NO167292C - Fremgangsmaate ved fremstilling av cefuroksim 1-acetoksyetylester. - Google Patents

Fremgangsmaate ved fremstilling av cefuroksim 1-acetoksyetylester.

Info

Publication number: NO167292C
Authority: NO; Norway
Prior art keywords: acetoxylyl; cefuroxim; este; procedure; preparation
Prior art date: 1983-07-29

Application number

NO843055A

Other languages

English (en)

Norwegian (no)

Other versions

NO843055L (no

NO167292B (no

Inventor

Harold Alfred Crisp

Michael Wright

John Peter Turnbull

John Francis Oughton

Original Assignee

Glaxo Group Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1983-07-29

Filing date

1984-07-27

Publication date

1991-10-23

1984-07-27 Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd

1985-01-30 Publication of NO843055L publication Critical patent/NO843055L/no

1991-07-15 Publication of NO167292B publication Critical patent/NO167292B/no

1991-10-23 Publication of NO167292C publication Critical patent/NO167292C/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
- C07D501/46—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by carboxylic acids containing hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/26—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
- C07D501/34—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by carboxylic acids containing hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Cephalosporin Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

NO843055A 1983-07-29 1984-07-27 Fremgangsmaate ved fremstilling av cefuroksim 1-acetoksyetylester. NO167292C (no)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB838320521A GB8320521D0 (en)	1983-07-29	1983-07-29	Chemical process

Publications (3)

Publication Number	Publication Date
NO843055L NO843055L (no)	1985-01-30
NO167292B NO167292B (no)	1991-07-15
NO167292C true NO167292C (no)	1991-10-23

Family

ID=10546505

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO843055A NO167292C (no)	1983-07-29	1984-07-27	Fremgangsmaate ved fremstilling av cefuroksim 1-acetoksyetylester.

Country Status (21)

Country	Link
JP (1)	JPH0613526B2 (pt)
KR (1)	KR910008377B1 (pt)
AT (1)	AT392470B (pt)
AU (2)	AU582121B2 (pt)
BE (1)	BE900241A (pt)
CA (1)	CA1265511A (pt)
CH (1)	CH662121A5 (pt)
DE (1)	DE3427828A1 (pt)
DK (1)	DK165505C (pt)
ES (1)	ES534695A0 (pt)
FI (1)	FI76808C (pt)
FR (1)	FR2549837B1 (pt)
GB (2)	GB8320521D0 (pt)
IE (1)	IE57726B1 (pt)
IL (1)	IL72536A (pt)
NL (1)	NL8402372A (pt)
NO (1)	NO167292C (pt)
NZ (1)	NZ209046A (pt)
PT (1)	PT78985B (pt)
SE (1)	SE463263B (pt)
ZA (1)	ZA845830B (pt)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8400024D0 (en) *	1984-01-03	1984-02-08	Glaxo Group Ltd	Cephalosporin antibiotics
GB8524001D0 (en) *	1985-09-30	1985-11-06	Glaxo Group Ltd	Pharmaceutical composition
US5063224A (en) *	1990-07-09	1991-11-05	Eli Lilly And Company	R-cefuroxime axetil
IT1277426B1 (it) *	1995-08-03	1997-11-10	Acs Dobfar Spa	Forma cristallina biodisponibile del cefuroxima axetil
CN1111537C (zh) *	1997-05-15	2003-06-18	第一制糖株式会社	高纯晶形头孢呋辛1－乙酰氧乙酯的制备方法
KR100228264B1 (ko) *	1997-08-02	1999-11-01	김선진	결정형 세푸록심 악세틸의 제조방법
CA2209868C (en) *	1997-08-15	2001-08-14	Bernard Charles Sherman	Pharmaceutical compositions comprising cefuroxime axetil
IN186539B (pt) *	1997-09-29	2001-09-29	Ranbaxy Lab Ltd
PT937727E (pt) *	1998-02-20	2002-07-31	Fako Ilaclari A S	Processo para a producao de cefuroxima azetil cristalina soluvel
IN190849B (pt)	2000-07-17	2003-08-23	Ranbaxy Lab Ltd
AT411996B (de)	2000-09-11	2004-08-26	Sandoz Ag	Verfahren zur herstellung von cefuroxim in der form seines n-butylammoniumsalzes
ITMI20011763A1 (it) *	2001-08-10	2003-02-10	Antibioticos Spa	Processo di preparazione di cefuroxime axelite ad elevata purezza
ITMI20011925A1 (it) *	2001-09-14	2003-03-14	Antibioticos Spa	Metodo applicabile su scala industriale per la preparazione di cefuroxime axetile cristallino
TWI328006B (en) *	2003-12-26	2010-08-01	Nissan Chemical Ind Ltd	Crystal form of quinoline compound and process for its production
CN100448879C (zh) *	2004-07-22	2009-01-07	北京化工大学	一种无定型头孢呋辛酯的制备方法
DE102005019458A1 (de)	2005-04-25	2006-10-26	Grünenthal GmbH	Darreichungsform mit verbesserter Freisetzung von Cefuroximaxetil
CN118561870A (zh) *	2024-05-15	2024-08-30	广东立国制药有限公司	一种制备头孢呋辛酸的方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1571683A (en) *	1976-02-16	1980-07-16	Glaxo Operations Ltd	Ester derivatives of cefuroxime
CA1094545A (en) *	1976-02-16	1981-01-27	Michael Gregson	Cephalosporin antibiotics
GB1598568A (en) *	1977-04-19	1981-09-23	Glaxo Lab Ltd	Esters of(6r,7r)-3-carbamoyloxymethyl-7-((z)-2-(fur-2-yl)-2-methoxyiminoacetamido)-ceph-3-em-4-carboxylic acid
JPS577485A (en) *	1980-06-13	1982-01-14	Takeda Chem Ind Ltd	Cephalosporin
YU44680B (en) *	1982-07-30	1990-12-31	Glaxo Lab Ltd	Process for obtaining very pure amorphous form of cephuroxim axetile
GB8400024D0 (en) *	1984-01-03	1984-02-08	Glaxo Group Ltd	Cephalosporin antibiotics

1983
- 1983-07-29 GB GB838320521A patent/GB8320521D0/en active Pending
1984
- 1984-07-27 NO NO843055A patent/NO167292C/no not_active IP Right Cessation
- 1984-07-27 FI FI843011A patent/FI76808C/fi not_active IP Right Cessation
- 1984-07-27 DE DE19843427828 patent/DE3427828A1/de not_active Ceased
- 1984-07-27 AU AU31256/84A patent/AU582121B2/en not_active Ceased
- 1984-07-27 SE SE8403897A patent/SE463263B/sv not_active IP Right Cessation
- 1984-07-27 DK DK366684A patent/DK165505C/da not_active IP Right Cessation
- 1984-07-27 JP JP59155694A patent/JPH0613526B2/ja not_active Expired - Lifetime
- 1984-07-27 AT AT2444/84A patent/AT392470B/de not_active IP Right Cessation
- 1984-07-27 ZA ZA845830A patent/ZA845830B/xx unknown
- 1984-07-27 ES ES534695A patent/ES534695A0/es active Granted
- 1984-07-27 IE IE1938/84A patent/IE57726B1/en not_active IP Right Cessation
- 1984-07-27 FR FR8412011A patent/FR2549837B1/fr not_active Expired
- 1984-07-27 BE BE0/213398A patent/BE900241A/fr not_active IP Right Cessation
- 1984-07-27 KR KR1019840004465A patent/KR910008377B1/ko not_active IP Right Cessation
- 1984-07-27 NL NL8402372A patent/NL8402372A/nl not_active Application Discontinuation
- 1984-07-27 PT PT78985A patent/PT78985B/pt unknown
- 1984-07-27 CH CH3672/84A patent/CH662121A5/de not_active IP Right Cessation
- 1984-07-27 GB GB08419202A patent/GB2145409B/en not_active Expired
- 1984-07-27 CA CA000459929A patent/CA1265511A/en not_active Expired - Fee Related
- 1984-07-29 IL IL72536A patent/IL72536A/xx not_active IP Right Cessation
- 1984-07-30 NZ NZ209046A patent/NZ209046A/en unknown
1989
- 1989-06-16 AU AU36601/89A patent/AU634965B2/en not_active Ceased

Also Published As

Publication number	Publication date
ZA845830B (en)	1986-03-26
CH662121A5 (de)	1987-09-15
AU3125684A (en)	1985-01-31
GB2145409B (en)	1987-02-18
FI76808C (fi)	1988-12-12
DK366684A (da)	1985-01-30
IL72536A (en)	1988-01-31
AU3660189A (en)	1989-10-05
FI76808B (fi)	1988-08-31
PT78985A (en)	1984-08-01
AU634965B2 (en)	1993-03-11
IL72536A0 (en)	1984-11-30
GB2145409A (en)	1985-03-27
DE3427828A1 (de)	1985-02-14
BE900241A (fr)	1985-01-28
AU582121B2 (en)	1989-03-16
IE841938L (en)	1985-01-29
GB8320521D0 (en)	1983-09-01
KR910008377B1 (ko)	1991-10-12
DK366684D0 (da)	1984-07-27
GB8419202D0 (en)	1984-08-30
CA1265511A (en)	1990-02-06
SE8403897L (sv)	1985-01-30
AT392470B (de)	1991-04-10
FI843011A0 (fi)	1984-07-27
SE463263B (sv)	1990-10-29
NO843055L (no)	1985-01-30
DK165505B (da)	1992-12-07
JPH0613526B2 (ja)	1994-02-23
FI843011A (fi)	1985-01-30
DK165505C (da)	1993-04-19
PT78985B (en)	1986-10-23
ES8601869A1 (es)	1985-11-01
FR2549837A1 (fr)	1985-02-01
NO167292B (no)	1991-07-15
JPS6075484A (ja)	1985-04-27
ATA244484A (de)	1990-09-15
IE57726B1 (en)	1993-03-24
NZ209046A (en)	1988-02-29
SE8403897D0 (sv)	1984-07-27
ES534695A0 (es)	1985-11-01
NL8402372A (nl)	1985-02-18
FR2549837B1 (fr)	1986-12-26
KR850001221A (ko)	1985-03-16

Publication	Publication Date	Title
NO820083L (no)	1982-07-14	Fremgangsmaate ved fremstilling av d-fenylalanyl-l-propyl-l-argininaldehydsulfat
NO843956L (no)	1985-04-09	Fremgangsmaate for fremstilling av karboksyalkenamido-cefalosporiner
NO852124L (no)	1985-12-02	Fremgangsmaate ved fremstilling av kinolonderivater.
NO821137L (no)	1982-10-11	Fremgangsmaate for fremstilling av tertiaere alkyletere
NO170071C (no)	1992-09-09	Fremgangsmaate ved fremstilling av klordioksyd.
NO167292C (no)	1991-10-23	Fremgangsmaate ved fremstilling av cefuroksim 1-acetoksyetylester.
FI822748A0 (fi)	1982-08-06	Foerfarande foer framstaellning av substituerade pyridazinderivat
NO166032C (no)	1991-05-22	Fremgangsmaate ved fremstilling av triklormonosilan.
NO844631L (no)	1985-05-28	Fremgangsmaate for fremstilling av tremasse
NO884665D0 (no)	1988-10-20	Fremgangsmaate ved fremstilling av 9-oh-alkoksyguanin.
NO170019C (no)	1992-09-02	Fremgangsmaate for fremstilling av deglucoteicoplanin (antibiotikum l 17392)
NO845207L (no)	1985-06-24	Fremgangsmaate for fremstilling av diaminopolyalkenyletere
NO820281L (no)	1982-08-03	Fremgangsmaate ved fremstilling av n-(halogenmethyl)-acylamider
NO157735C (no)	1988-05-11	Fremgangsmaate for fremstilling av alfa-arylalkansyrer.
NO855067L (no)	1986-06-18	Fremgangsmaate for fremstilling av n-formyl-alfa-aspartyl-fenylalanin.
NO165676C (no)	1991-03-20	Fremgangsmaate ved fremstilling av pyrrolidonderivater.
NO852810L (no)	1986-01-14	Fremgangsmaate ved fremstilling av fluorallylaminderivater.
NO166931C (no)	1991-09-18	Fremgangsmaate ved fremstilling av klordioksyd.
NO165405C (no)	1991-02-06	Fremgangsmaate for fremstilling av tixotrope vaskemidler.
NO163061C (no)	1990-03-28	Fremgangsmaate til fremstilling av ferromangan.
NO165637C (no)	1991-03-13	Fremgangsmaate for fremstilling av etoksylert lignitt.
NO840535L (no)	1984-08-16	Fremgangsmaate ved fremstilling av aroylimidazoloner
NO864386D0 (no)	1986-11-03	Fremgangsmaate ved fremstilling av uretaner.
NO165538C (no)	1991-02-27	Fremgangsmaate ved fremstilling av klordioksyd.
NO824072L (no)	1983-06-06	Fremgangsmaate ved fremstilling av anti-bakterielle p-oxooxazolidinylbenzen-sulfonamider

Legal Events

Date	Code	Title	Description
2003-03-10	MM1K	Lapsed by not paying the annual fees	Free format text: LAPSED IN JANUARY 2003