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MA23452A1 - Procede de preparation d'agents antiparasitaires consistant en derives d'avermectines et de milbemycines. - Google Patents

Procede de preparation d'agents antiparasitaires consistant en derives d'avermectines et de milbemycines.

Info

Publication number
MA23452A1
MA23452A1 MA23780A MA23780A MA23452A1 MA 23452 A1 MA23452 A1 MA 23452A1 MA 23780 A MA23780 A MA 23780A MA 23780 A MA23780 A MA 23780A MA 23452 A1 MA23452 A1 MA 23452A1
Authority
MA
Morocco
Prior art keywords
avmectins
milbemycins
derivatives
antiparasitic agents
agents consisting
Prior art date
Application number
MA23780A
Other languages
English (en)
Inventor
Nigel Derek Arthur Walshe
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MA23452A1 publication Critical patent/MA23452A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Dentistry (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Plant Pathology (AREA)
  • Molecular Biology (AREA)
  • Pest Control & Pesticides (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Wood Science & Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
MA23780A 1994-02-16 1995-02-15 Procede de preparation d'agents antiparasitaires consistant en derives d'avermectines et de milbemycines. MA23452A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB9402916A GB9402916D0 (en) 1994-02-16 1994-02-16 Antiparasitic agents

Publications (1)

Publication Number Publication Date
MA23452A1 true MA23452A1 (fr) 1995-10-01

Family

ID=10750420

Family Applications (1)

Application Number Title Priority Date Filing Date
MA23780A MA23452A1 (fr) 1994-02-16 1995-02-15 Procede de preparation d'agents antiparasitaires consistant en derives d'avermectines et de milbemycines.

Country Status (30)

Country Link
US (1) US5723488A (fr)
EP (1) EP0745089B1 (fr)
JP (2) JP3194959B2 (fr)
KR (1) KR100196751B1 (fr)
CN (1) CN1043996C (fr)
AP (1) AP547A (fr)
AT (1) ATE174340T1 (fr)
AU (1) AU686326B2 (fr)
CA (1) CA2183453C (fr)
CZ (1) CZ241496A3 (fr)
DE (1) DE69506525T2 (fr)
DK (1) DK0745089T3 (fr)
EG (1) EG20774A (fr)
ES (1) ES2124529T3 (fr)
FI (1) FI963201A0 (fr)
GB (1) GB9402916D0 (fr)
HU (1) HUT76521A (fr)
IL (1) IL112596A0 (fr)
MA (1) MA23452A1 (fr)
MX (1) MX9603486A (fr)
NO (1) NO963389L (fr)
NZ (1) NZ279494A (fr)
OA (1) OA10309A (fr)
PL (1) PL315902A1 (fr)
RU (1) RU2134272C1 (fr)
SI (1) SI9520021A (fr)
SK (1) SK106096A3 (fr)
WO (1) WO1995022552A1 (fr)
YU (1) YU8795A (fr)
ZA (1) ZA951218B (fr)

Families Citing this family (184)

* Cited by examiner, † Cited by third party
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US8754053B2 (en) 2010-02-17 2014-06-17 Syngenta Crop Protection Llc Isoxazoline derivatives as insecticides
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CN103534237B (zh) 2011-05-18 2016-06-15 先正达参股股份有限公司 基于芳硫基乙酰胺衍生物的杀虫化合物
UY34104A (es) 2011-05-31 2013-01-03 Syngenta Participations Ag ?compuestos derivados benzamídicos heterocíclicos, procesos e intermedios para su preparación, composiciones y métodos para su uso?.
WO2012163948A1 (fr) 2011-05-31 2012-12-06 Syngenta Participations Ag Mélanges pesticides comprenant des dérivés d'isoxazoline
WO2012175474A1 (fr) 2011-06-20 2012-12-27 Syngenta Participations Ag Pesticides à base de 1,2,3-triazole
WO2013026726A1 (fr) 2011-08-22 2013-02-28 Syngenta Participations Ag Dérivés de dihydrofurane en tant que composés insecticides
US20140343049A1 (en) 2011-08-22 2014-11-20 Syngenta Participations Ag Dihydrofuran derivatives as insecticidal compounds
CN103781356A (zh) 2011-08-25 2014-05-07 先正达参股股份有限公司 作为杀虫化合物的异噁唑啉衍生物
US9247740B2 (en) 2011-08-25 2016-02-02 Syngenta Participations Ag Isoxazoline derivatives as insecticidal compounds
WO2013026695A1 (fr) 2011-08-25 2013-02-28 Syngenta Participations Ag Dérivés d'isoxazoline en tant que composés insecticides
BR112014003730A2 (pt) 2011-08-25 2017-03-14 Syngenta Participations Ag processo para a preparação de derivados de tietano
WO2013026929A1 (fr) 2011-08-25 2013-02-28 Syngenta Participations Ag Dérivés de dihydropyrrole en tant que composés insecticides
BR112014005683B1 (pt) 2011-09-13 2018-12-04 Syngenta Participations Ag derivados isotiazolina como compostos inseticidas
US9023873B2 (en) 2011-10-03 2015-05-05 Syngenta Participations Ag Insecticidal 2-methoxybenzamide derivatives
US20140243375A1 (en) 2011-10-03 2014-08-28 Syngenta Participations Ag Isoxazoline derivatives as insecticidal compounds
WO2013135674A1 (fr) 2012-03-12 2013-09-19 Syngenta Participations Ag Composés de 2-aryl-acétamide insecticides
WO2014001121A1 (fr) 2012-06-25 2014-01-03 Syngenta Participations Ag Dérivés d'isothiazole en tant que composés insecticides
WO2014001120A1 (fr) 2012-06-25 2014-01-03 Syngenta Participations Ag Dérivés d'isothiazole en tant que composés insecticides
WO2014067838A1 (fr) 2012-10-31 2014-05-08 Syngenta Participations Ag Composés insecticides
WO2014079935A1 (fr) 2012-11-21 2014-05-30 Syngenta Participations Ag Composés insecticides à base de dérivés d'arylthioacétamide
BR112015025203B1 (pt) 2013-04-02 2020-11-24 Syngenta Participations Ag compostos, processo para a produção de compostos, método de uso de compostos, métodos para controle de insetos, ácaros, nematódeos ou moluscos e para a proteção de plantas úteis e composição
CN105102433B (zh) 2013-04-02 2017-12-15 先正达参股股份有限公司 杀虫化合物
CN104231022B (zh) * 2013-06-14 2018-10-09 南开大学 一种大环内酯类化合物的制备及应用
CN103421065B (zh) * 2013-07-03 2016-05-18 大庆志飞生物化工有限公司 一类新型阿维菌素衍生物及其制备方法
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CN105849084B (zh) 2013-12-23 2018-07-20 先正达参股股份有限公司 杀虫化合物
CN103896961A (zh) * 2014-03-25 2014-07-02 武汉大学 一种米尔贝肟类化合物及其制备方法
SI3206486T1 (sl) 2014-10-14 2023-04-28 ICB Pharma Pesticidne formulacije, ki imajo fizikalen način delovanja
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CN104447920A (zh) * 2014-11-28 2015-03-25 大庆志飞生物化工有限公司 一种阿维菌素氯代物及其制备方法和用途
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HUE050030T2 (hu) 2015-10-02 2020-11-30 Syngenta Participations Ag Mikrobiocid oxadiazol-származékok
CN108347936B (zh) 2015-10-28 2021-04-20 先正达参股股份有限公司 杀微生物的噁二唑衍生物
CN108349915A (zh) 2015-11-04 2018-07-31 先正达参股股份有限公司 杀微生物的苯胺衍生物
JP6930972B2 (ja) 2015-12-02 2021-09-01 シンジェンタ パーティシペーションズ アーゲー 殺微生物性オキサジアゾール誘導体
CN108368099B (zh) 2015-12-17 2021-11-12 先正达参股股份有限公司 杀微生物的噁二唑衍生物
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WO2017162868A1 (fr) 2016-03-24 2017-09-28 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
CN109068652A (zh) 2016-04-08 2018-12-21 先正达参股股份有限公司 杀微生物的噁二唑衍生物
JP2019516670A (ja) 2016-04-12 2019-06-20 シンジェンタ パーティシペーションズ アーゲー 殺微生物性オキサジアゾール誘導体
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WO2018029242A1 (fr) 2016-08-11 2018-02-15 Syngenta Participations Ag Dérivés d'oxadiazole microbicides
WO2018055133A1 (fr) 2016-09-23 2018-03-29 Syngenta Participations Ag Dérivés de tétrazolone microbiocides
BR112019005656A2 (pt) 2016-09-23 2019-06-04 Syngenta Participations Ag derivados oxadiazol microbiocidas
PL3522715T3 (pl) 2016-10-06 2021-06-28 Syngenta Participations Ag Mikrobiocydowe pochodne oksadiazolowe
UY37623A (es) 2017-03-03 2018-09-28 Syngenta Participations Ag Derivados de oxadiazol tiofeno fungicidas
JP2020514340A (ja) 2017-03-10 2020-05-21 シンジェンタ パーティシペーションズ アーゲー 殺微生物オキサジアゾール誘導体
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BR112019020756B1 (pt) 2017-04-05 2023-11-28 Syngenta Participations Ag Compostos derivados de oxadiazol microbicidas, composição agroquímica compreendendo os mesmos, método para controlar ou prevenir a infestação de plantas úteis por microrganismos fitopatogênicos e uso desses compostos
BR112019020735B1 (pt) 2017-04-05 2023-12-05 Syngenta Participations Ag Compostos derivados de oxadiazol microbiocidas e seu uso, composição agroquímica e método para controlar ou prevenir a infestação de plantas úteis por microrganismos fitopatogênicos
WO2018184986A1 (fr) 2017-04-05 2018-10-11 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
WO2018184988A1 (fr) 2017-04-05 2018-10-11 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
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WO2018185211A1 (fr) 2017-04-06 2018-10-11 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
WO2018206419A1 (fr) 2017-05-12 2018-11-15 Syngenta Participations Ag Dérivés hétérobicycliques microbiocides
CN110709395A (zh) 2017-06-02 2020-01-17 先正达参股股份有限公司 杀微生物的噁二唑衍生物
CN107021990B (zh) * 2017-06-14 2019-07-12 博瑞生物医药(苏州)股份有限公司 高纯度塞拉菌素的制备方法
CN107118247B (zh) * 2017-06-14 2019-07-26 博瑞生物医药(苏州)股份有限公司 塞拉菌素的制备方法
BR112020000465B1 (pt) 2017-07-11 2024-02-20 Syngenta Participations Ag Derivados oxadiazol microbiocidas
WO2019011926A1 (fr) 2017-07-11 2019-01-17 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
WO2019011929A1 (fr) 2017-07-11 2019-01-17 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
WO2019011928A1 (fr) 2017-07-11 2019-01-17 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
BR112020000371A2 (pt) 2017-07-12 2020-07-14 Syngenta Participations Ag derivados de oxadiazol microbiocidas
BR112020000414A2 (pt) 2017-07-12 2020-07-21 Syngenta Participations Ag derivados de oxadiazol microbicidas
WO2019012003A1 (fr) 2017-07-13 2019-01-17 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
CN107266511B (zh) * 2017-07-25 2019-08-20 中国农业大学 一类新颖的5-肟酯B2a结构的化合物及其制备方法与应用
JP7202366B2 (ja) 2017-09-13 2023-01-11 シンジェンタ パーティシペーションズ アーゲー 殺微生物性キノリン(チオ)カルボキサミド誘導体
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JP7150009B2 (ja) 2017-09-13 2022-10-07 シンジェンタ パーティシペーションズ アーゲー 殺微生物性キノリン(チオ)カルボキサミド誘導体
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WO2019097054A1 (fr) 2017-11-20 2019-05-23 Syngenta Participations Ag Dérivés d'oxadiazole microbiocides
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WO2020007658A1 (fr) 2018-07-02 2020-01-09 Syngenta Crop Protection Ag Dérivés de 3-(2-thiényl)-5-(trifluorométhyl) -1,2,4-oxadiazole en tant que fongicides agrochimiques
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GB201812692D0 (en) 2018-08-03 2018-09-19 Syngenta Participations Ag Microbiocidal compounds
WO2020058207A1 (fr) 2018-09-19 2020-03-26 Syngenta Crop Protection Ag Dérivés de quinoléine carboxamide microbiocides
WO2020070132A1 (fr) 2018-10-06 2020-04-09 Syngenta Participations Ag Dérivés de quinoléine dihydro-(thiazine) oxazine microbiocides
EP3860993B1 (fr) 2018-10-06 2022-08-10 Syngenta Participations Ag Dérivés de quinoléine dihydro-(thiazine)oxazine microbiocides
WO2020078732A1 (fr) 2018-10-17 2020-04-23 Syngenta Crop Protection Ag Dérivés d'oxadiazole microbiocides
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AP547A (en) 1996-10-30
OA10309A (en) 1997-10-07
DE69506525T2 (de) 1999-05-06
ZA951218B (en) 1996-08-15
YU8795A (sh) 1997-12-05
SI9520021A (en) 1997-04-30
CA2183453A1 (fr) 1995-08-24
EP0745089A1 (fr) 1996-12-04
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JPH11263791A (ja) 1999-09-28
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NO963389D0 (no) 1996-08-14
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