DE69906580D1 - Verfahren zur herstellung von 5-cyanophthalid - Google Patents

Verfahren zur herstellung von 5-cyanophthalid

Info

Publication number: DE69906580D1
Authority: DE; Germany
Prior art keywords: cyanophthalide; producing
Prior art date: 1998-12-23
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired - Lifetime

Application number

DE69906580T

Other languages

English (en)

Other versions

DE69906580T2 (de

Inventor

Hans Petersen

Nielsen Poul Dahlberg

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

H Lundbeck AS

Original Assignee

H Lundbeck AS

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-12-23

Filing date

1999-12-22

Publication date

2003-05-08

1999-12-22 Application filed by H Lundbeck AS filed Critical H Lundbeck AS

2003-05-08 Publication of DE69906580D1 publication Critical patent/DE69906580D1/de

2004-02-12 Application granted granted Critical

2004-02-12 Publication of DE69906580T2 publication Critical patent/DE69906580T2/de

2019-12-23 Anticipated expiration legal-status Critical

Status Expired - Lifetime legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Furan Compounds (AREA)

DE69906580T 1998-12-23 1999-12-22 Verfahren zur herstellung von 5-cyanophthalid Expired - Lifetime DE69906580T2 (de)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DKPA199801718		1998-12-23
DK171898		1998-12-23
PCT/DK1999/000728 WO2000039112A1 (en)	1998-12-23	1999-12-22	Method for the preparation of 5-cyanophthalide

Publications (2)

Publication Number	Publication Date
DE69906580D1 true DE69906580D1 (de)	2003-05-08
DE69906580T2 DE69906580T2 (de)	2004-02-12

Family

ID=8107494

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DE69906580T Expired - Lifetime DE69906580T2 (de)	1998-12-23	1999-12-22	Verfahren zur herstellung von 5-cyanophthalid

Country Status (31)

Country	Link
US (1)	US6392060B2 (de)
EP (1)	EP1140886B1 (de)
JP (1)	JP2002533450A (de)
KR (1)	KR100454008B1 (de)
CN (1)	CN1149208C (de)
AR (1)	AR019791A1 (de)
AT (1)	ATE236145T1 (de)
AU (1)	AU764161B2 (de)
BG (1)	BG64986B1 (de)
BR (1)	BR9916955A (de)
CA (1)	CA2356188C (de)
CZ (1)	CZ300408B6 (de)
DE (1)	DE69906580T2 (de)
DK (1)	DK1140886T3 (de)
EA (1)	EA003057B1 (de)
ES (1)	ES2195644T3 (de)
HK (1)	HK1043130B (de)
HU (1)	HUP0104856A3 (de)
IL (1)	IL143422A0 (de)
IS (1)	IS2261B (de)
IT (1)	IT1315269B1 (de)
NO (1)	NO326516B1 (de)
NZ (1)	NZ512073A (de)
PL (1)	PL203275B1 (de)
PT (1)	PT1140886E (de)
SI (1)	SI1140886T1 (de)
SK (1)	SK285530B6 (de)
TR (1)	TR200101796T2 (de)
UA (1)	UA70979C2 (de)
WO (1)	WO2000039112A1 (de)
ZA (1)	ZA200104262B (de)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JP3892667B2 (ja)	1998-10-20	2007-03-14	ハー・ルンドベック・アクチエゼルスカベット	シタロプラムの製造方法
SK285530B6 (sk)	1998-12-23	2007-03-01	H. Lundbeck A/S	Spôsob prípravy 5-kyanoftalidu
AR022329A1 (es) *	1999-01-29	2002-09-04	Lundbeck & Co As H	Metodo para la preparacion de 5-cianoftalida
CA2291129C (en)	1999-04-14	2002-10-22	H. Lundbeck A/S	Method for the preparation of citalopram
ITMI991581A1 (it) *	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
ITMI991579A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
TR200101874T1 (tr)	1999-10-25	2002-02-21	H. Lundbeck A/S	Sitalopram hazırlanması için yöntem
DE19983836C1 (de)	1999-10-25	2003-10-23	Lundbeck As Valby H	Verfahren zur Herstellung von Citalopram, 4-[1-(4- Fluorphenyl)-methanoyl]-benzonitril-Derivate und Verfahren zu deren Herstellung und deren Verwendung
AR026063A1 (es)	1999-11-01	2002-12-26	Lundbeck & Co As H	Metodo para la preparacion de 5-carboxiftalida.
CA2395404A1 (en)	1999-12-28	2001-07-05	H. Lundbeck A/S	Method for the preparation of citalopram
DK1246813T3 (da)	1999-12-30	2004-03-01	Lundbeck & Co As H	Fremgangsmåde til fremstilling af Citalopram
HUP0300343A2 (hu)	2000-01-14	2003-06-28	H. Lundbeck A/S	Eljárás 5-cianoftalid előállítására
FR2805812A1 (fr)	2000-02-24	2001-09-07	Lundbeck & Co As H	Procede de preparation du citalopram
NL1017417C1 (nl)	2000-03-03	2001-03-16	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
JP2003527385A (ja)	2000-03-13	2003-09-16	ハー・ルンドベック・アクチエゼルスカベット	５−置換された１−（４−フルオロフェニル）−１，３−ジヒドロイソベンゾフランの段階的アルキル化法
KR20020080481A (ko)	2000-03-13	2002-10-23	하. 룬트벡 아크티에 셀스카브	시탈로프람의 제조 방법
IES20010206A2 (en)	2000-03-13	2002-03-06	Lundbeck & Co As H	Method for the preparation of citalopram
AU2001239213A1 (en)	2000-03-14	2001-09-24	H Lundbeck A/S	Method for the preparation of citalopram
AT5093U1 (de) *	2000-03-16	2002-03-25	Lundbeck & Co As H	Verfahren zur herstellung von
AR032455A1 (es)	2000-05-12	2003-11-12	Lundbeck & Co As H	Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
FI20011622L (fi) *	2000-08-18	2002-02-19	Lundbeck & Co As H	Menetelmä sitalopraamin valmistamiseksi
BR0106272A (pt)	2000-12-22	2004-06-15	Lundbeck & Co As H	Processo para preparação de citalopram puro
DK1181272T3 (da)	2000-12-28	2002-12-30	Lundbeck & Co As H	Fremgangsmåde til fremstilling af rent citalopram
EP1321464A1 (de) *	2001-12-21	2003-06-25	ICROM S.p.A.	Verfahren zur Herstellung von 5-Cyanphthalid und dafür benötigte Zwischenprodeukte
CA2519629A1 (en)	2003-03-21	2004-09-30	H. Lundbeck A/S	Intermediates for the preparation of citalopram and escitalopram
AU2003223105A1 (en) *	2003-03-24	2004-10-18	Hetero Drugs Limited	Novel crystalline forms of (s)-citalopram oxalate
EP1777221A1 (de) *	2005-10-14	2007-04-25	Adorkem Technology SpA	Procédé pour la préparation du 5-cyanophtalide à partir du 5-carboxyphtalide

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1143702A (de)	1965-03-18
GB1526331A (en)	1976-01-14	1978-09-27	Kefalas As	Phthalanes
GB8419963D0 (en) *	1984-08-06	1984-09-12	Lundbeck & Co As H	Intermediate compound and method
GB8814057D0 (en)	1988-06-14	1988-07-20	Lundbeck & Co As H	New enantiomers & their isolation
DK213290D0 (da)	1990-09-06	1990-09-06	Lundbeck & Co As H	Treatment of cerebrovascular disorders
DE19626659A1 (de)	1996-07-03	1998-01-08	Basf Ag	Verfahren zur Herstellung von Phthaliden
DE19627697A1 (de)	1996-07-10	1998-01-15	Basf Ag	Verfahren zur Herstellung von Phthaliden
ZA9711376B (en)	1996-12-20	1998-07-21	Lundbeck & Co As H	Indole or dihydroindole derivatives
ES2148120T3 (es) *	1997-07-08	2002-01-16	Lundbeck & Co As H	Metodo para la preparacion de citalopram.
UA62985C2 (en)	1997-11-10	2004-01-15	Lunnbeck As H	A method for the preparation of citalopram
TR200001341T2 (tr)	1997-11-11	2000-11-21	H. Lundbeck A/S	Sitalopramın hazırlandığı metot
JP3892667B2 (ja)	1998-10-20	2007-03-14	ハー・ルンドベック・アクチエゼルスカベット	シタロプラムの製造方法
SK285530B6 (sk)	1998-12-23	2007-03-01	H. Lundbeck A/S	Spôsob prípravy 5-kyanoftalidu
AR022329A1 (es)	1999-01-29	2002-09-04	Lundbeck & Co As H	Metodo para la preparacion de 5-cianoftalida
CA2291129C (en)	1999-04-14	2002-10-22	H. Lundbeck A/S	Method for the preparation of citalopram
ITMI991579A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
ITMI991581A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
TR200101874T1 (tr)	1999-10-25	2002-02-21	H. Lundbeck A/S	Sitalopram hazırlanması için yöntem
US6310222B1 (en)	1999-11-01	2001-10-30	Sumika Fine Chemicals Co., Ltd.	Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate

1999
- 1999-12-22 SK SK896-2001A patent/SK285530B6/sk unknown
- 1999-12-22 EA EA200100696A patent/EA003057B1/ru not_active IP Right Cessation
- 1999-12-22 IL IL14342299A patent/IL143422A0/xx not_active IP Right Cessation
- 1999-12-22 PT PT99960958T patent/PT1140886E/pt unknown
- 1999-12-22 HU HU0104856A patent/HUP0104856A3/hu unknown
- 1999-12-22 ES ES99960958T patent/ES2195644T3/es not_active Expired - Lifetime
- 1999-12-22 PL PL348608A patent/PL203275B1/pl not_active IP Right Cessation
- 1999-12-22 NZ NZ512073A patent/NZ512073A/en not_active IP Right Cessation
- 1999-12-22 KR KR10-2001-7007686A patent/KR100454008B1/ko not_active IP Right Cessation
- 1999-12-22 SI SI9930278T patent/SI1140886T1/xx unknown
- 1999-12-22 TR TR2001/01796T patent/TR200101796T2/xx unknown
- 1999-12-22 CA CA002356188A patent/CA2356188C/en not_active Expired - Fee Related
- 1999-12-22 DK DK99960958T patent/DK1140886T3/da active
- 1999-12-22 WO PCT/DK1999/000728 patent/WO2000039112A1/en active IP Right Grant
- 1999-12-22 JP JP2000591023A patent/JP2002533450A/ja active Pending
- 1999-12-22 UA UA2001064498A patent/UA70979C2/uk unknown
- 1999-12-22 CZ CZ20012335A patent/CZ300408B6/cs not_active IP Right Cessation
- 1999-12-22 DE DE69906580T patent/DE69906580T2/de not_active Expired - Lifetime
- 1999-12-22 CN CNB998150002A patent/CN1149208C/zh not_active Expired - Fee Related
- 1999-12-22 EP EP99960958A patent/EP1140886B1/de not_active Expired - Lifetime
- 1999-12-22 AU AU17742/00A patent/AU764161B2/en not_active Ceased
- 1999-12-22 AT AT99960958T patent/ATE236145T1/de not_active IP Right Cessation
- 1999-12-22 BR BR9916955-0A patent/BR9916955A/pt not_active IP Right Cessation
- 1999-12-23 IT IT1999MI002696A patent/IT1315269B1/it active
- 1999-12-23 AR ARP990106726A patent/AR019791A1/es active IP Right Grant
2001
- 2001-05-22 IS IS5952A patent/IS2261B/is unknown
- 2001-05-24 ZA ZA200104262A patent/ZA200104262B/en unknown
- 2001-06-22 US US09/888,067 patent/US6392060B2/en not_active Expired - Fee Related
- 2001-06-22 NO NO20013150A patent/NO326516B1/no not_active IP Right Cessation
- 2001-06-27 BG BG105655A patent/BG64986B1/bg unknown
2002
- 2002-07-05 HK HK02105040.7A patent/HK1043130B/zh not_active IP Right Cessation

Also Published As

Publication number	Publication date
HUP0104856A2 (hu)	2002-04-29
AU1774200A (en)	2000-07-31
KR100454008B1 (ko)	2004-10-20
NO20013150L (no)	2001-08-20
KR20010082370A (ko)	2001-08-29
AU764161B2 (en)	2003-08-14
ES2195644T3 (es)	2003-12-01
ITMI992696A0 (it)	1999-12-23
HUP0104856A3 (en)	2003-01-28
DE69906580T2 (de)	2004-02-12
IL143422A0 (en)	2002-04-21
UA70979C2 (uk)	2004-11-15
IT1315269B1 (it)	2003-02-03
IS5952A (is)	2001-05-22
BG64986B1 (bg)	2006-11-30
SK285530B6 (sk)	2007-03-01
EP1140886A1 (de)	2001-10-10
TR200101796T2 (tr)	2001-11-21
BR9916955A (pt)	2001-09-11
SK8962001A3 (en)	2003-03-04
DK1140886T3 (da)	2003-07-28
AR019791A1 (es)	2002-03-13
EA200100696A1 (ru)	2001-12-24
BG105655A (en)	2002-01-31
US20020019546A1 (en)	2002-02-14
CZ300408B6 (cs)	2009-05-13
CN1149208C (zh)	2004-05-12
PL203275B1 (pl)	2009-09-30
CZ20012335A3 (cs)	2001-12-12
HK1043130A1 (en)	2002-09-06
JP2002533450A (ja)	2002-10-08
NZ512073A (en)	2003-10-31
US6392060B2 (en)	2002-05-21
WO2000039112A1 (en)	2000-07-06
CN1331686A (zh)	2002-01-16
EA003057B1 (ru)	2002-12-26
ZA200104262B (en)	2001-12-11
NO20013150D0 (no)	2001-06-22
CA2356188A1 (en)	2000-07-06
IS2261B (is)	2007-06-15
PT1140886E (pt)	2003-08-29
PL348608A1 (en)	2002-06-03
NO326516B1 (no)	2008-12-22
HK1043130B (zh)	2005-03-04
ATE236145T1 (de)	2003-04-15
SI1140886T1 (en)	2003-08-31
CA2356188C (en)	2006-05-23
EP1140886B1 (de)	2003-04-02
ITMI992696A1 (it)	2001-06-23

Publication	Publication Date	Title
ATE230738T1 (de)	2003-01-15	Verfahren zur herstellung von citalopram
ATE232524T1 (de)	2003-02-15	Verfahren zur herstellung von citalopram
ATE236145T1 (de)	2003-04-15	Verfahren zur herstellung von 5-cyanophthalid
DE69907037D1 (de)	2003-05-22	Verfahren zur herstellung von citalopram
DE69900891D1 (de)	2002-03-21	Verfahren zur herstellung von citalopram
ATE235478T1 (de)	2003-04-15	Verfahren zur herstellung von citalopram
DE60000364D1 (de)	2002-10-02	Verfahren zur herstellung von 5-cyanophthalid
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Legal Events

Date	Code	Title	Description
2004-04-29	8364	No opposition during term of opposition