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AR205579A1 - Procedimiento para preparar nuevos derivados de la metiltio-5 cloro-6 amino-2 (piperazina-1-il)-4-pirimidina - Google Patents

Procedimiento para preparar nuevos derivados de la metiltio-5 cloro-6 amino-2 (piperazina-1-il)-4-pirimidina

Info

Publication number
AR205579A1
AR205579A1 AR259942A AR25994275A AR205579A1 AR 205579 A1 AR205579 A1 AR 205579A1 AR 259942 A AR259942 A AR 259942A AR 25994275 A AR25994275 A AR 25994275A AR 205579 A1 AR205579 A1 AR 205579A1
Authority
AR
Argentina
Prior art keywords
methylthi
piperazine
pyrimidine
chloro
amino
Prior art date
Application number
AR259942A
Other languages
English (en)
Spanish (es)
Original Assignee
Ugine Kuhlmann
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ugine Kuhlmann filed Critical Ugine Kuhlmann
Application granted granted Critical
Publication of AR205579A1 publication Critical patent/AR205579A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AR259942A 1974-08-09 1975-01-01 Procedimiento para preparar nuevos derivados de la metiltio-5 cloro-6 amino-2 (piperazina-1-il)-4-pirimidina AR205579A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7427671A FR2281117A2 (fr) 1974-08-09 1974-08-09 Nouvelles piperazino-pyrimidines utilisables comme medicaments

Publications (1)

Publication Number Publication Date
AR205579A1 true AR205579A1 (es) 1976-05-14

Family

ID=9142279

Family Applications (1)

Application Number Title Priority Date Filing Date
AR259942A AR205579A1 (es) 1974-08-09 1975-01-01 Procedimiento para preparar nuevos derivados de la metiltio-5 cloro-6 amino-2 (piperazina-1-il)-4-pirimidina

Country Status (13)

Country Link
JP (2) JPS51125089A (no)
AR (1) AR205579A1 (no)
BE (1) BE832277R (no)
CA (1) CA1036598A (no)
CH (1) CH609692A5 (no)
DE (1) DE2534963A1 (no)
ES (1) ES440153A2 (no)
FR (1) FR2281117A2 (no)
GB (1) GB1512101A (no)
LU (1) LU73175A1 (no)
NL (1) NL7509184A (no)
NO (1) NO752586L (no)
ZA (1) ZA755118B (no)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2417507A2 (fr) * 1977-07-28 1979-09-14 Ugine Kuhlmann Diamino-2,4 (ou -4,6) methylthio-5 pyrimidines herbicides
FR2503162A1 (fr) * 1981-04-07 1982-10-08 Pharmindustrie Nouveaux derives de piperazino-2 pyrimidine, procedes pour leur preparation et leur utilisation comme medicaments ou comme intermediaires pour la fabrication de medicaments
JPS5973573A (ja) * 1982-09-09 1984-04-25 ワ−ナ−−ランバ−ト・コンパニ− ジアミノピリミジン化合物
US6825198B2 (en) 2001-06-21 2004-11-30 Pfizer Inc 5-HT receptor ligands and uses thereof
MXPA06000051A (es) 2003-07-02 2006-03-21 Vertex Pharma Pirimidinas utiles como moduladores de canales ionicos dependientes de voltaje.
JP5388574B2 (ja) 2005-05-31 2014-01-15 バーテックス ファーマシューティカルズ インコーポレイテッド イオンチャネルのモジュレーターとして有用なヘテロ環式類

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2119234A5 (en) * 1970-12-24 1972-08-04 Ugine Kuhlmann 5-alkylthio amino halopyrimidines - fungicides herbicides insecticides and bactericides
FR2173746B1 (no) * 1972-03-01 1975-04-25 Ugine Kuhlmann

Also Published As

Publication number Publication date
JPS58150571A (ja) 1983-09-07
JPS51125089A (en) 1976-11-01
ES440153A2 (es) 1977-07-01
LU73175A1 (no) 1976-03-02
ZA755118B (en) 1976-07-28
DE2534963A1 (de) 1976-02-19
GB1512101A (en) 1978-05-24
BE832277R (fr) 1976-02-09
FR2281117A2 (fr) 1976-03-05
NL7509184A (nl) 1976-02-11
JPS5946943B2 (ja) 1984-11-15
NO752586L (no) 1976-02-10
FR2281117B2 (no) 1978-07-28
CH609692A5 (en) 1979-03-15
CA1036598A (fr) 1978-08-15

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