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CY1114563T1 - Υδροχλωριδια και ενυδρα συμπλεγματα της 1-[(3-κυανο-πυριδιν-2-υλο)μεθυλο]-3-μεθυλο-7-(2-βουτιν-1-υλο)-8-(3-αμινο-πιπεριδιν-1-υλο)ξανθινης, η παραγωγη αυτων και η χρηση αυτων ως φαρμακευτικα μεσα - Google Patents

Υδροχλωριδια και ενυδρα συμπλεγματα της 1-[(3-κυανο-πυριδιν-2-υλο)μεθυλο]-3-μεθυλο-7-(2-βουτιν-1-υλο)-8-(3-αμινο-πιπεριδιν-1-υλο)ξανθινης, η παραγωγη αυτων και η χρηση αυτων ως φαρμακευτικα μεσα

Info

Publication number
CY1114563T1
CY1114563T1 CY20131100819T CY131100819T CY1114563T1 CY 1114563 T1 CY1114563 T1 CY 1114563T1 CY 20131100819 T CY20131100819 T CY 20131100819T CY 131100819 T CY131100819 T CY 131100819T CY 1114563 T1 CY1114563 T1 CY 1114563T1
Authority
CY
Cyprus
Prior art keywords
methyl
butin
pyridin
hydrates
cyano
Prior art date
Application number
CY20131100819T
Other languages
English (en)
Inventor
Waldemar Pfrengle
Peter Sieger
Original Assignee
Boehringer Ingelheim International Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37102454&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1114563(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim International Gmbh filed Critical Boehringer Ingelheim International Gmbh
Publication of CY1114563T1 publication Critical patent/CY1114563T1/el

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
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Abstract

Η εφεύρεση σχετίζεται με άλατα της 1-[(3-κυανο-πυριδιν-2-υλο)μεθυλο]-3-μεθυλο-7-(2-βουτιν-1-υλο)-8-[3-αμινο-πιπεριδιν-1-υλο]-ξανθίνης με υδροχλωρικό οξύ, καθώς και με τα εναντιομερή αυτών, μείγματα αυτών και ένυδρα συμπλέγματα αυτών.
CY20131100819T 2005-07-30 2013-09-18 Υδροχλωριδια και ενυδρα συμπλεγματα της 1-[(3-κυανο-πυριδιν-2-υλο)μεθυλο]-3-μεθυλο-7-(2-βουτιν-1-υλο)-8-(3-αμινο-πιπεριδιν-1-υλο)ξανθινης, η παραγωγη αυτων και η χρηση αυτων ως φαρμακευτικα μεσα CY1114563T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102005035891A DE102005035891A1 (de) 2005-07-30 2005-07-30 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
EP06777973.6A EP1912990B1 (de) 2005-07-30 2006-07-26 Hydrochloride und hydrate von 1-[(3-cyano-pyridin-2-yl) methyl]-3-methyl-7-(2-butin-1-yl)-8-(3-amino-piperidin-1-yl)-xanthin, deren herstellung und deren verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
CY1114563T1 true CY1114563T1 (el) 2016-10-05

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
CY20131100819T CY1114563T1 (el) 2005-07-30 2013-09-18 Υδροχλωριδια και ενυδρα συμπλεγματα της 1-[(3-κυανο-πυριδιν-2-υλο)μεθυλο]-3-μεθυλο-7-(2-βουτιν-1-υλο)-8-(3-αμινο-πιπεριδιν-1-υλο)ξανθινης, η παραγωγη αυτων και η χρηση αυτων ως φαρμακευτικα μεσα

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EP (2) EP2540724B1 (el)
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