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HK1119174A1 - N4-phenyl-quinazoline-4 -amine derivatives and related compounds as erbb type i receptor tyrosine kinase inhibitors for the treatment of hyperproliferative diseases - Google Patents

N4-phenyl-quinazoline-4 -amine derivatives and related compounds as erbb type i receptor tyrosine kinase inhibitors for the treatment of hyperproliferative diseases Download PDF

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Publication number
HK1119174A1
HK1119174A1 HK08113123.5A HK08113123A HK1119174A1 HK 1119174 A1 HK1119174 A1 HK 1119174A1 HK 08113123 A HK08113123 A HK 08113123A HK 1119174 A1 HK1119174 A1 HK 1119174A1
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HK
Hong Kong
Prior art keywords
alkyl
saturated
partially unsaturated
heteroaryl
aryl
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HK08113123.5A
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German (de)
English (en)
French (fr)
Chinese (zh)
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HK1119174B (en
Inventor
Joseph P. Lyssikatos
Fredrik P. Marmsater
Qian Zhao
Julie Marie Greschuk
Original Assignee
Array Biopharma Inc.
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38022019&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1119174(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Array Biopharma Inc. filed Critical Array Biopharma Inc.
Priority to HK09109538.1A priority Critical patent/HK1129678B/en
Publication of HK1119174A1 publication Critical patent/HK1119174A1/en
Publication of HK1119174B publication Critical patent/HK1119174B/en

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  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Hospice & Palliative Care (AREA)
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  • Hematology (AREA)
  • Mycology (AREA)
  • Microbiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychiatry (AREA)
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  • Pain & Pain Management (AREA)
HK08113123.5A 2005-11-15 2006-11-15 N4-phenyl-quinazoline-4 -amine derivatives and related compounds as erbb type i receptor tyrosine kinase inhibitors for the treatment of hyperproliferative diseases HK1119174B (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
HK09109538.1A HK1129678B (en) 2005-11-15 2008-12-02 Processes and intermediates for the preparation of n4-phenyl-quinazoline-4-amine derivatives

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US73628905P 2005-11-15 2005-11-15
US60/736,289 2005-11-15
US81701906P 2006-06-28 2006-06-28
US60/817,019 2006-06-28
PCT/US2006/044431 WO2007059257A2 (en) 2005-11-15 2006-11-15 N4-phenyl-quinaz0line-4 -amine derivatives and related compounds as erbb type i receptor tyrosine kinase inhibitors for the treatment of hyperproliferative diseases

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
HK09109538.1A Division HK1129678B (en) 2005-11-15 2008-12-02 Processes and intermediates for the preparation of n4-phenyl-quinazoline-4-amine derivatives

Related Child Applications (1)

Application Number Title Priority Date Filing Date
HK09109538.1A Addition HK1129678B (en) 2005-11-15 2008-12-02 Processes and intermediates for the preparation of n4-phenyl-quinazoline-4-amine derivatives

Publications (2)

Publication Number Publication Date
HK1119174A1 true HK1119174A1 (en) 2009-02-27
HK1119174B HK1119174B (en) 2010-01-15

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AU2006315383B2 (en) 2011-06-02
DE602006009968D1 (de) 2009-12-03
BR122018075851B1 (pt) 2022-01-11
CA2755268A1 (en) 2007-05-24
IL248993B (en) 2018-11-29
ATE507224T1 (de) 2011-05-15
FR21C1031I2 (fr) 2022-07-15
NO20082598L (no) 2008-08-06
RU2011122539A (ru) 2012-12-10
SG152230A1 (en) 2009-05-29
KR101086967B1 (ko) 2011-11-29
US20170252317A1 (en) 2017-09-07
CA2632194C (en) 2012-01-03
IL239149A (en) 2016-11-30
LUC00217I2 (ja) 2022-10-07
ZA200804498B (en) 2009-07-29
CA2755268C (en) 2013-12-31
CN101356171A (zh) 2009-01-28
WO2007059257A2 (en) 2007-05-24
EP2090575B1 (en) 2011-04-27
RU2008118417A (ru) 2009-12-27
AU2006315383A1 (en) 2007-05-24
AU2010202330B2 (en) 2012-07-19
JP5134548B2 (ja) 2013-01-30
RU2592703C2 (ru) 2016-07-27
EP1971601A2 (en) 2008-09-24
US20210008023A1 (en) 2021-01-14
CY2021019I2 (el) 2021-12-31
EP2090575A1 (en) 2009-08-19
CA2632194A1 (en) 2007-05-24
PL1971601T3 (pl) 2010-03-31
JP2010270154A (ja) 2010-12-02
ES2364901T3 (es) 2011-09-16
US20110034689A1 (en) 2011-02-10
LTPA2021516I1 (ja) 2021-08-10
PT1971601E (pt) 2010-01-26
BRPI0618668B1 (pt) 2021-09-21
CY2021019I1 (el) 2021-10-15
DK1971601T3 (da) 2010-02-08
CN102887891B (zh) 2016-03-09
AU2010202330A1 (en) 2010-07-01
NL301113I2 (nl) 2021-08-03
SI1971601T1 (sl) 2010-03-31
RU2592703C9 (ru) 2016-10-20
US8648087B2 (en) 2014-02-11
NL301113I1 (nl) 2021-07-01
HK1129678A1 (en) 2009-12-04
DK2090575T3 (da) 2011-05-23
RU2428421C2 (ru) 2011-09-10
US9693989B2 (en) 2017-07-04
ATE446294T1 (de) 2009-11-15
CY1110583T1 (el) 2015-04-29
FR21C1031I1 (ja) 2021-08-27
NO342413B1 (no) 2018-05-22
ES2335535T3 (es) 2010-03-29
JP2009515988A (ja) 2009-04-16
IL248993A0 (en) 2017-01-31
CN102887891A (zh) 2013-01-23
US20180271824A1 (en) 2018-09-27
FIC20210022I1 (fi) 2021-07-09
CY1112754T1 (el) 2016-02-10
EP1971601B1 (en) 2009-10-21
US20140023643A1 (en) 2014-01-23
HUS2100028I1 (hu) 2021-08-30
PL2090575T3 (pl) 2011-09-30
WO2007059257A8 (en) 2007-07-12
US10780073B2 (en) 2020-09-22
DE602006021645D1 (de) 2011-06-09
WO2007059257A3 (en) 2007-08-23
LTC1971601I2 (ja) 2022-10-25
US12171739B2 (en) 2024-12-24
PT2090575E (pt) 2011-06-06
US20230142839A1 (en) 2023-05-11
KR20080070064A (ko) 2008-07-29
JP5232841B2 (ja) 2013-07-10
BRPI0618668A2 (pt) 2011-09-06
IL239149A0 (en) 2015-07-30
SI2090575T1 (sl) 2011-08-31

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