DK1915375T3 - Derivater af 5-pyridinyl-1-azabicyclo[3,2,1]octan, fremgangsmåde til fremstilling deraf samt anvendelse deraf til terapi - Google Patents

Derivater af 5-pyridinyl-1-azabicyclo[3,2,1]octan, fremgangsmåde til fremstilling deraf samt anvendelse deraf til terapi

Info

Publication number: DK1915375T3
Authority: DK; Denmark
Prior art keywords: azabicyclo; pyridinyl; octane; therapy; derivatives
Prior art date: 2005-08-12

Application number

DK06794298.7T

Other languages

English (en)

Inventor

Frederic Galli

Odile Leclerc

Alistair Lochead

Julien Vache

Original Assignee

Sanofi Aventis

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-08-12

Filing date

2006-08-07

Publication date

2010-02-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36273387&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1915375(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2006-08-07 Application filed by Sanofi Aventis filed Critical Sanofi Aventis

2010-02-15 Application granted granted Critical

2010-02-15 Publication of DK1915375T3 publication Critical patent/DK1915375T3/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/18—Bridged systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Addiction (AREA)
Psychiatry (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Hospice & Palliative Care (AREA)
Dermatology (AREA)
Psychology (AREA)
Vascular Medicine (AREA)
Pain & Pain Management (AREA)
Epidemiology (AREA)
Rheumatology (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)

DK06794298.7T 2005-08-12 2006-08-07 Derivater af 5-pyridinyl-1-azabicyclo[3,2,1]octan, fremgangsmåde til fremstilling deraf samt anvendelse deraf til terapi DK1915375T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR0508528A FR2889701B1 (fr)	2005-08-12	2005-08-12	Derives de 5-pyridinyl-1-azabicyclo[3.2.1]octane, leur preparation en therapeutique.
PCT/FR2006/001912 WO2007020344A1 (fr)	2005-08-12	2006-08-07	DÉRIVÉS DE δ-PYRIDINYL-i-AZABICYCLO[3.2.1]OCTANE, A LEUR PRÉPARATION ET LEUR APPLICATION EN THÉRAPEUTIQUE

Publications (1)

Publication Number	Publication Date
DK1915375T3 true DK1915375T3 (da)	2010-02-15

Family

ID=36273387

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK06794298.7T DK1915375T3 (da)	2005-08-12	2006-08-07	Derivater af 5-pyridinyl-1-azabicyclo[3,2,1]octan, fremgangsmåde til fremstilling deraf samt anvendelse deraf til terapi

Country Status (41)

Country	Link
US (2)	US7863290B2 (da)
EP (1)	EP1915375B1 (da)
JP (1)	JP5164841B2 (da)
KR (1)	KR101299339B1 (da)
CN (1)	CN101238125B (da)
AT (1)	ATE444964T1 (da)
AU (1)	AU2006281341B2 (da)
BR (1)	BRPI0614623A2 (da)
CA (1)	CA2617828C (da)
CR (1)	CR9625A (da)
CY (1)	CY1109717T1 (da)
DE (1)	DE602006009668D1 (da)
DK (1)	DK1915375T3 (da)
DO (1)	DOP2006000180A (da)
EA (1)	EA014023B1 (da)
EC (1)	ECSP088170A (da)
ES (1)	ES2332472T3 (da)
FR (1)	FR2889701B1 (da)
GT (1)	GT200600368A (da)
HK (1)	HK1120788A1 (da)
HN (1)	HN2008000090A (da)
HR (1)	HRP20090677T1 (da)
IL (1)	IL188796A (da)
JO (1)	JO2583B1 (da)
MA (1)	MA30200B1 (da)
ME (1)	ME01750B (da)
MX (1)	MX2008001968A (da)
MY (1)	MY147846A (da)
NO (1)	NO20081151L (da)
NZ (1)	NZ565149A (da)
PE (1)	PE20070339A1 (da)
PL (1)	PL1915375T3 (da)
PT (1)	PT1915375E (da)
RS (1)	RS51068B (da)
SI (1)	SI1915375T1 (da)
TN (1)	TNSN07472A1 (da)
TW (1)	TWI324158B (da)
UA (1)	UA92917C2 (da)
UY (1)	UY29744A1 (da)
WO (1)	WO2007020344A1 (da)
ZA (1)	ZA200800958B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2912404B1 (fr) *	2007-02-09	2009-04-10	Sanofi Aventis Sa	Derives d'azabicycloalkane,leur preparation et leur application en therapeutique.
GB0817424D0 (en)	2008-09-24	2008-10-29	Medivir Ab	Protease inhibitors
JP2017114765A (ja) *	2014-04-25	2017-06-29	大正製薬株式会社	トリアゾリルで置換されたヘテロアリール化合物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5817679A (en) *	1993-04-01	1998-10-06	University Of Virginia	7-Azabicyclo 2.2.1!-heptane and -heptene derivatives as cholinergic receptor ligands
EP0664293A1 (en) *	1993-12-24	1995-07-26	Duphar International Research B.V	2-Phenyl-7-azabicycloheptanes and 6-phenyl-8-azabicyclo
JP4447663B2 (ja) *	1997-05-30	2010-04-07	ニューロサーチ、アクティーゼルスカブ	ニコチン性ａｃｈレセプターに於けるコリン作動性リガンドとしての８−アザビシクロ（３．２．１）オクト−２−エン及びオクタン誘導体
FR2834511B1 (fr) *	2002-01-07	2004-02-13	Sanofi Synthelabo	Derives de 5-(pyridin-3-yl)-1-azabicyclo[3.2.1]octane, leur preparation et leur application en therapeutique

2005
- 2005-08-12 FR FR0508528A patent/FR2889701B1/fr active Active
2006
- 2006-07-08 UA UAA200802988A patent/UA92917C2/uk unknown
- 2006-07-26 JO JO2006252A patent/JO2583B1/en active
- 2006-08-02 DO DO2006000180A patent/DOP2006000180A/es unknown
- 2006-08-07 PT PT06794298T patent/PT1915375E/pt unknown
- 2006-08-07 AT AT06794298T patent/ATE444964T1/de active
- 2006-08-07 KR KR1020087003271A patent/KR101299339B1/ko not_active IP Right Cessation
- 2006-08-07 ES ES06794298T patent/ES2332472T3/es active Active
- 2006-08-07 WO PCT/FR2006/001912 patent/WO2007020344A1/fr active Application Filing
- 2006-08-07 SI SI200630515T patent/SI1915375T1/sl unknown
- 2006-08-07 ZA ZA200800958A patent/ZA200800958B/xx unknown
- 2006-08-07 NZ NZ565149A patent/NZ565149A/en not_active IP Right Cessation
- 2006-08-07 AU AU2006281341A patent/AU2006281341B2/en not_active Ceased
- 2006-08-07 JP JP2008525599A patent/JP5164841B2/ja not_active Expired - Fee Related
- 2006-08-07 EP EP06794298A patent/EP1915375B1/fr active Active
- 2006-08-07 EA EA200800575A patent/EA014023B1/ru not_active IP Right Cessation
- 2006-08-07 PL PL06794298T patent/PL1915375T3/pl unknown
- 2006-08-07 ME MEP-2009-576A patent/ME01750B/me unknown
- 2006-08-07 MX MX2008001968A patent/MX2008001968A/es active IP Right Grant
- 2006-08-07 CA CA2617828A patent/CA2617828C/fr not_active Expired - Fee Related
- 2006-08-07 CN CN2006800291833A patent/CN101238125B/zh not_active Expired - Fee Related
- 2006-08-07 RS RSP-2009/0576A patent/RS51068B/sr unknown
- 2006-08-07 BR BRPI0614623-6A patent/BRPI0614623A2/pt not_active IP Right Cessation
- 2006-08-07 DK DK06794298.7T patent/DK1915375T3/da active
- 2006-08-07 DE DE602006009668T patent/DE602006009668D1/de active Active
- 2006-08-10 GT GT200600368A patent/GT200600368A/es unknown
- 2006-08-10 PE PE2006000974A patent/PE20070339A1/es not_active Application Discontinuation
- 2006-08-10 MY MYPI20063888A patent/MY147846A/en unknown
- 2006-08-11 TW TW095129651A patent/TWI324158B/zh not_active IP Right Cessation
- 2006-08-11 UY UY29744A patent/UY29744A1/es not_active Application Discontinuation
2007
- 2007-12-14 TN TNP2007000472A patent/TNSN07472A1/en unknown
- 2007-12-20 CR CR9625A patent/CR9625A/es unknown
2008
- 2008-01-15 IL IL188796A patent/IL188796A/en not_active IP Right Cessation
- 2008-01-22 HN HN2008000090A patent/HN2008000090A/es unknown
- 2008-02-11 US US12/028,999 patent/US7863290B2/en not_active Expired - Fee Related
- 2008-02-11 EC EC2008008170A patent/ECSP088170A/es unknown
- 2008-03-04 NO NO20081151A patent/NO20081151L/no not_active Application Discontinuation
- 2008-03-07 MA MA30724A patent/MA30200B1/fr unknown
- 2008-11-11 HK HK08112365.4A patent/HK1120788A1/xx not_active IP Right Cessation
2009
- 2009-12-17 HR HR20090677T patent/HRP20090677T1/hr unknown
2010
- 2010-01-05 CY CY20101100013T patent/CY1109717T1/el unknown
- 2010-11-29 US US12/955,389 patent/US8541440B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
WO2007020344A1 (fr)	2007-02-22
JO2583B1 (en)	2011-02-27
ME01750B (me)	2010-10-31
UY29744A1 (es)	2007-03-30
IL188796A0 (en)	2008-08-07
CA2617828C (fr)	2014-03-11
TWI324158B (en)	2010-05-01
ZA200800958B (en)	2009-04-29
US7863290B2 (en)	2011-01-04
RS51068B (sr)	2010-10-31
CN101238125A (zh)	2008-08-06
US20080146608A1 (en)	2008-06-19
PT1915375E (pt)	2009-11-26
EA200800575A1 (ru)	2008-06-30
CN101238125B (zh)	2012-07-04
IL188796A (en)	2012-09-24
DE602006009668D1 (de)	2009-11-19
MX2008001968A (es)	2008-03-26
UA92917C2 (uk)	2010-12-27
HRP20090677T1 (hr)	2010-01-31
EP1915375A1 (fr)	2008-04-30
ATE444964T1 (de)	2009-10-15
US8541440B2 (en)	2013-09-24
NZ565149A (en)	2011-05-27
SI1915375T1 (sl)	2010-01-29
EP1915375B1 (fr)	2009-10-07
ECSP088170A (es)	2008-03-26
NO20081151L (no)	2008-05-13
TNSN07472A1 (en)	2009-03-17
KR20080033378A (ko)	2008-04-16
JP2009505971A (ja)	2009-02-12
CY1109717T1 (el)	2014-08-13
DOP2006000180A (es)	2007-02-28
BRPI0614623A2 (pt)	2011-04-12
KR101299339B1 (ko)	2013-08-26
PE20070339A1 (es)	2007-04-18
HK1120788A1 (da)	2009-04-09
MY147846A (en)	2013-01-31
PL1915375T3 (pl)	2010-03-31
US20110077264A1 (en)	2011-03-31
EA014023B1 (ru)	2010-08-30
GT200600368A (es)	2007-07-06
ES2332472T3 (es)	2010-02-05
CR9625A (es)	2008-04-10
FR2889701A1 (fr)	2007-02-16
HN2008000090A (es)	2010-08-19
JP5164841B2 (ja)	2013-03-21
AU2006281341A1 (en)	2007-02-22
CA2617828A1 (fr)	2007-02-22
AU2006281341B2 (en)	2012-04-19
MA30200B1 (fr)	2009-02-02
FR2889701B1 (fr)	2007-10-05
TW200740810A (en)	2007-11-01

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EA200970149A1 (ru)	2009-06-30	Производные n-(аминогетероарил)-1h-индол-2-карбоксамидов, их получение и их применение в терапии
BRPI0412347A (pt)	2006-09-05	2-aminofenil-4-fenilpiridinas como inibidores de quinase
UY29857A1 (es)	2007-05-31	Derivados de la 4-amino-quinazolina, su preparación y su aplicación en terapéutica.
BRPI0418639A (pt)	2007-05-29	inibidores de dipeptidil peptidase
WO2007103187A3 (en)	2007-11-01	8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists
MX2010006799A (es)	2010-10-05	Benzofuropirimidinonas como inhibidores de la proteina cinasa.
WO2004087699A3 (en)	2004-12-09	Thiazoles useful as inhibitors of protein kinases
WO2008120725A1 (ja)	2008-10-09	新規ピロリノン誘導体およびそれを含有する医薬組成物
DK2041133T3 (da)	2011-02-07	Derivater af imadazol [1,2-A] pyridine-2-carboxamider, fremstilling deraf og anvendelse deraf i terapeutik
HRP20070577T3 (en)	2008-08-31	Quinazolinone derivatives useful as vanilloid antagonists
ECSP067111A (es)	2007-01-26	Derivados de pirido-pirimidina, su preparación, su aplicación en terapéutica
WO2008128009A3 (en)	2009-01-08	Aminopyrimidines useful as kinase inhibitors
UY29859A1 (es)	2007-05-31	Derivados de 1-amino-isiquinolina,su preparación y su aplicación terapéutica
RS20060239A (en)	2008-06-05	Arylalkylcarbamate derivatives, preparation method thereof and use of same in therapeutics
DK1915375T3 (da)	2010-02-15	Derivater af 5-pyridinyl-1-azabicyclo[3,2,1]octan, fremgangsmåde til fremstilling deraf samt anvendelse deraf til terapi
ZA200900165B (en)	2009-12-30	4-amino-3-arylamino-6-arylpyrazolo[3,4-D]pyrimidine derivatives, methods for their preparation and their use as antiviral agents
WO2009106750A3 (fr)	2010-02-25	Dérivés 6-heterocyclique-imidazo[1,2-a]pyrroine-2-carboxamides, leur préparation et leur application en thérapeutique
WO2006066044A3 (en)	2007-05-10	Processes for producing 4-aminoquinazolines
UA104302C2 (ru)	2014-01-27	Производные морфин-6-глюкуронида, их получение и их применение в терапии
WO2005123694A3 (en)	2006-04-13	Quinazolinone compounds for the treatment of cough
WO2010067008A3 (fr)	2011-07-07	Derives bicycliques de morphine-6-glucuronide, leur preparation et leur application en therapeutique