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FR08C0017I2 - Combinaisons à base d'inhibiteurs de DPP-IV et d'antidiabetiques - Google Patents

Combinaisons à base d'inhibiteurs de DPP-IV et d'antidiabetiques

Info

Publication number
FR08C0017I2
FR08C0017I2 FR08C0017C FR08C0017C FR08C0017I2 FR 08C0017 I2 FR08C0017 I2 FR 08C0017I2 FR 08C0017 C FR08C0017 C FR 08C0017C FR 08C0017 C FR08C0017 C FR 08C0017C FR 08C0017 I2 FR08C0017 I2 FR 08C0017I2
Authority
FR
France
Prior art keywords
inhibitors
insulin
glucose
fructose
nvp
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
FR08C0017C
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis Pharma AG
Original Assignee
Novartis Pharma AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27049636&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FR08C0017(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Pharma AG filed Critical Novartis Pharma AG
Publication of FR08C0017I1 publication Critical patent/FR08C0017I1/fr
Application granted granted Critical
Publication of FR08C0017I2 publication Critical patent/FR08C0017I2/fr
Active legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/12Drugs for disorders of the metabolism for electrolyte homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
FR08C0017C 2000-01-21 2008-05-14 Combinaisons à base d'inhibiteurs de DPP-IV et d'antidiabetiques Active FR08C0017I2 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US48923400A 2000-01-21 2000-01-21
US61926200A 2000-07-19 2000-07-19
EP01909661A EP1248604B2 (fr) 2000-01-21 2001-01-19 Combinaisons comprenant un inhibiteur de la dipeptidylpeptidase - iv

Publications (2)

Publication Number Publication Date
FR08C0017I1 FR08C0017I1 (fr) 2008-07-18
FR08C0017I2 true FR08C0017I2 (fr) 2010-12-31

Family

ID=27049636

Family Applications (1)

Application Number Title Priority Date Filing Date
FR08C0017C Active FR08C0017I2 (fr) 2000-01-21 2008-05-14 Combinaisons à base d'inhibiteurs de DPP-IV et d'antidiabetiques

Country Status (18)

Country Link
US (1) US20030139434A1 (fr)
EP (5) EP1743655B1 (fr)
JP (7) JP2003520226A (fr)
CN (3) CN102327614A (fr)
AT (2) ATE385421T1 (fr)
AU (1) AU2001237321A1 (fr)
BR (1) BRPI0107715B8 (fr)
CA (2) CA2397554C (fr)
CY (6) CY1106303T1 (fr)
DE (3) DE122008000018I1 (fr)
DK (5) DK1741447T3 (fr)
ES (5) ES2301142T3 (fr)
FR (1) FR08C0017I2 (fr)
HK (4) HK1102424A1 (fr)
LU (1) LU91436I2 (fr)
NL (1) NL300346I1 (fr)
PT (5) PT1741447E (fr)
WO (1) WO2001052825A2 (fr)

Families Citing this family (138)

* Cited by examiner, † Cited by third party
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EP1741447A3 (fr) 2007-01-17
DK1741446T3 (da) 2008-06-02
DK1248604T3 (da) 2007-02-19
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JP2003520226A (ja) 2003-07-02
CN1400908A (zh) 2003-03-05
JP2011162550A (ja) 2011-08-25
DK1741445T3 (da) 2013-11-04
ATE385421T1 (de) 2008-02-15
US20030139434A1 (en) 2003-07-24
ATE346613T1 (de) 2006-12-15
ES2275654T5 (es) 2012-06-07
WO2001052825A2 (fr) 2001-07-26
PT1741446E (pt) 2008-05-09
FR08C0017I1 (fr) 2008-07-18
CY1114593T1 (el) 2016-10-05
JP2014088435A (ja) 2014-05-15
EP1741446B1 (fr) 2008-02-06
BRPI0107715B1 (pt) 2016-07-05
DK1741447T3 (da) 2013-12-09
PT1741447E (pt) 2013-12-11
ES2275654T3 (es) 2007-06-16
EP1743655A1 (fr) 2007-01-17
PT1248604E (pt) 2007-01-31
HK1102424A1 (en) 2007-11-23
DK1743655T3 (da) 2014-08-18
HK1102405A1 (en) 2007-11-23
BR0107715A (pt) 2002-11-19
LU91436I2 (fr) 2008-07-09
LU91436I9 (fr) 2019-01-02
EP1741445A3 (fr) 2007-01-24
ES2301142T3 (es) 2008-06-16
JP6374995B2 (ja) 2018-08-15
ES2487897T3 (es) 2014-08-25
EP1741447B1 (fr) 2013-09-18
EP1248604B1 (fr) 2006-11-29
NL300346I1 (fr) 2008-07-01
JP6104331B2 (ja) 2017-03-29
JP5824224B2 (ja) 2015-11-25
EP1741446A2 (fr) 2007-01-10
CN1977842A (zh) 2007-06-13
CY1106303T1 (el) 2011-10-12
JP5835910B2 (ja) 2015-12-24
HK1102422A1 (en) 2007-11-23
JP2017081994A (ja) 2017-05-18
PT1743655E (pt) 2014-09-09
JP2011116772A (ja) 2011-06-16
CA2673615C (fr) 2013-07-16
WO2001052825A3 (fr) 2002-03-28
JP6095589B2 (ja) 2017-03-15
PT1741445E (pt) 2013-11-11
DE60124861T2 (de) 2007-05-10
EP1248604B2 (fr) 2012-02-29
CA2673615A1 (fr) 2001-07-26
EP1743655B1 (fr) 2014-06-25
EP1741445B1 (fr) 2013-08-14
DE122008000018I1 (de) 2008-08-14
CY1115449T1 (el) 2017-01-04
ES2433476T3 (es) 2013-12-11
JP2006273873A (ja) 2006-10-12
ES2436610T3 (es) 2014-01-03
CY2008010I2 (el) 2009-11-04
CY1107423T1 (el) 2010-07-28
BRPI0107715B8 (pt) 2021-05-25
DE60132723T2 (de) 2009-01-29
HK1108359A1 (en) 2008-05-09
AU2001237321A1 (en) 2001-07-31
CY2008010I1 (el) 2009-11-04
EP1741447A2 (fr) 2007-01-10
CY1114466T1 (el) 2016-10-05
CN102327614A (zh) 2012-01-25
EP1248604A2 (fr) 2002-10-16
CA2397554C (fr) 2009-09-22
CA2397554A1 (fr) 2001-07-26
DE60132723D1 (de) 2008-03-20

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