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CL2007003805A1 - Forma cristalina del compuesto 3-{[5-(acetidin-1-ilcarbonil)piracin-2-il]oxi}-5-[(1-metiletil)oxi]-n-1h-pirazol-3-ilbenzamida; procedimiento de preparacion; composicion farmaceutica que comprende a dicha forma; y uso para el tratamiento de la diabete - Google Patents

Forma cristalina del compuesto 3-{[5-(acetidin-1-ilcarbonil)piracin-2-il]oxi}-5-[(1-metiletil)oxi]-n-1h-pirazol-3-ilbenzamida; procedimiento de preparacion; composicion farmaceutica que comprende a dicha forma; y uso para el tratamiento de la diabete

Info

Publication number
CL2007003805A1
CL2007003805A1 CL200703805A CL2007003805A CL2007003805A1 CL 2007003805 A1 CL2007003805 A1 CL 2007003805A1 CL 200703805 A CL200703805 A CL 200703805A CL 2007003805 A CL2007003805 A CL 2007003805A CL 2007003805 A1 CL2007003805 A1 CL 2007003805A1
Authority
CL
Chile
Prior art keywords
oxi
methylety
ilcarbonil
ilbenzamida
piracin
Prior art date
Application number
CL200703805A
Other languages
English (en)
Inventor
James Tomkinson Gary Pe Mccabe
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39138920&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2007003805(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of CL2007003805A1 publication Critical patent/CL2007003805A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CL200703805A 2006-12-21 2007-12-21 Forma cristalina del compuesto 3-{[5-(acetidin-1-ilcarbonil)piracin-2-il]oxi}-5-[(1-metiletil)oxi]-n-1h-pirazol-3-ilbenzamida; procedimiento de preparacion; composicion farmaceutica que comprende a dicha forma; y uso para el tratamiento de la diabete CL2007003805A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US87125506P 2006-12-21 2006-12-21

Publications (1)

Publication Number Publication Date
CL2007003805A1 true CL2007003805A1 (es) 2008-08-01

Family

ID=39138920

Family Applications (1)

Application Number Title Priority Date Filing Date
CL200703805A CL2007003805A1 (es) 2006-12-21 2007-12-21 Forma cristalina del compuesto 3-{[5-(acetidin-1-ilcarbonil)piracin-2-il]oxi}-5-[(1-metiletil)oxi]-n-1h-pirazol-3-ilbenzamida; procedimiento de preparacion; composicion farmaceutica que comprende a dicha forma; y uso para el tratamiento de la diabete

Country Status (21)

Country Link
US (2) US20100094009A1 (es)
EP (1) EP2121666A1 (es)
JP (1) JP2010513445A (es)
KR (1) KR20090090390A (es)
CN (1) CN101595104A (es)
AR (1) AR064625A1 (es)
AU (1) AU2007336016A1 (es)
BR (1) BRPI0721143A2 (es)
CA (1) CA2671535A1 (es)
CL (1) CL2007003805A1 (es)
CO (1) CO6190522A2 (es)
EC (1) ECSP099427A (es)
MX (1) MX2009006729A (es)
NO (1) NO20092129L (es)
PE (1) PE20081396A1 (es)
RU (1) RU2009121756A (es)
SA (1) SA07280732B1 (es)
TW (1) TW200833339A (es)
UY (1) UY30822A1 (es)
WO (1) WO2008075073A1 (es)
ZA (1) ZA200904296B (es)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0102764D0 (sv) 2001-08-17 2001-08-17 Astrazeneca Ab Compounds
RU2392275C2 (ru) * 2004-02-18 2010-06-20 Астразенека Аб Бензамидные производные и их применение в качестве активирующих глюкокиназу агентов
TW200600086A (en) * 2004-06-05 2006-01-01 Astrazeneca Ab Chemical compound
TW200714597A (en) * 2005-05-27 2007-04-16 Astrazeneca Ab Chemical compounds
WO2007007041A1 (en) 2005-07-09 2007-01-18 Astrazeneca Ab Heteroaryl benzamide derivatives for use as glk activators in the treatment of diabetes
SA07280576B1 (ar) * 2006-10-26 2011-06-22 استرازينيكا ايه بي مركبات بنزويل أمينو سيكليل غير متجانسة بأعتبارها عوامل منشطة للجلوكوكيناز
PE20110568A1 (es) 2008-08-04 2011-09-07 Astrazeneca Ab Agentes terapeuticos 414
GB0902434D0 (en) * 2009-02-13 2009-04-01 Astrazeneca Ab Chemical process
GB0902406D0 (en) * 2009-02-13 2009-04-01 Astrazeneca Ab Crystalline polymorphic form
AR076221A1 (es) * 2009-04-09 2011-05-26 Astrazeneca Ab Derivado de pirazol [4,5-e] pirimidina y su uso para tratar diabetes y obesidad
AR076220A1 (es) 2009-04-09 2011-05-26 Astrazeneca Ab Derivados de pirazol [4,5 - e] pirimidina
WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
US8933024B2 (en) 2010-06-18 2015-01-13 Sanofi Azolopyridin-3-one derivatives as inhibitors of lipases and phospholipases
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
TW201215387A (en) 2010-07-05 2012-04-16 Sanofi Aventis Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
WO2013045413A1 (en) 2011-09-27 2013-04-04 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
GB201714777D0 (en) 2017-09-14 2017-11-01 Univ London Queen Mary Agent

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Also Published As

Publication number Publication date
AR064625A1 (es) 2009-04-15
EP2121666A1 (en) 2009-11-25
RU2009121756A (ru) 2011-01-27
BRPI0721143A2 (pt) 2014-03-11
KR20090090390A (ko) 2009-08-25
JP2010513445A (ja) 2010-04-30
ZA200904296B (en) 2010-04-28
NO20092129L (no) 2009-06-18
CA2671535A1 (en) 2008-06-26
US20080153800A1 (en) 2008-06-26
UY30822A1 (es) 2008-07-31
WO2008075073A1 (en) 2008-06-26
TW200833339A (en) 2008-08-16
CN101595104A (zh) 2009-12-02
PE20081396A1 (es) 2008-12-05
MX2009006729A (es) 2009-08-07
ECSP099427A (es) 2009-07-31
US20100094009A1 (en) 2010-04-15
SA07280732B1 (ar) 2011-08-20
US7696191B2 (en) 2010-04-13
AU2007336016A1 (en) 2008-06-26
CO6190522A2 (es) 2010-08-19

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