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MX344838B - Metodo para la produccion de polvos de nanoparticulas y microparticulas comerciales. - Google Patents

Metodo para la produccion de polvos de nanoparticulas y microparticulas comerciales.

Info

Publication number
MX344838B
MX344838B MX2011011216A MX2011011216A MX344838B MX 344838 B MX344838 B MX 344838B MX 2011011216 A MX2011011216 A MX 2011011216A MX 2011011216 A MX2011011216 A MX 2011011216A MX 344838 B MX344838 B MX 344838B
Authority
MX
Mexico
Prior art keywords
biologically active
production
powders
compositions
methods
Prior art date
Application number
MX2011011216A
Other languages
English (en)
Other versions
MX2011011216A (es
Inventor
Norret Marck
Dodd Aaron
Meiser Felix
Russell Adrian
H Bosch William
Original Assignee
Iceutica Pty Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from AU2009901747A external-priority patent/AU2009901747A0/en
Application filed by Iceutica Pty Ltd filed Critical Iceutica Pty Ltd
Publication of MX2011011216A publication Critical patent/MX2011011216A/es
Publication of MX344838B publication Critical patent/MX344838B/es

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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
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    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682—Processes
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    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/08—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing solids as carriers or diluents
    • A01N25/10—Macromolecular compounds
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    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
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    • A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
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    • A01N57/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds
    • A01N57/10—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds
    • A01N57/12—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds containing acyclic or cycloaliphatic radicals
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    • A01N57/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds
    • A01N57/18—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-carbon bonds
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Abstract

La presente invención se refiere a un método para disminuir la propensión de un material biológicamente activo a adherirse a un material seleccionado del grupo que consiste de acero inoxidable, vidrio, plástico, polietileno y polipropileno, caracterizado porque el método comprende: producir una composición que comprende el material biológicamente activo por molienda en seco del material biológicamente activo y una matriz de trituración molible en un molino que comprende una pluridad de cuerpos de molienda, por un periodo de entre 10 minutos y 2 horas, en donde la molienda en seco se lleva a cabo en ausencia de líquido, en donde el tamaño de las partículas del material biológicamente activo y el tamaño de las partículas de la matriz de trituración molible se reduce por molienda en seco, en donde el material biológicamente activo se selecciona del grupo que consiste de indometacina, meloxicam, diclofenaco ácido, naproxeno ácido, halusulfuron, metsulfuron, tribenuran, mancozeb, metaxalona, naproxeno sódico, ácido 2, 4-diclorofenoxiacético, glifosato, celecoxib, ciclosporina A, progesterona, salbutamol, ciprofloxacina, monohidrato de creatina, cilostazol, antraquinona, cacao en polvo, semillas de cacao, granos de café, jengibre, hojas de frambuesa, fenogreco, linaza, bayas de gojí, té verde, clavo, semilla de albaricoque, guisantes deshidratados, lavanda, mongostán, canela y cúrcuma, y en donde la matriz de trituración molible se selecciona del grupo que consiste de lactosa anhidra, lactosa mononidrato, lactosa monohidrato de calidad alimentaria, manito, dihitrato de citrato de trisodio, carbonato de calcio, xilito,, ácido málico, ácido tartárico, sorbitol, maltitol, sacarosa, suero en polvo y celulosa microcristalina.
MX2011011216A 2009-04-24 2010-04-23 Metodo para la produccion de polvos de nanoparticulas y microparticulas comerciales. MX344838B (es)

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AU2009901747A AU2009901747A0 (en) 2009-04-24 Method for the Production of Commercial Nanoparticle and Microparticle Powders
PCT/AU2010/000467 WO2010121323A1 (en) 2009-04-24 2010-04-23 Method for the production of commercial nanoparticle and microparticle powders

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