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AP2013007198A0 - Thieno [2,3-D] pyrimidine derivatives and their use to treat arrhythmia - Google Patents

Thieno [2,3-D] pyrimidine derivatives and their use to treat arrhythmia

Info

Publication number
AP2013007198A0
AP2013007198A0 AP2013007198A AP2013007198A AP2013007198A0 AP 2013007198 A0 AP2013007198 A0 AP 2013007198A0 AP 2013007198 A AP2013007198 A AP 2013007198A AP 2013007198 A AP2013007198 A AP 2013007198A AP 2013007198 A0 AP2013007198 A0 AP 2013007198A0
Authority
AP
ARIPO
Prior art keywords
thieno
pyrimidine derivatives
treat arrhythmia
arrhythmia
treat
Prior art date
Application number
AP2013007198A
Other languages
English (en)
Inventor
John Ford
Derek Edward John
Original Assignee
Xention Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44071904&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AP2013007198(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Xention Ltd filed Critical Xention Ltd
Publication of AP2013007198A0 publication Critical patent/AP2013007198A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AP2013007198A 2011-04-01 2012-03-29 Thieno [2,3-D] pyrimidine derivatives and their use to treat arrhythmia AP2013007198A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB1105659.5A GB201105659D0 (en) 2011-04-01 2011-04-01 Compounds
PCT/GB2012/050710 WO2012131379A1 (en) 2011-04-01 2012-03-29 Thieno [2, 3 -d] pyrimidine derivatives and their use to treat arrhythmia

Publications (1)

Publication Number Publication Date
AP2013007198A0 true AP2013007198A0 (en) 2013-10-31

Family

ID=44071904

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2013007198A AP2013007198A0 (en) 2011-04-01 2012-03-29 Thieno [2,3-D] pyrimidine derivatives and their use to treat arrhythmia

Country Status (42)

Country Link
US (1) US9249155B2 (xx)
EP (1) EP2694518B1 (xx)
JP (1) JP5826374B2 (xx)
KR (1) KR20140023332A (xx)
CN (1) CN103492392B (xx)
AP (1) AP2013007198A0 (xx)
AR (1) AR088735A1 (xx)
AU (1) AU2012235882B2 (xx)
BR (1) BR112013025236A2 (xx)
CA (1) CA2831493A1 (xx)
CL (1) CL2013002789A1 (xx)
CO (1) CO6801756A2 (xx)
CR (1) CR20130488A (xx)
CU (1) CU24173B1 (xx)
CY (1) CY1117025T1 (xx)
DK (1) DK2694518T3 (xx)
EA (1) EA201301111A1 (xx)
EC (1) ECSP13012988A (xx)
ES (1) ES2558563T3 (xx)
GB (1) GB201105659D0 (xx)
GT (1) GT201300225A (xx)
HR (1) HRP20151340T1 (xx)
HU (1) HUE028438T2 (xx)
IL (1) IL228555A0 (xx)
MA (1) MA35064B1 (xx)
ME (1) ME02314B (xx)
MX (1) MX335937B (xx)
NI (1) NI201300100A (xx)
PE (1) PE20141021A1 (xx)
PH (1) PH12013501952A1 (xx)
PL (1) PL2694518T3 (xx)
PT (1) PT2694518E (xx)
RS (1) RS54458B1 (xx)
RU (1) RU2013148627A (xx)
SG (1) SG193578A1 (xx)
SI (1) SI2694518T1 (xx)
SM (1) SMT201500322B (xx)
TN (1) TN2013000377A1 (xx)
TW (1) TWI516265B (xx)
UA (1) UA110131C2 (xx)
WO (1) WO2012131379A1 (xx)
ZA (1) ZA201307085B (xx)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2922858A4 (en) * 2012-11-20 2016-06-15 Univ Mcgill THIENOPYRIMIDININHIBITORS OF FARNESYL AND / OR GERANYL GERANYL PYROPHOSPHATE SYNTHASE
EP3394056B1 (en) 2015-12-22 2021-04-14 Shy Therapeutics LLC Compounds for the treatment of cancer and inflammatory disease
CN106727587A (zh) * 2016-11-28 2017-05-31 李娜 一种治疗心律失常的药物组合物
MA49458A (fr) * 2017-06-21 2020-04-29 SHY Therapeutics LLC Composés interagissant avec la superfamille ras destinés à être utilisés dans le traitement de cancers, de maladies inflammatoires, de rasopathies et de maladies fibrotiques

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Also Published As

Publication number Publication date
NZ615621A (en) 2015-01-30
CA2831493A1 (en) 2012-10-04
CO6801756A2 (es) 2013-11-29
ECSP13012988A (es) 2013-12-31
EP2694518A1 (en) 2014-02-12
PT2694518E (pt) 2016-02-05
PH12013501952A1 (en) 2018-04-11
KR20140023332A (ko) 2014-02-26
UA110131C2 (ru) 2015-11-25
GT201300225A (es) 2014-12-30
MX2013011301A (es) 2014-04-16
ES2558563T3 (es) 2016-02-05
CN103492392B (zh) 2015-11-25
DK2694518T3 (en) 2015-11-09
HK1193096A1 (zh) 2014-09-12
RU2013148627A (ru) 2015-05-10
TN2013000377A1 (en) 2015-01-20
US20140206703A1 (en) 2014-07-24
PL2694518T3 (pl) 2016-03-31
GB201105659D0 (en) 2011-05-18
CU24173B1 (es) 2016-04-25
CY1117025T1 (el) 2017-04-05
ZA201307085B (en) 2015-04-29
NI201300100A (es) 2014-01-07
EA201301111A1 (ru) 2014-02-28
HUE028438T2 (en) 2017-02-28
PE20141021A1 (es) 2014-08-30
HRP20151340T1 (hr) 2016-02-26
JP5826374B2 (ja) 2015-12-02
HK1193806A1 (zh) 2014-10-03
JP2014509637A (ja) 2014-04-21
AR088735A1 (es) 2014-07-02
CN103492392A (zh) 2014-01-01
MX335937B (es) 2016-01-04
IL228555A0 (en) 2013-12-31
TW201244720A (en) 2012-11-16
CL2013002789A1 (es) 2014-07-18
BR112013025236A2 (pt) 2019-09-24
MA35064B1 (fr) 2014-04-03
CR20130488A (es) 2013-12-06
US9249155B2 (en) 2016-02-02
SI2694518T1 (sl) 2016-02-29
CU20130124A7 (es) 2014-01-29
EP2694518B1 (en) 2015-10-07
WO2012131379A1 (en) 2012-10-04
ME02314B (me) 2016-06-20
TWI516265B (zh) 2016-01-11
AU2012235882B2 (en) 2015-08-06
SG193578A1 (en) 2013-10-30
RS54458B1 (en) 2016-06-30
SMT201500322B (it) 2016-02-25
AU2012235882A1 (en) 2013-05-02

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