NO934493L - Imidazo(2,1-b)(3)benzazepinderivater, sammensetninger og anvendel ses-metoder - Google Patents

Imidazo(2,1-b)(3)benzazepinderivater, sammensetninger og anvendel ses-metoder

Info

Publication number: NO934493L
Authority: NO; Norway
Prior art keywords: 4alkyl; substituted; hydroxycarbonyl; represents hydrogen; 4alkyloxy
Prior art date: 1991-06-13

Application number

NO934493A

Other languages

English (en)

Other versions

NO300689B1 (no

Inventor

Frans Eduard Janssens

Gaston Stanislas Marcell Diels

Joseph Elisabeth Leenaerts

Ludwig Paul Cooymans

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-06-13

Filing date

1993-12-09

Publication date

1994-01-04

1993-12-09 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

1994-01-04 Publication of NO934493L publication Critical patent/NO934493L/no

1997-07-07 Publication of NO300689B1 publication Critical patent/NO300689B1/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Pulmonology (AREA)
Animal Behavior & Ethology (AREA)
Immunology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Paper (AREA)
Detergent Compositions (AREA)
Fats And Perfumes (AREA)
Lubricants (AREA)
Solid-Sorbent Or Filter-Aiding Compositions (AREA)

NO934493A 1991-06-13 1993-12-09 Imidazo£2,1-b|£3|benzazepinderivater og sammensetninger NO300689B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US71448791A	1991-06-13	1991-06-13
PCT/EP1992/001331 WO1992022553A1 (en)	1991-06-13	1992-06-09	IMIDAZO[1,2-a](PYRROLO, THIENO OR FURANO)[3,2-d]AZEPINE DERIVATIVES, COMPOSITIONS AND METHODS OF USE

Publications (2)

Publication Number	Publication Date
NO934493L true NO934493L (no)	1994-01-04
NO300689B1 NO300689B1 (no)	1997-07-07

Family

ID=24870247

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
NO934493A NO300689B1 (no)	1991-06-13	1993-12-09	Imidazo£2,1-b\|£3\|benzazepinderivater og sammensetninger
NO934493D NO934493D0 (no)	1991-06-13	1993-12-09	Imidazo[2,1-b](pyrrolo, tieno eller furano)[3,2-d]-azepinderivater, sammensetninger og anvendelsesmetode

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
NO934493D NO934493D0 (no)	1991-06-13	1993-12-09	Imidazo[2,1-b](pyrrolo, tieno eller furano)[3,2-d]-azepinderivater, sammensetninger og anvendelsesmetode

Country Status (26)

Country	Link
US (1)	US5461050A (no)
EP (2)	EP0518434A1 (no)
JP (1)	JP3182421B2 (no)
KR (1)	KR100247504B1 (no)
CN (1)	CN1033587C (no)
AT (1)	ATE247118T1 (no)
AU (1)	AU652841B2 (no)
CA (1)	CA2102889C (no)
DE (1)	DE69233161T2 (no)
ES (1)	ES2204892T3 (no)
FI (1)	FI104077B (no)
HR (1)	HRP920156A2 (no)
HU (1)	HU221013B1 (no)
IE (1)	IE921919A1 (no)
IL (1)	IL101851A (no)
MA (1)	MA22554A1 (no)
MX (1)	MX9202860A (no)
NO (2)	NO300689B1 (no)
NZ (1)	NZ242775A (no)
PL (1)	PL170376B1 (no)
SI (1)	SI9200104A (no)
TN (1)	TNSN92049A1 (no)
TW (1)	TW218382B (no)
WO (1)	WO1992022553A1 (no)
ZA (1)	ZA924327B (no)
ZM (1)	ZM2892A1 (no)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL101850A (en) *	1991-06-13	1996-01-31	Janssen Pharmaceutica Nv	History 11-) 4-Pipridinyl (-Imidazo] B-1, 2 [] 3 [Benzazepine, their preparation and pharmaceutical preparations containing them
GR1001385B (el) *	1992-10-12	1993-10-29	Janssen Pharmaceutica Nv	Παράγωγα ιμιδαζο 1,2-α (πυρρολο,?ειενο η φουρανο) 3,2-d αζεπίνης συν?έσεις και μέ?οδοι χρήσεως.
KR100251296B1 (ko) *	1992-12-04	2000-05-01	디르크 반테	항앨러지성 트리아졸로(피롤로, 티에노 또는 푸라노)아제핀 유도체(Antiallergic triazolo(pyrrolo, thieno or furano)azepine derivatives)
PL176235B1 (pl) *	1992-12-04	1999-05-31	Janssen Pharmaceutica Nv	Nowe związki, pochodne imidazo[1,2-a] (tieno) [2,3-d] azepiny
KR100346802B1 (ko) *	1993-07-13	2002-11-29	얀센 파마슈티카 엔.브이.	항앨러지성이미다조아제핀
TW382017B (en)	1995-12-27	2000-02-11	Janssen Pharmaceutica Nv	1-(1,2-disubstituted piperidinyl)-4-(fused imidazole)-piperidine derivatives
TW527186B (en)	1996-03-19	2003-04-11	Janssen Pharmaceutica Nv	Fused imidazole derivatives as multidrug resistance modulators
JP3882224B2 (ja) *	1996-05-31	2007-02-14	旭硝子株式会社	パロキセチンの製造方法
US6544979B1 (en)	1997-09-18	2003-04-08	Janssen Pharmaceuticals, N.V.	Fused imidazole derivatives for improving oral bioavailability of pharmaceutical agents
NZ512870A (en)	1998-12-19	2003-11-28	Janssen Pharmaceutica Nv	Antihistaminic spiro compounds
TWI225488B (en) *	1999-12-21	2004-12-21	Janssen Pharmaceutica Nv	Derivatives of homopiperidinyl substituted benzimidazole analogues
WO2002100862A2 (en)	2001-06-12	2002-12-19	Janssen Pharmaceutica N.V.	Novel substituted tetracyclic imidazole derivatives, processes for their preparation, pharmaceutical compositions comprising them and their use as a medicine
AU2004259009A1 (en) *	2003-07-23	2005-02-03	Exelixis, Inc.	Azepine derivatives as pharmaceutical agents
AU2006221984C1 (en)	2005-03-08	2012-02-09	Janssen Pharmaceutica N.V.	Diaza-spiro-[4.4]-nonane derivatives as neurokinin (NK1) antagonists
TWI498115B (zh) *	2007-12-27	2015-09-01	Daiichi Sankyo Co Ltd	咪唑羰基化合物
CN103570731B (zh) *	2012-07-30	2016-05-18	中国科学院广州生物医药与健康研究院	嘧啶并三环或嘧啶并四环类化合物及其药用组合物和应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4148903A (en) *	1977-07-28	1979-04-10	Merck & Co., Inc.	Antipsychotic, antiserotonin and antihistaminic pyrrolo[2,1-b][3]benzazepines
GB8900380D0 (en) *	1989-01-09	1989-03-08	Janssen Pharmaceutica Nv	2-aminopyrimidinone derivatives
IL101850A (en) *	1991-06-13	1996-01-31	Janssen Pharmaceutica Nv	History 11-) 4-Pipridinyl (-Imidazo] B-1, 2 [] 3 [Benzazepine, their preparation and pharmaceutical preparations containing them

1992
- 1992-05-13 IL IL10185192A patent/IL101851A/en not_active IP Right Cessation
- 1992-05-15 NZ NZ242775A patent/NZ242775A/en unknown
- 1992-05-16 CN CN92104830A patent/CN1033587C/zh not_active Expired - Fee Related
- 1992-05-21 TW TW081103953A patent/TW218382B/zh active
- 1992-06-09 PL PL92301819A patent/PL170376B1/pl unknown
- 1992-06-09 WO PCT/EP1992/001331 patent/WO1992022553A1/en active IP Right Grant
- 1992-06-09 CA CA002102889A patent/CA2102889C/en not_active Expired - Fee Related
- 1992-06-09 AT AT92911643T patent/ATE247118T1/de not_active IP Right Cessation
- 1992-06-09 US US08/150,121 patent/US5461050A/en not_active Expired - Lifetime
- 1992-06-09 AU AU19011/92A patent/AU652841B2/en not_active Ceased
- 1992-06-09 EP EP92201665A patent/EP0518434A1/en active Pending
- 1992-06-09 KR KR1019930703789A patent/KR100247504B1/ko not_active IP Right Cessation
- 1992-06-09 EP EP92911643A patent/EP0588859B1/en not_active Expired - Lifetime
- 1992-06-09 ES ES92911643T patent/ES2204892T3/es not_active Expired - Lifetime
- 1992-06-09 HU HU9303554A patent/HU221013B1/hu not_active IP Right Cessation
- 1992-06-09 JP JP51073492A patent/JP3182421B2/ja not_active Expired - Fee Related
- 1992-06-09 DE DE69233161T patent/DE69233161T2/de not_active Expired - Fee Related
- 1992-06-10 HR HR920156A patent/HRP920156A2/hr not_active Application Discontinuation
- 1992-06-11 MA MA22844A patent/MA22554A1/fr unknown
- 1992-06-12 ZA ZA924327A patent/ZA924327B/xx unknown
- 1992-06-12 MX MX9202860A patent/MX9202860A/es not_active IP Right Cessation
- 1992-06-12 ZM ZM2892A patent/ZM2892A1/xx unknown
- 1992-06-12 SI SI19929200104A patent/SI9200104A/sl not_active IP Right Cessation
- 1992-06-15 TN TNTNSN92049A patent/TNSN92049A1/fr unknown
- 1992-07-01 IE IE191992A patent/IE921919A1/en not_active Application Discontinuation
1993
- 1993-12-09 NO NO934493A patent/NO300689B1/no not_active IP Right Cessation
- 1993-12-09 NO NO934493D patent/NO934493D0/no unknown
- 1993-12-10 FI FI935557A patent/FI104077B/fi active

Also Published As

Publication number	Publication date
IL101851A0 (en)	1992-12-30
EP0518434A1 (en)	1992-12-16
JP3182421B2 (ja)	2001-07-03
DE69233161T2 (de)	2004-05-27
NO934493D0 (no)	1993-12-09
CA2102889C (en)	2002-11-26
AU1901192A (en)	1993-01-12
FI104077B1 (fi)	1999-11-15
HU9303554D0 (en)	1994-04-28
CN1033587C (zh)	1996-12-18
ZA924327B (en)	1993-12-13
NO300689B1 (no)	1997-07-07
MA22554A1 (fr)	1992-12-31
MX9202860A (es)	1992-12-01
ZM2892A1 (en)	1994-05-25
ATE247118T1 (de)	2003-08-15
FI104077B (fi)	1999-11-15
CN1068116A (zh)	1993-01-20
EP0588859A1 (en)	1994-03-30
WO1992022553A1 (en)	1992-12-23
HU221013B1 (hu)	2002-07-29
KR100247504B1 (ko)	2000-05-01
IE921919A1 (en)	1992-12-16
DE69233161D1 (de)	2003-09-18
HRP920156A2 (en)	1995-12-31
TNSN92049A1 (fr)	1993-06-08
IL101851A (en)	1996-05-14
EP0588859B1 (en)	2003-08-13
CA2102889A1 (en)	1992-12-14
SI9200104A (en)	1992-12-31
HUT70428A (en)	1995-10-30
US5461050A (en)	1995-10-24
JPH06507890A (ja)	1994-09-08
AU652841B2 (en)	1994-09-08
TW218382B (no)	1994-01-01
FI935557A0 (fi)	1993-12-10
PL170376B1 (pl)	1996-12-31
ES2204892T3 (es)	2004-05-01
NZ242775A (en)	1995-03-28
FI935557A (fi)	1993-12-10

Publication	Publication Date	Title
NO934492D0 (no)	1993-12-09	Imidazo[2,1-b][3]benzazepinderivater, sammensetninger og anvendelses-metoder
NO934493L (no)	1994-01-04	Imidazo(2,1-b)(3)benzazepinderivater, sammensetninger og anvendel ses-metoder
PL300066A1 (en)	1994-02-21	Novel 7-(substituted)-8-(substituted)-9-(substituted amino)-6-demethyl-6-deoxy-tyetracyclines, methods of obtaining them and pharmaceutical composition
AU2174288A (en)	1989-03-09	Lactam derivatives
DE69332929D1 (de)	2003-06-05	ANTIALLERGISCHE IMIDAZO[1,2-a]THIENO[2,3-d]AZEPINDERIVATE

Legal Events

Date	Code	Title	Description
2005-04-25	MM1K	Lapsed by not paying the annual fees