JO2764B1 - Indole derivatives or benzimidazole derivatives to modify the enzyme AKP kinase - Google Patents

Indole derivatives or benzimidazole derivatives to modify the enzyme AKP kinase

Info

Publication number: JO2764B1
Authority: JO; Jordan
Prior art keywords: derivatives; modulating; ikappab kinase; benzimidazole; indole
Prior art date: 2002-08-17

Application number

JO200387A

Other languages

Arabic (ar)

English (en)

Inventor

ريتزيلر اولاف

هارد جيهين غير

Original Assignee

سانوفي - افانتيسي دويتشلاند جي ام بي اتش

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-08-17

Filing date

2003-07-23

Publication date

2014-03-15

2003-07-23 Application filed by سانوفي - افانتيسي دويتشلاند جي ام بي اتش filed Critical سانوفي - افانتيسي دويتشلاند جي ام بي اتش

2014-03-15 Application granted granted Critical

2014-03-15 Publication of JO2764B1 publication Critical patent/JO2764B1/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

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Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Physical Education & Sports Medicine (AREA)
Immunology (AREA)
Rheumatology (AREA)
Oncology (AREA)
Cardiology (AREA)
Orthopedic Medicine & Surgery (AREA)
Diabetes (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Heart & Thoracic Surgery (AREA)
Communicable Diseases (AREA)
Virology (AREA)
Pain & Pain Management (AREA)
Neurosurgery (AREA)
Tropical Medicine & Parasitology (AREA)
Obesity (AREA)
Dermatology (AREA)
Urology & Nephrology (AREA)
Hematology (AREA)
Endocrinology (AREA)
Hospice & Palliative Care (AREA)
Emergency Medicine (AREA)
AIDS & HIV (AREA)
Psychiatry (AREA)
Molecular Biology (AREA)

JO200387A 2002-08-17 2003-07-23 Indole derivatives or benzimidazole derivatives to modify the enzyme AKP kinase JO2764B1 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE10237722A DE10237722A1 (de)	2002-08-17	2002-08-17	Indol- oder Benzimidazolderivate zur Modulation der IKappaB-Kinase

Publications (1)

Publication Number	Publication Date
JO2764B1 true JO2764B1 (en)	2014-03-15

Family

ID=31968974

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
JO200387A JO2764B1 (en)	2002-08-17	2003-07-23	Indole derivatives or benzimidazole derivatives to modify the enzyme AKP kinase

Country Status (43)

Country	Link
US (2)	US7285560B2 (da)
EP (2)	EP1530568B1 (da)
JP (1)	JP4504812B2 (da)
KR (1)	KR101162046B1 (da)
CN (1)	CN1314683C (da)
AR (1)	AR040975A1 (da)
AT (2)	ATE557018T1 (da)
AU (1)	AU2003263196B2 (da)
BR (1)	BR0313562A (da)
CA (1)	CA2498559C (da)
CO (1)	CO5690586A2 (da)
CR (1)	CR7668A (da)
CY (2)	CY1111692T1 (da)
DE (2)	DE10237722A1 (da)
DK (2)	DK1530568T3 (da)
EC (1)	ECSP055612A (da)
ES (2)	ES2387954T3 (da)
HK (1)	HK1079509A1 (da)
HN (1)	HN2003000249A (da)
HR (1)	HRP20050042B1 (da)
IL (1)	IL166785A0 (da)
JO (1)	JO2764B1 (da)
MA (1)	MA27382A1 (da)
ME (1)	MEP60608A (da)
MX (1)	MXPA05001314A (da)
MY (1)	MY140074A (da)
NO (1)	NO330981B1 (da)
NZ (1)	NZ538296A (da)
OA (1)	OA12908A (da)
PA (1)	PA8580501A1 (da)
PE (1)	PE20040893A1 (da)
PL (1)	PL374229A1 (da)
PT (2)	PT1530568E (da)
RS (1)	RS51902B (da)
RU (1)	RU2318820C2 (da)
SI (2)	SI2233483T1 (da)
SV (1)	SV2004001599A (da)
TN (1)	TNSN05045A1 (da)
TW (1)	TWI290552B (da)
UA (1)	UA78591C2 (da)
UY (1)	UY27941A1 (da)
WO (1)	WO2004022553A1 (da)
ZA (1)	ZA200500322B (da)

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TW201221505A (en)	2010-07-05	2012-06-01	Sanofi Sa	Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
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Publication number	Publication date
US8778955B2 (en)	2014-07-15
MEP60608A (en)	2011-05-10
UY27941A1 (es)	2004-03-31
AU2003263196A1 (en)	2004-03-29
NO330981B1 (no)	2011-08-29
IL166785A0 (en)	2006-01-15
MA27382A1 (fr)	2005-06-01
DK1530568T3 (da)	2011-04-18
ECSP055612A (es)	2005-04-18
NZ538296A (en)	2007-03-30
MXPA05001314A (es)	2005-04-28
ES2358795T3 (es)	2011-05-13
CA2498559C (en)	2012-01-24
ATE557018T1 (de)	2012-05-15
ATE493402T1 (de)	2011-01-15
PA8580501A1 (es)	2004-04-23
DE10237722A1 (de)	2004-08-19
CN1314683C (zh)	2007-05-09
CY1112991T1 (el)	2016-04-13
HRP20050042B1 (hr)	2013-09-30
PT2233483E (pt)	2012-07-20
OA12908A (en)	2006-10-13
EP1530568A1 (de)	2005-05-18
HRP20050042A2 (en)	2006-03-31
CA2498559A1 (en)	2004-03-18
AU2003263196B2 (en)	2009-01-22
HN2003000249A (es)	2008-08-06
TWI290552B (en)	2007-12-01
RS51902B (sr)	2012-02-29
TNSN05045A1 (en)	2007-05-14
AR040975A1 (es)	2005-04-27
HK1079509A1 (en)	2006-04-07
KR101162046B1 (ko)	2012-07-04
RU2318820C2 (ru)	2008-03-10
ZA200500322B (en)	2006-07-26
WO2004022553A1 (de)	2004-03-18
RU2005107418A (ru)	2005-08-27
CR7668A (es)	2009-03-11
US7285560B2 (en)	2007-10-23
DK2233483T3 (da)	2012-08-20
SV2004001599A (es)	2004-02-26
NO20051337L (no)	2005-05-03
EP1530568B1 (de)	2010-12-29
BR0313562A (pt)	2006-06-13
JP4504812B2 (ja)	2010-07-14
KR20050058338A (ko)	2005-06-16
US20050197353A1 (en)	2005-09-08
UA78591C2 (en)	2007-04-10
DE50313372D1 (de)	2011-02-10
RS20050104A (en)	2007-06-04
EP2233483A1 (de)	2010-09-29
CY1111692T1 (el)	2015-10-07
US20070244139A1 (en)	2007-10-18
PL374229A1 (en)	2005-10-03
CN1675196A (zh)	2005-09-28
PT1530568E (pt)	2011-02-23
JP2005539054A (ja)	2005-12-22
EP2233483B1 (de)	2012-05-09
TW200418832A (en)	2004-10-01
SI1530568T1 (sl)	2011-05-31
MY140074A (en)	2009-11-30
PE20040893A1 (es)	2004-12-21
ES2387954T3 (es)	2012-10-04
CO5690586A2 (es)	2006-10-31
SI2233483T1 (sl)	2012-08-31

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NO20045589L (no)	2005-02-02	Nye forbindelser
HK1054039A1 (en)	2003-11-14	Substituded beta-carbolines
IL172942A0 (en)	2006-06-11	Pyrazoloisoquinoline derivatives as kinase inhibitors
SE0202241D0 (sv)	2002-07-17	Novel Compounds
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