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DK1296959T3 - Fremgangsmåder og præparater med anvendelse af quinazolinoner - Google Patents

Fremgangsmåder og præparater med anvendelse af quinazolinoner

Info

Publication number
DK1296959T3
DK1296959T3 DK01932769T DK01932769T DK1296959T3 DK 1296959 T3 DK1296959 T3 DK 1296959T3 DK 01932769 T DK01932769 T DK 01932769T DK 01932769 T DK01932769 T DK 01932769T DK 1296959 T3 DK1296959 T3 DK 1296959T3
Authority
DK
Denmark
Prior art keywords
quinazolinones
preparations
methods
associatged
formulae
Prior art date
Application number
DK01932769T
Other languages
English (en)
Inventor
Gustav Bergnes
David J Morgans Jr
Jeffrey T Finer
Bainian Feng
Whitney W Smith
John C Chabala
Original Assignee
Cytokinetics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cytokinetics Inc filed Critical Cytokinetics Inc
Application granted granted Critical
Publication of DK1296959T3 publication Critical patent/DK1296959T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/90—Oxygen atoms with acyclic radicals attached in position 2 or 3
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/91—Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Hospice & Palliative Care (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Paints Or Removers (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Fats And Perfumes (AREA)
  • Medicinal Preparation (AREA)
DK01932769T 2000-06-21 2001-04-27 Fremgangsmåder og præparater med anvendelse af quinazolinoner DK1296959T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US21310400P 2000-06-21 2000-06-21
US09/699,047 US6545004B1 (en) 1999-10-27 2000-10-24 Methods and compositions utilizing quinazolinones

Publications (1)

Publication Number Publication Date
DK1296959T3 true DK1296959T3 (da) 2006-07-31

Family

ID=26907773

Family Applications (1)

Application Number Title Priority Date Filing Date
DK01932769T DK1296959T3 (da) 2000-06-21 2001-04-27 Fremgangsmåder og præparater med anvendelse af quinazolinoner

Country Status (24)

Country Link
US (7) US6545004B1 (da)
EP (2) EP1296959B1 (da)
JP (1) JP4854906B2 (da)
KR (1) KR100847788B1 (da)
CN (1) CN1229353C (da)
AT (1) ATE323684T1 (da)
AU (3) AU5927001A (da)
BR (1) BR0111898A (da)
CA (1) CA2413426C (da)
CY (1) CY1105070T1 (da)
CZ (1) CZ303007B6 (da)
DE (1) DE60118921T2 (da)
DK (1) DK1296959T3 (da)
ES (1) ES2262649T3 (da)
HK (1) HK1053837A1 (da)
HU (1) HU229078B1 (da)
IL (1) IL153554A (da)
MX (1) MXPA02012627A (da)
NO (1) NO324440B1 (da)
NZ (1) NZ523233A (da)
PL (1) PL204525B1 (da)
PT (1) PT1296959E (da)
SI (1) SI1296959T1 (da)
WO (1) WO2001098278A1 (da)

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* Cited by examiner, † Cited by third party
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EP1296959A1 (en) 2003-04-02
PT1296959E (pt) 2006-07-31
PL358412A1 (en) 2004-08-09
PL204525B1 (pl) 2010-01-29
AU2006236024A1 (en) 2006-12-07
HUP0301201A3 (en) 2004-03-29
EP1707563A2 (en) 2006-10-04
AU5927001A (en) 2002-01-02
JP2004501140A (ja) 2004-01-15
EP1707563A3 (en) 2007-06-06
SI1296959T1 (sl) 2007-02-28
KR100847788B1 (ko) 2008-07-23
HK1053837A1 (en) 2003-11-07
US7105668B1 (en) 2006-09-12
DE60118921T2 (de) 2006-11-23
JP4854906B2 (ja) 2012-01-18
CA2413426C (en) 2011-01-04
NO20026172L (no) 2003-02-20
CN1437585A (zh) 2003-08-20
US6831085B1 (en) 2004-12-14
AU2001259270B2 (en) 2006-08-24
IL153554A (en) 2009-09-01
WO2001098278A1 (en) 2001-12-27
MXPA02012627A (es) 2003-09-25
US6630479B1 (en) 2003-10-07
US20040254203A1 (en) 2004-12-16
BR0111898A (pt) 2003-05-13
CZ20024178A3 (cs) 2003-05-14
NO324440B1 (no) 2007-10-15
IL153554A0 (en) 2003-07-06
ES2262649T3 (es) 2006-12-01
EP1296959B1 (en) 2006-04-19
ATE323684T1 (de) 2006-05-15
NO20026172D0 (no) 2002-12-20
KR20030047903A (ko) 2003-06-18
NZ523233A (en) 2004-10-29
US20040023996A1 (en) 2004-02-05
HU229078B1 (en) 2013-07-29
CZ303007B6 (cs) 2012-02-22
CA2413426A1 (en) 2001-12-27
US6562831B1 (en) 2003-05-13
HUP0301201A2 (hu) 2003-12-29
US6545004B1 (en) 2003-04-08
CN1229353C (zh) 2005-11-30
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CY1105070T1 (el) 2009-11-04
US7294634B2 (en) 2007-11-13

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