[go: up one dir, main page]

CR11441A - Producto de dispersion solida que contiene un compuesto a base de n-aril urea - Google Patents

Producto de dispersion solida que contiene un compuesto a base de n-aril urea

Info

Publication number
CR11441A
CR11441A CR11441A CR11441A CR11441A CR 11441 A CR11441 A CR 11441A CR 11441 A CR11441 A CR 11441A CR 11441 A CR11441 A CR 11441A CR 11441 A CR11441 A CR 11441A
Authority
CR
Costa Rica
Prior art keywords
urea
aril
based compound
product containing
solid dispersion
Prior art date
Application number
CR11441A
Other languages
English (en)
Inventor
Schroeder Rudolf
Heittermann Tanja
Original Assignee
Abbott Gmbh & Co Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Gmbh & Co Kg filed Critical Abbott Gmbh & Co Kg
Publication of CR11441A publication Critical patent/CR11441A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1635Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1652Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Un producto que comprende al menos un agente farmaceuticamente activo a base de N-aril urea o un agente de estructura relacionada que es obtenido mediante a) la preparacion de una mezcla liquida que contiene el al menos un agente activo
CR11441A 2007-10-19 2010-05-19 Producto de dispersion solida que contiene un compuesto a base de n-aril urea CR11441A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US99961307P 2007-10-19 2007-10-19

Publications (1)

Publication Number Publication Date
CR11441A true CR11441A (es) 2010-10-25

Family

ID=40089072

Family Applications (1)

Application Number Title Priority Date Filing Date
CR11441A CR11441A (es) 2007-10-19 2010-05-19 Producto de dispersion solida que contiene un compuesto a base de n-aril urea

Country Status (23)

Country Link
US (1) US20090143423A1 (es)
EP (1) EP2197426A2 (es)
JP (1) JP2011500647A (es)
KR (1) KR20100090689A (es)
CN (1) CN101827585A (es)
AR (1) AR068916A1 (es)
AU (1) AU2008313620A1 (es)
BR (1) BRPI0818339A2 (es)
CA (1) CA2699335A1 (es)
CL (1) CL2008003092A1 (es)
CO (1) CO6270303A2 (es)
CR (1) CR11441A (es)
DO (1) DOP2010000114A (es)
EC (1) ECSP10010184A (es)
GT (1) GT201000095A (es)
MX (1) MX2010004292A (es)
PE (1) PE20091041A1 (es)
RU (1) RU2010119924A (es)
TW (1) TW200922549A (es)
UA (1) UA100866C2 (es)
UY (1) UY31406A1 (es)
WO (1) WO2009050289A2 (es)
ZA (1) ZA201002130B (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2352726A1 (en) * 2008-10-17 2011-08-10 Abbott Laboratories Trpv1 antagonists
JP2012505908A (ja) * 2008-10-17 2012-03-08 アボット・ラボラトリーズ Trpv1アンタゴニスト
US20100210682A1 (en) * 2009-02-19 2010-08-19 Abbott Laboratories Repeated Dosing of TRPV1 Antagonists
CN102573755A (zh) * 2009-09-18 2012-07-11 巴斯夫欧洲公司 制备具有低水溶性的物质的制剂的方法
RU2013134339A (ru) 2010-12-23 2015-01-27 Эбботт Гмбх Унд Ко. Кг Твердые составы с замедленным действием на основе твердой дисперсии
CN103391770A (zh) 2011-01-10 2013-11-13 细胞基因公司 环丙烷羧酸{2-[(1s)-1-(3-乙氧基-4-甲氧基-苯基)-2-甲烷磺酰基-乙基]-3-氧代-2,3-二氢-1h-异吲哚-4-基}-酰胺的口服剂型
US9034832B2 (en) 2011-12-29 2015-05-19 Abbvie Inc. Solid compositions
EP2907505A3 (en) * 2011-12-29 2015-12-30 Abbvie Inc. Solid compositions comprising an HCV inhibitor
TW201431570A (zh) 2012-11-22 2014-08-16 Ucb Pharma Gmbh 用於經皮投服羅替戈汀(Rotigotine)之多天式貼片
HUE047777T2 (hu) 2013-01-31 2020-05-28 Gilead Pharmasset Llc Két vírusellenes vegyület kombinációs készítménye
BR112015021692A2 (pt) 2013-03-15 2017-07-18 Boehringer Ingelheim Int formulação de dosagem oral sólida de inibidor de hcv no estado amorfo
US10046151B2 (en) 2013-07-03 2018-08-14 Lts Lohmann Therapie-Systeme, Ag Transdermal therapeutic system with electronic component
PT3650014T (pt) 2013-08-27 2021-12-27 Gilead Pharmasset Llc Formulação combinada de dois compostos antivirais
JP6573913B2 (ja) * 2014-05-20 2019-09-11 エルテーエス ローマン テラピー−ジステーメ アーゲー ロチゴチンを含む経皮送達システム
JP6895755B2 (ja) 2014-05-20 2021-06-30 エルテーエス ローマン テラピー−ジステーメ アーゲー 経皮送達システムにおける活性薬剤の放出を調節するための方法
EP4238580A3 (en) 2014-05-20 2023-10-25 LTS Lohmann Therapie-Systeme AG Transdermal delivery system including an interface mediator
EP3307246A1 (en) 2015-06-09 2018-04-18 Capsugel Belgium NV Formulations to achieve rapid dissolution of drug from spray-dried dispersions in capsules
US12186314B2 (en) * 2015-12-22 2025-01-07 Arizona Board Of Regents On Behalf Of The University Of Arizona Compositions and methods for treatment, amelioration, and prevention of anesthesia-induced hypothermia
EP3873443A4 (en) * 2018-10-30 2022-07-27 Peloton Therapeutics, Inc. SOLID DISPERSIONS AND PHARMACEUTICAL COMPOSITIONS WITH A SUBSTITUTED INDAN AND PROCESSES FOR THEIR PREPARATION AND USE THEREOF
EP4019485B1 (en) 2019-08-23 2024-08-07 Mochida Pharmaceutical Co., Ltd. Method for producing heterocyclidene acetamide derivatives
MX2022002017A (es) 2019-08-23 2022-03-11 Mochida Pharm Co Ltd Metodo para producir derivado de heterociclideno acetamida.

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5362878A (en) * 1991-03-21 1994-11-08 Pfizer Inc. Intermediates for making N-aryl and N-heteroarylamide and urea derivatives as inhibitors of acyl coenzyme A: cholesterol acyl transferase (ACAT)
RU94046149A (ru) * 1992-05-28 1996-11-27 Пфайзер Инк. (US) Новые n-арил и n-гетероарил производные мочевины как ингибиторы ацил кофермента а:холестерин ацил трансферазы (асат) фармацевтическая композиция, способ ингибирования (асат)
CN1273526A (zh) * 1998-07-14 2000-11-15 Em工业股份有限公司 微分散给药系统
US7015233B2 (en) * 2003-06-12 2006-03-21 Abbott Laboratories Fused compounds that inhibit vanilloid subtype 1 (VR1) receptor
TWI389688B (zh) * 2004-06-08 2013-03-21 Vertex Pharma Vx-950之形態與調配物及其製備方法與用途
CN101048140B (zh) * 2004-08-27 2013-06-19 拜尔保健公司 用于治疗癌症的药物组合物
MX2007012947A (es) * 2005-04-18 2008-04-09 Rubicon Res Pvt Ltd Composiciones biomejoradas.
KR100715355B1 (ko) * 2005-09-30 2007-05-07 주식회사유한양행 프란루카스트를 함유하는 분무-건조 과립 및 그의 제조방법
CN101346128B (zh) * 2005-10-25 2013-10-02 雅培制药有限公司 包含低水溶解度药物的配方及其使用方法
WO2007066189A2 (en) * 2005-12-09 2007-06-14 Pfizer Products Inc. Salts, prodrugs and formulations of 1-[5-(4-amino-7-isopropyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-2-methoxy-phenyl]-3-(2,4-dichloro-phenyl)-urea
US7745448B2 (en) * 2005-12-28 2010-06-29 Abbott Laboratories Inc. Crystalline N-(4-(4-aminothieno[2,3-d]pyrimidin-5-yl)phenyl)-N′-(2-fluoro-5-(trifluoromethyl)phenyl)urea ethanolate
KR101418267B1 (ko) * 2006-02-09 2014-07-11 머크 샤프 앤드 돔 코포레이션 Cetp 억제제의 중합체 제형

Also Published As

Publication number Publication date
WO2009050289A3 (en) 2010-03-25
US20090143423A1 (en) 2009-06-04
GT201000095A (es) 2012-04-03
WO2009050289A2 (en) 2009-04-23
CO6270303A2 (es) 2011-04-20
BRPI0818339A2 (pt) 2015-04-22
KR20100090689A (ko) 2010-08-16
UY31406A1 (es) 2009-05-29
RU2010119924A (ru) 2011-11-27
UA100866C2 (ru) 2013-02-11
EP2197426A2 (en) 2010-06-23
CL2008003092A1 (es) 2009-11-27
ECSP10010184A (es) 2010-06-29
CN101827585A (zh) 2010-09-08
AU2008313620A1 (en) 2009-04-23
CA2699335A1 (en) 2009-04-23
AR068916A1 (es) 2009-12-16
MX2010004292A (es) 2010-08-02
PE20091041A1 (es) 2009-08-22
DOP2010000114A (es) 2010-05-15
TW200922549A (en) 2009-06-01
JP2011500647A (ja) 2011-01-06
ZA201002130B (en) 2011-11-30

Similar Documents

Publication Publication Date Title
CR11441A (es) Producto de dispersion solida que contiene un compuesto a base de n-aril urea
CU20060153A7 (es) Nueva forma cristalina v de agomelatina, procedimiento para su preparación y composiciones farmacéuticas que las contienen
CL2015001959A1 (es) (divisional solicitud 1567-2013) combinaciones de principios activos que comprenden piridiletilbenzamidas y otros principios activos
EA200971081A1 (ru) Пуриновые производные и их применение в качестве модуляторов толл-подобного рецептора 7
AR059350A1 (es) Formulacion farmaceutica para aerosoles con dos o mas principios activos y al menos una sustancia tensioactiva
WO2010041141A3 (en) Oil-based foamable carriers and formulations
MX2011006527A (es) Agentes medicinales unidos a dipeptido.
UA108641C2 (uk) Паразитицидна композиція, яка містить чотири активних агенти, та спосіб її застосування
BR112014000178A2 (pt) composições tópicas
MY151986A (en) Adamantyl diamide derivatives and uses of same
CL2010001642A1 (es) Composicion farmaceutica topica en gel que comprende a) 0,25 a 4,5% de un agente activo para el tratamiento de la queratosis actinica, b) un agente queratoliticamente activo, c) un formador de gel, d) un solvente organico, y menos de 5% en peso de agua; util para el tratamiento de la queratosis actinica.
BR112014011609A2 (pt) material de distribuição de fármaco polimérico, método para produção do mesmo, e método para distribuição de uma composição de distribuição de fármaco
CR11442A (es) Producto de dispersion solida de drogas basadas en n-aril urea
WO2010047592A3 (en) Preservation mixture and use thereof
BR112013028531A2 (pt) composição inseticida líquida
UY31059A1 (es) Formulaciones de aminoacido n-halogenado
TR200902923T2 (tr) Megestrol maddenin farmasötik olarak kararlı bir süspansiyonu.
CL2011001207A1 (es) Extruidos que contienen al menos una sustancia farmacéuticamente activa en forma de agujas, tal que la relación entre el tamaño de partículas de la sustancia farmacéuticamente activa con forma de agujas y el diámetro de la cadena es de al menos 1:20; composición farmacéutica; y su uso para preparar medicamentos.
DE602005025493D1 (de) Entzündungshemmende wirkstoffe
GT200500349A (es) Formulaciones de benzoxazoles substituidos
BR112012031471A2 (pt) mistura para tratamento de fertilizantes
MX2009005329A (es) Composiciones farmaceuticas anticonvulsivas.
ITMI20052515A1 (it) Formulazione farmaceutica per il trattamento della osteoartrite
MX2009003930A (es) Novedoso cristal de (s)-(+)-2-(2-clorofenil)-2-hidroxi-etil carbamato.
GT200400273A (es) Compuestos de haloalqueno, proceso para su produccion y pesticidas que los contienen.

Legal Events

Date Code Title Description
FA Abandonment or withdrawal (granting procedure)