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WO2004037768A3 - Phenethanolamine derivatives - Google Patents

Phenethanolamine derivatives Download PDF

Info

Publication number
WO2004037768A3
WO2004037768A3 PCT/EP2003/012038 EP0312038W WO2004037768A3 WO 2004037768 A3 WO2004037768 A3 WO 2004037768A3 EP 0312038 W EP0312038 W EP 0312038W WO 2004037768 A3 WO2004037768 A3 WO 2004037768A3
Authority
WO
WIPO (PCT)
Prior art keywords
phenethanolamine derivatives
phenethanolamine
derivatives
prophylaxis
therapy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/EP2003/012038
Other languages
French (fr)
Other versions
WO2004037768A2 (en
Inventor
Philip Charles Box
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Priority to AU2003293632A priority Critical patent/AU2003293632A1/en
Publication of WO2004037768A2 publication Critical patent/WO2004037768A2/en
Publication of WO2004037768A3 publication Critical patent/WO2004037768A3/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
    • C07C217/02—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C217/04—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C217/06—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted
    • C07C217/08—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to an acyclic carbon atom
    • C07C217/10—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to an acyclic carbon atom to an acyclic carbon atom of a hydrocarbon radical containing six-membered aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)

Abstract

The present invention relates to novel compounds of formula (I), to a process for their manufacture, to pharmaceutical compositions containing them, and to their use in therapy, in particular their use in the prophylaxis and treatment of respiratory diseases.
PCT/EP2003/012038 2002-10-28 2003-10-24 Phenethanolamine derivatives Ceased WO2004037768A2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2003293632A AU2003293632A1 (en) 2002-10-28 2003-10-24 Phenethanolamine derivatives

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB0225030.6 2002-10-28
GBGB0225030.6A GB0225030D0 (en) 2002-10-28 2002-10-28 Medicinal compounds

Publications (2)

Publication Number Publication Date
WO2004037768A2 WO2004037768A2 (en) 2004-05-06
WO2004037768A3 true WO2004037768A3 (en) 2004-07-29

Family

ID=9946704

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2003/012038 Ceased WO2004037768A2 (en) 2002-10-28 2003-10-24 Phenethanolamine derivatives

Country Status (3)

Country Link
AU (1) AU2003293632A1 (en)
GB (1) GB0225030D0 (en)
WO (1) WO2004037768A2 (en)

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Also Published As

Publication number Publication date
WO2004037768A2 (en) 2004-05-06
AU2003293632A1 (en) 2004-05-13
GB0225030D0 (en) 2002-12-04
AU2003293632A8 (en) 2004-05-13

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