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PT1048667E - Processo para preparacao de 8-ciclopentil-6-etil-3-(substituido)-5,8-di-hidro-4h-1,2,3a,7,8-pentaaza-as-indacenos e intermedi+arios uteis para esse fim - Google Patents

Processo para preparacao de 8-ciclopentil-6-etil-3-(substituido)-5,8-di-hidro-4h-1,2,3a,7,8-pentaaza-as-indacenos e intermedi+arios uteis para esse fim

Info

Publication number
PT1048667E
PT1048667E PT00302947T PT00302947T PT1048667E PT 1048667 E PT1048667 E PT 1048667E PT 00302947 T PT00302947 T PT 00302947T PT 00302947 T PT00302947 T PT 00302947T PT 1048667 E PT1048667 E PT 1048667E
Authority
PT
Portugal
Prior art keywords
cyclopentil
indacenes
pentaaza
dihydro
ethyl
Prior art date
Application number
PT00302947T
Other languages
English (en)
Inventor
Frank John Urban
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of PT1048667E publication Critical patent/PT1048667E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT00302947T 1999-04-30 2000-04-07 Processo para preparacao de 8-ciclopentil-6-etil-3-(substituido)-5,8-di-hidro-4h-1,2,3a,7,8-pentaaza-as-indacenos e intermedi+arios uteis para esse fim PT1048667E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US13194999P 1999-04-30 1999-04-30

Publications (1)

Publication Number Publication Date
PT1048667E true PT1048667E (pt) 2004-03-31

Family

ID=22451736

Family Applications (2)

Application Number Title Priority Date Filing Date
PT00302947T PT1048667E (pt) 1999-04-30 2000-04-07 Processo para preparacao de 8-ciclopentil-6-etil-3-(substituido)-5,8-di-hidro-4h-1,2,3a,7,8-pentaaza-as-indacenos e intermedi+arios uteis para esse fim
PT03024166T PT1380585E (pt) 1999-04-30 2000-04-07 Pirazolopiridinona como intermediario

Family Applications After (1)

Application Number Title Priority Date Filing Date
PT03024166T PT1380585E (pt) 1999-04-30 2000-04-07 Pirazolopiridinona como intermediario

Country Status (25)

Country Link
US (1) US6326495B2 (pt)
EP (1) EP1048667B1 (pt)
JP (1) JP3510560B2 (pt)
KR (1) KR100346619B1 (pt)
CN (2) CN1249064C (pt)
AR (1) AR029450A1 (pt)
AT (2) ATE282039T1 (pt)
AU (1) AU761391B2 (pt)
BR (1) BR0002070A (pt)
CA (1) CA2307080C (pt)
DE (2) DE60006026T2 (pt)
DK (2) DK1048667T3 (pt)
ES (2) ES2207464T3 (pt)
HK (2) HK1031881A1 (pt)
HU (1) HUP0001700A3 (pt)
ID (1) ID25705A (pt)
IL (1) IL135809A0 (pt)
IN (1) IN192746B (pt)
MX (1) MXPA00004214A (pt)
PL (1) PL339985A1 (pt)
PT (2) PT1048667E (pt)
RU (1) RU2189985C2 (pt)
TR (1) TR200001161A2 (pt)
TW (1) TWI256392B (pt)
ZA (1) ZA200002057B (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2287208B1 (en) 2009-08-13 2012-05-09 China Petroleum & Chemical Corporation A catalyst component for olefin polymerization and a catalyst comprising the same
TWI526421B (zh) 2010-09-08 2016-03-21 住友化學股份有限公司 製造嗒酮化合物的方法及其中間物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR9406946A (pt) 1993-07-06 1996-08-06 Pfizer Tetra-hidro-pirazolpiridinas bicíclicas
HUT77517A (hu) 1994-10-20 1998-05-28 Pfizer Inc. Biciklusos tetrahidro-pirazolo-piridin-származékok, alkalmazásuk és ilyen vegyületeket tartalmazó gyógyászati készítmények
DK0837860T3 (da) 1995-06-06 2002-05-27 Pfizer Tricykliske 5,6-dihydro-9H-pyrazolo[3,4-c]-1,2,4-triazolo-[4,3-alfa]pyridiner

Also Published As

Publication number Publication date
AR029450A1 (es) 2003-07-02
ID25705A (id) 2000-11-02
HU0001700D0 (en) 2000-07-28
CA2307080A1 (en) 2000-10-30
CA2307080C (en) 2003-12-23
AU761391B2 (en) 2003-06-05
ATE282039T1 (de) 2004-11-15
US20010039347A1 (en) 2001-11-08
IN192746B (pt) 2004-05-15
DK1380585T3 (da) 2005-03-07
ATE252582T1 (de) 2003-11-15
AU3018000A (en) 2000-11-02
ZA200002057B (en) 2001-10-26
DE60015819D1 (de) 2004-12-16
EP1048667A1 (en) 2000-11-02
US6326495B2 (en) 2001-12-04
CN1274724A (zh) 2000-11-29
HK1031881A1 (en) 2001-06-29
HK1062678A1 (en) 2004-11-19
PT1380585E (pt) 2005-03-31
EP1048667B1 (en) 2003-10-22
HUP0001700A2 (en) 2001-03-28
DE60006026D1 (de) 2003-11-27
CN1478779A (zh) 2004-03-03
RU2189985C2 (ru) 2002-09-27
ES2232805T3 (es) 2005-06-01
JP2000344771A (ja) 2000-12-12
CN1160353C (zh) 2004-08-04
KR100346619B1 (ko) 2002-07-26
CN1249064C (zh) 2006-04-05
HUP0001700A3 (en) 2001-05-28
DE60015819T2 (de) 2005-12-08
BR0002070A (pt) 2000-10-31
JP3510560B2 (ja) 2004-03-29
ES2207464T3 (es) 2004-06-01
IL135809A0 (en) 2001-05-20
TWI256392B (en) 2006-06-11
DK1048667T3 (da) 2004-03-01
KR20010029673A (ko) 2001-04-06
PL339985A1 (en) 2000-11-06
DE60006026T2 (de) 2004-06-17
TR200001161A2 (tr) 2000-12-21
MXPA00004214A (es) 2002-03-08

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