DK1758914T3 - Hidtil ukendte fluorglycosidderivater af pyrazoler, lægemidler indeholdende disse forbindelser og anvendelse heraf - Google Patents

Hidtil ukendte fluorglycosidderivater af pyrazoler, lægemidler indeholdende disse forbindelser og anvendelse heraf

Info

Publication number: DK1758914T3
Authority: DK; Denmark
Prior art keywords: pyrazoles; compounds; new; drugs containing; fluoroglycoside derivatives
Prior art date: 2004-06-11

Application number

DK05746637T

Other languages

Danish (da)

English (en)

Inventor

Harm Brummerhop

Wendelin Frick

Heiner Glombik

Oliver Plettenburg

Martin Bickel

Hubert Heuer

Stefan Theis

Original Assignee

Sanofi Aventis Deutschland

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2004-06-11

Filing date

2005-06-03

Publication date

2008-03-17

2005-06-03 Application filed by Sanofi Aventis Deutschland filed Critical Sanofi Aventis Deutschland

2008-03-17 Application granted granted Critical

2008-03-17 Publication of DK1758914T3 publication Critical patent/DK1758914T3/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Diabetes (AREA)
Hematology (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Immunology (AREA)
Neurosurgery (AREA)
Physical Education & Sports Medicine (AREA)
Rheumatology (AREA)
Molecular Biology (AREA)
Obesity (AREA)
Urology & Nephrology (AREA)
Psychiatry (AREA)
Genetics & Genomics (AREA)
Biotechnology (AREA)
Biochemistry (AREA)
Pulmonology (AREA)
Virology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Orthopedic Medicine & Surgery (AREA)
Ophthalmology & Optometry (AREA)
Dermatology (AREA)
Heart & Thoracic Surgery (AREA)
Vascular Medicine (AREA)
Emergency Medicine (AREA)

DK05746637T 2004-06-11 2005-06-03 Hidtil ukendte fluorglycosidderivater af pyrazoler, lægemidler indeholdende disse forbindelser og anvendelse heraf DK1758914T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE102004028241A DE102004028241B4 (de)	2004-06-11	2004-06-11	Neue Fluorglykosidderivate von Pyrazolen, diese Verbindungen enthaltende Arzneimittel und Herstellung dieser Arzneimittel
PCT/EP2005/005959 WO2005121161A1 (de)	2004-06-11	2005-06-03	Neue fluorglykosidderivate von pyrazolen, diese verbindungen enthaltende arzneimittel und deren verwendung

Publications (1)

Publication Number	Publication Date
DK1758914T3 true DK1758914T3 (da)	2008-03-17

Family

ID=35355753

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK05746637T DK1758914T3 (da)	2004-06-11	2005-06-03	Hidtil ukendte fluorglycosidderivater af pyrazoler, lægemidler indeholdende disse forbindelser og anvendelse heraf

Country Status (34)

Country	Link
US (1)	US7820804B2 (xx)
EP (1)	EP1758914B1 (xx)
JP (1)	JP4996464B2 (xx)
CN (1)	CN100582116C (xx)
AR (1)	AR049393A1 (xx)
AU (1)	AU2005252329B2 (xx)
BR (1)	BRPI0510770A (xx)
CA (1)	CA2570042C (xx)
CR (1)	CR8773A (xx)
CY (1)	CY1107426T1 (xx)
DE (2)	DE102004028241B4 (xx)
DK (1)	DK1758914T3 (xx)
EC (1)	ECSP067054A (xx)
ES (1)	ES2296180T3 (xx)
HK (1)	HK1100411A1 (xx)
HR (1)	HRP20080023T3 (xx)
IL (1)	IL179757A (xx)
MA (1)	MA28653B1 (xx)
MX (1)	MXPA06013513A (xx)
MY (1)	MY143565A (xx)
NO (1)	NO20070176L (xx)
NZ (1)	NZ551948A (xx)
PE (1)	PE20060297A1 (xx)
PL (1)	PL1758914T3 (xx)
PT (1)	PT1758914E (xx)
RS (1)	RS50541B (xx)
RU (1)	RU2370499C2 (xx)
SI (1)	SI1758914T1 (xx)
TN (1)	TNSN06409A1 (xx)
TW (1)	TWI382030B (xx)
UA (1)	UA89787C2 (xx)
UY (1)	UY28955A1 (xx)
WO (1)	WO2005121161A1 (xx)
ZA (1)	ZA200608832B (xx)

Families Citing this family (53)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW200637869A (en)	2005-01-28	2006-11-01	Chugai Pharmaceutical Co Ltd	The spiroketal derivatives and the use as therapeutical agent for diabetes of the same
DE102005026762A1 (de)	2005-06-09	2006-12-21	Sanofi-Aventis Deutschland Gmbh	Azolopyridin-2-on-derivate als Inhibitoren von Lipasen und Phospholipasen
PE20080251A1 (es)	2006-05-04	2008-04-25	Boehringer Ingelheim Int	Usos de inhibidores de dpp iv
WO2007136116A2 (en)	2006-05-19	2007-11-29	Taisho Pharmaceutical Co., Ltd.	C-phenyl glycitol compound for the treatment of diabetes
NZ573843A (en)	2006-06-29	2011-02-25	Taisho Pharmaceutical Co Ltd	C-phenyl 1-thioglucitol compound
KR20090047458A (ko)	2006-08-08	2009-05-12	사노피-아벤티스	아릴아미노아릴-알킬-치환된 이미다졸리딘-2,4-디온, 이의 제조방법, 이들 화합물을 포함하는 약제 및 이의 용도
DE102006053637B4 (de)	2006-11-14	2011-06-30	Sanofi-Aventis Deutschland GmbH, 65929	Neue mit Fluor substituierte 1,4-Benzothiepin-1,1-Dioxidderivate, diese Verbindungen enthaltende Arzneimittel und deren Verwendung
WO2008072726A1 (ja)	2006-12-14	2008-06-19	Taisho Pharmaceutical Co., Ltd.	１－フェニル１－チオ－ｄ－グルシト－ル誘導体
EP2025674A1 (de)	2007-08-15	2009-02-18	sanofi-aventis	Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
JP5272395B2 (ja) *	2007-12-12	2013-08-28	セントラル硝子株式会社	４−デオキシ−４−フルオロ−ｄ−グルコース誘導体の製造方法
WO2010003624A2 (en)	2008-07-09	2010-01-14	Sanofi-Aventis	Heterocyclic compounds, processes for their preparation, medicaments comprising these compounds, and the use thereof
WO2010023594A1 (en) *	2008-08-28	2010-03-04	Pfizer Inc.	Dioxa-bicyclo[3.2.1.]octane-2,3,4-triol derivatives
WO2010068601A1 (en)	2008-12-08	2010-06-17	Sanofi-Aventis	A crystalline heteroaromatic fluoroglycoside hydrate, processes for making, methods of use and pharmaceutical compositions thereof
ES2397086T3 (es)	2009-02-23	2013-03-04	Taisho Pharmaceutical Co., Ltd.	Compuestos de 4-isopropilfenil glucitol como inhibidores de SGLT1
CN102482312A (zh) *	2009-08-26	2012-05-30	赛诺菲	新颖的杂芳族氟代糖苷结晶水合物、含有这些化合物的药物和它们的用途
EP2298782A1 (en)	2009-08-26	2011-03-23	Sanofi-Aventis	Method for producing pyrazole glycoside derivatives
BR112012007349A2 (pt) *	2009-10-02	2019-09-24	Sanofi Sa	uso de composto com atividade inibidora de sglt-1/sglt-2 para produção de medicamentos para tratamento de doenças ósseas.
US8163704B2 (en)	2009-10-20	2012-04-24	Novartis Ag	Glycoside derivatives and uses thereof
DK2496583T3 (en)	2009-11-02	2015-02-02	Pfizer	Dioxa-bicyclo [3.2.1] octane-2,3,4-triol DERIVATIVES
AU2010319377B2 (en)	2009-11-13	2014-10-23	Astrazeneca Ab	Immediate release tablet formulations
CA2780938A1 (en)	2009-11-13	2011-05-19	Bristol-Myers Squibb Company	Reduced mass metformin formulations
EP2498758B1 (en)	2009-11-13	2018-07-25	AstraZeneca AB	Bilayer tablet formulations
WO2011107494A1 (de)	2010-03-03	2011-09-09	Sanofi	Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
WO2011157827A1 (de)	2010-06-18	2011-12-22	Sanofi	Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen
US8530413B2 (en)	2010-06-21	2013-09-10	Sanofi	Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201215387A (en)	2010-07-05	2012-04-16	Sanofi Aventis	Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament
TW201215388A (en)	2010-07-05	2012-04-16	Sanofi Sa	(2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
TW201221505A (en)	2010-07-05	2012-06-01	Sanofi Sa	Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
JP5532138B2 (ja)	2010-08-20	2014-06-25	大正製薬株式会社	４−イソプロピル−６−メトキシフェニルグルシトール化合物
RU2013112368A (ru)	2010-08-20	2014-09-27	Тайсо Фармасьютикал Ко., Лтд.	Кристаллическая форма 4-изопропилфенилглюцитольного соединения и способ ее получения
US20130224296A1 (en)	2010-09-03	2013-08-29	Bristol-Myers Squibb Company	Drug Formulations Using Water Soluble Antioxidants
RU2607480C2 (ru)	2011-02-01	2017-01-10	Бристол-Майерс Сквибб Компани	Фармацевтические композиции, содержащие аминосоединение
US8809325B2 (en)	2011-03-08	2014-08-19	Sanofi	Benzyl-oxathiazine derivatives substituted with adamantane and noradamantane, medicaments containing said compounds and use thereof
US8828995B2 (en)	2011-03-08	2014-09-09	Sanofi	Branched oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
WO2012120054A1 (de)	2011-03-08	2012-09-13	Sanofi	Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2012120052A1 (de)	2011-03-08	2012-09-13	Sanofi	Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
EP2683703B1 (de)	2011-03-08	2015-05-27	Sanofi	Neue substituierte phenyl-oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
WO2012120050A1 (de)	2011-03-08	2012-09-13	Sanofi	Neue substituierte phenyl-oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
EP2683699B1 (de)	2011-03-08	2015-06-24	Sanofi	Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2012120058A1 (de)	2011-03-08	2012-09-13	Sanofi	Mit benzyl- oder heteromethylengruppen substituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
EP2683700B1 (de)	2011-03-08	2015-02-18	Sanofi	Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
US8614195B2 (en) *	2011-04-14	2013-12-24	Novartis Ag	Glycoside derivatives and uses thereof
AR087701A1 (es) *	2011-08-31	2014-04-09	Japan Tobacco Inc	Derivados de pirazol con actividad inhibidora de sglt1
WO2013037390A1 (en)	2011-09-12	2013-03-21	Sanofi	6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
EP2760862B1 (en)	2011-09-27	2015-10-21	Sanofi	6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
UA113086C2 (xx) *	2012-05-10	2016-12-12		Піразольні сполуки як інгібітори sglt1
TW201425326A (zh)	2012-10-05	2014-07-01	Lilly Co Eli	新穎脲化合物
MX346453B (es)	2013-02-04	2017-03-17	Taisho Pharmaceutical Co Ltd	Medicamento profilactico o terapeutico para el estreñimiento.
EP2774619B1 (de)	2013-03-04	2016-05-18	BioActive Food GmbH	Zusammensetzung zur Behandlung von hyperglykämischen Erkrankungen
AR098670A1 (es)	2013-11-08	2016-06-08	Lilly Co Eli	Inhibidor de sglt1
EP2944311A1 (de)	2014-05-16	2015-11-18	BioActive Food GmbH	Kombination von biologisch aktiven Substanzen zur Behandlung von hyperglykämischen Erkrankungen
AU2019249560B2 (en) *	2018-04-04	2023-10-05	Japan Tobacco Inc.	Heteroaryl-substituted pyrazole compound and medicinal use thereof
EP3886854A4 (en)	2018-11-30	2022-07-06	Nuvation Bio Inc.	PYRROLE AND PYRAZOLE COMPOUNDS AND METHODS OF USE THERE

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0850948B1 (en) *	1996-12-26	2002-04-24	Tanabe Seiyaku Co., Ltd.	Propiophenone derivatives and process for preparing the same
AU782330B2 (en) *	1999-08-31	2005-07-21	Kissei Pharmaceutical Co. Ltd.	Glucopyranosyloxypyrazole derivatives, medicinal compositions containing the same and intermediates in the production thereof
PH12000002657B1 (en) *	1999-10-12	2006-02-21	Bristol Myers Squibb Co	C-aryl glucoside SGLT2 inhibitors
AU2002210990A1 (en) *	2000-11-02	2002-05-15	Ajinomoto Co. Inc.	Novel pyrazole derivatives and diabetes remedies containing the same
CA2438433A1 (en) *	2001-02-14	2002-08-22	Tularik Inc.	Methods for the diagnosis and treatment of tumors employing the hepsin gene
WO2004014932A1 (ja) *	2002-08-08	2004-02-19	Kissei Pharmaceutical Co., Ltd.	ピラゾール誘導体、それを含有する医薬組成物、その医薬用途及びその製造中間体
JP2004137245A (ja) *	2002-08-23	2004-05-13	Kissei Pharmaceut Co Ltd	ピラゾール誘導体、それを含有する医薬組成物、その医薬用途及びその製造中間体
JP4606876B2 (ja) *	2002-08-27	2011-01-05	キッセイ薬品工業株式会社	ピラゾール誘導体、それを含有する医薬組成物及びその医薬用途
EP1550668A4 (en) *	2002-10-04	2008-10-01	Kissei Pharmaceutical	PYRAZOLE DERIVATIVE, MEDICINAL COMPOSITION COMPRISING THE DERIVATIVE, MEDICINAL USE THEREOF, AND INTERMEDIATE ENTERING THE PRODUCTION THEREOF
AU2003289156A1 (en) *	2002-12-04	2004-06-23	Kissei Pharmaceutical Co., Ltd.	Preventive or remedy for diseases caused by hyperglycemia
DE10258008B4 (de) *	2002-12-12	2006-02-02	Sanofi-Aventis Deutschland Gmbh	Heterocyclische Fluorglycosidderivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zur Herstellung dieser Arzneimittel
CA2529878C (en) *	2003-06-20	2012-11-20	Kissei Pharmaceutical Co., Ltd.	Pyrazole derivative, drug composition containing the same and production intermediate therefor

2004
- 2004-06-11 DE DE102004028241A patent/DE102004028241B4/de not_active Expired - Fee Related
2005
- 2005-06-03 DK DK05746637T patent/DK1758914T3/da active
- 2005-06-03 AU AU2005252329A patent/AU2005252329B2/en not_active Ceased
- 2005-06-03 WO PCT/EP2005/005959 patent/WO2005121161A1/de active Application Filing
- 2005-06-03 RS RSP-2008/0017A patent/RS50541B/sr unknown
- 2005-06-03 DE DE502005002056T patent/DE502005002056D1/de active Active
- 2005-06-03 EP EP05746637A patent/EP1758914B1/de active Active
- 2005-06-03 PT PT05746637T patent/PT1758914E/pt unknown
- 2005-06-03 ES ES05746637T patent/ES2296180T3/es active Active
- 2005-06-03 CA CA2570042A patent/CA2570042C/en not_active Expired - Fee Related
- 2005-06-03 UA UAA200700259A patent/UA89787C2/ru unknown
- 2005-06-03 BR BRPI0510770-9A patent/BRPI0510770A/pt not_active IP Right Cessation
- 2005-06-03 RU RU2007101154/04A patent/RU2370499C2/ru not_active IP Right Cessation
- 2005-06-03 JP JP2007526254A patent/JP4996464B2/ja not_active Expired - Fee Related
- 2005-06-03 PL PL05746637T patent/PL1758914T3/pl unknown
- 2005-06-03 CN CN200580019067A patent/CN100582116C/zh not_active Expired - Fee Related
- 2005-06-03 NZ NZ551948A patent/NZ551948A/en not_active IP Right Cessation
- 2005-06-03 MX MXPA06013513A patent/MXPA06013513A/es active IP Right Grant
- 2005-06-03 SI SI200530142T patent/SI1758914T1/sl unknown
- 2005-06-09 MY MYPI20052616A patent/MY143565A/en unknown
- 2005-06-09 TW TW094118973A patent/TWI382030B/zh not_active IP Right Cessation
- 2005-06-10 UY UY28955A patent/UY28955A1/es unknown
- 2005-06-10 PE PE2005000666A patent/PE20060297A1/es not_active Application Discontinuation
- 2005-06-13 AR ARP050102406A patent/AR049393A1/es not_active Application Discontinuation
2006
- 2006-10-24 ZA ZA200608832A patent/ZA200608832B/en unknown
- 2006-11-27 CR CR8773A patent/CR8773A/es not_active Application Discontinuation
- 2006-11-30 IL IL179757A patent/IL179757A/en not_active IP Right Cessation
- 2006-12-05 MA MA29515A patent/MA28653B1/fr unknown
- 2006-12-06 US US11/567,410 patent/US7820804B2/en not_active Expired - Fee Related
- 2006-12-08 EC EC2006007054A patent/ECSP067054A/es unknown
- 2006-12-08 TN TNP2006000409A patent/TNSN06409A1/en unknown
2007
- 2007-01-10 NO NO20070176A patent/NO20070176L/no not_active Application Discontinuation
- 2007-07-31 HK HK07108324.3A patent/HK1100411A1/xx not_active IP Right Cessation
2008
- 2008-01-16 HR HR20080023T patent/HRP20080023T3/xx unknown
- 2008-02-04 CY CY20081100139T patent/CY1107426T1/el unknown

Also Published As

Publication number	Publication date
TW200610527A (en)	2006-04-01
RU2370499C2 (ru)	2009-10-20
CA2570042A1 (en)	2005-12-22
PL1758914T3 (pl)	2008-04-30
NO20070176L (no)	2007-03-09
CR8773A (es)	2008-02-28
JP2008501745A (ja)	2008-01-24
MA28653B1 (fr)	2007-06-01
DE102004028241A1 (de)	2006-01-05
CY1107426T1 (el)	2012-12-19
ES2296180T3 (es)	2008-04-16
RS50541B (sr)	2010-05-07
IL179757A0 (en)	2007-05-15
IL179757A (en)	2010-12-30
JP4996464B2 (ja)	2012-08-08
EP1758914A1 (de)	2007-03-07
AU2005252329A1 (en)	2005-12-22
MY143565A (en)	2011-05-31
HRP20080023T3 (en)	2008-06-30
CA2570042C (en)	2013-01-15
AU2005252329B2 (en)	2011-02-10
UY28955A1 (es)	2006-01-31
US20070197623A1 (en)	2007-08-23
CN100582116C (zh)	2010-01-20
CN1964984A (zh)	2007-05-16
DE102004028241B4 (de)	2007-09-13
ECSP067054A (es)	2007-01-26
NZ551948A (en)	2010-04-30
AR049393A1 (es)	2006-07-26
SI1758914T1 (sl)	2008-04-30
UA89787C2 (ru)	2010-03-10
PT1758914E (pt)	2008-01-31
US7820804B2 (en)	2010-10-26
DE502005002056D1 (de)	2008-01-03
ZA200608832B (en)	2008-05-28
TWI382030B (zh)	2013-01-11
BRPI0510770A (pt)	2007-11-20
TNSN06409A1 (en)	2008-02-22
PE20060297A1 (es)	2006-05-25
WO2005121161A1 (de)	2005-12-22
EP1758914B1 (de)	2007-11-21
HK1100411A1 (en)	2007-09-21
MXPA06013513A (es)	2007-03-01
RU2007101154A (ru)	2008-07-20

Publication	Publication Date	Title
DK1758914T3 (da)	2008-03-17	Hidtil ukendte fluorglycosidderivater af pyrazoler, lægemidler indeholdende disse forbindelser og anvendelse heraf
CY2013027I1 (el)	2024-09-20	Νεα παραγωγα ινσουλινης
NL350096I2 (nl)	2019-10-29	Isopyrazam of een tautomeer daarvan, en prothioconazole
DK1572708T3 (da)	2006-08-21	Hidtil ukendt, heterocycliske derivater af fluorglycosider, lægemidler indeholdende disse forbindelser og anvendelse deraf
DK1756064T3 (da)	2008-09-22	Pyrazolderivater, sammensætninger indeholdende sådanne forbindelser og anvendelsesmetoder
DK1656370T3 (da)	2012-11-26	Heterocykliske biarylforbindelser og fremgangsmåder til fremstilling og anvendelse af samme
NO20081604L (no)	2008-07-03	Nitrogeninneholdende heterocyklisk forbindelse og farmasøytisk anvendelse derav
DK1730131T3 (da)	2012-08-13	Glucopyranosyl-substituerede benzol-derivater, lægemiddel indeholdende disse forbindelser, deres anvendelse og fremgangsmåder til deres fremstilling
DK2057153T3 (da)	2012-10-15	(3-aryl-piperazin-1-yl)-derivater af 6,7 dialkoxyquinazolin, 6,7- dialkoxyphtalazin og 6,7-dialkoxyisoquinolin
DK1802579T3 (da)	2014-01-20	Derivater af 3-arylaminopyridin
DK1572707T3 (da)	2006-08-14	Hidtil ukendte aromatiske fluorglycosidderivater, lægemidler indeholdende disse forbindelser og anvendelse heraf
DK2508521T4 (da)	2022-10-03	Dimaleat af en aminocrotonylforbindelse og fremgangsmåde til fremstilling deraf
DK1913001T3 (da)	2013-10-21	(r)-n-methylnaltrexon, fremgangsmåder til syntese og farmaceutisk anvendelse heraf
DK1523488T3 (da)	2009-03-16	Nye thiophenglycosidderivater, fremgangsmåder til deres fremstilling, lægemidler indeholdende disse forbindelser og deres anvendelse
DK2617714T3 (da)	2016-06-27	Kemiske derivater af jasmonat, farmaceutiske præparater og fremgangsmåder til anvendelse deraf
BRPI0508259A (pt)	2007-07-31	derivado heterocìclico fundido, composição medicinal contendo o mesmo, e uso medicinal do mesmo
DK1805312T3 (da)	2009-10-19	Fremgangsmåder og midler til fremstilling af hyaluronan
CY2017048I1 (el)	2018-09-05	Νεες φαρμακευτικες χρησεις των παραγωγων σταυροσπορινης
DK1937664T3 (da)	2011-07-18	Hydrazidforbindelse og pesticid anvendelse af den samme
DK3305776T3 (da)	2019-12-09	Pyrrol-forbindelser som inhibitorer af erk-protein-kinaser og farmaceutiske sammensætninger, der indeholder disse forbindelser
DK2046715T3 (da)	2014-06-02	Substituerede 1,3-diphenylpropanderivater, præparater og anvendelser deraf
DK1939204T6 (da)	2022-09-05	Kondenseret heterocyklisk derivat, medicinalsammensætning indeholdende samme og medicinsk anvendelse deraf
DK1830850T3 (da)	2011-06-14	Quinolin-derivater til behandling af latent tuberkulose
NO20082256L (no)	2008-07-15	Pyrazolderivater, preparater som inneholder slike forbindelser, og fremgangsmåter for anvendelse
DK1601363T3 (da)	2012-09-03	Anvendelse som lægemiddel af derivater af cholest-4-en-3-on, farmaceutiske sammensætninger indeholdende disse og nye derivater