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UY25330A1 - Nuevos macrólidos - Google Patents

Nuevos macrólidos

Info

Publication number
UY25330A1
UY25330A1 UY25330A UY25330A UY25330A1 UY 25330 A1 UY25330 A1 UY 25330A1 UY 25330 A UY25330 A UY 25330A UY 25330 A UY25330 A UY 25330A UY 25330 A1 UY25330 A1 UY 25330A1
Authority
UY
Uruguay
Prior art keywords
new
birds
mammals
fish
macrolids
Prior art date
Application number
UY25330A
Other languages
English (en)
Inventor
John Philip Dirlam Y Mcarthur
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Priority to UY25574A priority Critical patent/UY25574A1/es
Publication of UY25330A1 publication Critical patent/UY25330A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

Se refiere a nuevas eritromicinas y azalidas útiles como agentes antibacterianas y antiprotozoos y en aplicaciones en mamíferos, incluyendo el ser humano, así como en peces y aves. También refiere a composiciones farmacéuticas conteniendo los nuevos compuestos y procedimientos para el tratamiento de las infecciones bacterianas y provocadas por protozoos en mamíferos, peces y aves, mediante administración de los nuevos compuestos a los mamíferos, peces y aves que necesitan dicho tratamiento.
UY25330A 1998-01-02 1998-12-30 Nuevos macrólidos UY25330A1 (es)

Priority Applications (1)

Application Number Priority Date Filing Date Title
UY25574A UY25574A1 (es) 1998-01-02 1999-06-18 Procedimiento para preparar nuevos macrolidos

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US7034398P 1998-01-02 1998-01-02

Publications (1)

Publication Number Publication Date
UY25330A1 true UY25330A1 (es) 2000-12-29

Family

ID=22094723

Family Applications (2)

Application Number Title Priority Date Filing Date
UY25330A UY25330A1 (es) 1998-01-02 1998-12-30 Nuevos macrólidos
UY25574A UY25574A1 (es) 1998-01-02 1999-06-18 Procedimiento para preparar nuevos macrolidos

Family Applications After (1)

Application Number Title Priority Date Filing Date
UY25574A UY25574A1 (es) 1998-01-02 1999-06-18 Procedimiento para preparar nuevos macrolidos

Country Status (34)

Country Link
US (2) US6472371B1 (es)
EP (1) EP1044207A1 (es)
JP (1) JP2002500230A (es)
KR (1) KR100352809B1 (es)
CN (1) CN1284081A (es)
AP (1) AP9801420A0 (es)
AR (4) AR014948A1 (es)
AU (1) AU756409B2 (es)
BG (1) BG104644A (es)
BR (1) BR9814601A (es)
CA (1) CA2316919C (es)
CO (1) CO4970821A1 (es)
CZ (1) CZ20002458A3 (es)
DZ (1) DZ2698A1 (es)
EA (1) EA200000594A1 (es)
GT (1) GT199800206A (es)
HR (1) HRP20000442A2 (es)
HU (1) HUP0100420A3 (es)
IL (1) IL137024A0 (es)
IS (1) IS5528A (es)
MA (1) MA24729A1 (es)
NO (1) NO20003347L (es)
NZ (1) NZ504986A (es)
OA (1) OA11438A (es)
PA (1) PA8465301A1 (es)
PE (1) PE20000049A1 (es)
PL (1) PL341642A1 (es)
SK (1) SK9782000A3 (es)
TN (1) TNSN98238A1 (es)
TW (1) TW520374B (es)
UY (2) UY25330A1 (es)
WO (1) WO1999035156A1 (es)
YU (1) YU41500A (es)
ZA (1) ZA9811939B (es)

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AP1060A (en) 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.
US6043227A (en) * 1998-08-19 2000-03-28 Pfizer Inc. C11 carbamates of macrolide antibacterials
EP1437360A3 (en) * 1998-08-19 2005-04-06 Pfizer Products Inc. C11 Carbamates of macrolide antibacterials
EP1754700A3 (en) 1999-01-27 2007-05-09 Kosan Biosciences, Inc. Synthesis of oligoketides
US6451768B1 (en) 1999-04-16 2002-09-17 Kosan Biosciences, Inc. Macrolide antiinfective agents
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
CA2370743A1 (en) 1999-04-16 2000-10-26 Dennis Hlasta Ketolide antibacterials
CZ20013733A3 (cs) 1999-05-24 2002-11-13 Pfizer Products Inc. Deriváty 13-methylerythromycinu
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ATE406348T1 (de) 2004-09-23 2008-09-15 Schering Plough Ltd Bekämpfung von parasiten in tieren durch verwendung neuer trifluormethansulfonanilidoximetherderivate
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UA85937C2 (uk) 2004-12-21 2009-03-10 Пфайзер Продактс Інк. Макроліди
AR054380A1 (es) * 2005-06-09 2007-06-20 Schering Plough Ltd Control de parasitos en animales con derivados de n- ((feniloxi) fenil) -1,1,1-trifluorometansulfonamida y de n-(fenilsulfanil) fenil) -1,1,1-trifluorometansulfonamida
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
US20070238700A1 (en) * 2006-04-10 2007-10-11 Winzenberg Kevin N N-phenyl-1,1,1-trifluoromethanesulfonamide hydrazone derivative compounds and their usage in controlling parasites
US8044230B2 (en) * 2006-12-13 2011-10-25 Intervet Inc. Water-soluble prodrugs of chloramphenicol, thiamphenicol, and analogs thereof
WO2008076259A1 (en) * 2006-12-13 2008-06-26 Schering-Plough Ltd. Water-soluble prodrugs of florfenicol and its analogs
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
ES2666187T3 (es) 2007-06-27 2018-05-03 E. I. Du Pont De Nemours And Company Procedimiento de control de plagas en animales
WO2009064953A1 (en) * 2007-11-15 2009-05-22 Enanta Pharmaceuticals, Inc. Use of bridged macrolides or tylosin derivatives in treating inflammatory bowel diseases
TWI468407B (zh) 2008-02-06 2015-01-11 Du Pont 中離子農藥
EP2321269B1 (en) * 2008-07-30 2018-09-19 Intervet International B.V. Process for preparing oxazoline-protected aminodiol compounds useful as intermediates to florfenicol
KR20120047996A (ko) 2009-08-05 2012-05-14 이 아이 듀폰 디 네모아 앤드 캄파니 메소이온성 살충제
UA107804C2 (en) 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
BR112012002519A2 (pt) 2009-08-05 2019-09-24 Du Pont "pesticidas mesoiônicos"
UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
JP5933530B2 (ja) 2010-05-27 2016-06-08 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニーＥ．Ｉ．Ｄｕ Ｐｏｎｔ Ｄｅ Ｎｅｍｏｕｒｓ Ａｎｄ Ｃｏｍｐａｎｙ ４−［５−［３−クロロ−５−（トリフルオロメチル）フェニル］−４，５−ジヒドロ−５−（トリフルオロメチル）−３−イソオキサゾリル］−ｎ−［２−オキソ−２−［（２，２，２−トリフルオロエチル）アミノ］エチル］−１−ナフタレンカルボキサミドの結晶質形態
WO2012087630A1 (en) 2010-12-20 2012-06-28 E.I. Du Pont De Nemours And Company Pyridine and pyrimidine compounds for controlling invertebrate
WO2012105562A1 (ja) * 2011-01-31 2012-08-09 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 新規マクロライド誘導体
MX2013014326A (es) 2011-06-20 2014-01-23 Du Pont Compuestos heterociclicos para tratar infecciones por helmintos.
CN102260306B (zh) * 2011-07-22 2012-07-18 山东鲁抗舍里乐药业有限公司 一种制备泰拉霉素的方法
JP2015502936A (ja) 2011-11-28 2015-01-29 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニーＥ．Ｉ．Ｄｕ Ｐｏｎｔ Ｄｅ Ｎｅｍｏｕｒｓ Ａｎｄ Ｃｏｍｐａｎｙ スルホンアミド駆虫薬
WO2013158422A1 (en) 2012-04-17 2013-10-24 E. I. Du Pont De Nemours And Company Heterocyclic compounds for controlling invertebrate pests
WO2014099837A1 (en) 2012-12-18 2014-06-26 E. I. Du Pont De Nemours And Company Sulfonamide anthelmintics
CN105669798B (zh) * 2013-08-23 2019-07-26 普莱柯生物工程股份有限公司 一种大环内酯类化合物
CN103965273B (zh) * 2013-08-23 2016-05-25 普莱柯生物工程股份有限公司 一种大环内酯类化合物

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Also Published As

Publication number Publication date
TNSN98238A1 (fr) 2005-03-15
AR020551A2 (es) 2002-05-15
CO4970821A1 (es) 2000-11-07
AR019787A2 (es) 2002-03-13
CN1284081A (zh) 2001-02-14
HRP20000442A2 (en) 2001-04-30
KR100352809B1 (ko) 2002-11-01
AR020851A2 (es) 2002-05-29
WO1999035156B1 (en) 1999-10-21
SK9782000A3 (en) 2001-12-03
WO1999035156A1 (en) 1999-07-15
YU41500A (sh) 2003-02-28
HUP0100420A2 (hu) 2001-07-30
US20040092459A1 (en) 2004-05-13
CA2316919A1 (en) 1999-07-15
BR9814601A (pt) 2000-10-17
AR014948A1 (es) 2001-04-11
PA8465301A1 (es) 2000-09-29
UY25574A1 (es) 1999-09-27
MA24729A1 (fr) 1999-07-01
EA200000594A1 (ru) 2001-04-23
NO20003347D0 (no) 2000-06-27
KR20010024818A (ko) 2001-03-26
NO20003347L (no) 2000-08-28
US6472371B1 (en) 2002-10-29
NZ504986A (en) 2003-03-28
AP9801420A0 (en) 1998-12-31
OA11438A (en) 2004-04-30
HUP0100420A3 (en) 2003-07-28
BG104644A (en) 2001-01-31
CA2316919C (en) 2004-10-26
JP2002500230A (ja) 2002-01-08
CZ20002458A3 (cs) 2001-10-17
EP1044207A1 (en) 2000-10-18
US7015203B2 (en) 2006-03-21
ZA9811939B (en) 2000-06-30
DZ2698A1 (fr) 2003-03-29
GT199800206A (es) 2000-06-21
AU1444799A (en) 1999-07-26
PL341642A1 (en) 2001-04-23
TW520374B (en) 2003-02-11
IL137024A0 (en) 2001-06-14
PE20000049A1 (es) 2000-02-07
IS5528A (is) 2000-06-09
AU756409B2 (en) 2003-01-09

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