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BRPI0514076A - processo de preparação da n-aminopiperidina e de seus sais - Google Patents

processo de preparação da n-aminopiperidina e de seus sais

Info

Publication number
BRPI0514076A
BRPI0514076A BRPI0514076-5A BRPI0514076A BRPI0514076A BR PI0514076 A BRPI0514076 A BR PI0514076A BR PI0514076 A BRPI0514076 A BR PI0514076A BR PI0514076 A BRPI0514076 A BR PI0514076A
Authority
BR
Brazil
Prior art keywords
aminopiperidine
salts
preparation
preparing
formula
Prior art date
Application number
BRPI0514076-5A
Other languages
English (en)
Inventor
Pierre Jean Grossi
Raphaul Sole
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of BRPI0514076A publication Critical patent/BRPI0514076A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/28Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/28Nitrogen atoms
    • C07D295/30Nitrogen atoms non-acylated
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/92Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with a hetero atom directly attached to the ring nitrogen atom
    • C07D211/98Nitrogen atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

PROCESSO DE PREPARAçãO DA N-AMINOPIPERIDINA E DE SEUS SAIS. A presente invenção refere-se a um novo processo de preparação da N-aminopiperidina de fórmula:
BRPI0514076-5A 2004-08-05 2005-08-02 processo de preparação da n-aminopiperidina e de seus sais BRPI0514076A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0408700A FR2874013B1 (fr) 2004-08-05 2004-08-05 Procede de preparation de la n-aminopiperidine et de ses sels
PCT/FR2005/002016 WO2006024778A1 (fr) 2004-08-05 2005-08-02 Procede de preparation de la n-aminopiperedine et de ses sels

Publications (1)

Publication Number Publication Date
BRPI0514076A true BRPI0514076A (pt) 2008-05-27

Family

ID=34947045

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0514076-5A BRPI0514076A (pt) 2004-08-05 2005-08-02 processo de preparação da n-aminopiperidina e de seus sais

Country Status (16)

Country Link
US (2) US20070173648A1 (pt)
EP (1) EP1776341A1 (pt)
JP (1) JP2008509114A (pt)
KR (1) KR20070048765A (pt)
CN (1) CN101001839A (pt)
AR (1) AR050089A1 (pt)
AU (1) AU2005279087A1 (pt)
BR (1) BRPI0514076A (pt)
CA (1) CA2576718A1 (pt)
FR (1) FR2874013B1 (pt)
IL (1) IL180870A0 (pt)
MX (1) MX2007001140A (pt)
RU (1) RU2373196C2 (pt)
TW (1) TW200621713A (pt)
UY (1) UY29045A1 (pt)
WO (1) WO2006024778A1 (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2864081B1 (fr) * 2003-12-17 2006-04-28 Isochem Sa Procede de synthese de derives de cycloalkyl-hydrazines exocycliques et de derives d'heterocycloalkyl-hydrazines exocycliques.

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE338609C (de) 1919-10-15 1921-06-22 Fritz Sommer Dr Verfahren zur Darstellung von Hydrazin und dessen Alkyl- oder Arylsubstitutionsprodukten
US3317607A (en) * 1959-07-30 1967-05-02 Fmc Corp Chemical reduction of nitrosamines
DE4138142C2 (de) * 1991-11-20 1996-04-25 Cassella Ag Verfahren zur Herstellung von 1-Amino-2,6-dimethylpiperidin
US5977360A (en) * 1996-12-27 1999-11-02 Japan Hydrazine Co., Ltd. Process for producing cyclic hydrazine derivatives, tetra-hydropyridazine and hexahydropyridazine
JP4118559B2 (ja) * 2001-12-19 2008-07-16 日本曹達株式会社 脂環式ヒドラジンの製造方法
JP2004137181A (ja) * 2002-10-17 2004-05-13 Nippon Soda Co Ltd N−アミノピペリジンの製造法
JP2004137182A (ja) * 2002-10-17 2004-05-13 Nippon Soda Co Ltd N−アミノピペリジンの製造方法

Also Published As

Publication number Publication date
IL180870A0 (en) 2009-02-11
JP2008509114A (ja) 2008-03-27
RU2373196C2 (ru) 2009-11-20
UY29045A1 (es) 2006-03-31
WO2006024778A1 (fr) 2006-03-09
FR2874013B1 (fr) 2006-09-29
FR2874013A1 (fr) 2006-02-10
AR050089A1 (es) 2006-09-27
CA2576718A1 (fr) 2006-03-09
TW200621713A (en) 2006-07-01
CN101001839A (zh) 2007-07-18
KR20070048765A (ko) 2007-05-09
RU2007107806A (ru) 2008-09-10
US20070173648A1 (en) 2007-07-26
EP1776341A1 (fr) 2007-04-25
US20080306274A1 (en) 2008-12-11
AU2005279087A1 (en) 2006-03-09
US7951952B2 (en) 2011-05-31
MX2007001140A (es) 2007-04-19

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2158 DE 15/05/2012.