ZA200707408B - Boron-containing small molecules - Google Patents

Boron-containing small molecules

Info

Publication number: ZA200707408B
Authority: ZA; South Africa
Prior art keywords: boron; small molecules; containing small; molecules; small
Prior art date: 2005-02-16

Application number

ZA200707408A

Other languages

English (en)

Inventor

Stephen J Baker

Akama Tsutomu

Bellinger-Kawahara Carolyn

Vincent S Hernandez

Karin M Hold

James J Leyden

Kirk R Maples

Jacob J Plattner

Sanders Virginia

Zhang Yong-Kang

Original Assignee

Anacor Pharmaceuticals Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-02-16

Filing date

2006-02-16

Publication date

2009-11-25

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36917059&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200707408(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2006-02-16 Application filed by Anacor Pharmaceuticals Inc filed Critical Anacor Pharmaceuticals Inc

2009-11-25 Publication of ZA200707408B publication Critical patent/ZA200707408B/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/05—Cyclic compounds having at least one ring containing boron but no carbon in the ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/69—Boron compounds
- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
- A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
- A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
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- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/027—Organoboranes and organoborohydrides
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Virology (AREA)
Oncology (AREA)
Engineering & Computer Science (AREA)
Communicable Diseases (AREA)
Bioinformatics & Cheminformatics (AREA)
Molecular Biology (AREA)
Tropical Medicine & Parasitology (AREA)
Epidemiology (AREA)
Dermatology (AREA)
Biotechnology (AREA)
Pulmonology (AREA)
Immunology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Neurology (AREA)
AIDS & HIV (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Ophthalmology & Optometry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

ZA200707408A 2005-02-16 2006-02-16 Boron-containing small molecules ZA200707408B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US65406005P	2005-02-16	2005-02-16

Publications (1)

Publication Number	Publication Date
ZA200707408B true ZA200707408B (en)	2009-11-25

Family

ID=36917059

Family Applications (4)

Application Number	Title	Priority Date	Filing Date
ZA200707408A ZA200707408B (en)	2005-02-16	2006-02-16	Boron-containing small molecules
ZA2009/05950A ZA200905950B (en)	2005-02-16	2009-08-27	Boron-containing small molecules
ZA2010/05380A ZA201005380B (en)	2005-02-16	2010-07-28	Boron-containing small molecules
ZA2015/06944A ZA201506944B (en)	2005-02-16	2015-09-17	Boron-containing small molecules

Family Applications After (3)

Application Number	Title	Priority Date	Filing Date
ZA2009/05950A ZA200905950B (en)	2005-02-16	2009-08-27	Boron-containing small molecules
ZA2010/05380A ZA201005380B (en)	2005-02-16	2010-07-28	Boron-containing small molecules
ZA2015/06944A ZA201506944B (en)	2005-02-16	2015-09-17	Boron-containing small molecules

Country Status (26)

Country	Link
US (11)	US7582621B2 (xx)
EP (4)	EP1853251B1 (xx)
JP (6)	JP5038912B2 (xx)
KR (4)	KR101337045B1 (xx)
CN (2)	CN101914109B (xx)
AU (3)	AU2006214247C1 (xx)
BR (1)	BRPI0608431B8 (xx)
CA (1)	CA2597982C (xx)
CY (3)	CY1120695T1 (xx)
DK (3)	DK3424932T3 (xx)
ES (4)	ES2414095T3 (xx)
FR (1)	FR20C1024I2 (xx)
HK (3)	HK1109735A1 (xx)
HU (4)	HUE026021T2 (xx)
IL (2)	IL185080A (xx)
LT (1)	LTC2343304I2 (xx)
LU (1)	LUC00157I2 (xx)
MX (1)	MX369262B (xx)
NL (1)	NL301049I2 (xx)
NZ (3)	NZ598441A (xx)
PL (4)	PL2987796T3 (xx)
PT (4)	PT1853251E (xx)
RU (3)	RU2414906C2 (xx)
SI (3)	SI2987796T1 (xx)
WO (1)	WO2006089067A2 (xx)
ZA (4)	ZA200707408B (xx)

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Publication number	Publication date
NZ598441A (en)	2013-07-26
RU2606947C2 (ru)	2017-01-10
US8889656B2 (en)	2014-11-18
IL185080A0 (en)	2008-08-07
JP2008535781A (ja)	2008-09-04
WO2006089067A2 (en)	2006-08-24
AU2006214247A1 (en)	2006-08-24
US20130244980A1 (en)	2013-09-19
CY1124503T1 (el)	2022-07-22
JP5038912B2 (ja)	2012-10-03
ZA200905950B (en)	2010-11-24
US20210070780A1 (en)	2021-03-11
KR20070112390A (ko)	2007-11-23
CY1120695T1 (el)	2019-12-11
EP3424932B1 (en)	2021-04-07
HUS2000019I1 (hu)	2020-07-28
IL185080A (en)	2012-07-31
HK1160139A1 (en)	2012-08-10
IL207156A (en)	2014-04-30
EP3424932A1 (en)	2019-01-09
KR101337068B1 (ko)	2013-12-06
LUC00157I1 (xx)	2020-06-08
NL301049I2 (nl)	2020-09-10
WO2006089067A3 (en)	2007-07-19
CY2020027I2 (el)	2021-01-27
LTC2343304I2 (lt)	2022-11-10
PT2343304E (pt)	2015-08-26
CN101160124A (zh)	2008-04-09
RU2007134429A (ru)	2009-03-27
US20190330245A1 (en)	2019-10-31
BRPI0608431B1 (pt)	2020-09-15
ES2540966T3 (es)	2015-07-15
FR20C1024I2 (fr)	2021-07-09
AU2006214247C1 (en)	2012-11-08
US20100190748A1 (en)	2010-07-29
JP2016020374A (ja)	2016-02-04
US20140142064A1 (en)	2014-05-22
ZA201506944B (en)	2018-08-29
CN101914109B (zh)	2014-07-23
US20160108063A1 (en)	2016-04-21
KR101337045B1 (ko)	2013-12-05
CA2597982A1 (en)	2006-08-24
JP2010248265A (ja)	2010-11-04
US20110319361A1 (en)	2011-12-29
SI3424932T1 (sl)	2021-08-31
AU2010203096B2 (en)	2010-12-02
LUC00157I2 (xx)	2021-07-06
RU2414906C2 (ru)	2011-03-27
EP1853251A4 (en)	2010-01-13
DK2987796T3 (en)	2018-09-17
ZA201005380B (en)	2016-08-31
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RU2016145916A3 (xx)	2020-07-21
ES2686981T3 (es)	2018-10-23
LTPA2020524I1 (lt)	2020-09-10
RU2010133524A (ru)	2012-02-20
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EP1853251A2 (en)	2007-11-14
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PL2987796T3 (pl)	2018-12-31
KR101426220B1 (ko)	2014-08-05
US20060234981A1 (en)	2006-10-19
KR101456815B1 (ko)	2014-10-31
EP2343304B1 (en)	2015-06-10
JP6046876B2 (ja)	2016-12-21
MX369262B (es)	2019-11-04
ES2414095T3 (es)	2013-07-18
CY2020027I1 (el)	2021-01-27
US7582621B2 (en)	2009-09-01
JP2017105826A (ja)	2017-06-15
CN101914109A (zh)	2010-12-15
AU2010203096A1 (en)	2010-08-12
SI2987796T1 (sl)	2018-11-30
US8039451B2 (en)	2011-10-18
KR20130100019A (ko)	2013-09-06
ES2872962T3 (es)	2021-11-03
BRPI0608431B8 (pt)	2021-05-25
KR20100105869A (ko)	2010-09-30
CA2597982C (en)	2014-07-08
US8440642B2 (en)	2013-05-14
HUE040060T2 (hu)	2019-02-28
AU2010203096C1 (en)	2012-09-20
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PT3424932T (pt)	2021-05-19
EP2987796A1 (en)	2016-02-24
BRPI0608431A2 (pt)	2009-12-29
AU2011200994A1 (en)	2011-03-31
RU2016145916A (ru)	2018-05-23
SI2343304T1 (sl)	2015-08-31
JP2013018778A (ja)	2013-01-31
NL301049I1 (nl)	2020-07-01
HUE054365T2 (hu)	2021-09-28
DK3424932T3 (da)	2021-05-25
HK1221956A1 (zh)	2017-06-16
HUE026021T2 (en)	2016-05-30
HK1109735A1 (en)	2008-06-20
PL3424932T3 (pl)	2021-09-20
DK2343304T3 (en)	2015-06-29
US20170066788A1 (en)	2017-03-09
NZ560448A (en)	2009-08-28
PT2987796T (pt)	2018-10-18
AU2006214247B2 (en)	2010-08-05

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