ZA200502269B - Macrocyclic pyrimidines, the production thereof and the use of the same as medicaments - Google Patents
Macrocyclic pyrimidines, the production thereof and the use of the same as medicaments Download PDFInfo
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- ZA200502269B ZA200502269B ZA200502269A ZA200502269A ZA200502269B ZA 200502269 B ZA200502269 B ZA 200502269B ZA 200502269 A ZA200502269 A ZA 200502269A ZA 200502269 A ZA200502269 A ZA 200502269A ZA 200502269 B ZA200502269 B ZA 200502269B
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- alkyl
- heteroaryl
- aryl
- stands
- cycloalkyl
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Classifications
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- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
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- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
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- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/08—Bridged systems
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- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/08—Bridged systems
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| DE10239042A DE10239042A1 (de) | 2002-08-21 | 2002-08-21 | Makrozyclische Pyrimidine, deren Herstellung und Verwendung als Arzneimittel |
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Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1543541A (en) * | 1976-05-27 | 1979-04-04 | Nippon Kayaku Kk | Fibre reactive anthraquinone dyestuffs |
| GB9523675D0 (en) * | 1995-11-20 | 1996-01-24 | Celltech Therapeutics Ltd | Chemical compounds |
| GB9828511D0 (en) * | 1998-12-24 | 1999-02-17 | Zeneca Ltd | Chemical compounds |
| GB0004888D0 (en) | 2000-03-01 | 2000-04-19 | Astrazeneca Uk Ltd | Chemical compounds |
| GB0016877D0 (en) * | 2000-07-11 | 2000-08-30 | Astrazeneca Ab | Chemical compounds |
| GB0021726D0 (en) * | 2000-09-05 | 2000-10-18 | Astrazeneca Ab | Chemical compounds |
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2002
- 2002-08-21 DE DE10239042A patent/DE10239042A1/de not_active Ceased
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2003
- 2003-08-05 CA CA002492319A patent/CA2492319A1/en not_active Abandoned
- 2003-08-05 PL PL03374686A patent/PL374686A1/xx not_active Application Discontinuation
- 2003-08-05 HR HR20050240A patent/HRP20050240A2/xx not_active Application Discontinuation
- 2003-08-05 WO PCT/EP2003/008664 patent/WO2004026881A1/de active IP Right Grant
- 2003-08-05 MX MXPA05001526A patent/MXPA05001526A/es unknown
- 2003-08-05 PT PT03797225T patent/PT1530574E/pt unknown
- 2003-08-05 AU AU2003250212A patent/AU2003250212A1/en not_active Abandoned
- 2003-08-05 AT AT03797225T patent/ATE346073T1/de not_active IP Right Cessation
- 2003-08-05 EP EP03797225A patent/EP1530574B1/de not_active Expired - Lifetime
- 2003-08-05 EA EA200500303A patent/EA200500303A1/ru unknown
- 2003-08-05 BR BR0312874-1A patent/BR0312874A/pt not_active IP Right Cessation
- 2003-08-05 ES ES03797225T patent/ES2278222T3/es not_active Expired - Lifetime
- 2003-08-05 RS YUP-2005/0162A patent/RS20050162A/sr unknown
- 2003-08-05 KR KR1020057002784A patent/KR20050058360A/ko not_active Withdrawn
- 2003-08-05 JP JP2004536924A patent/JP2006501271A/ja active Pending
- 2003-08-05 DK DK03797225T patent/DK1530574T3/da active
- 2003-08-05 CN CNB038197901A patent/CN100357295C/zh not_active Expired - Fee Related
- 2003-08-05 DE DE50305774T patent/DE50305774D1/de not_active Expired - Fee Related
- 2003-08-20 US US10/644,076 patent/US7312225B2/en not_active Expired - Fee Related
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2004
- 2004-12-22 IL IL16591304A patent/IL165913A0/xx unknown
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2005
- 2005-03-17 ZA ZA200502269A patent/ZA200502269B/en unknown
- 2005-03-18 EC EC2005005690A patent/ECSP055690A/es unknown
- 2005-03-18 NO NO20051448A patent/NO20051448L/no not_active Application Discontinuation
- 2005-03-21 IS IS7762A patent/IS7762A/is unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MXPA05001526A (es) | 2005-04-19 |
| AU2003250212A1 (en) | 2004-04-08 |
| DE10239042A1 (de) | 2004-03-04 |
| US7312225B2 (en) | 2007-12-25 |
| US20040209895A1 (en) | 2004-10-21 |
| DE50305774D1 (de) | 2007-01-04 |
| HRP20050240A2 (en) | 2005-06-30 |
| KR20050058360A (ko) | 2005-06-16 |
| RS20050162A (en) | 2007-06-04 |
| ATE346073T1 (de) | 2006-12-15 |
| JP2006501271A (ja) | 2006-01-12 |
| EP1530574A1 (de) | 2005-05-18 |
| CN1675225A (zh) | 2005-09-28 |
| PT1530574E (pt) | 2007-02-28 |
| WO2004026881A1 (de) | 2004-04-01 |
| BR0312874A (pt) | 2005-06-28 |
| NO20051448D0 (no) | 2005-03-18 |
| EP1530574B1 (de) | 2006-11-22 |
| IS7762A (is) | 2005-03-21 |
| CA2492319A1 (en) | 2004-04-01 |
| EA200500303A1 (ru) | 2005-08-25 |
| DK1530574T3 (da) | 2007-03-26 |
| IL165913A0 (en) | 2006-01-15 |
| ES2278222T3 (es) | 2007-08-01 |
| ECSP055690A (es) | 2005-05-30 |
| PL374686A1 (en) | 2005-10-31 |
| NO20051448L (no) | 2005-03-18 |
| CN100357295C (zh) | 2007-12-26 |
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