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CU24406B1 - 1-{[(2s,3s,4s)-3-etil-4-fluoro-5-oxopirrolidin-2-il]metoxi}-7 -metoxiisoquinolin-6-carboxamida - Google Patents

1-{[(2s,3s,4s)-3-etil-4-fluoro-5-oxopirrolidin-2-il]metoxi}-7 -metoxiisoquinolin-6-carboxamida

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Publication number
CU24406B1
CU24406B1 CU2016000149A CU20160149A CU24406B1 CU 24406 B1 CU24406 B1 CU 24406B1 CU 2016000149 A CU2016000149 A CU 2016000149A CU 20160149 A CU20160149 A CU 20160149A CU 24406 B1 CU24406 B1 CU 24406B1
Authority
CU
Cuba
Prior art keywords
fluoro
oxopirrolidin
metoxiisoquinolin
carboxamida
metoxi
Prior art date
Application number
CU2016000149A
Other languages
English (en)
Other versions
CU20160149A7 (es
Inventor
David Randolph Anderson
Mark Edward Bunnage
Kevin Joseph Curran
Christoph Martin Dehnhardt
Lori Krim Gavrin
Joel Adam Goldberg
Seungil Han
David Hepworth
Horng-Chih Huang
Arthur Lee
Katherine Lin Lee
Frank Eldridge Lovering
Michael Dennis Lowe
John Paul Mathias
Nikolaos Papaioannou
Akshay Patny
Betsy Susan Pierce
Eddine Saiah
Joseph Walter Strohbach
John David Trzupek
Richard Vargas
Xiaolun Wang
Stephen Wayne Wright
Christoph Wolfgang Zapf
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CU20160149A7 publication Critical patent/CU20160149A7/es
Publication of CU24406B1 publication Critical patent/CU24406B1/es

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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
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Abstract

<p>Se describe el compuesto 1-{[(2S,3S,4S)-3-etil-4-fluoro-5-oxopirrolidin-2-il]metoxi}-7-metoxiisoquinolin-6-carboxamida, útil por sus propiedades antiinflamatorias.</p>
CU2016000149A 2014-04-04 2015-03-26 1-{[(2s,3s,4s)-3-etil-4-fluoro-5-oxopirrolidin-2-il]metoxi}-7 -metoxiisoquinolin-6-carboxamida CU24406B1 (es)

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