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SI1523303T1 - Zdravila, ki vsebujejo vardenafil hidroklorid trihidrat in postopki za njihovo izdelavo - Google Patents

Zdravila, ki vsebujejo vardenafil hidroklorid trihidrat in postopki za njihovo izdelavo

Info

Publication number
SI1523303T1
SI1523303T1 SI200332114T SI200332114T SI1523303T1 SI 1523303 T1 SI1523303 T1 SI 1523303T1 SI 200332114 T SI200332114 T SI 200332114T SI 200332114 T SI200332114 T SI 200332114T SI 1523303 T1 SI1523303 T1 SI 1523303T1
Authority
SI
Slovenia
Prior art keywords
manufacture
processes
medicaments containing
hydrochloride trihydrate
trihydrate
Prior art date
Application number
SI200332114T
Other languages
English (en)
Inventor
Peter Serno
Alfons Grunenberg
Andreas Ohm
Rainer Bellinghausen
Eimer Vollers
Jan-Olav Henck
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=29796385&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI1523303(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of SI1523303T1 publication Critical patent/SI1523303T1/sl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2095Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2893Tablet coating processes
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Gynecology & Obstetrics (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SI200332114T 2002-07-16 2003-07-03 Zdravila, ki vsebujejo vardenafil hidroklorid trihidrat in postopki za njihovo izdelavo SI1523303T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10232113A DE10232113A1 (de) 2002-07-16 2002-07-16 Vardenafil Hydrochlorid Trihydrat enthaltende Arzneimittel
PCT/EP2003/007093 WO2004006894A1 (de) 2002-07-16 2003-07-03 Vardenafil hydrochlorid trihydrat enthaltende arzneimittel
EP03763695A EP1523303B1 (de) 2002-07-16 2003-07-03 Vardenafil hydrochlorid trihydrat enthaltende arzneimittel und deren herstellungsverfahren

Publications (1)

Publication Number Publication Date
SI1523303T1 true SI1523303T1 (sl) 2012-06-29

Family

ID=29796385

Family Applications (2)

Application Number Title Priority Date Filing Date
SI200332508A SI2272505T1 (sl) 2002-07-16 2003-07-03 Tablete, ki vsebujejo vardenafil hidroklorid trihidrat
SI200332114T SI1523303T1 (sl) 2002-07-16 2003-07-03 Zdravila, ki vsebujejo vardenafil hidroklorid trihidrat in postopki za njihovo izdelavo

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SI200332508A SI2272505T1 (sl) 2002-07-16 2003-07-03 Tablete, ki vsebujejo vardenafil hidroklorid trihidrat

Country Status (32)

Country Link
US (2) US8273876B2 (sl)
EP (2) EP1523303B1 (sl)
JP (2) JP5173113B2 (sl)
KR (2) KR101552418B1 (sl)
CN (2) CN1681481B (sl)
AT (1) ATE538777T1 (sl)
AU (1) AU2003249942B2 (sl)
BR (1) BRPI0305559B8 (sl)
CA (2) CA2805600C (sl)
CU (1) CU23473B7 (sl)
CY (2) CY1112460T1 (sl)
DE (1) DE10232113A1 (sl)
DK (2) DK1523303T3 (sl)
EC (1) ECSP055541A (sl)
ES (2) ES2378358T3 (sl)
HK (1) HK1084019A1 (sl)
HR (3) HRP20050143B1 (sl)
HU (1) HUE032362T2 (sl)
IL (2) IL166162A (sl)
LT (1) LT2272505T (sl)
MA (1) MA27320A1 (sl)
MX (1) MXPA05000554A (sl)
NO (2) NO335434B1 (sl)
NZ (1) NZ537698A (sl)
PH (1) PH12012501171A1 (sl)
PL (1) PL223341B1 (sl)
PT (2) PT2272505T (sl)
RU (1) RU2349306C2 (sl)
SI (2) SI2272505T1 (sl)
UA (1) UA85542C2 (sl)
WO (1) WO2004006894A1 (sl)
ZA (1) ZA200500268B (sl)

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PT1174431E (pt) * 1997-11-12 2012-07-24 Bayer Pharma AG Imidazotriazinonas 2-fenil-substituídas como inibidores de fosfodiesterase
WO2002089808A1 (de) * 2001-05-09 2002-11-14 Bayer Healthcare Ag Neue verwendung von 2-phenyl-substituierten imidazotriazinonen
DE10232113A1 (de) 2002-07-16 2004-01-29 Bayer Ag Vardenafil Hydrochlorid Trihydrat enthaltende Arzneimittel
DE102004023069A1 (de) * 2004-05-11 2005-12-08 Bayer Healthcare Ag Neue Darreichungsformen des PDE 5-Inhibitors Vardenafil
DE102005001989A1 (de) * 2005-01-15 2006-07-20 Bayer Healthcare Ag Intravenöse Formulierungen von PDE-Inhibitoren
DE102005009240A1 (de) * 2005-03-01 2006-09-07 Bayer Healthcare Ag Arzneiformen mit verbesserten pharmakokinetischen Eigenschaften
DE102005009241A1 (de) * 2005-03-01 2006-09-07 Bayer Healthcare Ag Arzneiformen mit kontrollierter Bioverfügbarkeit
EP1898879A1 (en) * 2005-06-23 2008-03-19 Schering Corporation Rapidly absorbing oral formulations of pde5 inhibitors
WO2007010337A2 (de) * 2005-07-15 2007-01-25 Proxomed Medizintechnik Gmbh Verwendung von phosphodiesterase typ 5-hemmern für die prävention und behandlung von adipositas, sowie abgabesysteme für dieselben
EP1931797A2 (en) * 2005-09-29 2008-06-18 Bayer HealthCare AG Pde inhibitors and combinations thereof for the treatment of urological disorders
US7977478B2 (en) * 2006-03-13 2011-07-12 Dr. Reddy's Laboratories Limited Polymorphic forms of vardenafil
DE102007027067A1 (de) * 2007-06-12 2008-12-18 Ratiopharm Gmbh Verfahren zur Herstellung eines Arzneimittels enthaltend Vardenafil Hydrochlorid Trihydrat
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PL390079A1 (pl) 2009-12-30 2011-07-04 Zakłady Farmaceutyczne POLPHARMA Spółka Akcyjna Sposób otrzymywania wardenafilu i jego izolacji jako soli z kwasem cytrynowym oraz krystaliczna postać tej soli
CZ303877B6 (cs) 2011-11-24 2013-06-05 Zentiva, K.S. Zpusob prípravy a izolace solí vardenafilu s kyselinami
CN103372014B (zh) * 2012-04-26 2015-10-21 齐鲁制药有限公司 一种能快速溶出、稳定的盐酸伐地那非口服固体制剂及其制备方法
CZ307091B6 (cs) 2012-09-14 2018-01-10 Zentiva, K.S. Stabilní farmaceutický přípravek obsahující Vardenafil hydrochlorid
JP6594303B2 (ja) * 2013-11-19 2019-10-23 シガ・テクノロジーズ・インコーポレーテッド 微粒子化テコビリマット一水和物の再水和
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JP7336241B2 (ja) * 2019-04-02 2023-08-31 富士化学工業株式会社 バルデナフィル含有錠剤の製造方法
CN110507626B (zh) * 2019-09-19 2020-08-18 山东创新药物研发有限公司 一种稳定的盐酸伐地那非三水合物药物组合物的制备方法

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EP1523303A1 (de) 2005-04-20
CN1681481B (zh) 2010-12-15
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US20130078306A1 (en) 2013-03-28
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CN1681481A (zh) 2005-10-12
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IL166162A (en) 2014-05-28
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CN102210689B (zh) 2014-07-30
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IL232538A0 (en) 2014-06-30
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