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UY26958A1 - Nuevos agentes anticolinérgicos que se pueden emplear como medicamentos así como procedimiento para su preparación - Google Patents

Nuevos agentes anticolinérgicos que se pueden emplear como medicamentos así como procedimiento para su preparación

Info

Publication number
UY26958A1
UY26958A1 UY26958A UY26958A UY26958A1 UY 26958 A1 UY26958 A1 UY 26958A1 UY 26958 A UY26958 A UY 26958A UY 26958 A UY26958 A UY 26958A UY 26958 A1 UY26958 A1 UY 26958A1
Authority
UY
Uruguay
Prior art keywords
procedure
preparation
well
agents
polynergic
Prior art date
Application number
UY26958A
Other languages
English (en)
Inventor
Dr Georg Speck
Dr Rolf Banholzer
Helmut Meissner
Gerd Morschhauser
Dr Michael-Paul Pieper
Dr Gerald Pohl
Dr Richard Reichl
Original Assignee
Boehringer Ingelheim Pharma
Co Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma, Co Kg filed Critical Boehringer Ingelheim Pharma
Publication of UY26958A1 publication Critical patent/UY26958A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/10—Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

El presente invento se refiere a nuevos agentes anticolinérgicos de la Fórmula general 1 en la que A, X y los radicales R1, R2, R3, R4, R5, R6 y R7 pueden tener los significados mencionados en las reivindicaciones y en la memoria descriptiva, a un procedimiento para su preparación, así como a su utilización como medicamentos.
UY26958A 2000-10-14 2001-10-10 Nuevos agentes anticolinérgicos que se pueden emplear como medicamentos así como procedimiento para su preparación UY26958A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10050994A DE10050994A1 (de) 2000-10-14 2000-10-14 Neue als Arneimittel einsetzbare Anticholinergika sowie Verfahren zu deren Herstellung

Publications (1)

Publication Number Publication Date
UY26958A1 true UY26958A1 (es) 2002-06-20

Family

ID=7659808

Family Applications (1)

Application Number Title Priority Date Filing Date
UY26958A UY26958A1 (es) 2000-10-14 2001-10-10 Nuevos agentes anticolinérgicos que se pueden emplear como medicamentos así como procedimiento para su preparación

Country Status (38)

Country Link
EP (2) EP1325001B1 (es)
JP (2) JP4109106B2 (es)
KR (1) KR100830359B1 (es)
CN (1) CN1275962C (es)
AR (1) AR035589A1 (es)
AT (1) ATE259805T1 (es)
AU (2) AU2002213975B2 (es)
BG (1) BG66225B1 (es)
BR (1) BR0114635A (es)
CA (1) CA2425557C (es)
DE (2) DE10050994A1 (es)
DK (1) DK1325001T3 (es)
EA (1) EA005816B1 (es)
EC (1) ECSP034542A (es)
EE (1) EE05179B1 (es)
ES (1) ES2215147T3 (es)
HK (1) HK1060566A1 (es)
HR (1) HRP20030278B1 (es)
HU (1) HUP0301203A3 (es)
IL (2) IL155334A0 (es)
ME (1) MEP39908A (es)
MX (1) MXPA03003160A (es)
MY (1) MY127144A (es)
NO (1) NO328207B1 (es)
NZ (1) NZ525836A (es)
PE (1) PE20020433A1 (es)
PL (1) PL207311B1 (es)
PT (1) PT1325001E (es)
RS (1) RS50464B (es)
SA (1) SA01220414B1 (es)
SI (1) SI1325001T1 (es)
SK (1) SK287138B6 (es)
TR (1) TR200400376T4 (es)
TW (1) TWI306098B (es)
UA (1) UA73804C2 (es)
UY (1) UY26958A1 (es)
WO (1) WO2002032899A1 (es)
ZA (1) ZA200302914B (es)

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Also Published As

Publication number Publication date
EP1382606A3 (de) 2004-10-13
CA2425557A1 (en) 2003-04-11
SA01220414B1 (ar) 2007-01-20
JP2004511557A (ja) 2004-04-15
EE200300151A (et) 2003-06-16
WO2002032899A1 (de) 2002-04-25
TR200400376T4 (tr) 2004-03-22
MY127144A (en) 2006-11-30
BR0114635A (pt) 2004-02-10
ZA200302914B (en) 2003-11-14
DK1325001T3 (da) 2004-06-21
BG66225B1 (bg) 2012-06-29
SI1325001T1 (en) 2004-08-31
TWI306098B (en) 2009-02-11
ATE259805T1 (de) 2004-03-15
NO20031693D0 (no) 2003-04-11
ECSP034542A (es) 2003-06-25
NO20031693L (no) 2003-05-28
PE20020433A1 (es) 2002-06-28
HRP20030278B1 (en) 2006-02-28
KR20030041165A (ko) 2003-05-23
EA005816B1 (ru) 2005-06-30
EP1382606A2 (de) 2004-01-21
HUP0301203A2 (hu) 2003-10-28
PL207311B1 (pl) 2010-11-30
CA2425557C (en) 2007-11-13
CN1468236A (zh) 2004-01-14
NO328207B1 (no) 2010-01-11
JP4109106B2 (ja) 2008-07-02
BG107688A (bg) 2003-09-30
KR100830359B1 (ko) 2008-05-20
EE05179B1 (et) 2009-06-15
AR035589A1 (es) 2004-06-16
HK1060566A1 (en) 2004-08-13
CN1275962C (zh) 2006-09-20
AU2002213975B2 (en) 2006-11-09
PT1325001E (pt) 2004-07-30
UA73804C2 (en) 2005-09-15
MEP39908A (en) 2011-02-10
RS50464B (sr) 2010-03-02
YU29503A (sh) 2006-03-03
EP1325001B1 (de) 2004-02-18
HUP0301203A3 (en) 2006-05-29
PL360673A1 (en) 2004-09-20
EP1325001A1 (de) 2003-07-09
SK4352003A3 (en) 2003-08-05
IL155334A0 (en) 2003-11-23
JP2008120834A (ja) 2008-05-29
AU1397502A (en) 2002-04-29
DE10050994A1 (de) 2002-04-18
EA200300459A1 (ru) 2003-10-30
DE50101524D1 (de) 2004-03-25
HRP20030278A2 (en) 2005-02-28
MXPA03003160A (es) 2005-09-09
SK287138B6 (sk) 2010-01-07
ES2215147T3 (es) 2004-10-01
NZ525836A (en) 2004-09-24
IL155334A (en) 2009-02-11

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