
  • AIDS & HIV (AREA)
  • Psychiatry (AREA)
  • Molecular Biology (AREA)
OA1200500047A 2002-08-17 2003-08-05 Indole or benzimidazole derivatives for modulatingIKB-kinase. OA12908A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10237722A DE10237722A1 (de) 2002-08-17 2002-08-17 Indol- oder Benzimidazolderivate zur Modulation der IKappaB-Kinase

Publications (1)

Publication Number Publication Date
OA12908A true OA12908A (en) 2006-10-13

Family

ID=31968974

Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200500047A OA12908A (en) 2002-08-17 2003-08-05 Indole or benzimidazole derivatives for modulatingIKB-kinase.

Country Status (43)

Country Link
US (2) US7285560B2 (fr)
EP (2) EP1530568B1 (fr)
JP (1) JP4504812B2 (fr)
KR (1) KR101162046B1 (fr)
CN (1) CN1314683C (fr)
AR (1) AR040975A1 (fr)
AT (2) ATE557018T1 (fr)
AU (1) AU2003263196B2 (fr)
BR (1) BR0313562A (fr)
CA (1) CA2498559C (fr)
CO (1) CO5690586A2 (fr)
CR (1) CR7668A (fr)
CY (2) CY1111692T1 (fr)
DE (2) DE10237722A1 (fr)
DK (2) DK1530568T3 (fr)
EC (1) ECSP055612A (fr)
ES (2) ES2387954T3 (fr)
HK (1) HK1079509A1 (fr)
HN (1) HN2003000249A (fr)
HR (1) HRP20050042B1 (fr)
IL (1) IL166785A0 (fr)
JO (1) JO2764B1 (fr)
MA (1) MA27382A1 (fr)
ME (1) MEP60608A (fr)
MX (1) MXPA05001314A (fr)
MY (1) MY140074A (fr)
NO (1) NO330981B1 (fr)
NZ (1) NZ538296A (fr)
OA (1) OA12908A (fr)
PA (1) PA8580501A1 (fr)
PE (1) PE20040893A1 (fr)
PL (1) PL374229A1 (fr)
PT (2) PT1530568E (fr)
RS (1) RS51902B (fr)
RU (1) RU2318820C2 (fr)
SI (2) SI2233483T1 (fr)
SV (1) SV2004001599A (fr)
TN (1) TNSN05045A1 (fr)
TW (1) TWI290552B (fr)
UA (1) UA78591C2 (fr)
UY (1) UY27941A1 (fr)
WO (1) WO2004022553A1 (fr)
ZA (1) ZA200500322B (fr)

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