SG11202004260YA - Process for preparing antihelmintic 4-amino-quinoline-3-carboxamide derivatives - Google Patents
Process for preparing antihelmintic 4-amino-quinoline-3-carboxamide derivativesInfo
- Publication number
- SG11202004260YA SG11202004260YA SG11202004260YA SG11202004260YA SG11202004260YA SG 11202004260Y A SG11202004260Y A SG 11202004260YA SG 11202004260Y A SG11202004260Y A SG 11202004260YA SG 11202004260Y A SG11202004260Y A SG 11202004260YA SG 11202004260Y A SG11202004260Y A SG 11202004260YA
- Authority
- SG
- Singapore
- Prior art keywords
- antihelmintic
- quinoline
- amino
- preparing
- carboxamide derivatives
- Prior art date
Links
- BIPPNESAFWTABU-UHFFFAOYSA-N 4-aminoquinoline-3-carboxamide Chemical class C1=CC=CC2=C(N)C(C(=O)N)=CN=C21 BIPPNESAFWTABU-UHFFFAOYSA-N 0.000 title 1
- 230000000507 anthelmentic effect Effects 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J23/00—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00
- B01J23/38—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00 of noble metals
- B01J23/40—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00 of noble metals of the platinum group metals
- B01J23/44—Palladium
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Materials Engineering (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Tropical Medicine & Parasitology (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Quinoline Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP17207586 | 2017-12-15 | ||
PCT/EP2018/084964 WO2019115768A1 (en) | 2017-12-15 | 2018-12-14 | Process for preparing antihelmintic 4-amino-quinoline-3-carboxamide derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
SG11202004260YA true SG11202004260YA (en) | 2020-06-29 |
Family
ID=60673654
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG11202004260YA SG11202004260YA (en) | 2017-12-15 | 2018-12-14 | Process for preparing antihelmintic 4-amino-quinoline-3-carboxamide derivatives |
Country Status (17)
Country | Link |
---|---|
US (1) | US11505544B2 (he) |
EP (1) | EP3692037A1 (he) |
JP (1) | JP7516245B2 (he) |
KR (1) | KR20200099548A (he) |
CN (1) | CN111448192B (he) |
AU (1) | AU2018382999B2 (he) |
CA (1) | CA3085675A1 (he) |
CL (1) | CL2020001589A1 (he) |
CO (1) | CO2020007222A2 (he) |
DO (1) | DOP2020000118A (he) |
IL (1) | IL275216A (he) |
MX (1) | MX2020006185A (he) |
PH (1) | PH12020550905A1 (he) |
SG (1) | SG11202004260YA (he) |
TW (1) | TWI809018B (he) |
UY (1) | UY38009A (he) |
WO (1) | WO2019115768A1 (he) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2020014068A1 (en) | 2018-07-09 | 2020-01-16 | Boehringer Ingelheim Animal Health USA Inc. | Anthelminthic heterocyclic compounds |
MX2021007540A (es) * | 2018-12-18 | 2021-10-13 | Elanco Tiergesundheit Ag | Derivados biciclicos. |
CR20210477A (es) | 2019-03-19 | 2022-01-06 | Boehringer Ingelheim Animal Health Usa Inc | Compuestos de aza-benzotiofeno y aza-benzofurano como antihelmínticos |
CN115667221A (zh) * | 2020-04-09 | 2023-01-31 | 拜耳动物保健有限责任公司 | 作为驱虫化合物的取代的稠合嗪类 |
WO2021242581A1 (en) | 2020-05-29 | 2021-12-02 | Boehringer Ingelheim Animal Health USA Inc. | Anthelmintic heterocyclic compounds |
EP4148052A1 (en) * | 2021-09-09 | 2023-03-15 | Bayer Animal Health GmbH | New quinoline derivatives |
KR20240112282A (ko) | 2021-11-01 | 2024-07-18 | 베링거잉겔하임베트메디카게엠베하 | 구충제 피롤로피리다진 화합물 |
KR20240154881A (ko) | 2023-04-19 | 2024-10-28 | 오신희 | 내진 및 제진구조를 갖는 각종 시설물 지지행거 |
WO2025027117A1 (en) | 2023-08-02 | 2025-02-06 | Intervet International B.V. | Carboxamide-4-quinoline compounds with anthelmintic activity |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1999032450A1 (en) * | 1997-12-22 | 1999-07-01 | Pharmacia & Upjohn Company | 4-hydroxyquinoline-3-carboxamides and hydrazides as antiviral agents |
MXPA02006474A (es) | 1999-12-28 | 2002-11-29 | Eisai Co Ltd | Compuestos heterociclicos que contienen sulfonamida. |
KR100767000B1 (ko) | 2000-02-03 | 2007-10-15 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 인테그린 발현 저해제 |
JP2008214323A (ja) | 2007-03-08 | 2008-09-18 | Kyowa Hakko Kogyo Co Ltd | 皮膚疾患の治療及び/または予防剤 |
US9006257B2 (en) | 2012-02-09 | 2015-04-14 | Glenmark Pharmaceuticals S.A. | Bicyclic compounds as mPGES-1 inhibitors |
AR098475A1 (es) * | 2013-11-26 | 2016-06-01 | Bayer Cropscience Ag | Compuestos pesticidas y usos |
CA2943100C (en) | 2014-03-24 | 2017-04-04 | Hao Wu | Quinoline derivatives as smo inhibitors |
TW201733988A (zh) | 2015-12-17 | 2017-10-01 | 阿斯特克斯治療有限公司 | 化學化合物 |
PT3538512T (pt) * | 2016-11-11 | 2021-08-16 | Bayer Animal Health Gmbh | Novos derivados de quinolina-3-carboxamida anti-helmínticos |
-
2018
- 2018-12-14 AU AU2018382999A patent/AU2018382999B2/en active Active
- 2018-12-14 MX MX2020006185A patent/MX2020006185A/es unknown
- 2018-12-14 KR KR1020207020010A patent/KR20200099548A/ko active Pending
- 2018-12-14 WO PCT/EP2018/084964 patent/WO2019115768A1/en active Application Filing
- 2018-12-14 CA CA3085675A patent/CA3085675A1/en active Pending
- 2018-12-14 JP JP2020531937A patent/JP7516245B2/ja active Active
- 2018-12-14 CN CN201880080813.2A patent/CN111448192B/zh active Active
- 2018-12-14 SG SG11202004260YA patent/SG11202004260YA/en unknown
- 2018-12-14 TW TW107145129A patent/TWI809018B/zh active
- 2018-12-14 US US16/772,680 patent/US11505544B2/en active Active
- 2018-12-14 UY UY0001038009A patent/UY38009A/es not_active Application Discontinuation
- 2018-12-14 EP EP18815237.5A patent/EP3692037A1/en active Pending
-
2020
- 2020-06-08 IL IL275216A patent/IL275216A/he unknown
- 2020-06-12 CO CONC2020/0007222A patent/CO2020007222A2/es unknown
- 2020-06-12 CL CL2020001589A patent/CL2020001589A1/es unknown
- 2020-06-15 DO DO2020000118A patent/DOP2020000118A/es unknown
- 2020-06-15 PH PH12020550905A patent/PH12020550905A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
US20200308153A1 (en) | 2020-10-01 |
JP2021506774A (ja) | 2021-02-22 |
RU2020123282A (ru) | 2022-01-17 |
PH12020550905A1 (en) | 2021-05-17 |
TW201927773A (zh) | 2019-07-16 |
CL2020001589A1 (es) | 2020-11-20 |
JP7516245B2 (ja) | 2024-07-16 |
IL275216A (he) | 2020-07-30 |
DOP2020000118A (es) | 2020-08-31 |
MX2020006185A (es) | 2020-09-03 |
KR20200099548A (ko) | 2020-08-24 |
CN111448192A (zh) | 2020-07-24 |
TWI809018B (zh) | 2023-07-21 |
AU2018382999A1 (en) | 2020-05-28 |
UY38009A (es) | 2019-07-31 |
CA3085675A1 (en) | 2019-06-20 |
CO2020007222A2 (es) | 2020-11-20 |
EP3692037A1 (en) | 2020-08-12 |
US11505544B2 (en) | 2022-11-22 |
CN111448192B (zh) | 2024-04-12 |
WO2019115768A1 (en) | 2019-06-20 |
AU2018382999B2 (en) | 2023-11-23 |
BR112020011901A2 (pt) | 2020-11-24 |
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