FI962445L - Paroksetiinitabletteja ja menetelmä niiden valmistamiseksi - Google Patents

Paroksetiinitabletteja ja menetelmä niiden valmistamiseksi Download PDF

Info

Publication number: FI962445L
Authority: FI; Finland
Prior art keywords: preparation; paroxetine tablets; paroxetine; tablets
Prior art date: 1993-12-15

Application number

FI962445A

Other languages

English (en)

Swedish (sv)

Other versions

FI962445A0 (fi

Inventor

Ram Dutta Pathak

David George Doughty

Original Assignee

Smithkline Beecham Plc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1993-12-15

Filing date

1996-06-12

Publication date

1996-06-12

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10746644&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI962445(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1996-06-12 Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc

1996-06-12 Publication of FI962445L publication Critical patent/FI962445L/fi

1996-06-12 Publication of FI962445A0 publication Critical patent/FI962445A0/fi

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4525—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with oxygen as a ring hetero atom
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Pain & Pain Management (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Psychiatry (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Plural Heterocyclic Compounds (AREA)

FI962445A 1993-12-15 1996-06-12 Paroksetiinitabletteja ja menetelmä niiden valmistamiseksi FI962445A0 (fi)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB939325644A GB9325644D0 (en)	1993-12-15	1993-12-15	Novel formulation
PCT/EP1994/004164 WO1995016448A1 (en)	1993-12-15	1994-12-14	Paroxetine tablets and process to prepare them

Publications (2)

Publication Number	Publication Date
FI962445L true FI962445L (fi)	1996-06-12
FI962445A0 FI962445A0 (fi)	1996-06-12

Family

ID=10746644

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI962445A FI962445A0 (fi)	1993-12-15	1996-06-12	Paroksetiinitabletteja ja menetelmä niiden valmistamiseksi

Country Status (36)

Country	Link
US (1)	US6113944A (fi)
EP (1)	EP0734260B2 (fi)
JP (1)	JP3037757B2 (fi)
KR (1)	KR100367796B1 (fi)
CN (1)	CN1071116C (fi)
AP (1)	AP540A (fi)
AT (1)	ATE180973T1 (fi)
AU (1)	AU697982B2 (fi)
BG (1)	BG62755B1 (fi)
BR (1)	BR9408219A (fi)
CA (4)	CA2274387A1 (fi)
CZ (1)	CZ287891B6 (fi)
DE (1)	DE69419033T2 (fi)
DK (1)	DK0734260T4 (fi)
DZ (1)	DZ1835A1 (fi)
ES (1)	ES2132610T5 (fi)
FI (1)	FI962445A0 (fi)
GB (1)	GB9325644D0 (fi)
GR (1)	GR3031047T3 (fi)
HK (1)	HK1012285A1 (fi)
HU (1)	HUT75880A (fi)
IL (1)	IL111978A (fi)
MA (1)	MA23395A1 (fi)
MY (1)	MY112123A (fi)
NO (1)	NO307366B1 (fi)
NZ (1)	NZ277790A (fi)
OA (1)	OA10297A (fi)
PL (1)	PL314980A1 (fi)
RO (1)	RO115413B1 (fi)
RU (1)	RU2146141C1 (fi)
SA (1)	SA94150373B1 (fi)
SI (1)	SI0734260T2 (fi)
SK (1)	SK282620B6 (fi)
UA (1)	UA42745C2 (fi)
WO (1)	WO1995016448A1 (fi)
ZA (1)	ZA949900B (fi)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US20020086053A1 (en) *	1993-12-15	2002-07-04	Smithkline Beecham Plc	Formulations, tablets of paroxetine and process to prepare them
SK283608B6 (sk) *	1995-02-06	2003-10-07	Smithkline Beecham Plc	Bezvodý hydrochlorid paroxetínu, spôsob jeho výroby a použitie
US6548084B2 (en)	1995-07-20	2003-04-15	Smithkline Beecham Plc	Controlled release compositions
GB9605828D0 (en) *	1996-03-20	1996-05-22	Smithkline Beecham Plc	Treatment method
US6638948B1 (en)	1996-09-09	2003-10-28	Pentech Pharmaceuticals, Inc.	Amorphous paroxetine composition
EP1078925A1 (en)	1997-06-10	2001-02-28	Synthon B.V.	4-Phenylpiperidine compounds
US5955475A (en) *	1997-06-30	1999-09-21	Endo Pharmaceuticals Inc.	Process for manufacturing paroxetine solid dispersions
US6699882B2 (en)	1998-03-24	2004-03-02	Smithkline Beecham P.L.C.	Paroxetine compositions
US6168805B1 (en)	1998-05-07	2001-01-02	Endo Pharmaceuticals, Inc.	Aqueous process for manufacturing paroxetine solid dispersions
GB9810181D0 (en) *	1998-05-13	1998-07-08	Smithkline Beecham Plc	Novel formulations
DE19821625C1 (de) *	1998-05-15	2000-01-05	Merck Patent Gmbh	Pharmazeutische Zubereitung
CH689805A8 (fr) *	1998-07-02	2000-02-29	Smithkline Beecham Plc	Méthanesulfonate de paroxétine, procédé pour sa préparation et compositions pharmaceutiques le contenant.
WO2000078290A2 (en) *	1999-06-22	2000-12-28	Smithkline Beecham P.L.C.	Pharmaceutical composition comprising a salt of paroxetine
GB0003232D0 (en) *	2000-02-11	2000-04-05	Smithkline Beecham Plc	Novel composition
EP1313474A2 (en) *	2000-08-28	2003-05-28	Synthon B.V.	Paroxetine compositions and processes for making the same
DE20100529U1 (de) *	2001-01-11	2001-05-10	Synthon Bv	Pharmazeutische Tablette umfassend Paroxetinmesylat
HUP0401946A2 (hu)	2001-07-31	2005-01-28	H. Lundbeck A/S	Escitalopramot tartalmazó kristályos gyógyszerkészítmény
NZ532432A (en) *	2001-10-22	2005-02-25	Synthon Bv	N-formyl paroxetine compounds and their use in a synthetic route for obtaining paroxetine
AU2002359857B8 (en) *	2001-12-28	2009-01-08	Teva Pharmaceutical Industries Ltd.	A stable pharmaceutical formulation of paroxetine hydrochloride anhydrous and a process for preparation thereof
US20040220153A1 (en) *	2002-09-24	2004-11-04	Jost-Price Edward Roydon	Methods and reagents for the treatment of diseases and disorders associated with increased levels of proinflammatory cytokines
US20050266082A1 (en) *	2004-05-26	2005-12-01	Patel Satishkumar A	Preparation of stable paroxetine HC1 ER tablets using a melt granulation process
US20080032959A1 (en) *	2004-06-23	2008-02-07	Alves Stephen E	Estrogen Receptor Modulators
US20060063737A1 (en) *	2004-08-18	2006-03-23	Holmdahl Lisa K	Liquid paroxetine compositions
EP1791531A1 (en) *	2004-08-20	2007-06-06	Alpharma, Inc.	Paroxetine formulations
US20060216345A1 (en) *	2005-03-24	2006-09-28	Sun Pharmaceutical Industries Limited	Oral pharmaceutical composition including paroxetine
CA2629514A1 (en) *	2005-11-14	2007-05-24	Auspex Pharmaceuticals, Inc.	Substituted phenylpiperidines with serotoninergic activity and enhanced therapeutic properties
US20080033050A1 (en)	2006-08-04	2008-02-07	Richards Patricia Allison Tewe	Method of treating thermoregulatory disfunction with paroxetine
US9138430B2 (en) *	2007-12-27	2015-09-22	Mylan Specialty L.P.	Formulation and method for the release of paroxetine in the large intestine
CA2937365C (en)	2016-03-29	2018-09-18	F. Hoffmann-La Roche Ag	Granulate formulation of 5-methyl-1-phenyl-2-(1h)-pyridone and method of making the same
CN109771381B (zh) *	2017-11-13	2021-02-19	北京福元医药股份有限公司	一种帕罗西汀药物制剂

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS50116401A (fi) *	1974-03-04	1975-09-11
ZA813205B (en) *	1980-12-05	1983-03-30	Smith Kline French Lab	Dosage units
GB8430581D0 (en) *	1984-12-04	1985-01-09	Ferrosan As	Treatment
DE3680184D1 (de) *	1985-08-10	1991-08-14	Beecham Group Plc	Verfahren zur herstellung von arylpiperidincarbinol.
GB8520154D0 (en) *	1985-08-10	1985-09-18	Beecham Group Plc	Chemical process
DE3688827T2 (de) *	1985-10-25	1994-03-31	Beecham Group Plc	Piperidinderivat, seine Herstellung und seine Verwendung als Arzneimittel.
GB8626936D0 (en) *	1986-11-11	1986-12-10	Ferrosan As	Treatment
GB8714707D0 (en) *	1987-06-23	1987-07-29	Beecham Group Plc	Chemical process
JPH06502854A (ja) *	1990-11-24	1994-03-31	ビーチャム・グループ・パブリック・リミテッド・カンパニー	老年痴呆、過食症、片頭痛または食欲不振の治療用のパロキセチンの使用
GB9209687D0 (en) *	1992-05-06	1992-06-17	Smithkline Beecham Plc	Novel process
US5776969A (en) *	1997-02-27	1998-07-07	Eli Lilly And Company	Treatment of sleep disorders

1993
- 1993-12-15 GB GB939325644A patent/GB9325644D0/en active Pending
1994
- 1994-12-13 ZA ZA949900A patent/ZA949900B/xx unknown
- 1994-12-13 MA MA23723A patent/MA23395A1/fr unknown
- 1994-12-13 SA SA94150373A patent/SA94150373B1/ar unknown
- 1994-12-13 AP APAP/P/1994/000704A patent/AP540A/en active
- 1994-12-13 MY MYPI94003326A patent/MY112123A/en unknown
- 1994-12-13 DZ DZ940132A patent/DZ1835A1/fr active
- 1994-12-14 NZ NZ277790A patent/NZ277790A/en not_active IP Right Cessation
- 1994-12-14 RO RO96-01196A patent/RO115413B1/ro unknown
- 1994-12-14 IL IL11197894A patent/IL111978A/xx unknown
- 1994-12-14 CN CN94194457A patent/CN1071116C/zh not_active Expired - Fee Related
- 1994-12-14 CA CA002274387A patent/CA2274387A1/en not_active Abandoned
- 1994-12-14 DK DK95904476T patent/DK0734260T4/da active
- 1994-12-14 KR KR1019960703153A patent/KR100367796B1/ko not_active Expired - Fee Related
- 1994-12-14 HU HU9601665A patent/HUT75880A/hu not_active Application Discontinuation
- 1994-12-14 UA UA96062355A patent/UA42745C2/uk unknown
- 1994-12-14 CA CA002274389A patent/CA2274389C/en not_active Expired - Fee Related
- 1994-12-14 JP JP07516534A patent/JP3037757B2/ja not_active Expired - Fee Related
- 1994-12-14 SI SI9430251T patent/SI0734260T2/sl not_active IP Right Cessation
- 1994-12-14 EP EP95904476A patent/EP0734260B2/en not_active Expired - Lifetime
- 1994-12-14 DE DE69419033T patent/DE69419033T2/de not_active Expired - Lifetime
- 1994-12-14 WO PCT/EP1994/004164 patent/WO1995016448A1/en active IP Right Grant
- 1994-12-14 SK SK756-96A patent/SK282620B6/sk not_active IP Right Cessation
- 1994-12-14 CZ CZ19961763A patent/CZ287891B6/cs not_active IP Right Cessation
- 1994-12-14 BR BR9408219A patent/BR9408219A/pt not_active Application Discontinuation
- 1994-12-14 ES ES95904476T patent/ES2132610T5/es not_active Expired - Lifetime
- 1994-12-14 CA CA002214575A patent/CA2214575C/en not_active Expired - Fee Related
- 1994-12-14 PL PL94314980A patent/PL314980A1/xx unknown
- 1994-12-14 CA CA002178637A patent/CA2178637C/en not_active Expired - Fee Related
- 1994-12-14 AU AU13145/95A patent/AU697982B2/en not_active Ceased
- 1994-12-14 AT AT95904476T patent/ATE180973T1/de not_active IP Right Cessation
- 1994-12-14 RU RU96114954A patent/RU2146141C1/ru not_active IP Right Cessation
1996
- 1996-06-06 BG BG100648A patent/BG62755B1/bg unknown
- 1996-06-12 FI FI962445A patent/FI962445A0/fi not_active Application Discontinuation
- 1996-06-14 OA OA60845A patent/OA10297A/en unknown
- 1996-06-14 NO NO962547A patent/NO307366B1/no not_active IP Right Cessation
1998
- 1998-06-30 US US09/108,138 patent/US6113944A/en not_active Expired - Fee Related
- 1998-12-16 HK HK98113624A patent/HK1012285A1/xx not_active IP Right Cessation
1999
- 1999-08-19 GR GR990402125T patent/GR3031047T3/el unknown

Also Published As

Publication number	Publication date
AU697982B2 (en)	1998-10-22
SA94150373B1 (ar)	2006-05-27
PL314980A1 (en)	1996-09-30
CA2178637A1 (en)	1995-06-22
CA2274389A1 (en)	1995-06-22
EP0734260B2 (en)	2008-07-09
ES2132610T3 (es)	1999-08-16
SK282620B6 (sk)	2002-10-08
HUT75880A (en)	1997-05-28
EP0734260A1 (en)	1996-10-02
SI0734260T1 (en)	1999-08-31
CN1137236A (zh)	1996-12-04
AU1314595A (en)	1995-07-03
EP0734260B1 (en)	1999-06-09
CZ287891B6 (cs)	2001-03-14
WO1995016448A1 (en)	1995-06-22
NZ277790A (en)	1998-02-26
SA94150373A (ar)	2005-12-03
CA2274387A1 (en)	1995-06-22
CN1071116C (zh)	2001-09-19
JPH09506602A (ja)	1997-06-30
CA2178637C (en)	1997-12-23
IL111978A0 (en)	1995-03-15
ES2132610T5 (es)	2008-12-16
NO962547L (no)	1996-06-14
JP3037757B2 (ja)	2000-05-08
GB9325644D0 (en)	1994-02-16
AP9400704A0 (en)	1995-01-31
NO307366B1 (no)	2000-03-27
BG62755B1 (bg)	2000-07-31
DK0734260T3 (da)	1999-11-15
MA23395A1 (fr)	1995-07-01
BG100648A (bg)	1997-02-28
KR100367796B1 (ko)	2003-07-22
FI962445A0 (fi)	1996-06-12
HU9601665D0 (en)	1996-08-28
GR3031047T3 (en)	1999-12-31
US6113944A (en)	2000-09-05
UA42745C2 (uk)	2001-11-15
SI0734260T2 (sl)	2008-12-31
DK0734260T4 (da)	2008-09-29
BR9408219A (pt)	1997-08-26
DE69419033D1 (de)	1999-07-15
NO962547D0 (no)	1996-06-14
CA2214575A1 (en)	1995-06-22
HK1012285A1 (en)	1999-07-30
ATE180973T1 (de)	1999-06-15
CZ176396A3 (en)	1996-09-11
ZA949900B (en)	1995-10-10
CA2274389C (en)	2004-09-14
CA2214575C (en)	1999-12-07
IL111978A (en)	2000-07-16
RO115413B1 (ro)	2000-02-28
RU2146141C1 (ru)	2000-03-10
DZ1835A1 (fr)	2002-02-17
DE69419033T2 (de)	1999-11-25
AP540A (en)	1996-09-20
OA10297A (en)	1997-10-07
SK75696A3 (en)	1996-11-06
MY112123A (en)	2001-04-30

Publication	Publication Date	Title
FI962445L (fi)	1996-06-12	Paroksetiinitabletteja ja menetelmä niiden valmistamiseksi
FI956270L (fi)	1995-12-27	Piperdiinijohdannaisia ja menetelmä niiden valmistamiseksi
FI940585L (fi)	1994-08-11	Pinnoittamattomat tabletit ja menetelmä niiden valmistamiseksi
FI951305L (fi)	1995-03-20	Lääketieteellinen materiaali ja menetelmä sen valmistamiseksi
FI941137L (fi)	1994-09-12	2-debentsoyyli-2-asyylitaksolijohdannaisia ja menetelmiä niiden valmistamiseksi
FI945476L (fi)	1995-05-24	Hitaasti vapautuvat koostumukset ja menetelmä farmaseuttisten koostumusten valmistamiseksi
FI964028L (fi)	1996-10-08	Uusi farmaseuttinen formulaatio ja menetelmä
FI944961L (fi)	1994-10-21	Farmaseuttinen valmiste ja menetelmä sen valmistamiseksi
FI942745L (fi)	1994-12-12	Fluoreeniyhdisteitä ja valmistusmenetelmä
FI954246L (fi)	1995-09-11	Uusia A83543-yhdisteitä ja menetelmä niiden valmistamiseksi
FI944452L (fi)	1995-03-29	Gelatiinikapseli ja menetelmä sen valmistamiseksi
FI960948L (fi)	1996-02-29	Pakkaus ja menetelmä mainitun pakkauksen tuottamiseksi
EE9500064A (et)	1996-06-17	Asendatud 1H-imidasoolid, nende valmistamismeetodid ja farmatseutilised kompositsioonid
FI956080L (fi)	1996-01-17	Kuidutettu selluloosatuote ja menetelmä sen valmistamiseksi
FI943532L (fi)	1994-07-27	Revinnäismassa ja menetelmä revinnäismassan valmistamiseksi
FI962486L (fi)	1996-08-12	Pakkaus ja menetelmä sekä laite sen valmistamiseksi
FI942932L (fi)	1994-06-17	Farmaseuttinen koostumus ja menetelmä sen valmistamiseksi
FI952324A0 (fi)	1995-05-12	Heterosykliset karbamaatit, menetelmä niiden valmistamiseksi ja lääkkeet
FI954499L (fi)	1995-09-22	Menetelmä ja analyysi
FI944713L (fi)	1994-12-02	4-difenyylimetyylipiperidiinijohdannaisia ja menetelmä niiden valmistamiseksi
FI931232L (fi)	1994-09-20	Makeutusaine, menetelmä sen valmistamiseksi ja sen käyttö
EE9800164A (et)	1998-12-15	Farmatseutiline kompositsioon ja meetod epitelioomi raviks
FI941914A0 (fi)	1994-04-25	2-amino-4-kinoliinidihydropyridiinejä, menetelmiä niiden valmistamiseksi ja niiden käyttö
FI942298L (fi)	1995-11-18	Menetelmä ja sovitelma tilaelementtien siirtämiseksi
FI955123A0 (fi)	1995-10-27	Kolestyramiinia sisältävä koostumus ja menetelmä tämän valmistamiseksi

Legal Events

Date	Code	Title	Description
2010-06-07	FD	Application lapsed