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HN1998000159A - Derivados de 9- amino - 3 ceto eritromicina - Google Patents

Derivados de 9- amino - 3 ceto eritromicina

Info

Publication number
HN1998000159A
HN1998000159A HN1998000159A HN1998000159A HN1998000159A HN 1998000159 A HN1998000159 A HN 1998000159A HN 1998000159 A HN1998000159 A HN 1998000159A HN 1998000159 A HN1998000159 A HN 1998000159A HN 1998000159 A HN1998000159 A HN 1998000159A
Authority
HN
Honduras
Prior art keywords
eritromicina
ceto
derivatives
amino
present
Prior art date
Application number
HN1998000159A
Other languages
English (en)
Inventor
Pfizer Products Inc
Original Assignee
Monsanto Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Monsanto Co filed Critical Monsanto Co
Publication of HN1998000159A publication Critical patent/HN1998000159A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

LA PRESENTE INVENCION SE REFIERE A:
HN1998000159A 1997-10-29 1998-10-08 Derivados de 9- amino - 3 ceto eritromicina HN1998000159A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US6367697P 1997-10-29 1997-10-29

Publications (1)

Publication Number Publication Date
HN1998000159A true HN1998000159A (es) 1999-02-09

Family

ID=22050768

Family Applications (1)

Application Number Title Priority Date Filing Date
HN1998000159A HN1998000159A (es) 1997-10-29 1998-10-08 Derivados de 9- amino - 3 ceto eritromicina

Country Status (13)

Country Link
US (1) US6159945A (es)
AP (1) AP9801378A0 (es)
AR (1) AR017177A1 (es)
AU (1) AU9277698A (es)
CO (1) CO4810375A1 (es)
GT (1) GT199800163A (es)
HN (1) HN1998000159A (es)
HR (1) HRP980571A2 (es)
MA (1) MA26558A1 (es)
PA (1) PA8461701A1 (es)
PE (1) PE122499A1 (es)
TN (1) TNSN98194A1 (es)
WO (1) WO1999021866A1 (es)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6710033B1 (en) 1996-08-14 2004-03-23 Vanderbilt University Methods and treatment of multiple sclerosis
US6890526B2 (en) 1997-05-06 2005-05-10 Vanderbilt University Methods and reagents for the treatment of multiple sclerosis
AP9801420A0 (en) * 1998-01-02 1998-12-31 Pfizer Prod Inc Novel macrolides.
AU3439899A (en) 1998-06-03 1999-12-20 Pfizer Products Inc. Tricyclic 3-keto derivatives of 6-o-methylerythromycin
TR200102129T2 (tr) 1998-12-10 2002-01-21 Pfizer Products Inc. Karbamat ve karbazat ketolid antibiyotikleri.
EP1298138B1 (en) * 1998-12-10 2006-11-02 Pfizer Products Inc. Carbamate and Carbazate Ketolide Antibiotics
HK1042707A1 (zh) 1999-01-27 2002-08-23 辉瑞产品公司 酮內酯類抗生素
OA11945A (en) * 1999-05-24 2006-04-13 Pfizer Prod Inc 13-Methyl erythromycin derivatives.
ID27331A (id) * 1999-09-29 2001-03-29 Pfizer Prod Inc Pembuatan antibiotik-antibiotik ketolida karbamat
US6498146B1 (en) * 1999-10-28 2002-12-24 Pfizer Inc Erythromycin derivatives
EP1146051A3 (en) * 2000-04-10 2001-10-31 Pfizer Products Inc. Erythromycin A derivatives
US20020115621A1 (en) * 2000-08-07 2002-08-22 Wei-Gu Su Macrolide antibiotics
US20040208842A1 (en) * 2001-09-18 2004-10-21 Ritchie Branson W. Antimicrobial cleansing compositions and methods of use
US20070003508A1 (en) * 2005-07-01 2007-01-04 Wooley Richard E Methods and compositions for promoting wound healing
US20040151765A1 (en) * 2001-09-18 2004-08-05 Ritchie Branson W. Methods and compositions for wound management
WO2004080391A2 (en) 2003-03-10 2004-09-23 Optimer Pharmaceuticals, Inc. Novel antibacterial agents
US20070185202A1 (en) * 2004-03-03 2007-08-09 University Of Georgia Research Foundation, Inc. Methods and compositions for ophthalmic treatment of fungal and bacterial infections
CA2591746A1 (en) * 2004-12-21 2006-06-29 Pfizer Products Inc. Macrolides
CN105732745A (zh) 2007-10-25 2016-07-06 森普拉制药公司 大环内酯类抗菌剂的制备方法
US9072759B2 (en) 2008-10-24 2015-07-07 Cempra Pharmaceuticals, Inc. Biodefenses using triazole-containing macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
EP2475253B1 (en) 2009-09-10 2016-10-26 Cempra Pharmaceuticals, Inc. Methods for treating malaria, tuberculosis and mac diseases
SI2550286T1 (sl) 2010-03-22 2016-04-29 Cempra Pharmaceuticals, Inc. Kristalne oblike makrolida in njihove uporabe
CA2799937A1 (en) 2010-05-20 2011-11-24 Cempra Pharmaceuticals, Inc. Processes for preparing macrolides and ketolides and intermediates therefor
JP6042334B2 (ja) 2010-09-10 2016-12-14 センプラ ファーマシューティカルズ,インコーポレイテッド 疾患治療のための水素結合形成フルオロケトライド
JP6208742B2 (ja) 2012-03-27 2017-10-04 センプラ ファーマシューティカルズ,インコーポレイテッド マクロライド抗生物質を投与するための非経口製剤
WO2014152326A1 (en) 2013-03-14 2014-09-25 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
RU2015138797A (ru) 2013-03-15 2017-04-24 Семпра Фармасьютикалс, Инк. Конвергентные способы получения макролидных антибактериальных агентов
CN111825733A (zh) * 2013-04-04 2020-10-27 哈佛大学的校长及成员们 大环内酯及其制备和使用方法
WO2016057798A1 (en) 2014-10-08 2016-04-14 President And Fellows Of Harvard College 14-membered ketolides and methods of their preparation and use
US10640528B2 (en) 2015-03-25 2020-05-05 President And Fellows Of Havard College Macrolides with modified desosamine sugars and uses thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL99995A (en) * 1990-11-21 1997-11-20 Roussel Uclaf Erythromycin derivatives, their preparation and pharmaceutical compositions containing them
US6060234A (en) * 1991-01-17 2000-05-09 Abbott Laboratories Polyketide derivatives and recombinant methods for making same
CA2118488C (en) * 1992-04-22 2002-11-05 Toshifumi Asaka 5-o-desosaminylerythronolide a derivative
US6162794A (en) * 1997-05-09 2000-12-19 Pfizer Inc. Erythromycin derivatives
CZ9904388A3 (cs) * 1997-06-11 2002-10-16 Pfizer Products Inc. 9-Oximové deriváty erythromycinu

Also Published As

Publication number Publication date
PE122499A1 (es) 1999-12-02
US6159945A (en) 2000-12-12
AR017177A1 (es) 2001-08-22
AU9277698A (en) 1999-05-17
WO1999021866A1 (en) 1999-05-06
AP9801378A0 (en) 2000-04-29
CO4810375A1 (es) 1999-06-30
HRP980571A2 (en) 1999-08-31
PA8461701A1 (es) 2000-05-24
MA26558A1 (fr) 2004-12-20
TNSN98194A1 (fr) 2005-03-15
GT199800163A (es) 2000-04-15

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