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FI954946L - Kinoksaliinit, menetelmä niiden valmistamiseksi ja niiden käyttö - Google Patents

Kinoksaliinit, menetelmä niiden valmistamiseksi ja niiden käyttö Download PDF

Info

Publication number
FI954946L
FI954946L FI954946A FI954946A FI954946L FI 954946 L FI954946 L FI 954946L FI 954946 A FI954946 A FI 954946A FI 954946 A FI954946 A FI 954946A FI 954946 L FI954946 L FI 954946L
Authority
FI
Finland
Prior art keywords
quinoxalines
preparation
Prior art date
Application number
FI954946A
Other languages
English (en)
Swedish (sv)
Other versions
FI954946A0 (fi
Inventor
Manfred Dr Roesner
Uta-Maria Billhardt-Troughton
Reinhard Dr Kirsch
Joerg-Peter Dr Kleim
Christoph Dr Meichsner
Guenther Dr Ries
Irvin Dr Winkler
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of FI954946A0 publication Critical patent/FI954946A0/fi
Publication of FI954946L publication Critical patent/FI954946L/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/36Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
    • C07D241/38Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
    • C07D241/40Benzopyrazines
    • C07D241/44Benzopyrazines with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Dental Preparations (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Compounds Of Unknown Constitution (AREA)
FI954946A 1994-10-19 1995-10-17 Kinoksaliinit, menetelmä niiden valmistamiseksi ja niiden käyttö FI954946L (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4437406A DE4437406A1 (de) 1994-10-19 1994-10-19 Chinoxaline, Verfahren zu ihrer Herstellung und ihre Verwendung

Publications (2)

Publication Number Publication Date
FI954946A0 FI954946A0 (fi) 1995-10-17
FI954946L true FI954946L (fi) 1996-04-20

Family

ID=6531202

Family Applications (1)

Application Number Title Priority Date Filing Date
FI954946A FI954946L (fi) 1994-10-19 1995-10-17 Kinoksaliinit, menetelmä niiden valmistamiseksi ja niiden käyttö

Country Status (28)

Country Link
US (1) US5723461A (fi)
EP (1) EP0708093B1 (fi)
JP (1) JPH08225544A (fi)
KR (1) KR960014108A (fi)
CN (1) CN1094930C (fi)
AT (1) ATE198747T1 (fi)
AU (1) AU708293B2 (fi)
BR (1) BR9504456A (fi)
CA (1) CA2160859A1 (fi)
CZ (1) CZ271295A3 (fi)
DE (2) DE4437406A1 (fi)
DK (1) DK0708093T3 (fi)
ES (1) ES2154311T3 (fi)
FI (1) FI954946L (fi)
GR (1) GR3035673T3 (fi)
HK (1) HK1011988A1 (fi)
HR (1) HRP950524B1 (fi)
HU (1) HUT73485A (fi)
IL (1) IL115641A0 (fi)
MY (1) MY132057A (fi)
NO (1) NO306615B1 (fi)
NZ (1) NZ280258A (fi)
PL (1) PL184860B1 (fi)
PT (1) PT708093E (fi)
SI (1) SI9500329A (fi)
SK (1) SK128495A3 (fi)
TW (1) TW328954B (fi)
ZA (1) ZA958783B (fi)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6369057B1 (en) * 1991-04-15 2002-04-09 Aventis Pharma Deutschland Gmbh Quinoxalines, processes for their preparation and their use
US6015800A (en) * 1997-09-03 2000-01-18 Warner-Lambert Company Substituted quinoxaline-2-ones as glutamate receptor antagonists
WO1999025327A2 (en) * 1997-11-14 1999-05-27 Warner-Lambert Company Small molecule intervention in hiv-1 replication
GB9901795D0 (en) * 1999-01-28 1999-03-17 Glaxo Group Ltd Chemical compounds
GB9911887D0 (en) * 1999-05-21 1999-07-21 Glaxo Group Ltd Methods and medicaments for post exposure prophylaxis of an hiv infection
WO2002087500A2 (en) * 2001-04-27 2002-11-07 Newbiotics, Inc. Viral enzyme activated prototoxophores and use of same to treat viral infections
WO2005018531A2 (fr) * 2003-08-26 2005-03-03 'chemical Diversity Research Institute', Ltd. Compositions pharmaceutiques, composes azo-heterocycliques et procedes de fabrication et d'utilisation correspondants
US7351709B2 (en) * 2004-06-09 2008-04-01 Wyeth Estrogen receptor ligands
BR112014026703B1 (pt) 2012-04-24 2022-10-25 Vertex Pharmaceuticals Incorporated Inibidores de dna-pk e seus usos, composição farmacêutica e seus usos, e método de sensibilização de uma célula
HRP20211855T1 (hr) 2013-03-12 2022-03-04 Vertex Pharmaceuticals Incorporated Inhibitori dnk-pk
LT3424920T (lt) 2013-10-17 2020-08-10 Vertex Pharmaceuticals Incorporated (s)-n-metil-8-(1-((2`-metil-[4,5`-bipirimidin]-6-il)amino)propan-2-il)chinolin-4-karboksamido ir jo deuterintų darinių, kaip dnr-pk inhibitorių, bendri kristalai
KR20190062485A (ko) 2016-09-27 2019-06-05 버텍스 파마슈티칼스 인코포레이티드 Dna-손상제 및 dna-pk 저해제의 조합을 사용한 암 치료 방법

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0509398B1 (de) * 1991-04-15 2001-09-19 Aventis Pharma Deutschland GmbH Chinoxaline, Verfahren zu ihrer Herstellung und ihre Verwendung
DE4342024A1 (de) * 1993-12-09 1995-06-14 Hoechst Ag Kombinationspräparate, enthaltend ein Chinoxalin und ein Nukleosid

Also Published As

Publication number Publication date
IL115641A0 (en) 1996-01-19
AU708293B2 (en) 1999-07-29
ZA958783B (en) 1996-05-09
MY132057A (en) 2007-09-28
TW328954B (en) 1998-04-01
HRP950524B1 (en) 2002-06-30
SI9500329A (en) 1996-04-30
CZ271295A3 (en) 1996-08-14
HK1011988A1 (en) 1999-07-23
JPH08225544A (ja) 1996-09-03
PT708093E (pt) 2001-06-29
GR3035673T3 (en) 2001-06-29
NZ280258A (en) 1997-09-22
NO954139D0 (no) 1995-10-18
PL311016A1 (en) 1996-04-29
CN1094930C (zh) 2002-11-27
HRP950524A2 (en) 1997-10-31
BR9504456A (pt) 1997-05-20
CA2160859A1 (en) 1996-04-20
SK128495A3 (en) 1996-06-05
NO306615B1 (no) 1999-11-29
PL184860B1 (pl) 2003-01-31
EP0708093B1 (de) 2001-01-17
CN1135483A (zh) 1996-11-13
NO954139L (no) 1996-04-22
EP0708093A1 (de) 1996-04-24
ES2154311T3 (es) 2001-04-01
DE59508969D1 (de) 2001-02-22
FI954946A0 (fi) 1995-10-17
HU9503005D0 (en) 1995-12-28
HUT73485A (en) 1996-08-28
DK0708093T3 (da) 2001-04-30
ATE198747T1 (de) 2001-02-15
AU3431695A (en) 1996-05-02
KR960014108A (ko) 1996-05-22
US5723461A (en) 1998-03-03
DE4437406A1 (de) 1996-04-25

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