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MX373867B - Amidas heterocíclicas como inhibidores de cinasas. - Google Patents

Amidas heterocíclicas como inhibidores de cinasas.

Info

Publication number
MX373867B
MX373867B MX2018008312A MX2018008312A MX373867B MX 373867 B MX373867 B MX 373867B MX 2018008312 A MX2018008312 A MX 2018008312A MX 2018008312 A MX2018008312 A MX 2018008312A MX 373867 B MX373867 B MX 373867B
Authority
MX
Mexico
Prior art keywords
kinase inhibitors
heterocyclic amides
amides
heterocyclic
kinase
Prior art date
Application number
MX2018008312A
Other languages
English (en)
Inventor
Deepak Bandyopadhyay
Sehon Clark A
Patrick M Eidam
Peter J Gough
Philip Anthony Harris
Jae U Jeong
Jianxing Kang
Bryan Wayne King
Shah Ami Lakdawala
Lara Kathryn Leister
Robert W Marquis Jr
Attiq Rahman
Joshi M Ramanjulu
Robert Singhaus Jr
Daohua Zhang
Original Assignee
Glaxosmithkline Ip Dev Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Ip Dev Ltd filed Critical Glaxosmithkline Ip Dev Ltd
Publication of MX373867B publication Critical patent/MX373867B/es

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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Abstract

Se desvelan compuestos que tienen la fórmula (I) en donde X, Y, Z1, Z2, Z3, Z4, R5, RA, m, A, L y B son como se definen en el presente documento, y procedimientos de preparación y uso de los mismos.
MX2018008312A 2013-02-15 2014-02-14 Amidas heterocíclicas como inhibidores de cinasas. MX373867B (es)

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