ES440153A2 - Un procedimiento para la preparacion de nuevas piperazino- pirimidinas. - Google Patents
Un procedimiento para la preparacion de nuevas piperazino- pirimidinas.Info
- Publication number
- ES440153A2 ES440153A2 ES440153A ES440153A ES440153A2 ES 440153 A2 ES440153 A2 ES 440153A2 ES 440153 A ES440153 A ES 440153A ES 440153 A ES440153 A ES 440153A ES 440153 A2 ES440153 A2 ES 440153A2
- Authority
- ES
- Spain
- Prior art keywords
- formula
- preparation
- see formula
- alkyl group
- carbon atoms
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7427671A FR2281117A2 (fr) | 1974-08-09 | 1974-08-09 | Nouvelles piperazino-pyrimidines utilisables comme medicaments |
Publications (1)
Publication Number | Publication Date |
---|---|
ES440153A2 true ES440153A2 (es) | 1977-07-01 |
Family
ID=9142279
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES440153A Expired ES440153A2 (es) | 1974-08-09 | 1975-08-08 | Un procedimiento para la preparacion de nuevas piperazino- pirimidinas. |
Country Status (13)
Country | Link |
---|---|
JP (2) | JPS51125089A (no) |
AR (1) | AR205579A1 (no) |
BE (1) | BE832277R (no) |
CA (1) | CA1036598A (no) |
CH (1) | CH609692A5 (no) |
DE (1) | DE2534963A1 (no) |
ES (1) | ES440153A2 (no) |
FR (1) | FR2281117A2 (no) |
GB (1) | GB1512101A (no) |
LU (1) | LU73175A1 (no) |
NL (1) | NL7509184A (no) |
NO (1) | NO752586L (no) |
ZA (1) | ZA755118B (no) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2417507A2 (fr) * | 1977-07-28 | 1979-09-14 | Ugine Kuhlmann | Diamino-2,4 (ou -4,6) methylthio-5 pyrimidines herbicides |
FR2503162A1 (fr) * | 1981-04-07 | 1982-10-08 | Pharmindustrie | Nouveaux derives de piperazino-2 pyrimidine, procedes pour leur preparation et leur utilisation comme medicaments ou comme intermediaires pour la fabrication de medicaments |
JPS5973573A (ja) * | 1982-09-09 | 1984-04-25 | ワ−ナ−−ランバ−ト・コンパニ− | ジアミノピリミジン化合物 |
US6825198B2 (en) | 2001-06-21 | 2004-11-30 | Pfizer Inc | 5-HT receptor ligands and uses thereof |
MXPA06000051A (es) | 2003-07-02 | 2006-03-21 | Vertex Pharma | Pirimidinas utiles como moduladores de canales ionicos dependientes de voltaje. |
JP5388574B2 (ja) | 2005-05-31 | 2014-01-15 | バーテックス ファーマシューティカルズ インコーポレイテッド | イオンチャネルのモジュレーターとして有用なヘテロ環式類 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2119234A5 (en) * | 1970-12-24 | 1972-08-04 | Ugine Kuhlmann | 5-alkylthio amino halopyrimidines - fungicides herbicides insecticides and bactericides |
FR2173746B1 (no) * | 1972-03-01 | 1975-04-25 | Ugine Kuhlmann |
-
1974
- 1974-08-09 FR FR7427671A patent/FR2281117A2/fr active Granted
-
1975
- 1975-01-01 AR AR259942A patent/AR205579A1/es active
- 1975-07-21 NO NO752586A patent/NO752586L/no unknown
- 1975-08-01 NL NL7509184A patent/NL7509184A/xx not_active Application Discontinuation
- 1975-08-05 DE DE19752534963 patent/DE2534963A1/de not_active Withdrawn
- 1975-08-07 LU LU73175A patent/LU73175A1/xx unknown
- 1975-08-08 JP JP50096602A patent/JPS51125089A/ja active Pending
- 1975-08-08 CA CA233,149A patent/CA1036598A/fr not_active Expired
- 1975-08-08 GB GB33132/75A patent/GB1512101A/en not_active Expired
- 1975-08-08 ES ES440153A patent/ES440153A2/es not_active Expired
- 1975-08-08 BE BE159072A patent/BE832277R/xx not_active IP Right Cessation
- 1975-08-08 ZA ZA00755118A patent/ZA755118B/xx unknown
- 1975-08-11 CH CH1044275A patent/CH609692A5/xx not_active IP Right Cessation
-
1983
- 1983-02-04 JP JP58017292A patent/JPS5946943B2/ja not_active Expired
Also Published As
Publication number | Publication date |
---|---|
JPS58150571A (ja) | 1983-09-07 |
JPS51125089A (en) | 1976-11-01 |
LU73175A1 (no) | 1976-03-02 |
ZA755118B (en) | 1976-07-28 |
DE2534963A1 (de) | 1976-02-19 |
GB1512101A (en) | 1978-05-24 |
BE832277R (fr) | 1976-02-09 |
AR205579A1 (es) | 1976-05-14 |
FR2281117A2 (fr) | 1976-03-05 |
NL7509184A (nl) | 1976-02-11 |
JPS5946943B2 (ja) | 1984-11-15 |
NO752586L (no) | 1976-02-10 |
FR2281117B2 (no) | 1978-07-28 |
CH609692A5 (en) | 1979-03-15 |
CA1036598A (fr) | 1978-08-15 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ES378367A1 (es) | Procedimiento para la preparacion de nucleosidos. | |
ES8500244A1 (es) | "un procedimiento para preparar derivados de pirazinona" | |
ES468501A1 (es) | Un procedimiento para la preparacion de derivados de imida- zodiacepina. | |
ES440153A2 (es) | Un procedimiento para la preparacion de nuevas piperazino- pirimidinas. | |
ES385627A2 (es) | Procedimiento para la preparacion de derivados de morfoli- na. | |
ES450380A1 (es) | Procedimiento para preparar derivados de acido indanacetico. | |
ES418113A1 (es) | Un procedimiento para la preparacion de nuevas piperacino- pirimidinas. | |
ES438364A1 (es) | Procedimiento para la obtencion de nuevos derivados de gen- tamicina. | |
ES451466A1 (es) | Procedimiento para la preparacion de nuevos derivados de 5- tiazol-metanoamina. | |
ES443421A1 (es) | Un procedimiento para la preparacion de una composicion far-macologica que contiene una 11-desoxi-gamma-pentanorprosta- glandina. | |
ES465346A1 (es) | Procedimiento para preparar imidazoles 4,5-disustituidos. | |
ES435351A1 (es) | Procedimiento para preparar 1-(3-fenil-propil)-4-furoilpi- perazinas. | |
ES438736A1 (es) | Procedimiento para preparar esteres del acido dihidro-16, 17 apovincaminico. | |
ES386969A1 (es) | Un metodo para preparar una amidinourea. | |
CH614940A5 (en) | Process for the preparation of new terpenoaromatic amidines | |
ES465761A1 (es) | Procedimiento para la obtencion de compuestos de acido 3-ha-logenosulfonil-tiofen-carboxilico. | |
ES386567A1 (es) | Procedimiento para la obtencion de derivados de piridazona. | |
ES439180A1 (es) | Procedimiento para la preparacion de derivados de piperido- na. | |
ES401239A1 (es) | Procedimiento para la obtencion de compuestos heterocicli- cos. | |
ES423560A1 (es) | Un procedimiento para preparar dibencilperoxidicarbonatos. | |
ES405275A1 (es) | Procedimiento para la preparacion de 2h, 5, 6-dihidro-1,4- oxazinas y 2h, 5, 6-dihidro-1, 4-tiazinas. | |
ES440004A1 (es) | Procedimiento para la preparacion de derivados de proscila- ridina. | |
ES438050A1 (es) | Procedimiento para la produccion de nuevos derivados de pi- razol. | |
ES379624A1 (es) | Procedimiento para producir compuestos de pirazol-diazepi- nona. | |
ES469913A1 (es) | Un procedimiento para la preparacion de nuevos derivados de 6,11-dihidrobenzo-(b.e.)-tiepin-11-ona. |