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AR040130A1 - Esteres de etonogestrel, su uso como anticopceptivo y para el tratamiento de desordenes ginecologicos - Google Patents

Esteres de etonogestrel, su uso como anticopceptivo y para el tratamiento de desordenes ginecologicos

Info

Publication number
AR040130A1
AR040130A1 ARP030101859A ARP030101859A AR040130A1 AR 040130 A1 AR040130 A1 AR 040130A1 AR P030101859 A ARP030101859 A AR P030101859A AR P030101859 A ARP030101859 A AR P030101859A AR 040130 A1 AR040130 A1 AR 040130A1
Authority
AR
Argentina
Prior art keywords
anticopceptive
esteres
etonogestrel
treatment
gynecological disorders
Prior art date
Application number
ARP030101859A
Other languages
English (en)
Inventor
Nijs Henrik De
Der Voort Hendrikus Adrianus Antonius Van
Arij Jan Grootenhuis
Dirk Leysen
Original Assignee
Akzo Nobel Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv
Publication of AR040130A1 publication Critical patent/AR040130A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0096—Alkynyl derivatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16—Masculine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/34—Gestagens

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Endocrinology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Epidemiology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Ésteres de progestógenos y los usos de ellos como anticonceptivo.
ARP030101859A 2002-05-30 2003-05-28 Esteres de etonogestrel, su uso como anticopceptivo y para el tratamiento de desordenes ginecologicos AR040130A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP02077119 2002-05-30

Publications (1)

Publication Number Publication Date
AR040130A1 true AR040130A1 (es) 2005-03-16

Family

ID=29595014

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP030101859A AR040130A1 (es) 2002-05-30 2003-05-28 Esteres de etonogestrel, su uso como anticopceptivo y para el tratamiento de desordenes ginecologicos

Country Status (31)

Country Link
US (1) US7323454B2 (es)
EP (1) EP1513861B1 (es)
JP (1) JP4716726B2 (es)
KR (1) KR20050009723A (es)
CN (2) CN1314701C (es)
AR (1) AR040130A1 (es)
AT (1) ATE349458T1 (es)
AU (1) AU2003238081B2 (es)
BR (1) BR0311254A (es)
CA (1) CA2487722C (es)
CO (1) CO5631449A2 (es)
DE (1) DE60310714T2 (es)
DK (1) DK1513861T3 (es)
ES (1) ES2277085T3 (es)
HK (1) HK1072609A1 (es)
HR (1) HRP20041101A2 (es)
IL (1) IL165087A0 (es)
IS (1) IS2421B (es)
MX (1) MXPA04011797A (es)
NO (1) NO20044898L (es)
NZ (1) NZ536619A (es)
PE (1) PE20040068A1 (es)
PL (1) PL373855A1 (es)
PT (1) PT1513861E (es)
RS (1) RS97604A (es)
RU (1) RU2325910C2 (es)
SI (1) SI1513861T1 (es)
TW (1) TW200403065A (es)
UA (1) UA80126C2 (es)
WO (1) WO2003102012A2 (es)
ZA (1) ZA200410410B (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200400041A (en) * 2002-05-30 2004-01-01 Akzo Nobel Nv Use of new etonogestrel esters
WO2007011708A2 (en) 2005-07-15 2007-01-25 Micell Technologies, Inc. Stent with polymer coating containing amorphous rapamycin
ES2691646T3 (es) 2005-07-15 2018-11-28 Micell Technologies, Inc. Revestimientos poliméricos que contienen polvo de fármaco de morfología controlada
WO2007127363A2 (en) 2006-04-26 2007-11-08 Micell Technologies, Inc. Coatings containing multiple drugs
WO2008086369A1 (en) 2007-01-08 2008-07-17 Micell Technologies, Inc. Stents having biodegradable layers
US11426494B2 (en) 2007-01-08 2022-08-30 MT Acquisition Holdings LLC Stents having biodegradable layers
CN102083397B (zh) 2008-04-17 2013-12-25 米歇尔技术公司 具有生物可吸收层的支架
WO2011009096A1 (en) 2009-07-16 2011-01-20 Micell Technologies, Inc. Drug delivery medical device
US9486431B2 (en) 2008-07-17 2016-11-08 Micell Technologies, Inc. Drug delivery medical device
US20100239635A1 (en) 2009-03-23 2010-09-23 Micell Technologies, Inc. Drug delivery medical device
CN102481195B (zh) 2009-04-01 2015-03-25 米歇尔技术公司 涂覆支架
EP3366326A1 (en) 2009-04-17 2018-08-29 Micell Technologies, Inc. Stents having controlled elution
WO2011097103A1 (en) 2010-02-02 2011-08-11 Micell Technologies, Inc. Stent and stent delivery system with improved deliverability
EP2560576B1 (en) 2010-04-22 2018-07-18 Micell Technologies, Inc. Stents and other devices having extracellular matrix coating
CA2805631C (en) 2010-07-16 2018-07-31 Micell Technologies, Inc. Drug delivery medical device
CA2841360A1 (en) 2011-07-15 2013-01-24 Micell Technologies, Inc. Drug delivery medical device
US10188772B2 (en) 2011-10-18 2019-01-29 Micell Technologies, Inc. Drug delivery medical device
CA2905419C (en) 2013-03-12 2020-04-28 Micell Technologies, Inc. Bioabsorbable biomedical implants
EP2996629B1 (en) 2013-05-15 2021-09-22 Micell Technologies, Inc. Bioabsorbable biomedical implants
RU2595818C1 (ru) * 2015-05-25 2016-08-27 Федеральное государственное бюджетное научное учреждение "Научный центр проблем здоровья семьи и репродукции человека" Способ комплексного лечения дисфункции яичников при применении гормонального контрацептива имплантата "импланона"
CN111057120B (zh) * 2019-12-27 2021-04-27 苏州翔实医药发展有限公司 一种依托孕烯衍生物a及其制备方法和用途

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB845442A (en) 1956-03-22 1960-08-24 Schering Ag Manufacture of steroid compounds
DE1013284B (de) 1956-03-22 1957-08-08 Schering Ag Verfahren zur Einfuehrung der Reste wenig reaktionsfaehiger Carbonsaeuren, insbesondere des ª‰-Cyclopentyl-propionylrestes, in die 17ª‡-staendige Oxygruppe solcher Steroide, die am Kohlenstoffatom 17 neben der Oxygruppe eine Acetylgruppe tragen
GB8313921D0 (en) * 1983-05-19 1983-06-22 World Health Org Contraceptive compositions
DE4227989A1 (de) * 1992-08-21 1994-06-09 Schering Ag Mittel zur transdermalen Applikation enthaltend 3-Keto-desogestrel
DE4240806A1 (de) 1992-12-01 1994-06-09 Schering Ag Mittel zur transdermalen Applikation enthaltend 14alpha,17alpha-Ethanoestra-1,3,5(10)-trien-3,17beta-diol
JPH07101884A (ja) 1993-10-01 1995-04-18 Sanei Gen F F I Inc 水溶性ヘミセルロースを含有する製剤
CN1135716A (zh) 1993-12-27 1996-11-13 阿克佐诺贝尔公司 经皮吸收的药用制剂
EP0848620A1 (de) * 1995-07-17 1998-06-24 Schering Aktiengesellschaft Mittel zur transdermalen applikation enthaltend ester des 3-ketodegestrel
DE19613698A1 (de) 1995-07-17 1997-01-23 Schering Ag Mittel zur transdermalen Applikation enthaltend Ester des 13-Ethyl-17ß-hydroxy-11-methylen-18,19-dinor-17alpha-pregn-4-en-20-yn-3-ons
EP1087986B1 (en) 1998-06-19 2002-04-10 Akzo Nobel N.V. 7.alpha.-methyl 19-nortestosterone undecanoate with androgenic activity
AU4513099A (en) 1998-06-19 2000-01-10 Akzo Nobel N.V. Cycloalkyl-carboxylic acid esters of 7.alpha.methyl-estr-4-en-3-one 17.beta.-ol (19-nor 7.alpha.-methyltestosterone)
US6180682B1 (en) * 1999-01-26 2001-01-30 Virgil A. Place Buccal drug delivery system for use in male contraception
TW200400041A (en) * 2002-05-30 2004-01-01 Akzo Nobel Nv Use of new etonogestrel esters

Also Published As

Publication number Publication date
WO2003102012A2 (en) 2003-12-11
PT1513861E (pt) 2007-03-30
CO5631449A2 (es) 2006-04-28
KR20050009723A (ko) 2005-01-25
AU2003238081A1 (en) 2003-12-19
RU2004138807A (ru) 2005-05-27
US20050222113A1 (en) 2005-10-06
AU2003238081B2 (en) 2008-09-18
WO2003102012A3 (en) 2004-04-22
HRP20041101A2 (en) 2004-12-31
BR0311254A (pt) 2005-03-15
WO2003102012A9 (en) 2005-01-13
HK1072609A1 (en) 2005-09-02
CN1314701C (zh) 2007-05-09
DE60310714T2 (de) 2007-10-11
EP1513861A2 (en) 2005-03-16
PL373855A1 (en) 2005-09-19
CN1692122A (zh) 2005-11-02
CA2487722A1 (en) 2003-12-11
NO20044898L (no) 2005-02-25
ES2277085T3 (es) 2007-07-01
PE20040068A1 (es) 2004-02-18
DE60310714D1 (de) 2007-02-08
JP4716726B2 (ja) 2011-07-06
ATE349458T1 (de) 2007-01-15
RS97604A (en) 2006-10-27
RU2325910C2 (ru) 2008-06-10
CA2487722C (en) 2011-07-19
CN101100480A (zh) 2008-01-09
MXPA04011797A (es) 2005-03-31
ZA200410410B (en) 2006-02-22
IL165087A0 (en) 2005-12-18
SI1513861T1 (sl) 2007-06-30
US7323454B2 (en) 2008-01-29
TW200403065A (en) 2004-03-01
DK1513861T3 (da) 2007-04-10
IS2421B (is) 2008-10-15
NZ536619A (en) 2007-09-28
UA80126C2 (en) 2007-08-27
EP1513861B1 (en) 2006-12-27
IS7528A (is) 2004-11-15
JP2005532350A (ja) 2005-10-27

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