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MX2015007900A - Esteroides neuroactivos sustituidos con 19-alcoxi-17, profarmacos de los mismos, y metodos de tratamiento usando los mismos. - Google Patents

Esteroides neuroactivos sustituidos con 19-alcoxi-17, profarmacos de los mismos, y metodos de tratamiento usando los mismos.

Info

Publication number
MX2015007900A
MX2015007900A MX2015007900A MX2015007900A MX2015007900A MX 2015007900 A MX2015007900 A MX 2015007900A MX 2015007900 A MX2015007900 A MX 2015007900A MX 2015007900 A MX2015007900 A MX 2015007900A MX 2015007900 A MX2015007900 A MX 2015007900A
Authority
MX
Mexico
Prior art keywords
neuroactive
alkoxy
treatment
prodrugs
methods
Prior art date
Application number
MX2015007900A
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English (en)
Other versions
MX365644B (es
Inventor
Douglas Covey
Albert Jean Robichaud
Original Assignee
Univ Washington
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Washington filed Critical Univ Washington
Publication of MX2015007900A publication Critical patent/MX2015007900A/es
Publication of MX365644B publication Critical patent/MX365644B/es

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    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
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    • C07—ORGANIC CHEMISTRY
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Abstract

La descripción actual se dirige generalmente a esteroides neuroactivos sustituidos con 19-alcoxi-17 como se hace referencia en la presente, y sales farmacéuticamente aceptables de los mismos, para uso como, por ejemplo, un anestésico, y/o en el tratamiento de trastornos relacionados a la función y actividad GABA. La descripción actual se dirige además a composiciones farmacéuticas que comprenden tales compuestos.
MX2015007900A 2012-12-18 2013-12-18 Esteroides neuroactivos sustituidos con 19-alcoxi-17, profarmacos de los mismos, y metodos de tratamiento usando los mismos. MX365644B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261738822P 2012-12-18 2012-12-18
PCT/US2013/076214 WO2014100228A1 (en) 2012-12-18 2013-12-18 Neuroactive 19-alkoxy-17-substituted steroids, prodrugs thereof, and methods of treatment using same

Publications (2)

Publication Number Publication Date
MX2015007900A true MX2015007900A (es) 2016-02-05
MX365644B MX365644B (es) 2019-06-10

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MX2019006739A MX388946B (es) 2012-12-18 2013-12-18 Esteroides neuroactivos sustituidos con 19-alcoxi-17, profarmacos de los mismos, y metodos de tratamiento usando los mismos.
MX2015007900A MX365644B (es) 2012-12-18 2013-12-18 Esteroides neuroactivos sustituidos con 19-alcoxi-17, profarmacos de los mismos, y metodos de tratamiento usando los mismos.

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Publication number Priority date Publication date Assignee Title
EA017290B1 (ru) 2005-11-28 2012-11-30 Домейн Раша Инвестментс Лимитед Композиции на основе ганаксолона
SMT202300232T1 (it) 2011-09-08 2023-09-06 Sage Therapeutics Inc Steroidi neuroattivi, composizioni e relativi usi
AU2012323888A1 (en) 2011-10-14 2014-05-29 Sage Therapeutics, Inc. 3,3 disubstituted 19-nor pregnane compounds, compositions, and uses thereof
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