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PL3268372T3 - Inhibitory kv1.3 i ich zastosowanie medyczne - Google Patents

Inhibitory kv1.3 i ich zastosowanie medyczne

Info

Publication number
PL3268372T3
PL3268372T3 PL16709798T PL16709798T PL3268372T3 PL 3268372 T3 PL3268372 T3 PL 3268372T3 PL 16709798 T PL16709798 T PL 16709798T PL 16709798 T PL16709798 T PL 16709798T PL 3268372 T3 PL3268372 T3 PL 3268372T3
Authority
PL
Poland
Prior art keywords
inhibitors
medical application
medical
application
Prior art date
Application number
PL16709798T
Other languages
English (en)
Inventor
Stefan Tasler
Ilga KRIMMELBEIN
Original Assignee
4Sc Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 4Sc Ag filed Critical 4Sc Ag
Publication of PL3268372T3 publication Critical patent/PL3268372T3/pl

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • C07D491/048—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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    • A61K31/33—Heterocyclic compounds
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    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
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    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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    • C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14—Ortho-condensed systems
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    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
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    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Obesity (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Oncology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Toxicology (AREA)
  • Endocrinology (AREA)
  • Biochemistry (AREA)
  • Emergency Medicine (AREA)
PL16709798T 2015-03-13 2016-03-14 Inhibitory kv1.3 i ich zastosowanie medyczne PL3268372T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP15159083 2015-03-13
EP16709798.9A EP3268372B9 (en) 2015-03-13 2016-03-14 Kv1.3 inhibitors and their medical application
PCT/EP2016/055441 WO2016146575A1 (en) 2015-03-13 2016-03-14 Kv1.3 inhibitors and their medical application

Publications (1)

Publication Number Publication Date
PL3268372T3 true PL3268372T3 (pl) 2020-11-30

Family

ID=52684083

Family Applications (1)

Application Number Title Priority Date Filing Date
PL16709798T PL3268372T3 (pl) 2015-03-13 2016-03-14 Inhibitory kv1.3 i ich zastosowanie medyczne

Country Status (29)

Country Link
US (2) US10399991B2 (pl)
EP (1) EP3268372B9 (pl)
JP (1) JP6506410B2 (pl)
KR (1) KR20170137055A (pl)
CN (1) CN107548396B (pl)
AU (1) AU2016232330B2 (pl)
BR (1) BR112017019386A2 (pl)
CA (1) CA2979501A1 (pl)
CY (1) CY1123797T1 (pl)
DK (1) DK3268372T3 (pl)
EA (1) EA036935B1 (pl)
ES (1) ES2818102T3 (pl)
HK (1) HK1243998A1 (pl)
HR (1) HRP20201425T1 (pl)
HU (1) HUE050606T2 (pl)
IL (1) IL254390B (pl)
LT (1) LT3268372T (pl)
MX (1) MX378039B (pl)
PH (1) PH12017501653B1 (pl)
PL (1) PL3268372T3 (pl)
PT (1) PT3268372T (pl)
RS (1) RS60800B1 (pl)
SG (1) SG11201707282RA (pl)
SI (1) SI3268372T1 (pl)
SM (1) SMT202000475T1 (pl)
TW (1) TWI698438B (pl)
UA (1) UA121494C2 (pl)
WO (1) WO2016146575A1 (pl)
ZA (1) ZA201705676B (pl)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3156981A1 (en) * 2019-10-07 2021-04-15 D.E. Shaw Research, Llc Aryl heterobicyclic compounds as kv1.3 potassium shaker channel blockers

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