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DK1971601T3 - N4-phenyl-quinazolin-4-aminderivater og beslægtede forbindelser som ERBB Type 1-receptortyrosinkinase-inhibitorer til behandling af hyperproliferative sygdomme - Google Patents

N4-phenyl-quinazolin-4-aminderivater og beslægtede forbindelser som ERBB Type 1-receptortyrosinkinase-inhibitorer til behandling af hyperproliferative sygdomme

Info

Publication number
DK1971601T3
DK1971601T3 DK06837728.2T DK06837728T DK1971601T3 DK 1971601 T3 DK1971601 T3 DK 1971601T3 DK 06837728 T DK06837728 T DK 06837728T DK 1971601 T3 DK1971601 T3 DK 1971601T3
Authority
DK
Denmark
Prior art keywords
treatment
tyrosine kinase
kinase inhibitors
receptor tyrosine
phenylquinazoline
Prior art date
Application number
DK06837728.2T
Other languages
English (en)
Inventor
Qian Zhao
Joseph P Lyssikatos
Julie Marie Greschuk
Fredrik P Marmsater
Original Assignee
Array Biopharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38022019&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1971601(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Array Biopharma Inc filed Critical Array Biopharma Inc
Application granted granted Critical
Publication of DK1971601T3 publication Critical patent/DK1971601T3/da

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    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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DK06837728.2T 2005-11-15 2006-11-15 N4-phenyl-quinazolin-4-aminderivater og beslægtede forbindelser som ERBB Type 1-receptortyrosinkinase-inhibitorer til behandling af hyperproliferative sygdomme DK1971601T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US73628905P 2005-11-15 2005-11-15
US81701906P 2006-06-28 2006-06-28
PCT/US2006/044431 WO2007059257A2 (en) 2005-11-15 2006-11-15 N4-phenyl-quinaz0line-4 -amine derivatives and related compounds as erbb type i receptor tyrosine kinase inhibitors for the treatment of hyperproliferative diseases

Publications (1)

Publication Number Publication Date
DK1971601T3 true DK1971601T3 (da) 2010-02-08

Family

ID=38022019

Family Applications (2)

Application Number Title Priority Date Filing Date
DK09157031.7T DK2090575T3 (da) 2005-11-15 2006-11-15 Fremgangsmåder og mellemprodukter til fremstillingen af N4 phenylquinazolin-4-aminderivater
DK06837728.2T DK1971601T3 (da) 2005-11-15 2006-11-15 N4-phenyl-quinazolin-4-aminderivater og beslægtede forbindelser som ERBB Type 1-receptortyrosinkinase-inhibitorer til behandling af hyperproliferative sygdomme

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK09157031.7T DK2090575T3 (da) 2005-11-15 2006-11-15 Fremgangsmåder og mellemprodukter til fremstillingen af N4 phenylquinazolin-4-aminderivater

Country Status (28)

Country Link
US (6) US8648087B2 (da)
EP (2) EP2090575B1 (da)
JP (2) JP5134548B2 (da)
KR (1) KR101086967B1 (da)
CN (2) CN102887891B (da)
AT (2) ATE507224T1 (da)
AU (2) AU2006315383B2 (da)
BR (2) BRPI0618668B1 (da)
CA (2) CA2755268C (da)
CY (3) CY1110583T1 (da)
DE (2) DE602006021645D1 (da)
DK (2) DK2090575T3 (da)
ES (2) ES2364901T3 (da)
FI (1) FIC20210022I1 (da)
FR (1) FR21C1031I2 (da)
HU (1) HUS2100028I1 (da)
IL (2) IL239149A (da)
LT (1) LTC1971601I2 (da)
LU (1) LUC00217I2 (da)
NL (1) NL301113I2 (da)
NO (1) NO342413B1 (da)
PL (2) PL2090575T3 (da)
PT (2) PT2090575E (da)
RU (2) RU2428421C2 (da)
SG (1) SG152230A1 (da)
SI (2) SI2090575T1 (da)
WO (1) WO2007059257A2 (da)
ZA (1) ZA200804498B (da)

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US7501427B2 (en) 2003-08-14 2009-03-10 Array Biopharma, Inc. Quinazoline analogs as receptor tyrosine kinase inhibitors
GB0420722D0 (en) 2004-09-17 2004-10-20 Addex Pharmaceuticals Sa Novel allosteric modulators
ATE507224T1 (de) 2005-11-15 2011-05-15 Array Biopharma Inc Verfahren und zwischenverbindungen zur herstellung von n4-phenyl-quinazolin-4-amin derivaten
TWI417095B (zh) 2006-03-15 2013-12-01 Janssen Pharmaceuticals Inc １，４-二取代之３-氰基-吡啶酮衍生物及其作為ｍＧｌｕＲ２-受體之正向異位性調節劑之用途
US7547781B2 (en) 2006-09-11 2009-06-16 Curis, Inc. Quinazoline based EGFR inhibitors containing a zinc binding moiety
JP5580592B2 (ja) 2006-09-11 2014-08-27 キュリス，インコーポレイテッド 亜鉛結合部分を含むキナゾリン系ｅｇｆｒインヒビター
JP2010502743A (ja) * 2006-09-11 2010-01-28 キュリス，インコーポレイテッド 抗増殖薬剤としての多機能性低分子
TW200900065A (en) 2007-03-07 2009-01-01 Janssen Pharmaceutica Nv 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives
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EP2162445B1 (en) * 2007-06-05 2013-11-27 Takeda Pharmaceutical Company Limited Heterobicyclic compounds as kinase inhibitors
US9114138B2 (en) 2007-09-14 2015-08-25 Janssen Pharmaceuticals, Inc. 1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′] bipyridinyl-2′-ones
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DE602006021645D1 (de) 2011-06-09
WO2007059257A3 (en) 2007-08-23
LTC1971601I2 (da) 2022-10-25
US12171739B2 (en) 2024-12-24
PT2090575E (pt) 2011-06-06
US20230142839A1 (en) 2023-05-11
KR20080070064A (ko) 2008-07-29
JP5232841B2 (ja) 2013-07-10
BRPI0618668A2 (pt) 2011-09-06
IL239149A0 (en) 2015-07-30
SI2090575T1 (sl) 2011-08-31

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