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NO951812L - Pyrrolderivater, deres fremstilling og anvendelse - Google Patents

Pyrrolderivater, deres fremstilling og anvendelse

Info

Publication number
NO951812L
NO951812L NO951812A NO951812A NO951812L NO 951812 L NO951812 L NO 951812L NO 951812 A NO951812 A NO 951812A NO 951812 A NO951812 A NO 951812A NO 951812 L NO951812 L NO 951812L
Authority
NO
Norway
Prior art keywords
group
branched
alkyl
pyrrole derivatives
preparation
Prior art date
Application number
NO951812A
Other languages
English (en)
Other versions
NO951812D0 (no
Inventor
Manuel Bedoya Zurita
Juan Antonio Diaz Martin
Gregorio Del Sol Moreno
Ulpiano Martin Escudero Perez
Maria Dolores Jimenez Bargueno
Magali Romanach Ferrer
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of NO951812D0 publication Critical patent/NO951812D0/no
Publication of NO951812L publication Critical patent/NO951812L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

5,6-dihydro-4H-tieno[3,4-c]pyrrolderivater med generell formel (D £OY> yT H N---' (I) hvor R! enten representerer en cyanogruppe, C}_4 alkoksy, C^ alkyltio, C:_t alkylsulfonyl, pyridyl, 3,4-dimetoksyfenyl eller cyklopropyl som eventuelt er substituert med en eller to alkylgrupper, eller en gruppe COR hvor R er en C^.^ alkyl- gruppe, fenyl eller piperidinyl, eller en benzylgruppe som er substituert med et eller flere halogenatomer og/eller rett- kjedet eller forgrenet C^ alkyl, rettkjedet eller forgrenet C^ alkoksy eller C02R' hvor R' er en rettkjedet eller forgrenet C1.4 alkylgruppe, eller en naftylmetylgruppe, og deres addisjonssalter med farmasøytisk tålbare syrer. Derivatene har terapeutisk anvendelse.
NO951812A 1994-05-10 1995-05-09 Pyrrolderivater, deres fremstilling og anvendelse NO951812L (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9405716A FR2719844B1 (fr) 1994-05-10 1994-05-10 Dérivés de 5,6-dihydro-4h-thiéno[3,4-c]pyrrole, leur préparation et leur application en thérapeutique.

Publications (2)

Publication Number Publication Date
NO951812D0 NO951812D0 (no) 1995-05-09
NO951812L true NO951812L (no) 1995-11-13

Family

ID=9463059

Family Applications (1)

Application Number Title Priority Date Filing Date
NO951812A NO951812L (no) 1994-05-10 1995-05-09 Pyrrolderivater, deres fremstilling og anvendelse

Country Status (17)

Country Link
EP (1) EP0682028A1 (no)
JP (1) JPH0853457A (no)
KR (1) KR950032205A (no)
CN (1) CN1117970A (no)
AU (1) AU1793395A (no)
CA (1) CA2148880A1 (no)
CZ (1) CZ119695A3 (no)
FI (1) FI952250L (no)
FR (1) FR2719844B1 (no)
HU (1) HUT72667A (no)
IL (1) IL113673A0 (no)
NO (1) NO951812L (no)
NZ (1) NZ272090A (no)
PL (1) PL308516A1 (no)
RU (1) RU95107154A (no)
SK (1) SK59795A3 (no)
ZA (1) ZA953749B (no)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19514579A1 (de) * 1995-04-20 1996-10-24 Boehringer Ingelheim Kg Verwendung von alpha¶1¶¶L¶-Agonisten zur Behandlung der Harninkontinenz
FR2733750B1 (fr) * 1995-05-03 1997-06-13 Synthelabo Derives de l'acide gamma-oxo-alpha-(phenylmethyl)-5,6- dihydro-4h-thieno(3,4-c)pyrrole-5-butanoique, leur preparation et leur application en therapeutique
CA2327543A1 (en) 1998-05-06 1999-11-11 Duke University Method of treating bladder and lower urinary tract syndromes

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8529546D0 (en) * 1985-11-30 1986-01-08 Beecham Group Plc Compounds
JPH06510760A (ja) * 1991-08-27 1994-12-01 ジ・アップジョン・カンパニー 代謝障害および代謝の治療法
EP0599697A1 (fr) * 1992-11-24 1994-06-01 Synthelabo Dérivés de pyrrole, leur préparation et leur application en thérapeutique

Also Published As

Publication number Publication date
HUT72667A (en) 1996-05-28
JPH0853457A (ja) 1996-02-27
FI952250L (fi) 1995-11-11
IL113673A0 (en) 1995-08-31
ZA953749B (en) 1996-04-02
EP0682028A1 (fr) 1995-11-15
AU1793395A (en) 1995-11-16
CA2148880A1 (fr) 1995-11-11
NZ272090A (en) 1996-03-26
RU95107154A (ru) 1997-03-20
FI952250A0 (fi) 1995-05-09
PL308516A1 (en) 1995-11-13
SK59795A3 (en) 1995-12-06
NO951812D0 (no) 1995-05-09
FR2719844B1 (fr) 1996-06-07
FR2719844A1 (fr) 1995-11-17
CN1117970A (zh) 1996-03-06
CZ119695A3 (en) 1995-11-15
KR950032205A (ko) 1995-12-20

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