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EA201101187A1 - Антидиабетические лекарственные средства, содержащие ингибитор dpp-4 (линаглиптин) необязательно в комбинации с другими антидиабетическими средствами - Google Patents

Антидиабетические лекарственные средства, содержащие ингибитор dpp-4 (линаглиптин) необязательно в комбинации с другими антидиабетическими средствами

Info

Publication number
EA201101187A1
EA201101187A1 EA201101187A EA201101187A EA201101187A1 EA 201101187 A1 EA201101187 A1 EA 201101187A1 EA 201101187 A EA201101187 A EA 201101187A EA 201101187 A EA201101187 A EA 201101187A EA 201101187 A1 EA201101187 A1 EA 201101187A1
Authority
EA
Eurasian Patent Office
Prior art keywords
diabetic
linagliptin
inhibitor
optional
combination
Prior art date
Application number
EA201101187A
Other languages
English (en)
Other versions
EA029759B1 (ru
Inventor
Эва Ульрике Грэфе-Моди
Ханс-Юрген Вёрле
Original Assignee
Бёрингер Ингельхайм Интернациональ Гмбх
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42174359&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201101187(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Бёрингер Ингельхайм Интернациональ Гмбх filed Critical Бёрингер Ингельхайм Интернациональ Гмбх
Publication of EA201101187A1 publication Critical patent/EA201101187A1/ru
Publication of EA029759B1 publication Critical patent/EA029759B1/ru

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    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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    • A61K31/52—Purines, e.g. adenine
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Abstract

В заявке описаны антидиабетические агенты, которые можно использовать для лечения или профилактики одного или более состояний, выбранных из группы, включающей в том числе сахарный диабет типа 1, сахарный диабет типа 2, нарушенную толерантность к глюкозе и гипергликемию. Кроме того, в заявке описаны способы профилактики или лечения метаболических нарушений и связанных с ними состояний.
EA201101187A 2009-02-13 2010-02-12 Антидиабетические лекарственные средства, содержащие ингибитор dpp-4 (линаглиптин) необязательно в комбинации с другими антидиабетическими средствами EA029759B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP09152869 2009-02-13
PCT/EP2010/051817 WO2010092163A2 (en) 2009-02-13 2010-02-12 Antidiabetic medications

Publications (2)

Publication Number Publication Date
EA201101187A1 true EA201101187A1 (ru) 2012-10-30
EA029759B1 EA029759B1 (ru) 2018-05-31

Family

ID=42174359

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201101187A EA029759B1 (ru) 2009-02-13 2010-02-12 Антидиабетические лекарственные средства, содержащие ингибитор dpp-4 (линаглиптин) необязательно в комбинации с другими антидиабетическими средствами

Country Status (14)

Country Link
US (6) US20120094894A1 (ru)
EP (1) EP2395988A2 (ru)
JP (3) JP2012517977A (ru)
KR (2) KR20160143897A (ru)
CN (3) CN117547538A (ru)
AU (1) AU2010212823B2 (ru)
BR (1) BRPI1013639A2 (ru)
CA (1) CA2752437C (ru)
CL (1) CL2011001853A1 (ru)
EA (1) EA029759B1 (ru)
IL (1) IL213716A0 (ru)
MX (2) MX2011008416A (ru)
NZ (2) NZ594044A (ru)
WO (1) WO2010092163A2 (ru)

Families Citing this family (106)

* Cited by examiner, † Cited by third party
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US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
US7772191B2 (en) 2005-05-10 2010-08-10 Boehringer Ingelheim International Gmbh Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
PE20110235A1 (es) 2006-05-04 2011-04-14 Boehringer Ingelheim Int Combinaciones farmaceuticas que comprenden linagliptina y metmorfina
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US20120094894A1 (en) 2012-04-19
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