HRP20041101A2 - New etonogestrel esters - Google Patents

New etonogestrel esters

Info

Publication number: HRP20041101A2
Authority: HR; Croatia
Prior art keywords: new; etonogestrel esters; esters; new etonogestrel; etonogestrel
Prior art date: 2002-05-30

Application number

Other languages

English (en)

Inventor

Henrik De Nijs

Hendrikus Adrianus Anton Voort

Dirk Leysen

Arij Jan Grootenhuis

Original Assignee

Akzo Nobel Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-05-30

Filing date

2003-05-22

Publication date

2004-12-31

2003-05-22 Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv

2004-12-31 Publication of HRP20041101A2 publication Critical patent/HRP20041101A2/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0081—Substituted in position 17 alfa and 17 beta
- C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
- C07J1/0096—Alkynyl derivatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/16—Masculine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/34—Gestagens

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Endocrinology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Reproductive Health (AREA)
Diabetes (AREA)
Gynecology & Obstetrics (AREA)
Epidemiology (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

HRP20041101 2002-05-30 2003-05-22 New etonogestrel esters HRP20041101A2 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP02077119		2002-05-30
PCT/EP2003/050187 WO2003102012A2 (en)	2002-05-30	2003-05-22	New etonogestrel esters

Publications (1)

Publication Number	Publication Date
HRP20041101A2 true HRP20041101A2 (en)	2004-12-31

Family

ID=29595014

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HRP20041101 HRP20041101A2 (en)	2002-05-30	2003-05-22	New etonogestrel esters

Country Status (30)

Country	Link
US (1)	US7323454B2 (es)
EP (1)	EP1513861B1 (es)
JP (1)	JP4716726B2 (es)
KR (1)	KR20050009723A (es)
CN (2)	CN101100480A (es)
AR (1)	AR040130A1 (es)
AT (1)	ATE349458T1 (es)
AU (1)	AU2003238081B2 (es)
BR (1)	BR0311254A (es)
CA (1)	CA2487722C (es)
CO (1)	CO5631449A2 (es)
DE (1)	DE60310714T2 (es)
DK (1)	DK1513861T3 (es)
ES (1)	ES2277085T3 (es)
HR (1)	HRP20041101A2 (es)
IL (1)	IL165087A0 (es)
IS (1)	IS2421B (es)
MX (1)	MXPA04011797A (es)
NO (1)	NO20044898L (es)
NZ (1)	NZ536619A (es)
PE (1)	PE20040068A1 (es)
PL (1)	PL373855A1 (es)
PT (1)	PT1513861E (es)
RS (1)	RS97604A (es)
RU (1)	RU2325910C2 (es)
SI (1)	SI1513861T1 (es)
TW (1)	TW200403065A (es)
UA (1)	UA80126C2 (es)
WO (1)	WO2003102012A2 (es)
ZA (1)	ZA200410410B (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW200400041A (en) *	2002-05-30	2004-01-01	Akzo Nobel Nv	Use of new etonogestrel esters
WO2007011707A2 (en)	2005-07-15	2007-01-25	Micell Technologies, Inc.	Polymer coatings containing drug powder of controlled morphology
US20090062909A1 (en)	2005-07-15	2009-03-05	Micell Technologies, Inc.	Stent with polymer coating containing amorphous rapamycin
ES2540059T3 (es)	2006-04-26	2015-07-08	Micell Technologies, Inc.	Recubrimientos que contienen múltiples fármacos
JP5603598B2 (ja)	2007-01-08	2014-10-08	ミセルテクノロジーズ、インコーポレイテッド	生物分解層を有するステント
US11426494B2 (en)	2007-01-08	2022-08-30	MT Acquisition Holdings LLC	Stents having biodegradable layers
NZ588549A (en)	2008-04-17	2013-05-31	Micell Technologies Inc	Stents having bioabsorbable layers
WO2011009096A1 (en)	2009-07-16	2011-01-20	Micell Technologies, Inc.	Drug delivery medical device
CN102159257B (zh)	2008-07-17	2015-11-25	米歇尔技术公司	药物递送医疗设备
WO2010111232A2 (en)	2009-03-23	2010-09-30	Micell Technologies, Inc.	Drug delivery medical device
CN102481195B (zh)	2009-04-01	2015-03-25	米歇尔技术公司	涂覆支架
EP2419058B1 (en)	2009-04-17	2018-02-28	Micell Technologies, Inc.	Stents having controlled elution
WO2011097103A1 (en)	2010-02-02	2011-08-11	Micell Technologies, Inc.	Stent and stent delivery system with improved deliverability
WO2011133655A1 (en)	2010-04-22	2011-10-27	Micell Technologies, Inc.	Stents and other devices having extracellular matrix coating
CA2805631C (en)	2010-07-16	2018-07-31	Micell Technologies, Inc.	Drug delivery medical device
WO2013012689A1 (en)	2011-07-15	2013-01-24	Micell Technologies, Inc.	Drug delivery medical device
US10188772B2 (en)	2011-10-18	2019-01-29	Micell Technologies, Inc.	Drug delivery medical device
KR20150143476A (ko)	2013-03-12	2015-12-23	미셀 테크놀로지즈, 인코포레이티드	생흡수성 생체의학적 임플란트
KR20180059584A (ko)	2013-05-15	2018-06-04	미셀 테크놀로지즈, 인코포레이티드	생흡수성 생체의학적 임플란트
RU2595818C1 (ru) *	2015-05-25	2016-08-27	Федеральное государственное бюджетное научное учреждение "Научный центр проблем здоровья семьи и репродукции человека"	Способ комплексного лечения дисфункции яичников при применении гормонального контрацептива имплантата "импланона"
CN111057120B (zh) *	2019-12-27	2021-04-27	苏州翔实医药发展有限公司	一种依托孕烯衍生物a及其制备方法和用途

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1013284B (de)	1956-03-22	1957-08-08	Schering Ag	Verfahren zur Einfuehrung der Reste wenig reaktionsfaehiger Carbonsaeuren, insbesondere des ª‰-Cyclopentyl-propionylrestes, in die 17ª‡-staendige Oxygruppe solcher Steroide, die am Kohlenstoffatom 17 neben der Oxygruppe eine Acetylgruppe tragen
GB845442A (en)	1956-03-22	1960-08-24	Schering Ag	Manufacture of steroid compounds
GB8313921D0 (en) *	1983-05-19	1983-06-22	World Health Org	Contraceptive compositions
DE4227989A1 (de) *	1992-08-21	1994-06-09	Schering Ag	Mittel zur transdermalen Applikation enthaltend 3-Keto-desogestrel
DE4240806A1 (de)	1992-12-01	1994-06-09	Schering Ag	Mittel zur transdermalen Applikation enthaltend 14alpha,17alpha-Ethanoestra-1,3,5(10)-trien-3,17beta-diol
JPH07101884A (ja)	1993-10-01	1995-04-18	Sanei Gen F F I Inc	水溶性ヘミセルロースを含有する製剤
BR9408457A (pt) *	1993-12-27	1997-08-05	Akzo Nobel Nv	Preparação farmacêutica percutânia
DE19613698A1 (de)	1995-07-17	1997-01-23	Schering Ag	Mittel zur transdermalen Applikation enthaltend Ester des 13-Ethyl-17ß-hydroxy-11-methylen-18,19-dinor-17alpha-pregn-4-en-20-yn-3-ons
WO1997003709A1 (de)	1995-07-17	1997-02-06	Schering Aktiengesellschaft	Mittel zur transdermalen applikation enthaltend ester des 3-ketodegestrel
DE19531936A1 (de) *	1995-08-17	1997-02-20	Schering Ag	Kombinationspräparat zur Kontrazeption, Kits diese enthaltend und eine Methode diese verwendend
DE19540253C2 (de) *	1995-10-28	1998-06-04	Jenapharm Gmbh	Mehrphasenpräparat zur Kontrazeption auf der Basis natürlicher Estrogene
TR200003743T2 (tr)	1998-06-19	2001-07-23	Akzo Nobel N.V.	Testosteron türevi.
AU4513099A (en)	1998-06-19	2000-01-10	Akzo Nobel N.V.	Cycloalkyl-carboxylic acid esters of 7.alpha.methyl-estr-4-en-3-one 17.beta.-ol (19-nor 7.alpha.-methyltestosterone)
US6180682B1 (en) *	1999-01-26	2001-01-30	Virgil A. Place	Buccal drug delivery system for use in male contraception
TW200400041A (en) *	2002-05-30	2004-01-01	Akzo Nobel Nv	Use of new etonogestrel esters

2003
- 2003-05-19 TW TW092113489A patent/TW200403065A/zh unknown
- 2003-05-22 US US10/516,402 patent/US7323454B2/en not_active Expired - Lifetime
- 2003-05-22 RU RU2004138807/15A patent/RU2325910C2/ru not_active IP Right Cessation
- 2003-05-22 KR KR10-2004-7019330A patent/KR20050009723A/ko not_active Ceased
- 2003-05-22 AU AU2003238081A patent/AU2003238081B2/en not_active Ceased
- 2003-05-22 NZ NZ536619A patent/NZ536619A/en unknown
- 2003-05-22 CN CNA2007101028610A patent/CN101100480A/zh active Pending
- 2003-05-22 PT PT03735713T patent/PT1513861E/pt unknown
- 2003-05-22 AT AT03735713T patent/ATE349458T1/de not_active IP Right Cessation
- 2003-05-22 CA CA2487722A patent/CA2487722C/en not_active Expired - Fee Related
- 2003-05-22 SI SI200330679T patent/SI1513861T1/sl unknown
- 2003-05-22 ES ES03735713T patent/ES2277085T3/es not_active Expired - Lifetime
- 2003-05-22 UA UA20041109287A patent/UA80126C2/uk unknown
- 2003-05-22 JP JP2004509703A patent/JP4716726B2/ja not_active Expired - Fee Related
- 2003-05-22 DE DE60310714T patent/DE60310714T2/de not_active Expired - Lifetime
- 2003-05-22 RS YU97604A patent/RS97604A/sr unknown
- 2003-05-22 EP EP03735713A patent/EP1513861B1/en not_active Expired - Lifetime
- 2003-05-22 MX MXPA04011797A patent/MXPA04011797A/es active IP Right Grant
- 2003-05-22 DK DK03735713T patent/DK1513861T3/da active
- 2003-05-22 HR HRP20041101 patent/HRP20041101A2/xx not_active Application Discontinuation
- 2003-05-22 PL PL03373855A patent/PL373855A1/xx unknown
- 2003-05-22 WO PCT/EP2003/050187 patent/WO2003102012A2/en active IP Right Grant
- 2003-05-22 BR BR0311254-3A patent/BR0311254A/pt not_active IP Right Cessation
- 2003-05-22 CN CNB038123754A patent/CN1314701C/zh not_active Expired - Fee Related
- 2003-05-28 AR ARP030101859A patent/AR040130A1/es unknown
- 2003-05-28 PE PE2003000517A patent/PE20040068A1/es not_active Application Discontinuation
2004
- 2004-11-08 IL IL16508704A patent/IL165087A0/xx unknown
- 2004-11-10 NO NO20044898A patent/NO20044898L/no not_active Application Discontinuation
- 2004-11-15 IS IS7528A patent/IS2421B/is unknown
- 2004-12-22 CO CO04127949A patent/CO5631449A2/es not_active Application Discontinuation
- 2004-12-23 ZA ZA200410410A patent/ZA200410410B/xx unknown

Also Published As

Publication number	Publication date
CA2487722C (en)	2011-07-19
IL165087A0 (en)	2005-12-18
KR20050009723A (ko)	2005-01-25
EP1513861B1 (en)	2006-12-27
CN101100480A (zh)	2008-01-09
WO2003102012A9 (en)	2005-01-13
IS2421B (is)	2008-10-15
IS7528A (is)	2004-11-15
AU2003238081B2 (en)	2008-09-18
BR0311254A (pt)	2005-03-15
DE60310714T2 (de)	2007-10-11
PE20040068A1 (es)	2004-02-18
ES2277085T3 (es)	2007-07-01
DK1513861T3 (da)	2007-04-10
US7323454B2 (en)	2008-01-29
PL373855A1 (en)	2005-09-19
EP1513861A2 (en)	2005-03-16
AR040130A1 (es)	2005-03-16
DE60310714D1 (de)	2007-02-08
CN1314701C (zh)	2007-05-09
TW200403065A (en)	2004-03-01
AU2003238081A1 (en)	2003-12-19
CN1692122A (zh)	2005-11-02
SI1513861T1 (sl)	2007-06-30
RU2325910C2 (ru)	2008-06-10
CO5631449A2 (es)	2006-04-28
PT1513861E (pt)	2007-03-30
JP4716726B2 (ja)	2011-07-06
ZA200410410B (en)	2006-02-22
RS97604A (en)	2006-10-27
JP2005532350A (ja)	2005-10-27
RU2004138807A (ru)	2005-05-27
NZ536619A (en)	2007-09-28
HK1072609A1 (en)	2005-09-02
NO20044898L (no)	2005-02-25
MXPA04011797A (es)	2005-03-31
WO2003102012A3 (en)	2004-04-22
WO2003102012A2 (en)	2003-12-11
UA80126C2 (en)	2007-08-27
CA2487722A1 (en)	2003-12-11
US20050222113A1 (en)	2005-10-06
ATE349458T1 (de)	2007-01-15

Publication	Publication Date	Title
AU2003249738A8 (en)	2004-01-23	Ostoscope
AU2003297193A8 (en)	2004-07-09	Meta-web
HRP20041101A2 (en)	2004-12-31	New etonogestrel esters
AU2003252028A8 (en)	2004-02-09	Heterodiamondoids
AU2003279495A8 (en)	2004-05-13	Alert-modeling
GB2400797B (en)	2006-12-20	Shelving
AU2003264900A8 (en)	2004-04-08	Cast-cutter
AU2002367810A8 (en)	2003-11-10	Bis-transition-metal-chelate-probes
IL165125A0 (en)	2005-12-18	Use of new etonogestrel esters
AU2003262681A8 (en)	2004-03-03	Hemo-aide
GB0310123D0 (en)	2003-06-04	Airfreshener combined luminair
AU2002341221A8 (en)	2004-04-19	Honey-brandy
AU2003253735A8 (en)	2004-01-06	Vacuolins
GB0215011D0 (en)	2002-08-07	Easy squeezy
GB0204882D0 (en)	2002-04-17	Pedestal
AU2328P (en)	2003-09-25	Archley Arctotis fastuosa
AU2327P (en)	2003-09-25	Archnah Arctotis fastuosa
AU2326P (en)	2003-09-25	Gavol Gazania rigens
AU150609S (en)	2003-02-11	Weephole former
PL113111U1 (en)	2003-10-06	Shelving
GB0214885D0 (en)	2002-08-07	Medicament
GB0211377D0 (en)	2002-06-26	Medicament
GB0227620D0 (en)	2003-01-08	Easy Klik
GB0210565D0 (en)	2002-06-19	Concept three
AU149787S (en)	2002-11-06	Pedestal

Legal Events

Date	Code	Title	Description
2004-12-31	A1OB	Publication of a patent application
2005-06-23	ARAI	Request for the grant of a patent on the basis of the submitted results of a substantive examination of a patent application
2006-12-12	PPPP	Transfer of rights	Owner name: N.V. ORGANON, NL
2008-05-06	ODRP	Renewal fee for the maintenance of a patent	Payment date: 20080506 Year of fee payment: 6
2009-11-25	OBST	Application withdrawn