IL147494A0 - Benzofuran derivatives - Google Patents

Benzofuran derivatives

Info

Publication number: IL147494A0
Authority: IL; Israel
Prior art keywords: benzofuran derivatives; benzofuran; derivatives
Prior art date: 1999-07-10

Application number

IL14749400A

Other languages

English (en)

Original Assignee

Merck Patent Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-07-10

Filing date

2000-06-29

Publication date

2002-08-14

2000-06-29 Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh

2002-08-14 Publication of IL147494A0 publication Critical patent/IL147494A0/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D307/84—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D307/85—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 2
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Neurology (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Furan Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

IL14749400A 1999-07-10 2000-06-29 Benzofuran derivatives IL147494A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE19932314A DE19932314A1 (de)	1999-07-10	1999-07-10	Benzofuranderivate
PCT/EP2000/006089 WO2001004112A2 (de)	1999-07-10	2000-06-29	Benzofuranderivate

Publications (1)

Publication Number	Publication Date
IL147494A0 true IL147494A0 (en)	2002-08-14

Family

ID=7914351

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
IL14749400A IL147494A0 (en)	1999-07-10	2000-06-29	Benzofuran derivatives
IL147494A IL147494A (en)	1999-07-10	2002-01-06	History of Benzoporn

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
IL147494A IL147494A (en)	1999-07-10	2002-01-06	History of Benzoporn

Country Status (29)

Country	Link
US (1)	US6531503B1 (uk)
EP (1)	EP1194426B1 (uk)
JP (1)	JP4908706B2 (uk)
KR (1)	KR100709378B1 (uk)
CN (1)	CN1178934C (uk)
AR (1)	AR024671A1 (uk)
AT (1)	ATE273973T1 (uk)
AU (1)	AU767413B2 (uk)
BR (1)	BRPI0012329B8 (uk)
CA (1)	CA2378603C (uk)
CZ (1)	CZ301441B6 (uk)
DE (2)	DE19932314A1 (uk)
DK (1)	DK1194426T3 (uk)
ES (1)	ES2226884T3 (uk)
HK (1)	HK1047275B (uk)
HU (1)	HU229135B1 (uk)
IL (2)	IL147494A0 (uk)
MX (1)	MXPA02000316A (uk)
MY (1)	MY122667A (uk)
NO (1)	NO328209B1 (uk)
PL (1)	PL196477B1 (uk)
PT (1)	PT1194426E (uk)
RU (1)	RU2278862C2 (uk)
SI (1)	SI1194426T1 (uk)
SK (1)	SK287360B6 (uk)
TR (1)	TR200200017T2 (uk)
UA (1)	UA73310C2 (uk)
WO (1)	WO2001004112A2 (uk)
ZA (1)	ZA200201085B (uk)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE102006060597A1 (de) *	2006-12-21	2008-06-26	Merck Patent Gmbh	Verfahren zur Herstellung von Benzofuran-2-carboxamiden
EP2110374A1 (en) *	2008-04-18	2009-10-21	Merck Sante	Benzofurane, benzothiophene, benzothiazol derivatives as FXR modulators
PE20120357A1 (es) *	2009-03-10	2012-05-03	Takeda Pharmaceutical	Derivados de benzofurano
CN102971311B (zh)	2010-05-06	2015-07-08	百时美施贵宝公司	作为gpr119调节剂的二环杂芳基化合物
US8729084B2 (en)	2010-05-06	2014-05-20	Bristol-Myers Squibb Company	Benzofuranyl analogues as GPR119 modulators
CN102964323B (zh) *	2012-11-13	2015-03-25	苏州永健生物医药有限公司	一种5-（哌嗪-1-基）苯并呋喃-2-甲酰胺的合成方法
AU2014279240A1 (en) *	2013-06-10	2016-01-07	Astellas Pharma Inc.	Bicyclic nitrogen-containing aromatic heterocyclic amide compound

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2724915A (en) *		1955-11-29		Snow remover
DE2757532A1 (de) *	1977-12-23	1979-07-05	Hoechst Ag	N,n'-disubstituiertes cyclisches diamin und verfahren zu dessen herstellung
CZ327795A3 (en) *	1993-06-14	1996-08-14	Pfizer	Secondary amines
DE4333254A1 (de)	1993-09-30	1995-04-06	Merck Patent Gmbh	Piperidine und Piperazine
DE19514567A1 (de) *	1995-04-20	1996-10-24	Merck Patent Gmbh	Benzofurane

1999
- 1999-07-10 DE DE19932314A patent/DE19932314A1/de not_active Withdrawn
2000
- 2000-06-29 SK SK6-2002A patent/SK287360B6/sk not_active IP Right Cessation
- 2000-06-29 TR TR2002/00017T patent/TR200200017T2/xx unknown
- 2000-06-29 MX MXPA02000316A patent/MXPA02000316A/es active IP Right Grant
- 2000-06-29 IL IL14749400A patent/IL147494A0/xx active IP Right Grant
- 2000-06-29 DK DK00949229T patent/DK1194426T3/da active
- 2000-06-29 PT PT00949229T patent/PT1194426E/pt unknown
- 2000-06-29 US US10/030,471 patent/US6531503B1/en not_active Expired - Lifetime
- 2000-06-29 ES ES00949229T patent/ES2226884T3/es not_active Expired - Lifetime
- 2000-06-29 JP JP2001509722A patent/JP4908706B2/ja not_active Expired - Fee Related
- 2000-06-29 CN CNB008093083A patent/CN1178934C/zh not_active Expired - Fee Related
- 2000-06-29 RU RU2002102234/04A patent/RU2278862C2/ru not_active IP Right Cessation
- 2000-06-29 HU HU0201903A patent/HU229135B1/hu not_active IP Right Cessation
- 2000-06-29 PL PL353157A patent/PL196477B1/pl not_active IP Right Cessation
- 2000-06-29 AU AU62665/00A patent/AU767413B2/en not_active Ceased
- 2000-06-29 KR KR1020017015565A patent/KR100709378B1/ko not_active IP Right Cessation
- 2000-06-29 DE DE50007501T patent/DE50007501D1/de not_active Expired - Lifetime
- 2000-06-29 UA UA2002021055A patent/UA73310C2/uk unknown
- 2000-06-29 CZ CZ20020011A patent/CZ301441B6/cs not_active IP Right Cessation
- 2000-06-29 CA CA2378603A patent/CA2378603C/en not_active Expired - Fee Related
- 2000-06-29 SI SI200030518T patent/SI1194426T1/xx unknown
- 2000-06-29 EP EP00949229A patent/EP1194426B1/de not_active Expired - Lifetime
- 2000-06-29 AT AT00949229T patent/ATE273973T1/de active
- 2000-06-29 BR BRPI0012329A patent/BRPI0012329B8/pt not_active IP Right Cessation
- 2000-06-29 WO PCT/EP2000/006089 patent/WO2001004112A2/de active IP Right Grant
- 2000-07-06 MY MYPI20003075A patent/MY122667A/en unknown
- 2000-07-07 AR ARP000103465A patent/AR024671A1/es active IP Right Grant
2002
- 2002-01-06 IL IL147494A patent/IL147494A/en not_active IP Right Cessation
- 2002-01-09 NO NO20020095A patent/NO328209B1/no not_active IP Right Cessation
- 2002-02-07 ZA ZA200201085A patent/ZA200201085B/en unknown
- 2002-11-29 HK HK02108676.2A patent/HK1047275B/zh unknown

Also Published As

Publication number	Publication date
EP1194426B1 (de)	2004-08-18
AR024671A1 (es)	2002-10-23
MY122667A (en)	2006-04-29
SK287360B6 (sk)	2010-08-09
ES2226884T3 (es)	2005-04-01
EP1194426A2 (de)	2002-04-10
HU229135B1 (en)	2013-08-28
HK1047275B (zh)	2005-09-02
HUP0201903A2 (en)	2002-10-28
JP2003504364A (ja)	2003-02-04
CZ301441B6 (cs)	2010-03-03
ATE273973T1 (de)	2004-09-15
RU2278862C2 (ru)	2006-06-27
AU767413B2 (en)	2003-11-06
JP4908706B2 (ja)	2012-04-04
ZA200201085B (en)	2003-07-30
WO2001004112A3 (de)	2001-08-02
WO2001004112A2 (de)	2001-01-18
TR200200017T2 (tr)	2002-05-21
KR100709378B1 (ko)	2007-04-20
NO20020095D0 (no)	2002-01-09
DE50007501D1 (de)	2004-09-23
CZ200211A3 (cs)	2002-04-17
CN1356996A (zh)	2002-07-03
CN1178934C (zh)	2004-12-08
HK1047275A1 (en)	2003-02-14
SK62002A3 (en)	2002-05-09
CA2378603C (en)	2010-05-11
NO20020095L (no)	2002-01-09
US6531503B1 (en)	2003-03-11
PL353157A1 (en)	2003-10-20
KR20020016815A (ko)	2002-03-06
NO328209B1 (no)	2010-01-11
MXPA02000316A (es)	2002-07-30
PL196477B1 (pl)	2008-01-31
CA2378603A1 (en)	2001-01-18
PT1194426E (pt)	2005-01-31
SI1194426T1 (en)	2005-02-28
AU6266500A (en)	2001-01-30
IL147494A (en)	2008-03-20
DE19932314A1 (de)	2001-01-11
BR0012329A (pt)	2002-03-19
DK1194426T3 (da)	2004-12-20
HUP0201903A3 (en)	2005-02-28
BR0012329B1 (pt)	2013-03-19
UA73310C2 (en)	2005-07-15
BRPI0012329B8 (pt)	2021-05-25

Publication	Publication Date	Title
EG23817A (en)	2007-09-19	4-Phenyl-pyridine derivatives
HUP0201535A2 (en)	2002-08-28	5-cyano-2-aminopyrimidine derivatives
IL148167A0 (en)	2002-09-12	Amino-triazolopyridine derivatives
GC0000183A (en)	2006-03-29	3-Phenyl-pyridine derivatives
IL145739A0 (en)	2002-07-25	13-methyl-erythromycin derivatives
GC0000338A (en)	2007-03-31	5-Phenyl-pyrimidine derivatives
HK1046400A1 (en)	2003-01-10	Substituted 2-dialkylaminoalkylbiphenyl derivatives
IL148837A0 (en)	2002-09-12	Isoxazolecarboxamide derivatives
GC0000191A (en)	2006-03-29	4-Phenyl-pyrimidine derivatives
GB0026485D0 (en)	2000-12-13	›-Carboline derivatives
CZ20012041A3 (cs)	2001-10-17	Benzofuranové deriváty
GC0000256A (en)	2006-11-01	Ethanesulfonyl-piperidine derivatives
IL150132A0 (en)	2002-12-01	Cyclopenteneone derivatives
IL147636A0 (en)	2002-08-14	3-amino-2-benzyl-1-phenyl-propane derivatives
IL147494A0 (en)	2002-08-14	Benzofuran derivatives
AP2001002327A0 (en)	2001-12-31	1-Trifluoromethyl-4-hydroxy-7- piperidinylaminomethy lchroman derivatives
IL144045A0 (en)	2002-04-21	Oxetanone derivatives
AU2049601A (en)	2001-07-03	Benzofuran derivatives
AU2049501A (en)	2001-07-03	Benzofuran derivatives
SI1222183T1 (en)	2003-10-31	Benzopyran derivatives
IL146282A0 (en)	2002-07-25	Thio-oxindole derivatives
GB9907134D0 (en)	1999-05-19	Antimor napthylcombretastatin derivatives
HK1043987A1 (zh)	2002-10-04	硫-羥吲衍生物

Legal Events

Date	Code	Title	Description
2008-11-03	FF	Patent granted
2008-11-27	KB	Patent renewed