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PT93629A - Processo para a preparacao de derivados de tieno-triazolo-diazepina - Google Patents

Processo para a preparacao de derivados de tieno-triazolo-diazepina

Info

Publication number
PT93629A
PT93629A PT93629A PT9362990A PT93629A PT 93629 A PT93629 A PT 93629A PT 93629 A PT93629 A PT 93629A PT 9362990 A PT9362990 A PT 9362990A PT 93629 A PT93629 A PT 93629A
Authority
PT
Portugal
Prior art keywords
tieno
triazolo
preparation
diazepine derivatives
diazepine
Prior art date
Application number
PT93629A
Other languages
English (en)
Other versions
PT93629B (pt
Inventor
Pierre Braquet
Andre Esanu
Jean-Pierre Laurent
Alian Rolland
Original Assignee
Scras
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Scras filed Critical Scras
Publication of PT93629A publication Critical patent/PT93629A/pt
Publication of PT93629B publication Critical patent/PT93629B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/22Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT93629A 1989-03-31 1990-03-30 Processo para a preparacao de derivados de tieno-triazolo-diazepina PT93629B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB898907256A GB8907256D0 (en) 1989-03-31 1989-03-31 New derivatives of hetrazepine as anti-asthmatic anti-allergic and gastro-intestinal protectors

Publications (2)

Publication Number Publication Date
PT93629A true PT93629A (pt) 1990-11-20
PT93629B PT93629B (pt) 1996-07-31

Family

ID=10654231

Family Applications (1)

Application Number Title Priority Date Filing Date
PT93629A PT93629B (pt) 1989-03-31 1990-03-30 Processo para a preparacao de derivados de tieno-triazolo-diazepina

Country Status (30)

Country Link
US (1) US5492906A (pt)
JP (1) JPH07103127B2 (pt)
KR (1) KR900014396A (pt)
AT (1) AT394561B (pt)
AU (1) AU622007B2 (pt)
BE (1) BE1003699A3 (pt)
CA (1) CA2013518C (pt)
CH (1) CH680365A5 (pt)
DE (1) DE4010316C2 (pt)
DK (1) DK80890A (pt)
ES (1) ES2019243A6 (pt)
FI (1) FI95036C (pt)
FR (2) FR2645022B1 (pt)
GB (2) GB8907256D0 (pt)
GR (1) GR1000394B (pt)
HK (1) HK95192A (pt)
IE (1) IE64564B1 (pt)
IN (1) IN174015B (pt)
IT (1) IT1240350B (pt)
LU (1) LU87710A1 (pt)
MA (1) MA21790A1 (pt)
MY (1) MY105538A (pt)
NL (1) NL194827C (pt)
NO (1) NO173784C (pt)
NZ (1) NZ233011A (pt)
OA (1) OA09442A (pt)
PT (1) PT93629B (pt)
SE (1) SE505417C2 (pt)
TN (1) TNSN90042A1 (pt)
ZA (1) ZA901765B (pt)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH30676A (en) * 1986-07-22 1997-09-16 Boehringer Ingelhein Kg Hetrazepine compounds which have useful pharmaceutical utility
US5382579A (en) * 1988-10-31 1995-01-17 Eisai Co., Ltd. Triazolo-1,4-diazepine derivatives and their use in pharmaceuticals
US5221671A (en) * 1988-10-31 1993-06-22 Eisai Co., Ltd. Triazolo-1,4-diazepine derivatives and their use in pharmaceuticals
US5304553A (en) * 1988-10-31 1994-04-19 Eisai Co., Ltd. 1,4-diazepine derivative and its pharmaceutical use
DE4027470A1 (de) * 1990-08-30 1992-03-05 Boehringer Ingelheim Kg Neue hetrazepinoide amide
ES2061406B1 (es) * 1993-05-07 1995-06-01 Uriach & Cia Sa J Nuevos derivados de la 2-(quinolina) con actividad farmacologica.
FI101989B (fi) * 1996-11-22 1998-09-30 Stora Enso Oyj Menetelmät neste- ja kaasutiiviin pakkauskartongin sekä pakkauksen val mistamiseksi sekä menetelmien mukaisesti valmistetut tuotteet
WO1998058930A1 (fr) 1997-06-25 1998-12-30 Nikken Chemicals Co., Ltd. Composes de triazolo-1,4-diazepine et composition medicinale les contenant
FR2779652B1 (fr) * 1998-06-15 2001-06-08 Sod Conseils Rech Applic Utilisation de diazepines pour la preparation de medicaments destines a traiter les etats pathologiques ou les maladies dans lesquels un des recepteurs de la somatostatine est implique
AU2001255708A1 (en) * 2000-04-28 2001-11-12 Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical College Synthesis and use of thienotriazolodiazepines
AU2004242777B2 (en) * 2003-05-30 2011-05-12 Ranbaxy Laboratories Limited Substituted pyrrole derivatives and their use as HMG-Co inhibitors
KR101329112B1 (ko) * 2005-11-08 2013-11-14 랜박시 래보러터리스 리미티드 (3r,5r)-7-〔2-(4-플루오로페닐)-5-이소프로필-3-페닐-4-〔(4-히드록시 메틸 페닐 아미노)카르보닐〕-피롤-1-일〕-3,5-디히드록시 헵탄산 헤미 칼슘염의 제조 방법
CL2007000667A1 (es) * 2006-03-14 2008-03-14 Ranbaxi Lab Ltd Composicion farmaceutica que comprende al acido 7-[2-(4-fluorofenil)-5-isopropil-3-fenil-4-[(4-hidroximetilfenilamino)carbonil]pirrol-1-il]-3,5-dihidroxi-heptanoico o una sal y al menos un agente estabilizante; procedimiento de preparacion, util en e
AU2007274724B2 (en) * 2006-07-14 2012-07-26 Ranbaxy Laboratories Limited Polymorphic forms of an HMG-CoA reductase inhibitor and uses thereof
KR101675984B1 (ko) * 2015-02-23 2016-11-14 한양대학교 에리카산학협력단 티에노디아제핀 유도체 또는 이의 약학적으로 허용가능한 염, 및 이를 유효성분으로 포함하는 약학적 조성물

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH30676A (en) * 1986-07-22 1997-09-16 Boehringer Ingelhein Kg Hetrazepine compounds which have useful pharmaceutical utility
US5028603A (en) * 1987-06-08 1991-07-02 Yoshitomi Pharmaceutical Industries, Ltd. Ester-substituted thienotriazolodiazepine compounds and pharmaceutical uses thereof
FI95708C (fi) * 1988-10-31 1996-03-11 Eisai Co Ltd Analogiamenetelmä 1,4-diatsepiinijohdannaisen ja sen farmaseuttisesti sopivan suolan valmistamiseksi
NL9000627A (nl) * 1990-03-29 1991-10-16 Scras Werkwijze ter bereiding van nieuwe thienotriazolo-diazepines.

Also Published As

Publication number Publication date
GR900100165A (en) 1990-07-31
BE1003699A3 (fr) 1992-05-26
GB2229723B (en) 1992-07-01
GB2229723A (en) 1990-10-03
JPH07103127B2 (ja) 1995-11-08
CA2013518A1 (en) 1990-09-30
IT9019884A1 (it) 1991-09-30
PT93629B (pt) 1996-07-31
DE4010316A1 (de) 1990-10-04
HK95192A (en) 1992-12-04
JPH02289582A (ja) 1990-11-29
ES2019243A6 (es) 1991-06-01
LU87710A1 (fr) 1990-07-24
KR900014396A (ko) 1990-10-23
OA09442A (fr) 1992-10-15
CH680365A5 (pt) 1992-08-14
FI901605A0 (fi) 1990-03-30
SE9000871L (sv) 1990-10-01
FI95036B (fi) 1995-08-31
IE900806L (en) 1990-09-30
NZ233011A (en) 1991-02-26
GR1000394B (el) 1992-06-30
DE4010316C2 (de) 2003-05-28
ATA56790A (de) 1991-10-15
NL194827C (nl) 2003-04-03
FR2645153B1 (fr) 1992-04-17
NO173784C (no) 1994-02-02
SE9000871D0 (sv) 1990-03-12
CA2013518C (en) 2004-02-24
IT9019884A0 (it) 1990-03-30
IE64564B1 (en) 1996-08-23
FR2645022A1 (fr) 1990-10-05
AU5242590A (en) 1990-11-01
US5492906A (en) 1996-02-20
AU622007B2 (en) 1992-03-26
SE505417C2 (sv) 1997-08-25
GB8907256D0 (en) 1989-05-17
FI95036C (fi) 1995-12-11
MA21790A1 (fr) 1990-10-01
FR2645153A1 (fr) 1990-10-05
NL194827B (nl) 2002-12-02
TNSN90042A1 (fr) 1991-03-05
AT394561B (de) 1992-05-11
MY105538A (en) 1994-10-31
ZA901765B (en) 1990-12-28
FR2645022B1 (fr) 1992-04-17
GB9007000D0 (en) 1990-05-30
DK80890D0 (da) 1990-03-30
NO901070L (no) 1990-10-01
NL9000626A (nl) 1990-10-16
DK80890A (da) 1990-10-01
NO901070D0 (no) 1990-03-07
IN174015B (pt) 1994-08-27
IT1240350B (it) 1993-12-07
NO173784B (no) 1993-10-25

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Legal Events

Date Code Title Description
FG3A Patent granted, date of granting

Effective date: 19960415