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CO4370082A1 - Procedimiento de obtencion de los compuestos 1-arilpirazoles substituidos de la formula ( i ) - Google Patents

Procedimiento de obtencion de los compuestos 1-arilpirazoles substituidos de la formula ( i )

Info

Publication number
CO4370082A1
CO4370082A1 CO94057545A CO94057545A CO4370082A1 CO 4370082 A1 CO4370082 A1 CO 4370082A1 CO 94057545 A CO94057545 A CO 94057545A CO 94057545 A CO94057545 A CO 94057545A CO 4370082 A1 CO4370082 A1 CO 4370082A1
Authority
CO
Colombia
Prior art keywords
alkyl
formula
phenyl
substituted
arylpirazoles
Prior art date
Application number
CO94057545A
Other languages
English (en)
Inventor
Joerg Stetter
Bernd Alig
Stefan Boehm
Achim Bertsch
Pieter Ooms
Christoph Erdelen
Juergen Hartwig
Ulrike Wachendorff-Neumann
Andreas Turberg
Norbert Mencke
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of CO4370082A1 publication Critical patent/CO4370082A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/30—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same unsaturated acyclic carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

1. 1-ARILPIRAZOLES SUBSTITUIDOS DE LA FORMULA GENERAL (I) EN LA QUE R1 SIGNIFICA HIDROGENO, CIANO, ALQUILO, ALCOXIAL- QUILO, ALQUILTIOALQUILO, HALOGENOALQUILO O CIANO- ALQUILO, R2 SIGNIFICA DIFLUOROETILO O TRIFLUORETILO, R3 SIGNIFICA HIDROGENO, AMINO, HALOGENO O SIGNIFI- CA UNA DE LAS AGRUPAMIENTOS SIGUIENTES DONDE R4 SIGNIFICA ALQUILO, HALOGENOALQUILO, ALCOXIAL- QUIL0 O FENILO EN CASO DADO SUBSTITUIDO, R5 SIGNI- FICA HIDROGENO O ALQUILO, R6 SIGNIFICA HIDROGENO, ALQUILO O FENILO EN CASO DADO SUBSTITUIDO Y R7 SIGNIFICA ALQUILO O R5 Y R6 JUNTO CON EL ATOMO DE CARBONO, CON EL QUE ESTAN ENLAZADOS, SIGNIFICAN UN HETEROCICLO EN CASO DADO SUBSTITUIDO, Ar SIGNIFICA FENILO O PIRIDILO EN CASO DADO SUBS- TITUIDOS Y n SIGNIFICA UNO DE LOS NUMEROS 0, 1 o 2. FIGURA 1
CO94057545A 1993-12-22 1994-12-20 Procedimiento de obtencion de los compuestos 1-arilpirazoles substituidos de la formula ( i ) CO4370082A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4343832A DE4343832A1 (de) 1993-12-22 1993-12-22 Substituierte 1-Arylpyrazole

Publications (1)

Publication Number Publication Date
CO4370082A1 true CO4370082A1 (es) 1996-10-07

Family

ID=6505768

Family Applications (1)

Application Number Title Priority Date Filing Date
CO94057545A CO4370082A1 (es) 1993-12-22 1994-12-20 Procedimiento de obtencion de los compuestos 1-arilpirazoles substituidos de la formula ( i )

Country Status (19)

Country Link
US (2) US5580843A (es)
EP (2) EP1293501B1 (es)
JP (1) JP3630458B2 (es)
CN (1) CN1061037C (es)
AT (2) ATE325792T1 (es)
AU (2) AU688401B2 (es)
BR (1) BR9405226A (es)
CA (1) CA2138452C (es)
CO (1) CO4370082A1 (es)
DE (3) DE4343832A1 (es)
DK (2) DK1293501T3 (es)
ES (2) ES2260375T3 (es)
HU (1) HU220274B (es)
NZ (1) NZ270191A (es)
PT (1) PT1293501E (es)
RU (1) RU2138485C1 (es)
TW (2) TW349843B (es)
UY (1) UY23857A1 (es)
ZA (1) ZA9410182B (es)

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JPH0987111A (ja) * 1995-09-27 1997-03-31 Sumitomo Chem Co Ltd 害虫駆除用毒餌剤
FR2739254B1 (fr) * 1995-09-29 1997-12-19 Rhone Merieux Composition antiparasitaire pour le traitement et la protection des animaux de compagnie
FR2739255B1 (fr) 1995-09-29 1998-09-04 Rhone Merieux Composition antiparasitaire pour le traitement et la protection des animaux de compagnie
TW362952B (en) 1996-01-30 1999-07-01 Takeda Chemical Industries Ltd Arylpyrazole insecticides
FR2745470B1 (fr) * 1996-03-04 1998-04-10 Rhone Poulenc Agrochimie Pyrazoles aphicides
EP0811615A1 (en) * 1996-06-03 1997-12-10 Rhone-Poulenc Agrochimie 1-Aryl-5-(substituted alkyl (thio) amido) pyrazoles and their use as pesticides
US6524603B1 (en) * 1996-07-23 2003-02-25 Rhone-Poulenc Agro Process and composition for the antiparasitic treatment of the surroundings of animals
US20050192319A1 (en) * 1996-09-19 2005-09-01 Albert Boeckh Spot-on formulations for combating parasites
EP0839809A1 (en) * 1996-11-01 1998-05-06 Rhone-Poulenc Agrochimie Pesticidal 1-arylpyrazole-5-sulfinilimine derivatives
DE19650197A1 (de) * 1996-12-04 1998-06-10 Bayer Ag 3-Thiocarbamoylpyrazol-Derivate
PL193231B1 (pl) * 1996-12-24 2007-01-31 Basf Ag Pochodna 3-acetylo-1-arylo-pirazolu i kompozycja szkodnikobójcza
ZA9711534B (en) 1996-12-24 1998-06-24 Rhone Poulenc Agrochimie Pesticidal 1-arylpyrazoles.
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US6506784B1 (en) 1999-07-01 2003-01-14 3-Dimensional Pharmaceuticals, Inc. Use of 1,3-substituted pyrazol-5-yl sulfonates as pesticides
US6409988B1 (en) 1999-07-01 2002-06-25 3-Dimensional Pharmaceuticals, Inc. Radiolabeled 1-aryl pyrazoles, the synthesis thereof and the use thereof as pest GABA receptor ligands
US6518266B1 (en) 1999-07-22 2003-02-11 3-Dimensional Pharmaceuticals 1- Aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides
FR2798042B1 (fr) * 1999-09-07 2003-04-25 Aventis Cropscience Sa Compositions insecticides dont la matiere active est de type phenyl-pyrazole et procede de lutte contre les insectes du sol
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CN1244564C (zh) * 2000-06-09 2006-03-08 拜尔农科股份有限公司 农药化合物的制备方法
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ES2515099T3 (es) * 2004-12-07 2014-10-29 Merial Limited 1-fenil-3-piperazin-pirazoles y composiciones pesticidas de los mismos
RU2312100C1 (ru) * 2006-08-28 2007-12-10 Общество с ограниченной ответственностью Научно-производственное предприятие "Ирбис" Инсектоакарицидная субстанция для борьбы с эктопаразитами собак и кошек
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IN2012DN00635A (es) 2009-07-23 2015-08-21 Bayer Cropscience Ag
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Also Published As

Publication number Publication date
AU718815B2 (en) 2000-04-20
AU688401B2 (en) 1998-03-12
ES2260375T3 (es) 2006-11-01
AU6065598A (en) 1998-06-18
DK1293501T3 (da) 2006-09-11
EP0659745A1 (de) 1995-06-28
TW349843B (en) 1999-01-11
EP1293501B1 (de) 2006-05-10
AU8043894A (en) 1995-07-06
ZA9410182B (en) 1995-08-25
USRE37495E1 (en) 2002-01-01
DE4343832A1 (de) 1995-06-29
TW520275B (en) 2003-02-11
EP1293501A1 (de) 2003-03-19
JP3630458B2 (ja) 2005-03-16
DE59410434D1 (de) 2006-06-14
DK0659745T3 (da) 2005-11-21
RU2138485C1 (ru) 1999-09-27
JPH0841031A (ja) 1996-02-13
CN1107842A (zh) 1995-09-06
PT1293501E (pt) 2006-07-31
CA2138452C (en) 2007-03-13
HU9403760D0 (en) 1995-02-28
NZ270191A (en) 1996-04-26
CN1061037C (zh) 2001-01-24
US5580843A (en) 1996-12-03
ATE300523T1 (de) 2005-08-15
DE59410411D1 (de) 2005-09-01
EP0659745B1 (de) 2005-07-27
ATE325792T1 (de) 2006-06-15
UY23857A1 (es) 1995-05-15
HUT71745A (en) 1996-01-29
RU94044348A (ru) 1996-09-27
ES2243921T3 (es) 2005-12-01
HU220274B (hu) 2001-11-28
CA2138452A1 (en) 1995-06-23
BR9405226A (pt) 1995-10-17

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